Index by author
July 01, 2005; Volume 33,Issue 7
A
Adelsberger, Jennifer
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Annaert, Pieter
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
B
Baillie, Thomas A.
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Barama, Azemi
- You have accessCYP3A5 GENETIC POLYMORPHISMS IN DIFFERENT ETHNIC POPULATIONSJean-Nicholas Roy, Julie Lajoie, Lynn S. Zijenah, Azemi Barama, Charles Poirier, Brian J. Ward and Michel RogerDrug Metabolism and Disposition July 2005, 33 (7) 884-887; DOI: https://doi.org/10.1124/dmd.105.003822
Baumann, Frank
- You have accessSYNTHESIS AND CHARACTERIZATION OF SOME NEW PHASE II METABOLITES OF THE ALKYLATOR BENDAMUSTINE AND THEIR IDENTIFICATION IN HUMAN BILE, URINE, AND PLASMA FROM PATIENTS WITH CHOLANGIOCARCINOMAJens Teichert, Reinhard Sohr, Frank Baumann, Lothar Hennig, Karlheinz Merkle, Karel Caca and Rainer PreissDrug Metabolism and Disposition July 2005, 33 (7) 984-992; DOI: https://doi.org/10.1124/dmd.105.003624
Beijnen, Jos H.
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
Benlhabib, E.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Bigler, Jeannette
- You have accessGLUCURONIDATION OF NONSTEROIDAL ANTI-INFLAMMATORY DRUGS: IDENTIFYING THE ENZYMES RESPONSIBLE IN HUMAN LIVER MICROSOMESGwendolyn E. Kuehl, Johanna W. Lampe, John D. Potter and Jeannette BiglerDrug Metabolism and Disposition July 2005, 33 (7) 1027-1035; DOI: https://doi.org/10.1124/dmd.104.002527
Blough, David
- You have accessCONTRIBUTION OF CYP3A5 TO HEPATIC AND RENAL IFOSFAMIDE N-DECHLOROETHYLATIONJeannine S. McCune, Linda J. Risler, Brian R. Phillips, Kenneth E. Thummel, David Blough and Danny D. ShenDrug Metabolism and Disposition July 2005, 33 (7) 1074-1081; DOI: https://doi.org/10.1124/dmd.104.002279
Boothe-Genthe, Catherine
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Borges, Silvana
- You have accessDEXTROMETHORPHAN TO DEXTRORPHAN URINARY METABOLIC RATIO DOES NOT REFLECT DEXTROMETHORPHAN ORAL CLEARANCESilvana Borges, Lang Li, Mitchell A. Hamman, David R. Jones, Stephen D. Hall and J. Christopher GorskiDrug Metabolism and Disposition July 2005, 33 (7) 1052-1055; DOI: https://doi.org/10.1124/dmd.104.003459
Bratton, Stacie
- You have accessLITHOCHOLIC ACID DECREASES EXPRESSION OF UGT2B7 IN CACO-2 CELLS: A POTENTIAL ROLE FOR A NEGATIVE FARNESOID X RECEPTOR RESPONSE ELEMENTYuan Lu, Jean-Marie Heydel, Xin Li, Stacie Bratton, Tim Lindblom and Anna Radominska-PandyaDrug Metabolism and Disposition July 2005, 33 (7) 937-946; DOI: https://doi.org/10.1124/dmd.104.003061
Brown, Cheri M.
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Brunner, Janice
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
C
Caca, Karel
- You have accessSYNTHESIS AND CHARACTERIZATION OF SOME NEW PHASE II METABOLITES OF THE ALKYLATOR BENDAMUSTINE AND THEIR IDENTIFICATION IN HUMAN BILE, URINE, AND PLASMA FROM PATIENTS WITH CHOLANGIOCARCINOMAJens Teichert, Reinhard Sohr, Frank Baumann, Lothar Hennig, Karlheinz Merkle, Karel Caca and Rainer PreissDrug Metabolism and Disposition July 2005, 33 (7) 984-992; DOI: https://doi.org/10.1124/dmd.105.003624
Caldwell, Stuart T.
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
Carlini, Edward
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Cascorbi, Ingolf
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
Catania, Viviana A.
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
Chen, Chuan
- You have accessTISSUE DISTRIBUTION AND ONTOGENY OF MOUSE ORGANIC ANION TRANSPORTING POLYPEPTIDES (OATPS)Xingguo Cheng, Jonathan Maher, Chuan Chen and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 1062-1073; DOI: https://doi.org/10.1124/dmd.105.003640
Cheng, Xingguo
- You have accessTISSUE DISTRIBUTION AND ONTOGENY OF MOUSE ORGANIC ANION TRANSPORTING POLYPEPTIDES (OATPS)Xingguo Cheng, Jonathan Maher, Chuan Chen and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 1062-1073; DOI: https://doi.org/10.1124/dmd.105.003640
- You have accessTISSUE DISTRIBUTION AND HEPATIC AND RENAL ONTOGENY OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) FAMILY IN MICEJonathan M. Maher, Angela L. Slitt, Nathan J. Cherrington, Xingguo Cheng and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 947-955; DOI: https://doi.org/10.1124/dmd.105.003780
- You have accessINDUCTION OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN FAMILY OF TRANSPORTERS BY CHEMICAL ACTIVATORS OF RECEPTOR-MEDIATED PATHWAYS IN MOUSE LIVERJonathan M. Maher, Xingguo Cheng, Angela L. Slitt, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 956-962; DOI: https://doi.org/10.1124/dmd.105.003798
Cherrington, Nathan J.
- You have accessTISSUE DISTRIBUTION AND HEPATIC AND RENAL ONTOGENY OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) FAMILY IN MICEJonathan M. Maher, Angela L. Slitt, Nathan J. Cherrington, Xingguo Cheng and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 947-955; DOI: https://doi.org/10.1124/dmd.105.003780
Chiba, Kan
- You have accessIDENTIFICATION OF HMG-CoA REDUCTASE INHIBITORS AS ACTIVATORS FOR HUMAN, MOUSE AND RAT CONSTITUTIVE ANDROSTANE RECEPTORKaoru Kobayashi, Yosuke Yamanaka, Norihiko Iwazaki, Ikumi Nakajo, Masakiyo Hosokawa, Masahiko Negishi and Kan ChibaDrug Metabolism and Disposition July 2005, 33 (7) 924-929; DOI: https://doi.org/10.1124/dmd.104.002741
Ciecko, Patrice
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Crocenzi, Fernando A.
