Index by author
March 01, 2006; Volume 34,Issue 3
A
Alnouti, Yazen
- You have accessTISSUE DISTRIBUTION AND ONTOGENY OF ORGANIC CATION TRANSPORTERS IN MICEYazen Alnouti, Jay S. Petrick and Curtis D. KlaassenDrug Metabolism and Disposition March 2006, 34 (3) 477-482; DOI: https://doi.org/10.1124/dmd.105.006932
Anand, Sathanandam S.
- You have accessONTOGENY OF HEPATIC AND PLASMA METABOLISM OF DELTAMETHRIN IN VITRO: ROLE IN AGE-DEPENDENT ACUTE NEUROTOXICITYSathanandam S. Anand, Kyu-Bong Kim, Stephanie Padilla, Srinivasa Muralidhara, Hyo J. Kim, Jeffrey W. Fisher and James V. BrucknerDrug Metabolism and Disposition March 2006, 34 (3) 389-397; DOI: https://doi.org/10.1124/dmd.105.007807
Anapolsky, Alexander
- You have accessTHE ROLE OF PREGNANE X RECEPTOR IN 2-ACETYLAMINOFLUORENE-MEDIATED INDUCTION OF DRUG TRANSPORT AND -METABOLIZING ENZYMES IN MICEAlexander Anapolsky, Shirley Teng, Santosh Dixit and Micheline Piquette-MillerDrug Metabolism and Disposition March 2006, 34 (3) 405-409; DOI: https://doi.org/10.1124/dmd.105.006197
Andreyev, Sergey
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
Antonovic, Leposava
- You have accessHEPATIC AND RENAL CYTOCHROME P450 GENE REGULATION DURING CITROBACTER RODENTIUM INFECTION IN WILD-TYPE AND TOLL-LIKE RECEPTOR 4 MUTANT MICETerrilyn A. Richardson, Melanie Sherman, Leposava Antonovic, Sean S. Kardar, Henry W. Strobel, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 354-360; DOI: https://doi.org/10.1124/dmd.105.007393
Arimori, Kazuhiko
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Aurang, Catherine
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
B
Balani, Suresh K.
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Ballent, M.
- You have accessMODULATION OF THE P-GLYCOPROTEIN-MEDIATED INTESTINAL SECRETION OF IVERMECTIN: IN VITRO AND IN VIVO ASSESSMENTSM. Ballent, A. Lifschitz, G. Virkel, J. Sallovitz and C. LanusseDrug Metabolism and Disposition March 2006, 34 (3) 457-463; DOI: https://doi.org/10.1124/dmd.105.007757
Block, Simone
- You have accessPURIFICATION AND CHARACTERIZATION OF AKR1B10 FROM HUMAN LIVER: ROLE IN CARBONYL REDUCTION OF XENOBIOTICSHans-Jörg Martin, Ursula Breyer-Pfaff, Vladimir Wsol, Simone Venz, Simone Block and Edmund MaserDrug Metabolism and Disposition March 2006, 34 (3) 464-470; DOI: https://doi.org/10.1124/dmd.105.007971
Breyer-Pfaff, Ursula
- You have accessPURIFICATION AND CHARACTERIZATION OF AKR1B10 FROM HUMAN LIVER: ROLE IN CARBONYL REDUCTION OF XENOBIOTICSHans-Jörg Martin, Ursula Breyer-Pfaff, Vladimir Wsol, Simone Venz, Simone Block and Edmund MaserDrug Metabolism and Disposition March 2006, 34 (3) 464-470; DOI: https://doi.org/10.1124/dmd.105.007971
Bruckner, James V.
- You have accessONTOGENY OF HEPATIC AND PLASMA METABOLISM OF DELTAMETHRIN IN VITRO: ROLE IN AGE-DEPENDENT ACUTE NEUROTOXICITYSathanandam S. Anand, Kyu-Bong Kim, Stephanie Padilla, Srinivasa Muralidhara, Hyo J. Kim, Jeffrey W. Fisher and James V. BrucknerDrug Metabolism and Disposition March 2006, 34 (3) 389-397; DOI: https://doi.org/10.1124/dmd.105.007807
Bugrim, Andrej
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
C
Chang, Yan
- You have accessNOVEL METABOLITES OF BUPRENORPHINE DETECTED IN HUMAN LIVER MICROSOMES AND HUMAN URINEYan Chang, David E. Moody and Elinore F. McCance-KatzDrug Metabolism and Disposition March 2006, 34 (3) 440-448; DOI: https://doi.org/10.1124/dmd.105.006148
Cheng, Peter T.
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
Costa, Arnaldo O.
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
D
Dalton, James T.
- You have accessPHARMACOKINETICS AND METABOLISM OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR IN RATS: IMPLICATION OF MOLECULAR PROPERTIES AND INTENSIVE METABOLIC PROFILE TO INVESTIGATE IDEAL PHARMACOKINETIC CHARACTERISTICS OF A PROPANAMIDE IN PRECLINICAL STUDYDi Wu, Zengru Wu, Jun Yang, Vipin A. Nair, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition March 2006, 34 (3) 483-494; DOI: https://doi.org/10.1124/dmd.105.006643
Daniel, Władysława A.
