Index by author
April 01, 2006; Volume 34,Issue 4
A
Abdelmegeed, Mohamed A.
- You have accessTHE MITOGEN-ACTIVATED PROTEIN KINASE KINASE (MEK) INHIBITOR PD98059 ELEVATES PRIMARY CULTURED RAT HEPATOCYTE GLUTATHIONE LEVELS INDEPENDENT OF INHIBITING MEKSang K. Kim, Mohamed A. Abdelmegeed and Raymond F. NovakDrug Metabolism and Disposition April 2006, 34 (4) 683-689; DOI: https://doi.org/10.1124/dmd.105.007666
Abildskov, Kirsten M.
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Alander, Sarah W.
- You have accessCYP2D6*36 GENE ARRANGEMENTS WITHIN THE CYP2D6 LOCUS: ASSOCIATION OF CYP2D6*36 WITH POOR METABOLIZER STATUSAndrea Gaedigk, L. DiAnne Bradford, Sarah W. Alander and J. Steven LeederDrug Metabolism and Disposition April 2006, 34 (4) 563-569; DOI: https://doi.org/10.1124/dmd.105.008292
Álvarez, Ana I.
- You have accessBREAST CANCER RESISTANCE PROTEIN (BCRP/ABCG2) TRANSPORTS FLUOROQUINOLONE ANTIBIOTICS AND AFFECTS THEIR ORAL AVAILABILITY, PHARMACOKINETICS, AND MILK SECRETIONGracia Merino, Ana I. Álvarez, Mivis M. Pulido, Antonio J. Molina, Alfred H. Schinkel and Julio G. PrietoDrug Metabolism and Disposition April 2006, 34 (4) 690-695; DOI: https://doi.org/10.1124/dmd.105.008219
Anderson, Bradley D.
- You have accessDEPENDENCE OF NELFINAVIR BRAIN UPTAKE ON DOSE AND TISSUE CONCENTRATIONS OF THE SELECTIVE P-GLYCOPROTEIN INHIBITOR ZOSUQUIDAR IN RATSBradley D. Anderson, Melissa J. May, Sherri Jordan, Lin Song, Michael J. Roberts and Markos LeggasDrug Metabolism and Disposition April 2006, 34 (4) 653-659; DOI: https://doi.org/10.1124/dmd.105.006536
Anderson, Gail D.
- You have accessINTERACTIONS OF AMOXICILLIN AND CEFACLOR WITH HUMAN RENAL ORGANIC ANION AND PEPTIDE TRANSPORTERSMeng Li, Gail D. Anderson, Brian R. Phillips, Wei Kong, Danny D. Shen and Joanne WangDrug Metabolism and Disposition April 2006, 34 (4) 547-555; DOI: https://doi.org/10.1124/dmd.105.006791
Arroyo, Sylvia E.
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Austin, R. P.
- You have accessRESPONSE TO “BINDING OF DRUGS TO HEPATIC MICROSOMES: COMMENT AND ASSESSMENT OF CURRENT PREDICTION METHODOLOGY WITH RECOMMENDATION FOR IMPROVEMENT”R. P. Austin, P. Barton and R. J. RileyDrug Metabolism and Disposition April 2006, 34 (4) 727; DOI: https://doi.org/10.1124/dmd.105.009142
B
Backes, Wayne L.
- You have accessAN EVALUATION OF METHODS FOR THE RECONSTITUTION OF CYTOCHROMES P450 AND NADPH P450 REDUCTASE INTO LIPID VESICLESJames R. Reed, Rusty W. Kelley and Wayne L. BackesDrug Metabolism and Disposition April 2006, 34 (4) 660-666; DOI: https://doi.org/10.1124/dmd.105.006825
Barton, P.
- You have accessRESPONSE TO “BINDING OF DRUGS TO HEPATIC MICROSOMES: COMMENT AND ASSESSMENT OF CURRENT PREDICTION METHODOLOGY WITH RECOMMENDATION FOR IMPROVEMENT”R. P. Austin, P. Barton and R. J. RileyDrug Metabolism and Disposition April 2006, 34 (4) 727; DOI: https://doi.org/10.1124/dmd.105.009142
Benzeroual, Kenza
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Bier, Dirk
- You have accessMETABOLISM OF THE A1 ADENOSINE RECEPTOR POSITRON EMISSION TOMOGRAPHY LIGAND [18F]8-CYCLOPENTYL-3-(3-FLUOROPROPYL)-1-PROPYLXANTHINE ([18F]CPFPX) IN RODENTS AND HUMANSDirk Bier, Marcus H. Holschbach, Walter Wutz, Ray A. Olsson and Heinz H. CoenenDrug Metabolism and Disposition April 2006, 34 (4) 570-576; DOI: https://doi.org/10.1124/dmd.105.006411
Biot, Christophe
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Bourrié, Martine
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Bowlin, Stephen
- You have accessIN VITRO METABOLIC ACTIVATION OF THIABENDAZOLE VIA 5-HYDROXYTHIABENDAZOLE: IDENTIFICATION OF A GLUTATHIONE CONJUGATE OF 5-HYDROXYTHIABENDAZOLEDeepak Dalvie, Evan Smith, Alan Deese and Stephen BowlinDrug Metabolism and Disposition April 2006, 34 (4) 709-717; DOI: https://doi.org/10.1124/dmd.105.008094
Bradford, L. DiAnne
- You have accessCYP2D6*36 GENE ARRANGEMENTS WITHIN THE CYP2D6 LOCUS: ASSOCIATION OF CYP2D6*36 WITH POOR METABOLIZER STATUSAndrea Gaedigk, L. DiAnne Bradford, Sarah W. Alander and J. Steven LeederDrug Metabolism and Disposition April 2006, 34 (4) 563-569; DOI: https://doi.org/10.1124/dmd.105.008292
Brocard, Jacques
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Brouwer, Kim L. R.