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
Crozier, Alan
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
D
D'Andrea, Vanesa
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
Dieter, Matthew Z.
- You have accessINDUCTION OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN FAMILY OF TRANSPORTERS BY CHEMICAL ACTIVATORS OF RECEPTOR-MEDIATED PATHWAYS IN MOUSE LIVERJonathan M. Maher, Xingguo Cheng, Angela L. Slitt, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 956-962; DOI: https://doi.org/10.1124/dmd.105.003798
Dong, Junxing
- You have accessMETABOLIC PROFILE OF 1,5-DICAFFEOYLQUINIC ACID IN RATS, AN IN VIVO AND IN VITRO STUDYBo Yang, Zhiyun Meng, Junxing Dong, Liangping Yan, Libo Zou, Zhongming Tang and Guifang DouDrug Metabolism and Disposition July 2005, 33 (7) 930-936; DOI: https://doi.org/10.1124/dmd.104.002154
Dou, Guifang
- You have accessMETABOLIC PROFILE OF 1,5-DICAFFEOYLQUINIC ACID IN RATS, AN IN VIVO AND IN VITRO STUDYBo Yang, Zhiyun Meng, Junxing Dong, Liangping Yan, Libo Zou, Zhongming Tang and Guifang DouDrug Metabolism and Disposition July 2005, 33 (7) 930-936; DOI: https://doi.org/10.1124/dmd.104.002154
Duthie, Garry G.
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
E
Edwards, Christine A.
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
Evans, Ronald M.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
F
Finel, Moshe
- You have accessKINETIC CHARACTERIZATION OF THE 1A SUBFAMILY OF RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESLeena Luukkanen, Jyrki Taskinen, Mika Kurkela, Risto Kostiainen, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition July 2005, 33 (7) 1017-1026; DOI: https://doi.org/10.1124/dmd.105.004093
Fuller, S.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Fusch, Christoph
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
Fuse, Eiichi
- You have accessP-GLYCOPROTEIN PLAYS A MAJOR ROLE IN THE EFFLUX OF FEXOFENADINE IN THE SMALL INTESTINE AND BLOOD-BRAIN BARRIER, BUT ONLY A LIMITED ROLE IN ITS BILIARY EXCRETIONHarunobu Tahara, Hiroyuki Kusuhara, Eiichi Fuse and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 963-968; DOI: https://doi.org/10.1124/dmd.105.004192
G
Gibson, Christopher R.
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Gorski, J. Christopher
- You have accessDEXTROMETHORPHAN TO DEXTRORPHAN URINARY METABOLIC RATIO DOES NOT REFLECT DEXTROMETHORPHAN ORAL CLEARANCESilvana Borges, Lang Li, Mitchell A. Hamman, David R. Jones, Stephen D. Hall and J. Christopher GorskiDrug Metabolism and Disposition July 2005, 33 (7) 1052-1055; DOI: https://doi.org/10.1124/dmd.104.003459
Gotoh, Yukiko
- You have accessREGULATION OF THE CELL SURFACE EXPRESSION OF HUMAN BCRP/ABCG2 BY THE PHOSPHORYLATION STATE OF AKT IN POLARIZED CELLSTappei Takada, Hiroshi Suzuki, Yukiko Gotoh and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 905-909; DOI: https://doi.org/10.1124/dmd.104.003228
Graf, Brigitte A.
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
Gräter, Frauke
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Gratz, Matthias
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
H
Haenisch, Sierk
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
Hall, Stephen D.
- You have accessDEXTROMETHORPHAN TO DEXTRORPHAN URINARY METABOLIC RATIO DOES NOT REFLECT DEXTROMETHORPHAN ORAL CLEARANCESilvana Borges, Lang Li, Mitchell A. Hamman, David R. Jones, Stephen D. Hall and J. Christopher GorskiDrug Metabolism and Disposition July 2005, 33 (7) 1052-1055; DOI: https://doi.org/10.1124/dmd.104.003459
Halpert, James R.
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Hamman, Mitchell A.
- You have accessDEXTROMETHORPHAN TO DEXTRORPHAN URINARY METABOLIC RATIO DOES NOT REFLECT DEXTROMETHORPHAN ORAL CLEARANCESilvana Borges, Lang Li, Mitchell A. Hamman, David R. Jones, Stephen D. Hall and J. Christopher GorskiDrug Metabolism and Disposition July 2005, 33 (7) 1052-1055; DOI: https://doi.org/10.1124/dmd.104.003459
Hartley, Richard C.
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
Hendrickx, Jan
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
Hennig, Lothar
- You have accessSYNTHESIS AND CHARACTERIZATION OF SOME NEW PHASE II METABOLITES OF THE ALKYLATOR BENDAMUSTINE AND THEIR IDENTIFICATION IN HUMAN BILE, URINE, AND PLASMA FROM PATIENTS WITH CHOLANGIOCARCINOMAJens Teichert, Reinhard Sohr, Frank Baumann, Lothar Hennig, Karlheinz Merkle, Karel Caca and Rainer PreissDrug Metabolism and Disposition July 2005, 33 (7) 984-992; DOI: https://doi.org/10.1124/dmd.105.003624
Heydel, Jean-Marie
- You have accessLITHOCHOLIC ACID DECREASES EXPRESSION OF UGT2B7 IN CACO-2 CELLS: A POTENTIAL ROLE FOR A NEGATIVE FARNESOID X RECEPTOR RESPONSE ELEMENTYuan Lu, Jean-Marie Heydel, Xin Li, Stacie Bratton, Tim Lindblom and Anna Radominska-PandyaDrug Metabolism and Disposition July 2005, 33 (7) 937-946; DOI: https://doi.org/10.1124/dmd.104.003061
Hirvonen, Jouni
- You have accessKINETIC CHARACTERIZATION OF THE 1A SUBFAMILY OF RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESLeena Luukkanen, Jyrki Taskinen, Mika Kurkela, Risto Kostiainen, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition July 2005, 33 (7) 1017-1026; DOI: https://doi.org/10.1124/dmd.105.004093
Hosokawa, Masakiyo
- You have accessIDENTIFICATION OF HMG-CoA REDUCTASE INHIBITORS AS ACTIVATORS FOR HUMAN, MOUSE AND RAT CONSTITUTIVE ANDROSTANE RECEPTORKaoru Kobayashi, Yosuke Yamanaka, Norihiko Iwazaki, Ikumi Nakajo, Masakiyo Hosokawa, Masahiko Negishi and Kan ChibaDrug Metabolism and Disposition July 2005, 33 (7) 924-929; DOI: https://doi.org/10.1124/dmd.104.002741
I
Iwazaki, Norihiko
- You have accessIDENTIFICATION OF HMG-CoA REDUCTASE INHIBITORS AS ACTIVATORS FOR HUMAN, MOUSE AND RAT CONSTITUTIVE ANDROSTANE RECEPTORKaoru Kobayashi, Yosuke Yamanaka, Norihiko Iwazaki, Ikumi Nakajo, Masakiyo Hosokawa, Masahiko Negishi and Kan ChibaDrug Metabolism and Disposition July 2005, 33 (7) 924-929; DOI: https://doi.org/10.1124/dmd.104.002741
J
Jacobs, Judith M.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Jedlitschky, Gabriele
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
Jiang, Hualiang
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Jones, David R.