- You have accessCHARACTERIZATION OF HUMAN CYTOCHROME P450 ENZYMES INVOLVED IN THE METABOLISM OF THE PIPERIDINE-TYPE PHENOTHIAZINE NEUROLEPTIC THIORIDAZINEJacek Wójcikowski, Patrick Maurel and Władysława A. DanielDrug Metabolism and Disposition March 2006, 34 (3) 471-476; DOI: https://doi.org/10.1124/dmd.105.006445
Daniels, J. Scott
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Dixit, Santosh
- You have accessTHE ROLE OF PREGNANE X RECEPTOR IN 2-ACETYLAMINOFLUORENE-MEDIATED INDUCTION OF DRUG TRANSPORT AND -METABOLIZING ENZYMES IN MICEAlexander Anapolsky, Shirley Teng, Santosh Dixit and Micheline Piquette-MillerDrug Metabolism and Disposition March 2006, 34 (3) 405-409; DOI: https://doi.org/10.1124/dmd.105.006197
Dworakowski, Wojciech
- You have accessINDUCIBILITY OF MALE-SPECIFIC ISOFORMS OF CYTOCHROME P450 BY SEX-DEPENDENT GROWTH HORMONE PROFILES IN HEPATOCYTE CULTURES FROM MALE BUT NOT FEMALE RATSChellappagounder Thangavel, Wojciech Dworakowski and Bernard H. ShapiroDrug Metabolism and Disposition March 2006, 34 (3) 410-419; DOI: https://doi.org/10.1124/dmd.105.007716
E
Ekins, Sean
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
Elliot, David J.
- You have accessSELECTIVITY OF SUBSTRATE (TRIFLUOPERAZINE) AND INHIBITOR (AMITRIPTYLINE, ANDROSTERONE, CANRENOIC ACID, HECOGENIN, PHENYLBUTAZONE, QUINIDINE, QUININE, AND SULFINPYRAZONE) “PROBES” FOR HUMAN UDP-GLUCURONOSYLTRANSFERASESVerawan Uchaipichat, Peter I. Mackenzie, David J. Elliot and John O. MinersDrug Metabolism and Disposition March 2006, 34 (3) 449-456; DOI: https://doi.org/10.1124/dmd.105.007369
Engeln, Katrin
- You have accessDIGITAL FLUORESCENCE IMAGING OF ORGANIC CATION TRANSPORT IN FRESHLY ISOLATED RAT PROXIMAL TUBULESFrank Pietruck, Markus Horbelt, Thorsten Feldkamp, Katrin Engeln, Stefan Herget-Rosenthal, Thomas Philipp and Andreas KribbenDrug Metabolism and Disposition March 2006, 34 (3) 339-342; DOI: https://doi.org/10.1124/dmd.105.006403
Everett, Donald W.
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
F
Falany, Charles N.
- You have accessSULFATION OF RALOXIFENE AND 4-HYDROXYTAMOXIFEN BY HUMAN CYTOSOLIC SULFOTRANSFERASESJosie L. Falany, Daniel E. Pilloff, Thomas S. Leyh and Charles N. FalanyDrug Metabolism and Disposition March 2006, 34 (3) 361-368; DOI: https://doi.org/10.1124/dmd.105.006551
Falany, Josie L.
- You have accessSULFATION OF RALOXIFENE AND 4-HYDROXYTAMOXIFEN BY HUMAN CYTOSOLIC SULFOTRANSFERASESJosie L. Falany, Daniel E. Pilloff, Thomas S. Leyh and Charles N. FalanyDrug Metabolism and Disposition March 2006, 34 (3) 361-368; DOI: https://doi.org/10.1124/dmd.105.006551
Feldkamp, Thorsten
- You have accessDIGITAL FLUORESCENCE IMAGING OF ORGANIC CATION TRANSPORT IN FRESHLY ISOLATED RAT PROXIMAL TUBULESFrank Pietruck, Markus Horbelt, Thorsten Feldkamp, Katrin Engeln, Stefan Herget-Rosenthal, Thomas Philipp and Andreas KribbenDrug Metabolism and Disposition March 2006, 34 (3) 339-342; DOI: https://doi.org/10.1124/dmd.105.006403
Fisher, Jeffrey W.
- You have accessONTOGENY OF HEPATIC AND PLASMA METABOLISM OF DELTAMETHRIN IN VITRO: ROLE IN AGE-DEPENDENT ACUTE NEUROTOXICITYSathanandam S. Anand, Kyu-Bong Kim, Stephanie Padilla, Srinivasa Muralidhara, Hyo J. Kim, Jeffrey W. Fisher and James V. BrucknerDrug Metabolism and Disposition March 2006, 34 (3) 389-397; DOI: https://doi.org/10.1124/dmd.105.007807
Fujita, Ken-Ichi
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Fukasawa, Yoshiki
- You have accessIN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTMasato Nakamura, Yasunori Kawakita, Akito Yasuhara, Yoshiki Fukasawa, Koji Yoshida, Kazunari Sakagami and Atsuro NakazatoDrug Metabolism and Disposition March 2006, 34 (3) 369-374; DOI: https://doi.org/10.1124/dmd.105.006213
G
Gaedigk, Andrea
- You have accessCOMMENTS ON HOSKINS ET AL. [(2005) DRUG METAB DISPOS 33:1564–1565]Andrea Gaedigk and J. Steven LeederDrug Metabolism and Disposition March 2006, 34 (3) 504-505; DOI: https://doi.org/10.1124/dmd.105.007799
Gan, Liang-Shang
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
H
Hamilton, Marta
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
Herget-Rosenthal, Stefan
- You have accessDIGITAL FLUORESCENCE IMAGING OF ORGANIC CATION TRANSPORT IN FRESHLY ISOLATED RAT PROXIMAL TUBULESFrank Pietruck, Markus Horbelt, Thorsten Feldkamp, Katrin Engeln, Stefan Herget-Rosenthal, Thomas Philipp and Andreas KribbenDrug Metabolism and Disposition March 2006, 34 (3) 339-342; DOI: https://doi.org/10.1124/dmd.105.006403
Hidaka, Muneaki
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Hollenberg, Paul F.