- You have accessCHARACTERIZATION OF TRANSPORT PROTEIN EXPRESSION IN MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) 2-DEFICIENT RATSBrendan M. Johnson, Peijin Zhang, John D. Schuetz and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 556-562; DOI: https://doi.org/10.1124/dmd.105.005793
- You have accessALTERED HEPATOBILIARY DISPOSITION OF 5 (AND 6)-CARBOXY-2′,7′-DICHLOROFLUORESCEIN IN Abcg2 (Bcrp1) AND Abcc2 (Mrp2) KNOCKOUT MICEKen-ichi Nezasa, Xianbin Tian, Maciej J. Zamek-Gliszczynski, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 718-723; DOI: https://doi.org/10.1124/dmd.105.007922
Brown, Simon
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
C
Camacho, Raquel
- You have accessEMPIRICAL VALIDATION OF A RAT IN VITRO ORGAN SLICE MODEL AS A TOOL FOR IN VIVO CLEARANCE PREDICTIONInge A. M. de Graaf, Ruben de Kanter, Marina H. de Jager, Raquel Camacho, Elise Langenkamp, Esther G. van de Kerkhof and Geny M. M. GroothuisDrug Metabolism and Disposition April 2006, 34 (4) 591-599; DOI: https://doi.org/10.1124/dmd.105.006726
Caspersen, Casper S.
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Cha, In-June
- You have accessINHIBITORY EFFECTS OF FRUIT JUICES ON CYP3A ACTIVITYHyunmi Kim, Yune-Jung Yoon, Ji-Hong Shon, In-June Cha, Jae-Gook Shin and Kwang-Hyeon LiuDrug Metabolism and Disposition April 2006, 34 (4) 521-523; DOI: https://doi.org/10.1124/dmd.105.007930
Chiron, Catherine
- You have accessIN VITRO AND IN VIVO INHIBITORY EFFECT OF STIRIPENTOL ON CLOBAZAM METABOLISMCarole Giraud, Jean-Marc Treluyer, Elisabeth Rey, Catherine Chiron, Jean Vincent, Gérard Pons and Agnès TranDrug Metabolism and Disposition April 2006, 34 (4) 608-611; DOI: https://doi.org/10.1124/dmd.105.007237
Chowdhury, Swapan K.
- You have accessIDENTIFICATION OF HUMAN LIVER CYTOCHROME P450 ENZYMES RESPONSIBLE FOR THE METABOLISM OF LONAFARNIB (SARASAR)Anima Ghosal, Swapan K. Chowdhury, Wei Tong, Neil Hapangama, Yuan Yuan, Ai-Duen Su and Shmuel ZbaidaDrug Metabolism and Disposition April 2006, 34 (4) 628-635; DOI: https://doi.org/10.1124/dmd.105.007906
Coenen, Heinz H.
- You have accessMETABOLISM OF THE A1 ADENOSINE RECEPTOR POSITRON EMISSION TOMOGRAPHY LIGAND [18F]8-CYCLOPENTYL-3-(3-FLUOROPROPYL)-1-PROPYLXANTHINE ([18F]CPFPX) IN RODENTS AND HUMANSDirk Bier, Marcus H. Holschbach, Walter Wutz, Ray A. Olsson and Heinz H. CoenenDrug Metabolism and Disposition April 2006, 34 (4) 570-576; DOI: https://doi.org/10.1124/dmd.105.006411
Cole, Susan P. C.
- You have accessMUTATIONAL ANALYSIS OF POLAR AMINO ACID RESIDUES WITHIN PREDICTED TRANSMEMBRANE HELICES 10 AND 16 OF MULTIDRUG RESISTANCE PROTEIN 1 (ABCC1): EFFECT ON SUBSTRATE SPECIFICITYDa-Wei Zhang, Kenichi Nunoya, Monika Vasa, Hong-Mei Gu, Susan P. C. Cole and Roger G. DeeleyDrug Metabolism and Disposition April 2006, 34 (4) 539-546; DOI: https://doi.org/10.1124/dmd.105.007740
D
Daher, Wassim
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Dalvie, Deepak
- You have accessIN VITRO METABOLIC ACTIVATION OF THIABENDAZOLE VIA 5-HYDROXYTHIABENDAZOLE: IDENTIFICATION OF A GLUTATHIONE CONJUGATE OF 5-HYDROXYTHIABENDAZOLEDeepak Dalvie, Evan Smith, Alan Deese and Stephen BowlinDrug Metabolism and Disposition April 2006, 34 (4) 709-717; DOI: https://doi.org/10.1124/dmd.105.008094
Daniel, Salha S.
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Deeley, Roger G.