- You have accessDEXTROMETHORPHAN TO DEXTRORPHAN URINARY METABOLIC RATIO DOES NOT REFLECT DEXTROMETHORPHAN ORAL CLEARANCESilvana Borges, Lang Li, Mitchell A. Hamman, David R. Jones, Stephen D. Hall and J. Christopher GorskiDrug Metabolism and Disposition July 2005, 33 (7) 1052-1055; DOI: https://doi.org/10.1124/dmd.104.003459
K
Kamel, Amin
- You have accessCHARACTERIZATION OF A NOVEL METABOLITE INTERMEDIATE OF ZIPRASIDONE IN HEPATIC CYTOSOLIC FRACTIONS OF RAT, DOG, AND HUMAN BY ESI-MS/MS, HYDROGEN/DEUTERIUM EXCHANGE, AND CHEMICAL DERIVATIZATIONZhuang Miao, Amin Kamel and Chandra PrakashDrug Metabolism and Disposition July 2005, 33 (7) 879-883; DOI: https://doi.org/10.1124/dmd.105.004036
Keyler, D. E.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Klaassen, Curtis D.
- You have accessTISSUE DISTRIBUTION AND ONTOGENY OF MOUSE ORGANIC ANION TRANSPORTING POLYPEPTIDES (OATPS)Xingguo Cheng, Jonathan Maher, Chuan Chen and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 1062-1073; DOI: https://doi.org/10.1124/dmd.105.003640
- You have accessTISSUE DISTRIBUTION AND HEPATIC AND RENAL ONTOGENY OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) FAMILY IN MICEJonathan M. Maher, Angela L. Slitt, Nathan J. Cherrington, Xingguo Cheng and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 947-955; DOI: https://doi.org/10.1124/dmd.105.003780
- You have accessINDUCTION OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN FAMILY OF TRANSPORTERS BY CHEMICAL ACTIVATORS OF RECEPTOR-MEDIATED PATHWAYS IN MOUSE LIVERJonathan M. Maher, Xingguo Cheng, Angela L. Slitt, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 956-962; DOI: https://doi.org/10.1124/dmd.105.003798
Kobayashi, Kaoru
- You have accessIDENTIFICATION OF HMG-CoA REDUCTASE INHIBITORS AS ACTIVATORS FOR HUMAN, MOUSE AND RAT CONSTITUTIVE ANDROSTANE RECEPTORKaoru Kobayashi, Yosuke Yamanaka, Norihiko Iwazaki, Ikumi Nakajo, Masakiyo Hosokawa, Masahiko Negishi and Kan ChibaDrug Metabolism and Disposition July 2005, 33 (7) 924-929; DOI: https://doi.org/10.1124/dmd.104.002741
Kostiainen, Risto
- You have accessKINETIC CHARACTERIZATION OF THE 1A SUBFAMILY OF RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESLeena Luukkanen, Jyrki Taskinen, Mika Kurkela, Risto Kostiainen, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition July 2005, 33 (7) 1017-1026; DOI: https://doi.org/10.1124/dmd.105.004093
Kostrubsky, Vsevolod E.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Kroemer, Heyo K.
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
Krolikowski, Paul
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Kuehl, Gwendolyn E.
- You have accessGLUCURONIDATION OF NONSTEROIDAL ANTI-INFLAMMATORY DRUGS: IDENTIFYING THE ENZYMES RESPONSIBLE IN HUMAN LIVER MICROSOMESGwendolyn E. Kuehl, Johanna W. Lampe, John D. Potter and Jeannette BiglerDrug Metabolism and Disposition July 2005, 33 (7) 1027-1035; DOI: https://doi.org/10.1124/dmd.104.002527
Kurkela, Mika
- You have accessKINETIC CHARACTERIZATION OF THE 1A SUBFAMILY OF RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESLeena Luukkanen, Jyrki Taskinen, Mika Kurkela, Risto Kostiainen, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition July 2005, 33 (7) 1017-1026; DOI: https://doi.org/10.1124/dmd.105.004093
Kusuhara, Hiroyuki
- You have accessP-GLYCOPROTEIN PLAYS A MAJOR ROLE IN THE EFFLUX OF FEXOFENADINE IN THE SMALL INTESTINE AND BLOOD-BRAIN BARRIER, BUT ONLY A LIMITED ROLE IN ITS BILIARY EXCRETIONHarunobu Tahara, Hiroyuki Kusuhara, Eiichi Fuse and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 963-968; DOI: https://doi.org/10.1124/dmd.105.004192
L
Lajoie, Julie
- You have accessCYP3A5 GENETIC POLYMORPHISMS IN DIFFERENT ETHNIC POPULATIONSJean-Nicholas Roy, Julie Lajoie, Lynn S. Zijenah, Azemi Barama, Charles Poirier, Brian J. Ward and Michel RogerDrug Metabolism and Disposition July 2005, 33 (7) 884-887; DOI: https://doi.org/10.1124/dmd.105.003822
Lampe, Johanna W.
- You have accessGLUCURONIDATION OF NONSTEROIDAL ANTI-INFLAMMATORY DRUGS: IDENTIFYING THE ENZYMES RESPONSIBLE IN HUMAN LIVER MICROSOMESGwendolyn E. Kuehl, Johanna W. Lampe, John D. Potter and Jeannette BiglerDrug Metabolism and Disposition July 2005, 33 (7) 1027-1035; DOI: https://doi.org/10.1124/dmd.104.002527
Le, C. T.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Lean, Michael E. J.