- You have accessSELECTIVE PATHWAYS FOR THE METABOLISM OF PHENCYCLIDINE BY CYTOCHROME P450 2B ENZYMES: IDENTIFICATION OF ELECTROPHILIC METABOLITES, GLUTATHIONE, AND N-ACETYL CYSTEINE ADDUCTSMohamad Shebley, Monica I. Jushchyshyn and Paul F. HollenbergDrug Metabolism and Disposition March 2006, 34 (3) 375-383; DOI: https://doi.org/10.1124/dmd.105.007047
Horbelt, Markus
- You have accessDIGITAL FLUORESCENCE IMAGING OF ORGANIC CATION TRANSPORT IN FRESHLY ISOLATED RAT PROXIMAL TUBULESFrank Pietruck, Markus Horbelt, Thorsten Feldkamp, Katrin Engeln, Stefan Herget-Rosenthal, Thomas Philipp and Andreas KribbenDrug Metabolism and Disposition March 2006, 34 (3) 339-342; DOI: https://doi.org/10.1124/dmd.105.006403
Humphreys, W. Griffith
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
I
Imai, Teruko
- You have accessFIRST-PASS HYDROLYSIS OF A PROPRANOLOL ESTER DERIVATIVE IN RAT SMALL INTESTINEKenji Masaki, Megumi Taketani and Teruko ImaiDrug Metabolism and Disposition March 2006, 34 (3) 398-404; DOI: https://doi.org/10.1124/dmd.105.007682
Iwakiri, Tomomi
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
J
Johnson, Kim A.
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
Jushchyshyn, Monica I.
- You have accessSELECTIVE PATHWAYS FOR THE METABOLISM OF PHENCYCLIDINE BY CYTOCHROME P450 2B ENZYMES: IDENTIFICATION OF ELECTROPHILIC METABOLITES, GLUTATHIONE, AND N-ACETYL CYSTEINE ADDUCTSMohamad Shebley, Monica I. Jushchyshyn and Paul F. HollenbergDrug Metabolism and Disposition March 2006, 34 (3) 375-383; DOI: https://doi.org/10.1124/dmd.105.007047
K
Kai, Hirofumi
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Kalman, Daniel
- You have accessEXPRESSION OF UDP-GLUCURONOSYLTRANSFERASE ISOFORM mRNAS DURING INFLAMMATION AND INFECTION IN MOUSE LIVER AND KIDNEYTerrilyn A. Richardson, Melanie Sherman, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 351-353; DOI: https://doi.org/10.1124/dmd.105.007435
- You have accessHEPATIC AND RENAL CYTOCHROME P450 GENE REGULATION DURING CITROBACTER RODENTIUM INFECTION IN WILD-TYPE AND TOLL-LIKE RECEPTOR 4 MUTANT MICETerrilyn A. Richardson, Melanie Sherman, Leposava Antonovic, Sean S. Kardar, Henry W. Strobel, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 354-360; DOI: https://doi.org/10.1124/dmd.105.007393
Kardar, Sean S.
- You have accessHEPATIC AND RENAL CYTOCHROME P450 GENE REGULATION DURING CITROBACTER RODENTIUM INFECTION IN WILD-TYPE AND TOLL-LIKE RECEPTOR 4 MUTANT MICETerrilyn A. Richardson, Melanie Sherman, Leposava Antonovic, Sean S. Kardar, Henry W. Strobel, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 354-360; DOI: https://doi.org/10.1124/dmd.105.007393
Kawakita, Yasunori
- You have accessIN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTMasato Nakamura, Yasunori Kawakita, Akito Yasuhara, Yoshiki Fukasawa, Koji Yoshida, Kazunari Sakagami and Atsuro NakazatoDrug Metabolism and Disposition March 2006, 34 (3) 369-374; DOI: https://doi.org/10.1124/dmd.105.006213
Kim, Hyo J.
- You have accessONTOGENY OF HEPATIC AND PLASMA METABOLISM OF DELTAMETHRIN IN VITRO: ROLE IN AGE-DEPENDENT ACUTE NEUROTOXICITYSathanandam S. Anand, Kyu-Bong Kim, Stephanie Padilla, Srinivasa Muralidhara, Hyo J. Kim, Jeffrey W. Fisher and James V. BrucknerDrug Metabolism and Disposition March 2006, 34 (3) 389-397; DOI: https://doi.org/10.1124/dmd.105.007807
Kim, Kyu-Bong
- You have accessONTOGENY OF HEPATIC AND PLASMA METABOLISM OF DELTAMETHRIN IN VITRO: ROLE IN AGE-DEPENDENT ACUTE NEUROTOXICITYSathanandam S. Anand, Kyu-Bong Kim, Stephanie Padilla, Srinivasa Muralidhara, Hyo J. Kim, Jeffrey W. Fisher and James V. BrucknerDrug Metabolism and Disposition March 2006, 34 (3) 389-397; DOI: https://doi.org/10.1124/dmd.105.007807
Kirillov, Eugene
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
Klaassen, Curtis D.
- You have accessTISSUE DISTRIBUTION AND ONTOGENY OF ORGANIC CATION TRANSPORTERS IN MICEYazen Alnouti, Jay S. Petrick and Curtis D. KlaassenDrug Metabolism and Disposition March 2006, 34 (3) 477-482; DOI: https://doi.org/10.1124/dmd.105.006932
Klausner, Mitch
- You have accessBENZO[A]PYRENE-INDUCED ORAL CARCINOGENESIS AND CHEMOPREVENTION: STUDIES IN BIOENGINEERED HUMAN TISSUEThomas Walle, U. Kristina Walle, David Sedmera and Mitch KlausnerDrug Metabolism and Disposition March 2006, 34 (3) 346-350; DOI: https://doi.org/10.1124/dmd.105.007948
Kribben, Andreas
- You have accessDIGITAL FLUORESCENCE IMAGING OF ORGANIC CATION TRANSPORT IN FRESHLY ISOLATED RAT PROXIMAL TUBULESFrank Pietruck, Markus Horbelt, Thorsten Feldkamp, Katrin Engeln, Stefan Herget-Rosenthal, Thomas Philipp and Andreas KribbenDrug Metabolism and Disposition March 2006, 34 (3) 339-342; DOI: https://doi.org/10.1124/dmd.105.006403
L
Lanusse, C.