- You have accessMUTATIONAL ANALYSIS OF POLAR AMINO ACID RESIDUES WITHIN PREDICTED TRANSMEMBRANE HELICES 10 AND 16 OF MULTIDRUG RESISTANCE PROTEIN 1 (ABCC1): EFFECT ON SUBSTRATE SPECIFICITYDa-Wei Zhang, Kenichi Nunoya, Monika Vasa, Hong-Mei Gu, Susan P. C. Cole and Roger G. DeeleyDrug Metabolism and Disposition April 2006, 34 (4) 539-546; DOI: https://doi.org/10.1124/dmd.105.007740
Deese, Alan
- You have accessIN VITRO METABOLIC ACTIVATION OF THIABENDAZOLE VIA 5-HYDROXYTHIABENDAZOLE: IDENTIFICATION OF A GLUTATHIONE CONJUGATE OF 5-HYDROXYTHIABENDAZOLEDeepak Dalvie, Evan Smith, Alan Deese and Stephen BowlinDrug Metabolism and Disposition April 2006, 34 (4) 709-717; DOI: https://doi.org/10.1124/dmd.105.008094
de Graaf, Inge A. M.
- You have accessEMPIRICAL VALIDATION OF A RAT IN VITRO ORGAN SLICE MODEL AS A TOOL FOR IN VIVO CLEARANCE PREDICTIONInge A. M. de Graaf, Ruben de Kanter, Marina H. de Jager, Raquel Camacho, Elise Langenkamp, Esther G. van de Kerkhof and Geny M. M. GroothuisDrug Metabolism and Disposition April 2006, 34 (4) 591-599; DOI: https://doi.org/10.1124/dmd.105.006726
de Jager, Marina H.
- You have accessEMPIRICAL VALIDATION OF A RAT IN VITRO ORGAN SLICE MODEL AS A TOOL FOR IN VIVO CLEARANCE PREDICTIONInge A. M. de Graaf, Ruben de Kanter, Marina H. de Jager, Raquel Camacho, Elise Langenkamp, Esther G. van de Kerkhof and Geny M. M. GroothuisDrug Metabolism and Disposition April 2006, 34 (4) 591-599; DOI: https://doi.org/10.1124/dmd.105.006726
de Kanter, Ruben
- You have accessEMPIRICAL VALIDATION OF A RAT IN VITRO ORGAN SLICE MODEL AS A TOOL FOR IN VIVO CLEARANCE PREDICTIONInge A. M. de Graaf, Ruben de Kanter, Marina H. de Jager, Raquel Camacho, Elise Langenkamp, Esther G. van de Kerkhof and Geny M. M. GroothuisDrug Metabolism and Disposition April 2006, 34 (4) 591-599; DOI: https://doi.org/10.1124/dmd.105.006726
Dive, Daniel
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Dreisbach, Annette
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
E
Eckstein, James A.
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Eikel, Daniel
- You have accessS-2-PENTYL-4-PENTYNOIC HYDROXAMIC ACID AND ITS METABOLITE S-2-PENTYL-4-PENTYNOIC ACID IN THE NMRI-EXENCEPHALY-MOUSE MODEL: PHARMACOKINETIC PROFILES, TERATOGENIC EFFECTS, AND HISTONE DEACETYLASE INHIBITION ABILITIES OF FURTHER VALPROIC ACID HYDROXAMATES AND AMIDESDaniel Eikel, Katrin Hoffmann, Karolin Zoll, Alfonso Lampen and Heinz NauDrug Metabolism and Disposition April 2006, 34 (4) 612-620; DOI: https://doi.org/10.1124/dmd.105.008078
F
Fabre, Gérard
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Farid, Nagy A.
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Fraisse, Laurent
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Fuchikami, Hiromi
- You have accessEFFECTS OF HERBAL EXTRACTS ON THE FUNCTION OF HUMAN ORGANIC ANION-TRANSPORTING POLYPEPTIDE OATP-BHiromi Fuchikami, Hiroki Satoh, Masayuki Tsujimoto, Shigehiro Ohdo, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition April 2006, 34 (4) 577-582; DOI: https://doi.org/10.1124/dmd.105.007872
Fusch, Christoph
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
G
Gaedigk, Andrea
- You have accessCYP2D6*36 GENE ARRANGEMENTS WITHIN THE CYP2D6 LOCUS: ASSOCIATION OF CYP2D6*36 WITH POOR METABOLIZER STATUSAndrea Gaedigk, L. DiAnne Bradford, Sarah W. Alander and J. Steven LeederDrug Metabolism and Disposition April 2006, 34 (4) 563-569; DOI: https://doi.org/10.1124/dmd.105.008292
Gallegos, Richard
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
Gan, Liang-Shang
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
Garland, Marianne
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Ghosal, Anima
- You have accessIDENTIFICATION OF HUMAN LIVER CYTOCHROME P450 ENZYMES RESPONSIBLE FOR THE METABOLISM OF LONAFARNIB (SARASAR)Anima Ghosal, Swapan K. Chowdhury, Wei Tong, Neil Hapangama, Yuan Yuan, Ai-Duen Su and Shmuel ZbaidaDrug Metabolism and Disposition April 2006, 34 (4) 628-635; DOI: https://doi.org/10.1124/dmd.105.007906
Giraud, Carole
- You have accessIN VITRO AND IN VIVO INHIBITORY EFFECT OF STIRIPENTOL ON CLOBAZAM METABOLISMCarole Giraud, Jean-Marc Treluyer, Elisabeth Rey, Catherine Chiron, Jean Vincent, Gérard Pons and Agnès TranDrug Metabolism and Disposition April 2006, 34 (4) 608-611; DOI: https://doi.org/10.1124/dmd.105.007237
Groothuis, Geny M. M.