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
LeSage, M. G.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Li, Lang
- You have accessDEXTROMETHORPHAN TO DEXTRORPHAN URINARY METABOLIC RATIO DOES NOT REFLECT DEXTROMETHORPHAN ORAL CLEARANCESilvana Borges, Lang Li, Mitchell A. Hamman, David R. Jones, Stephen D. Hall and J. Christopher GorskiDrug Metabolism and Disposition July 2005, 33 (7) 1052-1055; DOI: https://doi.org/10.1124/dmd.104.003459
Li, Weihua
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Li, Xin
- You have accessLITHOCHOLIC ACID DECREASES EXPRESSION OF UGT2B7 IN CACO-2 CELLS: A POTENTIAL ROLE FOR A NEGATIVE FARNESOID X RECEPTOR RESPONSE ELEMENTYuan Lu, Jean-Marie Heydel, Xin Li, Stacie Bratton, Tim Lindblom and Anna Radominska-PandyaDrug Metabolism and Disposition July 2005, 33 (7) 937-946; DOI: https://doi.org/10.1124/dmd.104.003061
Lin, Charles
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Lindblom, Tim
- You have accessLITHOCHOLIC ACID DECREASES EXPRESSION OF UGT2B7 IN CACO-2 CELLS: A POTENTIAL ROLE FOR A NEGATIVE FARNESOID X RECEPTOR RESPONSE ELEMENTYuan Lu, Jean-Marie Heydel, Xin Li, Stacie Bratton, Tim Lindblom and Anna Radominska-PandyaDrug Metabolism and Disposition July 2005, 33 (7) 937-946; DOI: https://doi.org/10.1124/dmd.104.003061
Linnemann, Knud
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
Liu, Hong
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Locuson, Charles W.
- You have accessTHREE-DIMENSIONAL QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP ANALYSIS OF CYTOCHROMES P450: EFFECT OF INCORPORATING HIGHER-AFFINITY LIGANDS AND POTENTIAL NEW APPLICATIONSCharles W. Locuson and Jan L. WahlstromDrug Metabolism and Disposition July 2005, 33 (7) 873-878; DOI: https://doi.org/10.1124/dmd.105.004325
Lu, Yuan
- You have accessLITHOCHOLIC ACID DECREASES EXPRESSION OF UGT2B7 IN CACO-2 CELLS: A POTENTIAL ROLE FOR A NEGATIVE FARNESOID X RECEPTOR RESPONSE ELEMENTYuan Lu, Jean-Marie Heydel, Xin Li, Stacie Bratton, Tim Lindblom and Anna Radominska-PandyaDrug Metabolism and Disposition July 2005, 33 (7) 937-946; DOI: https://doi.org/10.1124/dmd.104.003061
Luo, Xiaoming
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Luquita, Marcelo G.
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
Luu, Minh
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Luukkanen, Leena
- You have accessKINETIC CHARACTERIZATION OF THE 1A SUBFAMILY OF RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESLeena Luukkanen, Jyrki Taskinen, Mika Kurkela, Risto Kostiainen, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition July 2005, 33 (7) 1017-1026; DOI: https://doi.org/10.1124/dmd.105.004093
M
Maher, Jonathan
- You have accessTISSUE DISTRIBUTION AND ONTOGENY OF MOUSE ORGANIC ANION TRANSPORTING POLYPEPTIDES (OATPS)Xingguo Cheng, Jonathan Maher, Chuan Chen and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 1062-1073; DOI: https://doi.org/10.1124/dmd.105.003640
Maher, Jonathan M.
- You have accessTISSUE DISTRIBUTION AND HEPATIC AND RENAL ONTOGENY OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) FAMILY IN MICEJonathan M. Maher, Angela L. Slitt, Nathan J. Cherrington, Xingguo Cheng and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 947-955; DOI: https://doi.org/10.1124/dmd.105.003780
- You have accessINDUCTION OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN FAMILY OF TRANSPORTERS BY CHEMICAL ACTIVATORS OF RECEPTOR-MEDIATED PATHWAYS IN MOUSE LIVERJonathan M. Maher, Xingguo Cheng, Angela L. Slitt, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 956-962; DOI: https://doi.org/10.1124/dmd.105.003798
Mannens, Geert
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
McCune, Jeannine S.
- You have accessCONTRIBUTION OF CYP3A5 TO HEPATIC AND RENAL IFOSFAMIDE N-DECHLOROETHYLATIONJeannine S. McCune, Linda J. Risler, Brian R. Phillips, Kenneth E. Thummel, David Blough and Danny D. ShenDrug Metabolism and Disposition July 2005, 33 (7) 1074-1081; DOI: https://doi.org/10.1124/dmd.104.002279
Meng, Zhiyun
- You have accessMETABOLIC PROFILE OF 1,5-DICAFFEOYLQUINIC ACID IN RATS, AN IN VIVO AND IN VITRO STUDYBo Yang, Zhiyun Meng, Junxing Dong, Liangping Yan, Libo Zou, Zhongming Tang and Guifang DouDrug Metabolism and Disposition July 2005, 33 (7) 930-936; DOI: https://doi.org/10.1124/dmd.104.002154
Merkle, Karlheinz
- You have accessSYNTHESIS AND CHARACTERIZATION OF SOME NEW PHASE II METABOLITES OF THE ALKYLATOR BENDAMUSTINE AND THEIR IDENTIFICATION IN HUMAN BILE, URINE, AND PLASMA FROM PATIENTS WITH CHOLANGIOCARCINOMAJens Teichert, Reinhard Sohr, Frank Baumann, Lothar Hennig, Karlheinz Merkle, Karel Caca and Rainer PreissDrug Metabolism and Disposition July 2005, 33 (7) 984-992; DOI: https://doi.org/10.1124/dmd.105.003624
Meuldermans, Willem
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
Meyer zu Schwabedissen, Henriette E.