- You have accessMODULATION OF THE P-GLYCOPROTEIN-MEDIATED INTESTINAL SECRETION OF IVERMECTIN: IN VITRO AND IN VIVO ASSESSMENTSM. Ballent, A. Lifschitz, G. Virkel, J. Sallovitz and C. LanusseDrug Metabolism and Disposition March 2006, 34 (3) 457-463; DOI: https://doi.org/10.1124/dmd.105.007757
Lee, Frank W.
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Leeder, J. Steven
- You have accessCOMMENTS ON HOSKINS ET AL. [(2005) DRUG METAB DISPOS 33:1564–1565]Andrea Gaedigk and J. Steven LeederDrug Metabolism and Disposition March 2006, 34 (3) 504-505; DOI: https://doi.org/10.1124/dmd.105.007799
Leyh, Thomas S.
- You have accessSULFATION OF RALOXIFENE AND 4-HYDROXYTAMOXIFEN BY HUMAN CYTOSOLIC SULFOTRANSFERASESJosie L. Falany, Daniel E. Pilloff, Thomas S. Leyh and Charles N. FalanyDrug Metabolism and Disposition March 2006, 34 (3) 361-368; DOI: https://doi.org/10.1124/dmd.105.006551
Lifschitz, A.
- You have accessMODULATION OF THE P-GLYCOPROTEIN-MEDIATED INTESTINAL SECRETION OF IVERMECTIN: IN VITRO AND IN VIVO ASSESSMENTSM. Ballent, A. Lifschitz, G. Virkel, J. Sallovitz and C. LanusseDrug Metabolism and Disposition March 2006, 34 (3) 457-463; DOI: https://doi.org/10.1124/dmd.105.007757
Ling, Jie
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
Lum, Bert L.
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
M
Mackenzie, Peter I.
- You have accessSELECTIVITY OF SUBSTRATE (TRIFLUOPERAZINE) AND INHIBITOR (AMITRIPTYLINE, ANDROSTERONE, CANRENOIC ACID, HECOGENIN, PHENYLBUTAZONE, QUINIDINE, QUININE, AND SULFINPYRAZONE) “PROBES” FOR HUMAN UDP-GLUCURONOSYLTRANSFERASESVerawan Uchaipichat, Peter I. Mackenzie, David J. Elliot and John O. MinersDrug Metabolism and Disposition March 2006, 34 (3) 449-456; DOI: https://doi.org/10.1124/dmd.105.007369
Mahmood, Iftekhar
- You have accessCOMMENTS ON “A MATHEMATICAL DESCRIPTION OF THE FUNCTIONALITY OF CORRECTION FACTORS USED IN ALLOMETRY FOR PREDICTING HUMAN DRUG CLEARANCE”Iftekhar MahmoodDrug Metabolism and Disposition March 2006, 34 (3) 507-509; DOI: https://doi.org/10.1124/dmd.105.007187
Martin, Hans-Jörg
- You have accessPURIFICATION AND CHARACTERIZATION OF AKR1B10 FROM HUMAN LIVER: ROLE IN CARBONYL REDUCTION OF XENOBIOTICSHans-Jörg Martin, Ursula Breyer-Pfaff, Vladimir Wsol, Simone Venz, Simone Block and Edmund MaserDrug Metabolism and Disposition March 2006, 34 (3) 464-470; DOI: https://doi.org/10.1124/dmd.105.007971
Masaki, Kenji
- You have accessFIRST-PASS HYDROLYSIS OF A PROPRANOLOL ESTER DERIVATIVE IN RAT SMALL INTESTINEKenji Masaki, Megumi Taketani and Teruko ImaiDrug Metabolism and Disposition March 2006, 34 (3) 398-404; DOI: https://doi.org/10.1124/dmd.105.007682
Maser, Edmund
- You have accessPURIFICATION AND CHARACTERIZATION OF AKR1B10 FROM HUMAN LIVER: ROLE IN CARBONYL REDUCTION OF XENOBIOTICSHans-Jörg Martin, Ursula Breyer-Pfaff, Vladimir Wsol, Simone Venz, Simone Block and Edmund MaserDrug Metabolism and Disposition March 2006, 34 (3) 464-470; DOI: https://doi.org/10.1124/dmd.105.007971
Matsunaga, Naoya
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Maurel, Patrick
- You have accessCHARACTERIZATION OF HUMAN CYTOCHROME P450 ENZYMES INVOLVED IN THE METABOLISM OF THE PIPERIDINE-TYPE PHENOTHIAZINE NEUROLEPTIC THIORIDAZINEJacek Wójcikowski, Patrick Maurel and Władysława A. DanielDrug Metabolism and Disposition March 2006, 34 (3) 471-476; DOI: https://doi.org/10.1124/dmd.105.006445
Mayersohn, Michael
- You have accessRESPONSE TO COMMENTS ON “A MATHEMATICAL DESCRIPTION OF THE FUNCTIONALITY OF CORRECTION FACTORS USED IN ALLOMETRY FOR PREDICTING HUMAN DRUG CLEARANCE”Huadong Tang and Michael MayersohnDrug Metabolism and Disposition March 2006, 34 (3) 510-511; DOI: https://doi.org/10.1124/dmd.105.008359
McCance-Katz, Elinore F.
- You have accessNOVEL METABOLITES OF BUPRENORPHINE DETECTED IN HUMAN LIVER MICROSOMES AND HUMAN URINEYan Chang, David E. Moody and Elinore F. McCance-KatzDrug Metabolism and Disposition March 2006, 34 (3) 440-448; DOI: https://doi.org/10.1124/dmd.105.006148
Miao, Zhuang
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
Miller, Duane D.