- You have accessEMPIRICAL VALIDATION OF A RAT IN VITRO ORGAN SLICE MODEL AS A TOOL FOR IN VIVO CLEARANCE PREDICTIONInge A. M. de Graaf, Ruben de Kanter, Marina H. de Jager, Raquel Camacho, Elise Langenkamp, Esther G. van de Kerkhof and Geny M. M. GroothuisDrug Metabolism and Disposition April 2006, 34 (4) 591-599; DOI: https://doi.org/10.1124/dmd.105.006726
Grube, Markus
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
Gu, Hong-Mei
- You have accessMUTATIONAL ANALYSIS OF POLAR AMINO ACID RESIDUES WITHIN PREDICTED TRANSMEMBRANE HELICES 10 AND 16 OF MULTIDRUG RESISTANCE PROTEIN 1 (ABCC1): EFFECT ON SUBSTRATE SPECIFICITYDa-Wei Zhang, Kenichi Nunoya, Monika Vasa, Hong-Mei Gu, Susan P. C. Cole and Roger G. DeeleyDrug Metabolism and Disposition April 2006, 34 (4) 539-546; DOI: https://doi.org/10.1124/dmd.105.007740
Guillou, François
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
H
Hallifax, David
- You have accessBINDING OF DRUGS TO HEPATIC MICROSOMES: COMMENT AND ASSESSMENT OF CURRENT PREDICTION METHODOLOGY WITH RECOMMENDATION FOR IMPROVEMENTDavid Hallifax and J. Brian HoustonDrug Metabolism and Disposition April 2006, 34 (4) 724-726; DOI: https://doi.org/10.1124/dmd.105.007658
Hapangama, Neil
- You have accessIDENTIFICATION OF HUMAN LIVER CYTOCHROME P450 ENZYMES RESPONSIBLE FOR THE METABOLISM OF LONAFARNIB (SARASAR)Anima Ghosal, Swapan K. Chowdhury, Wei Tong, Neil Hapangama, Yuan Yuan, Ai-Duen Su and Shmuel ZbaidaDrug Metabolism and Disposition April 2006, 34 (4) 628-635; DOI: https://doi.org/10.1124/dmd.105.007906
Hashikura, Yasuhiko
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Heim, John B.
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Hoffmann, Katrin
- You have accessS-2-PENTYL-4-PENTYNOIC HYDROXAMIC ACID AND ITS METABOLITE S-2-PENTYL-4-PENTYNOIC ACID IN THE NMRI-EXENCEPHALY-MOUSE MODEL: PHARMACOKINETIC PROFILES, TERATOGENIC EFFECTS, AND HISTONE DEACETYLASE INHIBITION ABILITIES OF FURTHER VALPROIC ACID HYDROXAMATES AND AMIDESDaniel Eikel, Katrin Hoffmann, Karolin Zoll, Alfonso Lampen and Heinz NauDrug Metabolism and Disposition April 2006, 34 (4) 612-620; DOI: https://doi.org/10.1124/dmd.105.008078
Holschbach, Marcus H.
- You have accessMETABOLISM OF THE A1 ADENOSINE RECEPTOR POSITRON EMISSION TOMOGRAPHY LIGAND [18F]8-CYCLOPENTYL-3-(3-FLUOROPROPYL)-1-PROPYLXANTHINE ([18F]CPFPX) IN RODENTS AND HUMANSDirk Bier, Marcus H. Holschbach, Walter Wutz, Ray A. Olsson and Heinz H. CoenenDrug Metabolism and Disposition April 2006, 34 (4) 570-576; DOI: https://doi.org/10.1124/dmd.105.006411
Houston, J. Brian
- You have accessBINDING OF DRUGS TO HEPATIC MICROSOMES: COMMENT AND ASSESSMENT OF CURRENT PREDICTION METHODOLOGY WITH RECOMMENDATION FOR IMPROVEMENTDavid Hallifax and J. Brian HoustonDrug Metabolism and Disposition April 2006, 34 (4) 724-726; DOI: https://doi.org/10.1124/dmd.105.007658
I
Inada, Yoichi
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Isoherranen, Nina
- You have accessSTEREOCHEMICAL ASPECTS OF ITRACONAZOLE METABOLISM IN VITRO AND IN VIVOKent L. Kunze, Wendel L. Nelson, Evan D. Kharasch, Kenneth E. Thummel and Nina IsoherranenDrug Metabolism and Disposition April 2006, 34 (4) 583-590; DOI: https://doi.org/10.1124/dmd.105.008508
J
Jedlitschky, Gabriele
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
Johnson, Brendan M.