- You have accessVARIABLE EXPRESSION OF MRP2 (ABCC2) IN HUMAN PLACENTA: INFLUENCE OF GESTATIONAL AGE AND CELLULAR DIFFERENTIATIONHenriette E. Meyer zu Schwabedissen, Gabriele Jedlitschky, Matthias Gratz, Sierk Haenisch, Knud Linnemann, Christoph Fusch, Ingolf Cascorbi and Heyo K. KroemerDrug Metabolism and Disposition July 2005, 33 (7) 896-904; DOI: https://doi.org/10.1124/dmd.104.003335
Miao, Zhuang
- You have accessCHARACTERIZATION OF A NOVEL METABOLITE INTERMEDIATE OF ZIPRASIDONE IN HEPATIC CYTOSOLIC FRACTIONS OF RAT, DOG, AND HUMAN BY ESI-MS/MS, HYDROGEN/DEUTERIUM EXCHANGE, AND CHEMICAL DERIVATIZATIONZhuang Miao, Amin Kamel and Chandra PrakashDrug Metabolism and Disposition July 2005, 33 (7) 879-883; DOI: https://doi.org/10.1124/dmd.105.004036
Michael, Aimee
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Michel, Kimberly
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Mohutsky, Michael A.
- You have accessTHE USE OF A SUBSTRATE CASSETTE STRATEGY TO IMPROVE THE CAPACITY AND THROUGHPUT OF CYTOCHROME P450 INDUCTION STUDIES IN HUMAN HEPATOCYTESMichael A. Mohutsky, David M. Petullo and Steven A. WrightonDrug Metabolism and Disposition July 2005, 33 (7) 920-923; DOI: https://doi.org/10.1124/dmd.105.004291
Mottino, Aldo D.
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
Mullen, William
- You have accessDISPOSITION AND METABOLISM OF [2-14C]QUERCETIN-4′-GLUCOSIDE IN RATSBrigitte A. Graf, William Mullen, Stuart T. Caldwell, Richard C. Hartley, Garry G. Duthie, Michael E. J. Lean, Alan Crozier and Christine A. EdwardsDrug Metabolism and Disposition July 2005, 33 (7) 1036-1043; DOI: https://doi.org/10.1124/dmd.104.002691
N
Nakajo, Ikumi
- You have accessIDENTIFICATION OF HMG-CoA REDUCTASE INHIBITORS AS ACTIVATORS FOR HUMAN, MOUSE AND RAT CONSTITUTIVE ANDROSTANE RECEPTORKaoru Kobayashi, Yosuke Yamanaka, Norihiko Iwazaki, Ikumi Nakajo, Masakiyo Hosokawa, Masahiko Negishi and Kan ChibaDrug Metabolism and Disposition July 2005, 33 (7) 924-929; DOI: https://doi.org/10.1124/dmd.104.002741
Negishi, Masahiko
- You have accessIDENTIFICATION OF HMG-CoA REDUCTASE INHIBITORS AS ACTIVATORS FOR HUMAN, MOUSE AND RAT CONSTITUTIVE ANDROSTANE RECEPTORKaoru Kobayashi, Yosuke Yamanaka, Norihiko Iwazaki, Ikumi Nakajo, Masakiyo Hosokawa, Masahiko Negishi and Kan ChibaDrug Metabolism and Disposition July 2005, 33 (7) 924-929; DOI: https://doi.org/10.1124/dmd.104.002741
Nichols, Ralph C.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Noreault, Trisha L.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Noukens, Jan
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
O
Ochoa, J. Elena
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
P
Parikh, Mona
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Pellegrino, José M.
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
Pentel, P. R.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Petullo, David M.
- You have accessTHE USE OF A SUBSTRATE CASSETTE STRATEGY TO IMPROVE THE CAPACITY AND THROUGHPUT OF CYTOCHROME P450 INDUCTION STUDIES IN HUMAN HEPATOCYTESMichael A. Mohutsky, David M. Petullo and Steven A. WrightonDrug Metabolism and Disposition July 2005, 33 (7) 920-923; DOI: https://doi.org/10.1124/dmd.105.004291
Phillips, Brian R.
- You have accessCONTRIBUTION OF CYP3A5 TO HEPATIC AND RENAL IFOSFAMIDE N-DECHLOROETHYLATIONJeannine S. McCune, Linda J. Risler, Brian R. Phillips, Kenneth E. Thummel, David Blough and Danny D. ShenDrug Metabolism and Disposition July 2005, 33 (7) 1074-1081; DOI: https://doi.org/10.1124/dmd.104.002279
Poirier, Charles
- You have accessCYP3A5 GENETIC POLYMORPHISMS IN DIFFERENT ETHNIC POPULATIONSJean-Nicholas Roy, Julie Lajoie, Lynn S. Zijenah, Azemi Barama, Charles Poirier, Brian J. Ward and Michel RogerDrug Metabolism and Disposition July 2005, 33 (7) 884-887; DOI: https://doi.org/10.1124/dmd.105.003822
Potter, John D.
- You have accessGLUCURONIDATION OF NONSTEROIDAL ANTI-INFLAMMATORY DRUGS: IDENTIFYING THE ENZYMES RESPONSIBLE IN HUMAN LIVER MICROSOMESGwendolyn E. Kuehl, Johanna W. Lampe, John D. Potter and Jeannette BiglerDrug Metabolism and Disposition July 2005, 33 (7) 1027-1035; DOI: https://doi.org/10.1124/dmd.104.002527
Prakash, Chandra
- You have accessCHARACTERIZATION OF A NOVEL METABOLITE INTERMEDIATE OF ZIPRASIDONE IN HEPATIC CYTOSOLIC FRACTIONS OF RAT, DOG, AND HUMAN BY ESI-MS/MS, HYDROGEN/DEUTERIUM EXCHANGE, AND CHEMICAL DERIVATIZATIONZhuang Miao, Amin Kamel and Chandra PrakashDrug Metabolism and Disposition July 2005, 33 (7) 879-883; DOI: https://doi.org/10.1124/dmd.105.004036
Preiss, Rainer
- You have accessSYNTHESIS AND CHARACTERIZATION OF SOME NEW PHASE II METABOLITES OF THE ALKYLATOR BENDAMUSTINE AND THEIR IDENTIFICATION IN HUMAN BILE, URINE, AND PLASMA FROM PATIENTS WITH CHOLANGIOCARCINOMAJens Teichert, Reinhard Sohr, Frank Baumann, Lothar Hennig, Karlheinz Merkle, Karel Caca and Rainer PreissDrug Metabolism and Disposition July 2005, 33 (7) 984-992; DOI: https://doi.org/10.1124/dmd.105.003624
R
Raab, Conrad
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Radominska-Pandya, Anna
- You have accessLITHOCHOLIC ACID DECREASES EXPRESSION OF UGT2B7 IN CACO-2 CELLS: A POTENTIAL ROLE FOR A NEGATIVE FARNESOID X RECEPTOR RESPONSE ELEMENTYuan Lu, Jean-Marie Heydel, Xin Li, Stacie Bratton, Tim Lindblom and Anna Radominska-PandyaDrug Metabolism and Disposition July 2005, 33 (7) 937-946; DOI: https://doi.org/10.1124/dmd.104.003061
Richards, Karen
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Risler, Linda J.