- You have accessPHARMACOKINETICS AND METABOLISM OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR IN RATS: IMPLICATION OF MOLECULAR PROPERTIES AND INTENSIVE METABOLIC PROFILE TO INVESTIGATE IDEAL PHARMACOKINETIC CHARACTERISTICS OF A PROPANAMIDE IN PRECLINICAL STUDYDi Wu, Zengru Wu, Jun Yang, Vipin A. Nair, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition March 2006, 34 (3) 483-494; DOI: https://doi.org/10.1124/dmd.105.006643
Miners, John O.
- You have accessSELECTIVITY OF SUBSTRATE (TRIFLUOPERAZINE) AND INHIBITOR (AMITRIPTYLINE, ANDROSTERONE, CANRENOIC ACID, HECOGENIN, PHENYLBUTAZONE, QUINIDINE, QUININE, AND SULFINPYRAZONE) “PROBES” FOR HUMAN UDP-GLUCURONOSYLTRANSFERASESVerawan Uchaipichat, Peter I. Mackenzie, David J. Elliot and John O. MinersDrug Metabolism and Disposition March 2006, 34 (3) 449-456; DOI: https://doi.org/10.1124/dmd.105.007369
Miwa, Gerald T.
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Moody, David E.
- You have accessNOVEL METABOLITES OF BUPRENORPHINE DETECTED IN HUMAN LIVER MICROSOMES AND HUMAN URINEYan Chang, David E. Moody and Elinore F. McCance-KatzDrug Metabolism and Disposition March 2006, 34 (3) 440-448; DOI: https://doi.org/10.1124/dmd.105.006148
Morgan, Edward T.
- You have accessEXPRESSION OF UDP-GLUCURONOSYLTRANSFERASE ISOFORM mRNAS DURING INFLAMMATION AND INFECTION IN MOUSE LIVER AND KIDNEYTerrilyn A. Richardson, Melanie Sherman, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 351-353; DOI: https://doi.org/10.1124/dmd.105.007435
- You have accessHEPATIC AND RENAL CYTOCHROME P450 GENE REGULATION DURING CITROBACTER RODENTIUM INFECTION IN WILD-TYPE AND TOLL-LIKE RECEPTOR 4 MUTANT MICETerrilyn A. Richardson, Melanie Sherman, Leposava Antonovic, Sean S. Kardar, Henry W. Strobel, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 354-360; DOI: https://doi.org/10.1124/dmd.105.007393
Mosqueda-Garcia, Rogelio
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
Muralidhara, Srinivasa
- You have accessONTOGENY OF HEPATIC AND PLASMA METABOLISM OF DELTAMETHRIN IN VITRO: ROLE IN AGE-DEPENDENT ACUTE NEUROTOXICITYSathanandam S. Anand, Kyu-Bong Kim, Stephanie Padilla, Srinivasa Muralidhara, Hyo J. Kim, Jeffrey W. Fisher and James V. BrucknerDrug Metabolism and Disposition March 2006, 34 (3) 389-397; DOI: https://doi.org/10.1124/dmd.105.007807
N
Nagaraja, Nelamangala V.
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Nair, Vipin A.
- You have accessPHARMACOKINETICS AND METABOLISM OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR IN RATS: IMPLICATION OF MOLECULAR PROPERTIES AND INTENSIVE METABOLIC PROFILE TO INVESTIGATE IDEAL PHARMACOKINETIC CHARACTERISTICS OF A PROPANAMIDE IN PRECLINICAL STUDYDi Wu, Zengru Wu, Jun Yang, Vipin A. Nair, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition March 2006, 34 (3) 483-494; DOI: https://doi.org/10.1124/dmd.105.006643
Nakamura, Masato
- You have accessIN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTMasato Nakamura, Yasunori Kawakita, Akito Yasuhara, Yoshiki Fukasawa, Koji Yoshida, Kazunari Sakagami and Atsuro NakazatoDrug Metabolism and Disposition March 2006, 34 (3) 369-374; DOI: https://doi.org/10.1124/dmd.105.006213
Nakazato, Atsuro
- You have accessIN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTMasato Nakamura, Yasunori Kawakita, Akito Yasuhara, Yoshiki Fukasawa, Koji Yoshida, Kazunari Sakagami and Atsuro NakazatoDrug Metabolism and Disposition March 2006, 34 (3) 369-374; DOI: https://doi.org/10.1124/dmd.105.006213
Nikolskaya, Tatiana
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
O
Ogikubo, Tetsuya
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Okumura, Manabu
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
P
Padilla, Stephanie
- You have accessONTOGENY OF HEPATIC AND PLASMA METABOLISM OF DELTAMETHRIN IN VITRO: ROLE IN AGE-DEPENDENT ACUTE NEUROTOXICITYSathanandam S. Anand, Kyu-Bong Kim, Stephanie Padilla, Srinivasa Muralidhara, Hyo J. Kim, Jeffrey W. Fisher and James V. BrucknerDrug Metabolism and Disposition March 2006, 34 (3) 389-397; DOI: https://doi.org/10.1124/dmd.105.007807
Pai, Harish V.
- You have accessRESPONSE TO COMMENTS ON HOSKINS ET AL. [(2005) DRUG METAB DISPOS 33:1564–1565]Harish V. Pai and Vijayalakshmi RavindranathDrug Metabolism and Disposition March 2006, 34 (3) 506; DOI: https://doi.org/10.1124/dmd.105.008862
Pantze, Michael P.
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
Petrick, Jay S.