- You have accessCHARACTERIZATION OF TRANSPORT PROTEIN EXPRESSION IN MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) 2-DEFICIENT RATSBrendan M. Johnson, Peijin Zhang, John D. Schuetz and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 556-562; DOI: https://doi.org/10.1124/dmd.105.005793
Jordan, Sherri
- You have accessDEPENDENCE OF NELFINAVIR BRAIN UPTAKE ON DOSE AND TISSUE CONCENTRATIONS OF THE SELECTIVE P-GLYCOPROTEIN INHIBITOR ZOSUQUIDAR IN RATSBradley D. Anderson, Melissa J. May, Sherri Jordan, Lin Song, Michael J. Roberts and Markos LeggasDrug Metabolism and Disposition April 2006, 34 (4) 653-659; DOI: https://doi.org/10.1124/dmd.105.006536
Joshi, Meenal
- You have accessINDUCTION AND RECOVERY TIME COURSE OF RAT BRAIN CYP2E1 AFTER NICOTINE TREATMENTMeenal Joshi and Rachel F. TyndaleDrug Metabolism and Disposition April 2006, 34 (4) 647-652; DOI: https://doi.org/10.1124/dmd.105.008029
K
Kamiyoshi, Akiko
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Kapelioukh, Iouri
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
Karnes, Thomas H.
- You have accessEFFECT OF CHRONIC RENAL INSUFFICIENCY ON HEPATIC AND RENAL UDP-GLUCURONYLTRANSFERASES IN RATSChuanhui Yu, Joseph K. Ritter, Richard J. Krieg, Bhaskar Rege, Thomas H. Karnes and Mohamadi A. SarkarDrug Metabolism and Disposition April 2006, 34 (4) 621-627; DOI: https://doi.org/10.1124/dmd.105.006601
Kasper, Steve C.
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Kelley, Rusty W.
- You have accessAN EVALUATION OF METHODS FOR THE RECONSTITUTION OF CYTOCHROMES P450 AND NADPH P450 REDUCTASE INTO LIPID VESICLESJames R. Reed, Rusty W. Kelley and Wayne L. BackesDrug Metabolism and Disposition April 2006, 34 (4) 660-666; DOI: https://doi.org/10.1124/dmd.105.006825
Khalife, Jamal
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Kharasch, Evan D.
- You have accessSTEREOCHEMICAL ASPECTS OF ITRACONAZOLE METABOLISM IN VITRO AND IN VIVOKent L. Kunze, Wendel L. Nelson, Evan D. Kharasch, Kenneth E. Thummel and Nina IsoherranenDrug Metabolism and Disposition April 2006, 34 (4) 583-590; DOI: https://doi.org/10.1124/dmd.105.008508
Kim, Hyunmi
- You have accessINHIBITORY EFFECTS OF FRUIT JUICES ON CYP3A ACTIVITYHyunmi Kim, Yune-Jung Yoon, Ji-Hong Shon, In-June Cha, Jae-Gook Shin and Kwang-Hyeon LiuDrug Metabolism and Disposition April 2006, 34 (4) 521-523; DOI: https://doi.org/10.1124/dmd.105.007930
Kim, Sang K.
- You have accessTHE MITOGEN-ACTIVATED PROTEIN KINASE KINASE (MEK) INHIBITOR PD98059 ELEVATES PRIMARY CULTURED RAT HEPATOCYTE GLUTATHIONE LEVELS INDEPENDENT OF INHIBITING MEKSang K. Kim, Mohamed A. Abdelmegeed and Raymond F. NovakDrug Metabolism and Disposition April 2006, 34 (4) 683-689; DOI: https://doi.org/10.1124/dmd.105.007666
Kishida, Tomoyuki
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Kiu, Tung-wah
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Klieber, Sylvie
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Kong, Wei
- You have accessINTERACTIONS OF AMOXICILLIN AND CEFACLOR WITH HUMAN RENAL ORGANIC ANION AND PEPTIDE TRANSPORTERSMeng Li, Gail D. Anderson, Brian R. Phillips, Wei Kong, Danny D. Shen and Joanne WangDrug Metabolism and Disposition April 2006, 34 (4) 547-555; DOI: https://doi.org/10.1124/dmd.105.006791
Krieg, Richard J.
- You have accessEFFECT OF CHRONIC RENAL INSUFFICIENCY ON HEPATIC AND RENAL UDP-GLUCURONYLTRANSFERASES IN RATSChuanhui Yu, Joseph K. Ritter, Richard J. Krieg, Bhaskar Rege, Thomas H. Karnes and Mohamadi A. SarkarDrug Metabolism and Disposition April 2006, 34 (4) 621-627; DOI: https://doi.org/10.1124/dmd.105.006601
Kroemer, Heyo K.
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
Kunze, Kent L.