- You have accessCONTRIBUTION OF CYP3A5 TO HEPATIC AND RENAL IFOSFAMIDE N-DECHLOROETHYLATIONJeannine S. McCune, Linda J. Risler, Brian R. Phillips, Kenneth E. Thummel, David Blough and Danny D. ShenDrug Metabolism and Disposition July 2005, 33 (7) 1074-1081; DOI: https://doi.org/10.1124/dmd.104.002279
Ritter, Joseph K.
- You have accessDIFFERENTIAL RATES OF GLUCURONIDATION FOR 7-ETHYL-10-HYDROXY-CAMPTOTHECIN (SN-38) LACTONE AND CARBOXYLATE IN HUMAN AND RAT MICROSOMES AND RECOMBINANT UDP-GLUCURONOSYLTRANSFERASE ISOFORMSMelanie N. Tallman, Joseph K. Ritter and Philip C. SmithDrug Metabolism and Disposition July 2005, 33 (7) 977-983; DOI: https://doi.org/10.1124/dmd.104.003491
Rodrigues, A. David
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Roger, Michel
- You have accessCYP3A5 GENETIC POLYMORPHISMS IN DIFFERENT ETHNIC POPULATIONSJean-Nicholas Roy, Julie Lajoie, Lynn S. Zijenah, Azemi Barama, Charles Poirier, Brian J. Ward and Michel RogerDrug Metabolism and Disposition July 2005, 33 (7) 884-887; DOI: https://doi.org/10.1124/dmd.105.003822
Roiko, S. A.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Roy, Jean-Nicholas
- You have accessCYP3A5 GENETIC POLYMORPHISMS IN DIFFERENT ETHNIC POPULATIONSJean-Nicholas Roy, Julie Lajoie, Lynn S. Zijenah, Azemi Barama, Charles Poirier, Brian J. Ward and Michel RogerDrug Metabolism and Disposition July 2005, 33 (7) 884-887; DOI: https://doi.org/10.1124/dmd.105.003822
Roymans, Dirk
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
Rushmore, Thomas H.
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
S
Sánchez Pozzi, Enrique J.
- You have accessPREVENTION OF MRP2 ACTIVITY IMPAIRMENT IN ETHINYLESTRADIOL-INDUCED CHOLESTASIS BY URSODEOXYCHOLATE IN THE RATFernando A. Crocenzi, Vanesa D'Andrea, Viviana A. Catania, Marcelo G. Luquita, José M. Pellegrino, J. Elena Ochoa, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition July 2005, 33 (7) 888-891; DOI: https://doi.org/10.1124/dmd.104.003533
Schellens, Jan H. M.
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
Schinkel, Alfred H.
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
Scott, Emily E.
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Sensenhauser, Carlo
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
Shen, Danny D.
- You have accessCONTRIBUTION OF CYP3A5 TO HEPATIC AND RENAL IFOSFAMIDE N-DECHLOROETHYLATIONJeannine S. McCune, Linda J. Risler, Brian R. Phillips, Kenneth E. Thummel, David Blough and Danny D. ShenDrug Metabolism and Disposition July 2005, 33 (7) 1074-1081; DOI: https://doi.org/10.1124/dmd.104.002279
Shen, Jianhua
- You have accessPOSSIBLE PATHWAY(S) OF TESTOSTERONE EGRESS FROM THE ACTIVE SITE OF CYTOCHROME P450 2B1: A STEERED MOLECULAR DYNAMICS SIMULATIONWeihua Li, Hong Liu, Emily E. Scott, Frauke Gräter, James R. Halpert, Xiaoming Luo, Jianhua Shen and Hualiang JiangDrug Metabolism and Disposition July 2005, 33 (7) 910-919; DOI: https://doi.org/10.1124/dmd.105.004200
Silva, José
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
Sinclair, Jacqueline F.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Sinclair, Peter R.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Singh, Rominder
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Slitt, Angela L.
- You have accessTISSUE DISTRIBUTION AND HEPATIC AND RENAL ONTOGENY OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) FAMILY IN MICEJonathan M. Maher, Angela L. Slitt, Nathan J. Cherrington, Xingguo Cheng and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 947-955; DOI: https://doi.org/10.1124/dmd.105.003780
- You have accessINDUCTION OF THE MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN FAMILY OF TRANSPORTERS BY CHEMICAL ACTIVATORS OF RECEPTOR-MEDIATED PATHWAYS IN MOUSE LIVERJonathan M. Maher, Xingguo Cheng, Angela L. Slitt, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition July 2005, 33 (7) 956-962; DOI: https://doi.org/10.1124/dmd.105.003798
Smit, Johan W.
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
Smith, Philip C.
- You have accessDIFFERENTIAL RATES OF GLUCURONIDATION FOR 7-ETHYL-10-HYDROXY-CAMPTOTHECIN (SN-38) LACTONE AND CARBOXYLATE IN HUMAN AND RAT MICROSOMES AND RECOMBINANT UDP-GLUCURONOSYLTRANSFERASE ISOFORMSMelanie N. Tallman, Joseph K. Ritter and Philip C. SmithDrug Metabolism and Disposition July 2005, 33 (7) 977-983; DOI: https://doi.org/10.1124/dmd.104.003491
Sohr, Reinhard
- You have accessSYNTHESIS AND CHARACTERIZATION OF SOME NEW PHASE II METABOLITES OF THE ALKYLATOR BENDAMUSTINE AND THEIR IDENTIFICATION IN HUMAN BILE, URINE, AND PLASMA FROM PATIENTS WITH CHOLANGIOCARCINOMAJens Teichert, Reinhard Sohr, Frank Baumann, Lothar Hennig, Karlheinz Merkle, Karel Caca and Rainer PreissDrug Metabolism and Disposition July 2005, 33 (7) 984-992; DOI: https://doi.org/10.1124/dmd.105.003624
Sparidans, Rolf W.