- You have accessTISSUE DISTRIBUTION AND ONTOGENY OF ORGANIC CATION TRANSPORTERS IN MICEYazen Alnouti, Jay S. Petrick and Curtis D. KlaassenDrug Metabolism and Disposition March 2006, 34 (3) 477-482; DOI: https://doi.org/10.1124/dmd.105.006932
Philipp, Thomas
- You have accessDIGITAL FLUORESCENCE IMAGING OF ORGANIC CATION TRANSPORT IN FRESHLY ISOLATED RAT PROXIMAL TUBULESFrank Pietruck, Markus Horbelt, Thorsten Feldkamp, Katrin Engeln, Stefan Herget-Rosenthal, Thomas Philipp and Andreas KribbenDrug Metabolism and Disposition March 2006, 34 (3) 339-342; DOI: https://doi.org/10.1124/dmd.105.006403
Pietruck, Frank
- You have accessDIGITAL FLUORESCENCE IMAGING OF ORGANIC CATION TRANSPORT IN FRESHLY ISOLATED RAT PROXIMAL TUBULESFrank Pietruck, Markus Horbelt, Thorsten Feldkamp, Katrin Engeln, Stefan Herget-Rosenthal, Thomas Philipp and Andreas KribbenDrug Metabolism and Disposition March 2006, 34 (3) 339-342; DOI: https://doi.org/10.1124/dmd.105.006403
Pilloff, Daniel E.
- You have accessSULFATION OF RALOXIFENE AND 4-HYDROXYTAMOXIFEN BY HUMAN CYTOSOLIC SULFOTRANSFERASESJosie L. Falany, Daniel E. Pilloff, Thomas S. Leyh and Charles N. FalanyDrug Metabolism and Disposition March 2006, 34 (3) 361-368; DOI: https://doi.org/10.1124/dmd.105.006551
Piquette-Miller, Micheline
- You have accessTHE ROLE OF PREGNANE X RECEPTOR IN 2-ACETYLAMINOFLUORENE-MEDIATED INDUCTION OF DRUG TRANSPORT AND -METABOLIZING ENZYMES IN MICEAlexander Anapolsky, Shirley Teng, Santosh Dixit and Micheline Piquette-MillerDrug Metabolism and Disposition March 2006, 34 (3) 405-409; DOI: https://doi.org/10.1124/dmd.105.006197
Prakash, Chandra
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
Q
Qian, Mark G.
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
R
Rakhit, Ashok
- You have accessMETABOLISM AND EXCRETION OF ERLOTINIB, A SMALL MOLECULE INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE, IN HEALTHY MALE VOLUNTEERSJie Ling, Kim A. Johnson, Zhuang Miao, Ashok Rakhit, Michael P. Pantze, Marta Hamilton, Bert L. Lum and Chandra PrakashDrug Metabolism and Disposition March 2006, 34 (3) 420-426; DOI: https://doi.org/10.1124/dmd.105.007765
Rakhmatulin, Eugene A.
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
Ravindranath, Vijayalakshmi
- You have accessRESPONSE TO COMMENTS ON HOSKINS ET AL. [(2005) DRUG METAB DISPOS 33:1564–1565]Harish V. Pai and Vijayalakshmi RavindranathDrug Metabolism and Disposition March 2006, 34 (3) 506; DOI: https://doi.org/10.1124/dmd.105.008862
Richardson, Terrilyn A.
- You have accessEXPRESSION OF UDP-GLUCURONOSYLTRANSFERASE ISOFORM mRNAS DURING INFLAMMATION AND INFECTION IN MOUSE LIVER AND KIDNEYTerrilyn A. Richardson, Melanie Sherman, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 351-353; DOI: https://doi.org/10.1124/dmd.105.007435
- You have accessHEPATIC AND RENAL CYTOCHROME P450 GENE REGULATION DURING CITROBACTER RODENTIUM INFECTION IN WILD-TYPE AND TOLL-LIKE RECEPTOR 4 MUTANT MICETerrilyn A. Richardson, Melanie Sherman, Leposava Antonovic, Sean S. Kardar, Henry W. Strobel, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 354-360; DOI: https://doi.org/10.1124/dmd.105.007393
Ryabov, Andy
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
S
Sakagami, Kazunari
- You have accessIN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTMasato Nakamura, Yasunori Kawakita, Akito Yasuhara, Yoshiki Fukasawa, Koji Yoshida, Kazunari Sakagami and Atsuro NakazatoDrug Metabolism and Disposition March 2006, 34 (3) 369-374; DOI: https://doi.org/10.1124/dmd.105.006213
Sallovitz, J.
- You have accessMODULATION OF THE P-GLYCOPROTEIN-MEDIATED INTESTINAL SECRETION OF IVERMECTIN: IN VITRO AND IN VIVO ASSESSMENTSM. Ballent, A. Lifschitz, G. Virkel, J. Sallovitz and C. LanusseDrug Metabolism and Disposition March 2006, 34 (3) 457-463; DOI: https://doi.org/10.1124/dmd.105.007757
Sedmera, David
- You have accessBENZO[A]PYRENE-INDUCED ORAL CARCINOGENESIS AND CHEMOPREVENTION: STUDIES IN BIOENGINEERED HUMAN TISSUEThomas Walle, U. Kristina Walle, David Sedmera and Mitch KlausnerDrug Metabolism and Disposition March 2006, 34 (3) 346-350; DOI: https://doi.org/10.1124/dmd.105.007948
Setoguchi, Nao
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Shapiro, Bernard H.
- You have accessINDUCIBILITY OF MALE-SPECIFIC ISOFORMS OF CYTOCHROME P450 BY SEX-DEPENDENT GROWTH HORMONE PROFILES IN HEPATOCYTE CULTURES FROM MALE BUT NOT FEMALE RATSChellappagounder Thangavel, Wojciech Dworakowski and Bernard H. ShapiroDrug Metabolism and Disposition March 2006, 34 (3) 410-419; DOI: https://doi.org/10.1124/dmd.105.007716
Shebley, Mohamad
- You have accessSELECTIVE PATHWAYS FOR THE METABOLISM OF PHENCYCLIDINE BY CYTOCHROME P450 2B ENZYMES: IDENTIFICATION OF ELECTROPHILIC METABOLITES, GLUTATHIONE, AND N-ACETYL CYSTEINE ADDUCTSMohamad Shebley, Monica I. Jushchyshyn and Paul F. HollenbergDrug Metabolism and Disposition March 2006, 34 (3) 375-383; DOI: https://doi.org/10.1124/dmd.105.007047
Sherman, Melanie
- You have accessEXPRESSION OF UDP-GLUCURONOSYLTRANSFERASE ISOFORM mRNAS DURING INFLAMMATION AND INFECTION IN MOUSE LIVER AND KIDNEYTerrilyn A. Richardson, Melanie Sherman, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 351-353; DOI: https://doi.org/10.1124/dmd.105.007435
- You have accessHEPATIC AND RENAL CYTOCHROME P450 GENE REGULATION DURING CITROBACTER RODENTIUM INFECTION IN WILD-TYPE AND TOLL-LIKE RECEPTOR 4 MUTANT MICETerrilyn A. Richardson, Melanie Sherman, Leposava Antonovic, Sean S. Kardar, Henry W. Strobel, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 354-360; DOI: https://doi.org/10.1124/dmd.105.007393
Shimoga, Prakash R.