- You have accessSTEREOCHEMICAL ASPECTS OF ITRACONAZOLE METABOLISM IN VITRO AND IN VIVOKent L. Kunze, Wendel L. Nelson, Evan D. Kharasch, Kenneth E. Thummel and Nina IsoherranenDrug Metabolism and Disposition April 2006, 34 (4) 583-590; DOI: https://doi.org/10.1124/dmd.105.008508
Kurihara, Atsushi
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Kuroda, Junji
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
L
Lampen, Alfonso
- You have accessS-2-PENTYL-4-PENTYNOIC HYDROXAMIC ACID AND ITS METABOLITE S-2-PENTYL-4-PENTYNOIC ACID IN THE NMRI-EXENCEPHALY-MOUSE MODEL: PHARMACOKINETIC PROFILES, TERATOGENIC EFFECTS, AND HISTONE DEACETYLASE INHIBITION ABILITIES OF FURTHER VALPROIC ACID HYDROXAMATES AND AMIDESDaniel Eikel, Katrin Hoffmann, Karolin Zoll, Alfonso Lampen and Heinz NauDrug Metabolism and Disposition April 2006, 34 (4) 612-620; DOI: https://doi.org/10.1124/dmd.105.008078
Langenkamp, Elise
- You have accessEMPIRICAL VALIDATION OF A RAT IN VITRO ORGAN SLICE MODEL AS A TOOL FOR IN VIVO CLEARANCE PREDICTIONInge A. M. de Graaf, Ruben de Kanter, Marina H. de Jager, Raquel Camacho, Elise Langenkamp, Esther G. van de Kerkhof and Geny M. M. GroothuisDrug Metabolism and Disposition April 2006, 34 (4) 591-599; DOI: https://doi.org/10.1124/dmd.105.006726
Leeder, J. Steven
- You have accessCYP2D6*36 GENE ARRANGEMENTS WITHIN THE CYP2D6 LOCUS: ASSOCIATION OF CYP2D6*36 WITH POOR METABOLIZER STATUSAndrea Gaedigk, L. DiAnne Bradford, Sarah W. Alander and J. Steven LeederDrug Metabolism and Disposition April 2006, 34 (4) 563-569; DOI: https://doi.org/10.1124/dmd.105.008292
Leggas, Markos
- You have accessDEPENDENCE OF NELFINAVIR BRAIN UPTAKE ON DOSE AND TISSUE CONCENTRATIONS OF THE SELECTIVE P-GLYCOPROTEIN INHIBITOR ZOSUQUIDAR IN RATSBradley D. Anderson, Melissa J. May, Sherri Jordan, Lin Song, Michael J. Roberts and Markos LeggasDrug Metabolism and Disposition April 2006, 34 (4) 653-659; DOI: https://doi.org/10.1124/dmd.105.006536
Li, Meng
- You have accessINTERACTIONS OF AMOXICILLIN AND CEFACLOR WITH HUMAN RENAL ORGANIC ANION AND PEPTIDE TRANSPORTERSMeng Li, Gail D. Anderson, Brian R. Phillips, Wei Kong, Danny D. Shen and Joanne WangDrug Metabolism and Disposition April 2006, 34 (4) 547-555; DOI: https://doi.org/10.1124/dmd.105.006791
Li, Ping
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
Linnemann, Knud
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
Liu, Kwang-Hyeon
- You have accessINHIBITORY EFFECTS OF FRUIT JUICES ON CYP3A ACTIVITYHyunmi Kim, Yune-Jung Yoon, Ji-Hong Shon, In-June Cha, Jae-Gook Shin and Kwang-Hyeon LiuDrug Metabolism and Disposition April 2006, 34 (4) 521-523; DOI: https://doi.org/10.1124/dmd.105.007930
Lu, Chuang
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
M
Maffrand, Jean-Pierre
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Marechal, Jean-Didier
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
May, Melissa J.
- You have accessDEPENDENCE OF NELFINAVIR BRAIN UPTAKE ON DOSE AND TISSUE CONCENTRATIONS OF THE SELECTIVE P-GLYCOPROTEIN INHIBITOR ZOSUQUIDAR IN RATSBradley D. Anderson, Melissa J. May, Sherri Jordan, Lin Song, Michael J. Roberts and Markos LeggasDrug Metabolism and Disposition April 2006, 34 (4) 653-659; DOI: https://doi.org/10.1124/dmd.105.006536
Meissner, Konrad
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
Merino, Gracia
- You have accessBREAST CANCER RESISTANCE PROTEIN (BCRP/ABCG2) TRANSPORTS FLUOROQUINOLONE ANTIBIOTICS AND AFFECTS THEIR ORAL AVAILABILITY, PHARMACOKINETICS, AND MILK SECRETIONGracia Merino, Ana I. Álvarez, Mivis M. Pulido, Antonio J. Molina, Alfred H. Schinkel and Julio G. PrietoDrug Metabolism and Disposition April 2006, 34 (4) 690-695; DOI: https://doi.org/10.1124/dmd.105.008219
Meunier, Viviane
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Miwa, Gerald T.
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
Miyagawa, Shinichi
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Molina, Antonio J.
- You have accessBREAST CANCER RESISTANCE PROTEIN (BCRP/ABCG2) TRANSPORTS FLUOROQUINOLONE ANTIBIOTICS AND AFFECTS THEIR ORAL AVAILABILITY, PHARMACOKINETICS, AND MILK SECRETIONGracia Merino, Ana I. Álvarez, Mivis M. Pulido, Antonio J. Molina, Alfred H. Schinkel and Julio G. PrietoDrug Metabolism and Disposition April 2006, 34 (4) 690-695; DOI: https://doi.org/10.1124/dmd.105.008219
Murakami, Makoto
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
N
Nau, Heinz
- You have accessS-2-PENTYL-4-PENTYNOIC HYDROXAMIC ACID AND ITS METABOLITE S-2-PENTYL-4-PENTYNOIC ACID IN THE NMRI-EXENCEPHALY-MOUSE MODEL: PHARMACOKINETIC PROFILES, TERATOGENIC EFFECTS, AND HISTONE DEACETYLASE INHIBITION ABILITIES OF FURTHER VALPROIC ACID HYDROXAMATES AND AMIDESDaniel Eikel, Katrin Hoffmann, Karolin Zoll, Alfonso Lampen and Heinz NauDrug Metabolism and Disposition April 2006, 34 (4) 612-620; DOI: https://doi.org/10.1124/dmd.105.008078
Nelson, Wendel L.