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
St. Peter, J. V.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Stewart, S.
- You have accessMONOCLONAL NICOTINE-SPECIFIC ANTIBODIES REDUCE NICOTINE DISTRIBUTION TO BRAIN IN RATS: DOSE- AND AFFINITY-RESPONSE RELATIONSHIPSD. E. Keyler, S. A. Roiko, E. Benlhabib, M. G. LeSage, J. V. St. Peter, S. Stewart, S. Fuller, C. T. Le and P. R. PentelDrug Metabolism and Disposition July 2005, 33 (7) 1056-1061; DOI: https://doi.org/10.1124/dmd.105.004234
Strom, Stephen C.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Subramanian, Raju
- You have accessINDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Charles Lin, Rominder Singh, Cheri M. Brown, Karen Richards, Janice Brunner, Kimberly Michel, Jennifer Adelsberger, Edward Carlini, Catherine Boothe-Genthe, Conrad Raab, Minh Luu, Aimee Michael, Mona Parikh, Patrice Ciecko, Raju Subramanian, Paul Krolikowski, A. David Rodrigues, Thomas A. Baillie and Thomas H. RushmoreDrug Metabolism and Disposition July 2005, 33 (7) 1044-1051; DOI: https://doi.org/10.1124/dmd.105.003913
Sugiyama, Yuichi
- You have accessREGULATION OF THE CELL SURFACE EXPRESSION OF HUMAN BCRP/ABCG2 BY THE PHOSPHORYLATION STATE OF AKT IN POLARIZED CELLSTappei Takada, Hiroshi Suzuki, Yukiko Gotoh and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 905-909; DOI: https://doi.org/10.1124/dmd.104.003228
- You have accessP-GLYCOPROTEIN PLAYS A MAJOR ROLE IN THE EFFLUX OF FEXOFENADINE IN THE SMALL INTESTINE AND BLOOD-BRAIN BARRIER, BUT ONLY A LIMITED ROLE IN ITS BILIARY EXCRETIONHarunobu Tahara, Hiroyuki Kusuhara, Eiichi Fuse and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 963-968; DOI: https://doi.org/10.1124/dmd.105.004192
Suzuki, Hiroshi
- You have accessREGULATION OF THE CELL SURFACE EXPRESSION OF HUMAN BCRP/ABCG2 BY THE PHOSPHORYLATION STATE OF AKT IN POLARIZED CELLSTappei Takada, Hiroshi Suzuki, Yukiko Gotoh and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 905-909; DOI: https://doi.org/10.1124/dmd.104.003228
T
Tahara, Harunobu
- You have accessP-GLYCOPROTEIN PLAYS A MAJOR ROLE IN THE EFFLUX OF FEXOFENADINE IN THE SMALL INTESTINE AND BLOOD-BRAIN BARRIER, BUT ONLY A LIMITED ROLE IN ITS BILIARY EXCRETIONHarunobu Tahara, Hiroyuki Kusuhara, Eiichi Fuse and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 963-968; DOI: https://doi.org/10.1124/dmd.105.004192
Takada, Tappei
- You have accessREGULATION OF THE CELL SURFACE EXPRESSION OF HUMAN BCRP/ABCG2 BY THE PHOSPHORYLATION STATE OF AKT IN POLARIZED CELLSTappei Takada, Hiroshi Suzuki, Yukiko Gotoh and Yuichi SugiyamaDrug Metabolism and Disposition July 2005, 33 (7) 905-909; DOI: https://doi.org/10.1124/dmd.104.003228
Tallman, Melanie N.
- You have accessDIFFERENTIAL RATES OF GLUCURONIDATION FOR 7-ETHYL-10-HYDROXY-CAMPTOTHECIN (SN-38) LACTONE AND CARBOXYLATE IN HUMAN AND RAT MICROSOMES AND RECOMBINANT UDP-GLUCURONOSYLTRANSFERASE ISOFORMSMelanie N. Tallman, Joseph K. Ritter and Philip C. SmithDrug Metabolism and Disposition July 2005, 33 (7) 977-983; DOI: https://doi.org/10.1124/dmd.104.003491
Tang, Zhongming
- You have accessMETABOLIC PROFILE OF 1,5-DICAFFEOYLQUINIC ACID IN RATS, AN IN VIVO AND IN VITRO STUDYBo Yang, Zhiyun Meng, Junxing Dong, Liangping Yan, Libo Zou, Zhongming Tang and Guifang DouDrug Metabolism and Disposition July 2005, 33 (7) 930-936; DOI: https://doi.org/10.1124/dmd.104.002154
Taskinen, Jyrki
- You have accessKINETIC CHARACTERIZATION OF THE 1A SUBFAMILY OF RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASESLeena Luukkanen, Jyrki Taskinen, Mika Kurkela, Risto Kostiainen, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition July 2005, 33 (7) 1017-1026; DOI: https://doi.org/10.1124/dmd.105.004093
Teichert, Jens
- You have accessSYNTHESIS AND CHARACTERIZATION OF SOME NEW PHASE II METABOLITES OF THE ALKYLATOR BENDAMUSTINE AND THEIR IDENTIFICATION IN HUMAN BILE, URINE, AND PLASMA FROM PATIENTS WITH CHOLANGIOCARCINOMAJens Teichert, Reinhard Sohr, Frank Baumann, Lothar Hennig, Karlheinz Merkle, Karel Caca and Rainer PreissDrug Metabolism and Disposition July 2005, 33 (7) 984-992; DOI: https://doi.org/10.1124/dmd.105.003624
Thummel, Kenneth E.
- You have accessCONTRIBUTION OF CYP3A5 TO HEPATIC AND RENAL IFOSFAMIDE N-DECHLOROETHYLATIONJeannine S. McCune, Linda J. Risler, Brian R. Phillips, Kenneth E. Thummel, David Blough and Danny D. ShenDrug Metabolism and Disposition July 2005, 33 (7) 1074-1081; DOI: https://doi.org/10.1124/dmd.104.002279
Trask, Heidi W.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
U
Unadkat, Jashvant D.