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Sorokina, Svetlana
- You have accessA COMBINED APPROACH TO DRUG METABOLISM AND TOXICITY ASSESSMENTSean Ekins, Sergey Andreyev, Andy Ryabov, Eugene Kirillov, Eugene A. Rakhmatulin, Svetlana Sorokina, Andrej Bugrim and Tatiana NikolskayaDrug Metabolism and Disposition March 2006, 34 (3) 495-503; DOI: https://doi.org/10.1124/dmd.105.008458
Strobel, Henry W.
- You have accessHEPATIC AND RENAL CYTOCHROME P450 GENE REGULATION DURING CITROBACTER RODENTIUM INFECTION IN WILD-TYPE AND TOLL-LIKE RECEPTOR 4 MUTANT MICETerrilyn A. Richardson, Melanie Sherman, Leposava Antonovic, Sean S. Kardar, Henry W. Strobel, Daniel Kalman and Edward T. MorganDrug Metabolism and Disposition March 2006, 34 (3) 354-360; DOI: https://doi.org/10.1124/dmd.105.007393
Swaminathan, Arun
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
T
Taketani, Megumi
- You have accessFIRST-PASS HYDROLYSIS OF A PROPRANOLOL ESTER DERIVATIVE IN RAT SMALL INTESTINEKenji Masaki, Megumi Taketani and Teruko ImaiDrug Metabolism and Disposition March 2006, 34 (3) 398-404; DOI: https://doi.org/10.1124/dmd.105.007682
Tang, Huadong
- You have accessRESPONSE TO COMMENTS ON “A MATHEMATICAL DESCRIPTION OF THE FUNCTIONALITY OF CORRECTION FACTORS USED IN ALLOMETRY FOR PREDICTING HUMAN DRUG CLEARANCE”Huadong Tang and Michael MayersohnDrug Metabolism and Disposition March 2006, 34 (3) 510-511; DOI: https://doi.org/10.1124/dmd.105.008359
Teng, Shirley
- You have accessTHE ROLE OF PREGNANE X RECEPTOR IN 2-ACETYLAMINOFLUORENE-MEDIATED INDUCTION OF DRUG TRANSPORT AND -METABOLIZING ENZYMES IN MICEAlexander Anapolsky, Shirley Teng, Santosh Dixit and Micheline Piquette-MillerDrug Metabolism and Disposition March 2006, 34 (3) 405-409; DOI: https://doi.org/10.1124/dmd.105.006197
Thangavel, Chellappagounder
- You have accessINDUCIBILITY OF MALE-SPECIFIC ISOFORMS OF CYTOCHROME P450 BY SEX-DEPENDENT GROWTH HORMONE PROFILES IN HEPATOCYTE CULTURES FROM MALE BUT NOT FEMALE RATSChellappagounder Thangavel, Wojciech Dworakowski and Bernard H. ShapiroDrug Metabolism and Disposition March 2006, 34 (3) 410-419; DOI: https://doi.org/10.1124/dmd.105.007716
U
Uchaipichat, Verawan
- You have accessSELECTIVITY OF SUBSTRATE (TRIFLUOPERAZINE) AND INHIBITOR (AMITRIPTYLINE, ANDROSTERONE, CANRENOIC ACID, HECOGENIN, PHENYLBUTAZONE, QUINIDINE, QUININE, AND SULFINPYRAZONE) “PROBES” FOR HUMAN UDP-GLUCURONOSYLTRANSFERASESVerawan Uchaipichat, Peter I. Mackenzie, David J. Elliot and John O. MinersDrug Metabolism and Disposition March 2006, 34 (3) 449-456; DOI: https://doi.org/10.1124/dmd.105.007369
V
Venz, Simone
- You have accessPURIFICATION AND CHARACTERIZATION OF AKR1B10 FROM HUMAN LIVER: ROLE IN CARBONYL REDUCTION OF XENOBIOTICSHans-Jörg Martin, Ursula Breyer-Pfaff, Vladimir Wsol, Simone Venz, Simone Block and Edmund MaserDrug Metabolism and Disposition March 2006, 34 (3) 464-470; DOI: https://doi.org/10.1124/dmd.105.007971
Virkel, G.