- You have accessSTEREOCHEMICAL ASPECTS OF ITRACONAZOLE METABOLISM IN VITRO AND IN VIVOKent L. Kunze, Wendel L. Nelson, Evan D. Kharasch, Kenneth E. Thummel and Nina IsoherranenDrug Metabolism and Disposition April 2006, 34 (4) 583-590; DOI: https://doi.org/10.1124/dmd.105.008508
Nezasa, Ken-ichi
- You have accessALTERED HEPATOBILIARY DISPOSITION OF 5 (AND 6)-CARBOXY-2′,7′-DICHLOROFLUORESCEIN IN Abcg2 (Bcrp1) AND Abcc2 (Mrp2) KNOCKOUT MICEKen-ichi Nezasa, Xianbin Tian, Maciej J. Zamek-Gliszczynski, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 718-723; DOI: https://doi.org/10.1124/dmd.105.007922
Nishiyama, Masahiko
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Nix, Darrell
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
Novak, Raymond F.
- You have accessTHE MITOGEN-ACTIVATED PROTEIN KINASE KINASE (MEK) INHIBITOR PD98059 ELEVATES PRIMARY CULTURED RAT HEPATOCYTE GLUTATHIONE LEVELS INDEPENDENT OF INHIBITING MEKSang K. Kim, Mohamed A. Abdelmegeed and Raymond F. NovakDrug Metabolism and Disposition April 2006, 34 (4) 683-689; DOI: https://doi.org/10.1124/dmd.105.007666
Nunoya, Kenichi
- You have accessMUTATIONAL ANALYSIS OF POLAR AMINO ACID RESIDUES WITHIN PREDICTED TRANSMEMBRANE HELICES 10 AND 16 OF MULTIDRUG RESISTANCE PROTEIN 1 (ABCC1): EFFECT ON SUBSTRATE SPECIFICITYDa-Wei Zhang, Kenichi Nunoya, Monika Vasa, Hong-Mei Gu, Susan P. C. Cole and Roger G. DeeleyDrug Metabolism and Disposition April 2006, 34 (4) 539-546; DOI: https://doi.org/10.1124/dmd.105.007740
O
Ogawa, Shinichiro
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Ohdo, Shigehiro
- You have accessEFFECTS OF HERBAL EXTRACTS ON THE FUNCTION OF HUMAN ORGANIC ANION-TRANSPORTING POLYPEPTIDE OATP-BHiromi Fuchikami, Hiroki Satoh, Masayuki Tsujimoto, Shigehiro Ohdo, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition April 2006, 34 (4) 577-582; DOI: https://doi.org/10.1124/dmd.105.007872
Ohtani, Hisakazu
- You have accessEFFECTS OF HERBAL EXTRACTS ON THE FUNCTION OF HUMAN ORGANIC ANION-TRANSPORTING POLYPEPTIDE OATP-BHiromi Fuchikami, Hiroki Satoh, Masayuki Tsujimoto, Shigehiro Ohdo, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition April 2006, 34 (4) 577-582; DOI: https://doi.org/10.1124/dmd.105.007872
Olsson, Ray A.
- You have accessMETABOLISM OF THE A1 ADENOSINE RECEPTOR POSITRON EMISSION TOMOGRAPHY LIGAND [18F]8-CYCLOPENTYL-3-(3-FLUOROPROPYL)-1-PROPYLXANTHINE ([18F]CPFPX) IN RODENTS AND HUMANSDirk Bier, Marcus H. Holschbach, Walter Wutz, Ray A. Olsson and Heinz H. CoenenDrug Metabolism and Disposition April 2006, 34 (4) 570-576; DOI: https://doi.org/10.1124/dmd.105.006411
P
Paine, Mark. J. I.
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
Patel, Nita J.
- You have accessALTERED HEPATOBILIARY DISPOSITION OF 5 (AND 6)-CARBOXY-2′,7′-DICHLOROFLUORESCEIN IN Abcg2 (Bcrp1) AND Abcc2 (Mrp2) KNOCKOUT MICEKen-ichi Nezasa, Xianbin Tian, Maciej J. Zamek-Gliszczynski, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 718-723; DOI: https://doi.org/10.1124/dmd.105.007922
Pelinski, Lydie
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Phillips, Brian R.
- You have accessINTERACTIONS OF AMOXICILLIN AND CEFACLOR WITH HUMAN RENAL ORGANIC ANION AND PEPTIDE TRANSPORTERSMeng Li, Gail D. Anderson, Brian R. Phillips, Wei Kong, Danny D. Shen and Joanne WangDrug Metabolism and Disposition April 2006, 34 (4) 547-555; DOI: https://doi.org/10.1124/dmd.105.006791
Pikuleva, Irina A.
- You have accessCHOLESTEROL-METABOLIZING CYTOCHROMES P450Irina A. PikulevaDrug Metabolism and Disposition April 2006, 34 (4) 513-520; DOI: https://doi.org/10.1124/dmd.105.008789
Pons, Gérard
- You have accessIN VITRO AND IN VIVO INHIBITORY EFFECT OF STIRIPENTOL ON CLOBAZAM METABOLISMCarole Giraud, Jean-Marc Treluyer, Elisabeth Rey, Catherine Chiron, Jean Vincent, Gérard Pons and Agnès TranDrug Metabolism and Disposition April 2006, 34 (4) 608-611; DOI: https://doi.org/10.1124/dmd.105.007237
Prieto, Julio G.