- You have accessIDENTIFICATION OF CYTOCHROME P450 AND ARYLAMINE N-ACETYLTRANSFERASE ISOFORMS INVOLVED IN SULFADIAZINE METABOLISMHelen R. Winter and Jashvant D. UnadkatDrug Metabolism and Disposition July 2005, 33 (7) 969-976; DOI: https://doi.org/10.1124/dmd.104.002998
V
van der Kruijssen, Cornelia M. M.
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
van Herwaarden, Antonius E.
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
Van Houdt, Jos
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
Van Looveren, Cis
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
W
Wagenaar, Els
- You have accessMIDAZOLAM AND CYCLOSPORIN A METABOLISM IN TRANSGENIC MICE WITH LIVER-SPECIFIC EXPRESSION OF HUMAN CYP3A4Antonius E. van Herwaarden, Johan W. Smit, Rolf W. Sparidans, Els Wagenaar, Cornelia M. M. van der Kruijssen, Jan H. M. Schellens, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition July 2005, 33 (7) 892-895; DOI: https://doi.org/10.1124/dmd.105.004721
Wahlstrom, Jan L.
- You have accessTHREE-DIMENSIONAL QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP ANALYSIS OF CYTOCHROMES P450: EFFECT OF INCORPORATING HIGHER-AFFINITY LIGANDS AND POTENTIAL NEW APPLICATIONSCharles W. Locuson and Jan L. WahlstromDrug Metabolism and Disposition July 2005, 33 (7) 873-878; DOI: https://doi.org/10.1124/dmd.105.004325
Ward, Brian J.
- You have accessCYP3A5 GENETIC POLYMORPHISMS IN DIFFERENT ETHNIC POPULATIONSJean-Nicholas Roy, Julie Lajoie, Lynn S. Zijenah, Azemi Barama, Charles Poirier, Brian J. Ward and Michel RogerDrug Metabolism and Disposition July 2005, 33 (7) 884-887; DOI: https://doi.org/10.1124/dmd.105.003822
Weygers, Adri
- You have accessEXPRESSION AND INDUCTION POTENTIAL OF CYTOCHROMES P450 IN HUMAN CRYOPRESERVED HEPATOCYTESDirk Roymans, Pieter Annaert, Jos Van Houdt, Adri Weygers, Jan Noukens, Carlo Sensenhauser, José Silva, Cis Van Looveren, Jan Hendrickx, Geert Mannens and Willem MeuldermansDrug Metabolism and Disposition July 2005, 33 (7) 1004-1016; DOI: https://doi.org/10.1124/dmd.104.003046
Winter, Helen R.
- You have accessIDENTIFICATION OF CYTOCHROME P450 AND ARYLAMINE N-ACETYLTRANSFERASE ISOFORMS INVOLVED IN SULFADIAZINE METABOLISMHelen R. Winter and Jashvant D. UnadkatDrug Metabolism and Disposition July 2005, 33 (7) 969-976; DOI: https://doi.org/10.1124/dmd.104.002998
Wood, Sheryl G.
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Wrighton, Steven A.
- You have accessTHE USE OF A SUBSTRATE CASSETTE STRATEGY TO IMPROVE THE CAPACITY AND THROUGHPUT OF CYTOCHROME P450 INDUCTION STUDIES IN HUMAN HEPATOCYTESMichael A. Mohutsky, David M. Petullo and Steven A. WrightonDrug Metabolism and Disposition July 2005, 33 (7) 920-923; DOI: https://doi.org/10.1124/dmd.105.004291
- You have accessARSENITE DECREASES CYP3A4 AND RXRα IN PRIMARY HUMAN HEPATOCYTESTrisha L. Noreault, Vsevolod E. Kostrubsky, Sheryl G. Wood, Ralph C. Nichols, Stephen C. Strom, Heidi W. Trask, Steven A. Wrighton, Ronald M. Evans, Judith M. Jacobs, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition July 2005, 33 (7) 993-1003; DOI: https://doi.org/10.1124/dmd.105.003954
Y
Yamanaka, Yosuke
- You have accessIDENTIFICATION OF HMG-CoA REDUCTASE INHIBITORS AS ACTIVATORS FOR HUMAN, MOUSE AND RAT CONSTITUTIVE ANDROSTANE RECEPTORKaoru Kobayashi, Yosuke Yamanaka, Norihiko Iwazaki, Ikumi Nakajo, Masakiyo Hosokawa, Masahiko Negishi and Kan ChibaDrug Metabolism and Disposition July 2005, 33 (7) 924-929; DOI: https://doi.org/10.1124/dmd.104.002741
Yan, Liangping
- You have accessMETABOLIC PROFILE OF 1,5-DICAFFEOYLQUINIC ACID IN RATS, AN IN VIVO AND IN VITRO STUDYBo Yang, Zhiyun Meng, Junxing Dong, Liangping Yan, Libo Zou, Zhongming Tang and Guifang DouDrug Metabolism and Disposition July 2005, 33 (7) 930-936; DOI: https://doi.org/10.1124/dmd.104.002154
Yang, Bo
- You have accessMETABOLIC PROFILE OF 1,5-DICAFFEOYLQUINIC ACID IN RATS, AN IN VIVO AND IN VITRO STUDYBo Yang, Zhiyun Meng, Junxing Dong, Liangping Yan, Libo Zou, Zhongming Tang and Guifang DouDrug Metabolism and Disposition July 2005, 33 (7) 930-936; DOI: https://doi.org/10.1124/dmd.104.002154
Z
Zijenah, Lynn S.
- You have accessCYP3A5 GENETIC POLYMORPHISMS IN DIFFERENT ETHNIC POPULATIONSJean-Nicholas Roy, Julie Lajoie, Lynn S. Zijenah, Azemi Barama, Charles Poirier, Brian J. Ward and Michel RogerDrug Metabolism and Disposition July 2005, 33 (7) 884-887; DOI: https://doi.org/10.1124/dmd.105.003822
Zou, Libo
- You have accessMETABOLIC PROFILE OF 1,5-DICAFFEOYLQUINIC ACID IN RATS, AN IN VIVO AND IN VITRO STUDYBo Yang, Zhiyun Meng, Junxing Dong, Liangping Yan, Libo Zou, Zhongming Tang and Guifang DouDrug Metabolism and Disposition July 2005, 33 (7) 930-936; DOI: https://doi.org/10.1124/dmd.104.002154