- You have accessMODULATION OF THE P-GLYCOPROTEIN-MEDIATED INTESTINAL SECRETION OF IVERMECTIN: IN VITRO AND IN VIVO ASSESSMENTSM. Ballent, A. Lifschitz, G. Virkel, J. Sallovitz and C. LanusseDrug Metabolism and Disposition March 2006, 34 (3) 457-463; DOI: https://doi.org/10.1124/dmd.105.007757
W
Walle, Thomas
- You have accessBENZO[A]PYRENE-INDUCED ORAL CARCINOGENESIS AND CHEMOPREVENTION: STUDIES IN BIOENGINEERED HUMAN TISSUEThomas Walle, U. Kristina Walle, David Sedmera and Mitch KlausnerDrug Metabolism and Disposition March 2006, 34 (3) 346-350; DOI: https://doi.org/10.1124/dmd.105.007948
Walle, U. Kristina
- You have accessBENZO[A]PYRENE-INDUCED ORAL CARCINOGENESIS AND CHEMOPREVENTION: STUDIES IN BIOENGINEERED HUMAN TISSUEThomas Walle, U. Kristina Walle, David Sedmera and Mitch KlausnerDrug Metabolism and Disposition March 2006, 34 (3) 346-350; DOI: https://doi.org/10.1124/dmd.105.007948
Wang, Lifei
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
Wójcikowski, Jacek
- You have accessCHARACTERIZATION OF HUMAN CYTOCHROME P450 ENZYMES INVOLVED IN THE METABOLISM OF THE PIPERIDINE-TYPE PHENOTHIAZINE NEUROLEPTIC THIORIDAZINEJacek Wójcikowski, Patrick Maurel and Władysława A. DanielDrug Metabolism and Disposition March 2006, 34 (3) 471-476; DOI: https://doi.org/10.1124/dmd.105.006445
Wsol, Vladimir
- You have accessPURIFICATION AND CHARACTERIZATION OF AKR1B10 FROM HUMAN LIVER: ROLE IN CARBONYL REDUCTION OF XENOBIOTICSHans-Jörg Martin, Ursula Breyer-Pfaff, Vladimir Wsol, Simone Venz, Simone Block and Edmund MaserDrug Metabolism and Disposition March 2006, 34 (3) 464-470; DOI: https://doi.org/10.1124/dmd.105.007971
Wu, Di
- You have accessPHARMACOKINETICS AND METABOLISM OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR IN RATS: IMPLICATION OF MOLECULAR PROPERTIES AND INTENSIVE METABOLIC PROFILE TO INVESTIGATE IDEAL PHARMACOKINETIC CHARACTERISTICS OF A PROPANAMIDE IN PRECLINICAL STUDYDi Wu, Zengru Wu, Jun Yang, Vipin A. Nair, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition March 2006, 34 (3) 483-494; DOI: https://doi.org/10.1124/dmd.105.006643
Wu, Jing-Tao
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Wu, Shung
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
Wu, Zengru
- You have accessPHARMACOKINETICS AND METABOLISM OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR IN RATS: IMPLICATION OF MOLECULAR PROPERTIES AND INTENSIVE METABOLIC PROFILE TO INVESTIGATE IDEAL PHARMACOKINETIC CHARACTERISTICS OF A PROPANAMIDE IN PRECLINICAL STUDYDi Wu, Zengru Wu, Jun Yang, Vipin A. Nair, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition March 2006, 34 (3) 483-494; DOI: https://doi.org/10.1124/dmd.105.006643
X
Xue, Yongjun
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
Y
Yamasaki, Keishi
- You have accessTRANSIENT INHIBITION OF CYP3A IN RATS BY STAR FRUIT JUICEMuneaki Hidaka, Manabu Okumura, Tetsuya Ogikubo, Hirofumi Kai, Ken-Ichi Fujita, Tomomi Iwakiri, Keishi Yamasaki, Nao Setoguchi, Naoya Matsunaga and Kazuhiko ArimoriDrug Metabolism and Disposition March 2006, 34 (3) 343-345; DOI: https://doi.org/10.1124/dmd.105.006486
Yang, Hua
- You have accessEVALUATION OF MICRODOSING TO ASSESS PHARMACOKINETIC LINEARITY IN RATS USING LIQUID CHROMATOGRAPHY-TANDEM MASS SPECTROMETRYSuresh K. Balani, Nelamangala V. Nagaraja, Mark G. Qian, Arnaldo O. Costa, J. Scott Daniels, Hua Yang, Prakash R. Shimoga, Jing-Tao Wu, Liang-Shang Gan, Frank W. Lee and Gerald T. MiwaDrug Metabolism and Disposition March 2006, 34 (3) 384-388; DOI: https://doi.org/10.1124/dmd.105.007195
Yang, Jun
- You have accessPHARMACOKINETICS AND METABOLISM OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR IN RATS: IMPLICATION OF MOLECULAR PROPERTIES AND INTENSIVE METABOLIC PROFILE TO INVESTIGATE IDEAL PHARMACOKINETIC CHARACTERISTICS OF A PROPANAMIDE IN PRECLINICAL STUDYDi Wu, Zengru Wu, Jun Yang, Vipin A. Nair, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition March 2006, 34 (3) 483-494; DOI: https://doi.org/10.1124/dmd.105.006643
Yasuhara, Akito
- You have accessIN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTMasato Nakamura, Yasunori Kawakita, Akito Yasuhara, Yoshiki Fukasawa, Koji Yoshida, Kazunari Sakagami and Atsuro NakazatoDrug Metabolism and Disposition March 2006, 34 (3) 369-374; DOI: https://doi.org/10.1124/dmd.105.006213
Yoshida, Koji
- You have accessIN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTMasato Nakamura, Yasunori Kawakita, Akito Yasuhara, Yoshiki Fukasawa, Koji Yoshida, Kazunari Sakagami and Atsuro NakazatoDrug Metabolism and Disposition March 2006, 34 (3) 369-374; DOI: https://doi.org/10.1124/dmd.105.006213
Z
Zhang, Donglu
- You have accessGLUCURONIDATION AS A MAJOR METABOLIC CLEARANCE PATHWAY OF 14C-LABELED MURAGLITAZAR IN HUMANS: METABOLIC PROFILES IN SUBJECTS WITH OR WITHOUT BILE COLLECTIONLifei Wang, Donglu Zhang, Arun Swaminathan, Yongjun Xue, Peter T. Cheng, Shung Wu, Rogelio Mosqueda-Garcia, Catherine Aurang, Donald W. Everett and W. Griffith HumphreysDrug Metabolism and Disposition March 2006, 34 (3) 427-439; DOI: https://doi.org/10.1124/dmd.105.007617
In this issue

Advertisement