- You have accessBREAST CANCER RESISTANCE PROTEIN (BCRP/ABCG2) TRANSPORTS FLUOROQUINOLONE ANTIBIOTICS AND AFFECTS THEIR ORAL AVAILABILITY, PHARMACOKINETICS, AND MILK SECRETIONGracia Merino, Ana I. Álvarez, Mivis M. Pulido, Antonio J. Molina, Alfred H. Schinkel and Julio G. PrietoDrug Metabolism and Disposition April 2006, 34 (4) 690-695; DOI: https://doi.org/10.1124/dmd.105.008219
Pulido, Mivis M.
- You have accessBREAST CANCER RESISTANCE PROTEIN (BCRP/ABCG2) TRANSPORTS FLUOROQUINOLONE ANTIBIOTICS AND AFFECTS THEIR ORAL AVAILABILITY, PHARMACOKINETICS, AND MILK SECRETIONGracia Merino, Ana I. Álvarez, Mivis M. Pulido, Antonio J. Molina, Alfred H. Schinkel and Julio G. PrietoDrug Metabolism and Disposition April 2006, 34 (4) 690-695; DOI: https://doi.org/10.1124/dmd.105.008219
Pusalkar, Sandeepraj
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
R
Rankin, Elaine M.
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
Raub, Thomas J.
- You have accessALTERED HEPATOBILIARY DISPOSITION OF 5 (AND 6)-CARBOXY-2′,7′-DICHLOROFLUORESCEIN IN Abcg2 (Bcrp1) AND Abcc2 (Mrp2) KNOCKOUT MICEKen-ichi Nezasa, Xianbin Tian, Maciej J. Zamek-Gliszczynski, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 718-723; DOI: https://doi.org/10.1124/dmd.105.007922
Reed, James R.
- You have accessAN EVALUATION OF METHODS FOR THE RECONSTITUTION OF CYTOCHROMES P450 AND NADPH P450 REDUCTASE INTO LIPID VESICLESJames R. Reed, Rusty W. Kelley and Wayne L. BackesDrug Metabolism and Disposition April 2006, 34 (4) 660-666; DOI: https://doi.org/10.1124/dmd.105.006825
Rege, Bhaskar
- You have accessEFFECT OF CHRONIC RENAL INSUFFICIENCY ON HEPATIC AND RENAL UDP-GLUCURONYLTRANSFERASES IN RATSChuanhui Yu, Joseph K. Ritter, Richard J. Krieg, Bhaskar Rege, Thomas H. Karnes and Mohamadi A. SarkarDrug Metabolism and Disposition April 2006, 34 (4) 621-627; DOI: https://doi.org/10.1124/dmd.105.006601
Rehmel, Jessica L. Fayer
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Rey, Elisabeth
- You have accessIN VITRO AND IN VIVO INHIBITORY EFFECT OF STIRIPENTOL ON CLOBAZAM METABOLISMCarole Giraud, Jean-Marc Treluyer, Elisabeth Rey, Catherine Chiron, Jean Vincent, Gérard Pons and Agnès TranDrug Metabolism and Disposition April 2006, 34 (4) 608-611; DOI: https://doi.org/10.1124/dmd.105.007237
Reznik, Boris
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Riley, R. J.
- You have accessRESPONSE TO “BINDING OF DRUGS TO HEPATIC MICROSOMES: COMMENT AND ASSESSMENT OF CURRENT PREDICTION METHODOLOGY WITH RECOMMENDATION FOR IMPROVEMENT”R. P. Austin, P. Barton and R. J. RileyDrug Metabolism and Disposition April 2006, 34 (4) 727; DOI: https://doi.org/10.1124/dmd.105.009142
Ring, Barbara J.
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Ritter, Christoph A.
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
Ritter, Joseph K.
- You have accessEFFECT OF CHRONIC RENAL INSUFFICIENCY ON HEPATIC AND RENAL UDP-GLUCURONYLTRANSFERASES IN RATSChuanhui Yu, Joseph K. Ritter, Richard J. Krieg, Bhaskar Rege, Thomas H. Karnes and Mohamadi A. SarkarDrug Metabolism and Disposition April 2006, 34 (4) 621-627; DOI: https://doi.org/10.1124/dmd.105.006601
Roberts, Gordon C. K.
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
Roberts, Michael J.
- You have accessDEPENDENCE OF NELFINAVIR BRAIN UPTAKE ON DOSE AND TISSUE CONCENTRATIONS OF THE SELECTIVE P-GLYCOPROTEIN INHIBITOR ZOSUQUIDAR IN RATSBradley D. Anderson, Melissa J. May, Sherri Jordan, Lin Song, Michael J. Roberts and Markos LeggasDrug Metabolism and Disposition April 2006, 34 (4) 653-659; DOI: https://doi.org/10.1124/dmd.105.006536
S
Sadoun, Freddy
- You have accessIN VITRO METABOLISM OF FERROQUINE (SSR97193) IN ANIMAL AND HUMAN HEPATIC MODELS AND ANTIMALARIAL ACTIVITY OF MAJOR METABOLITES ON PLASMODIUM FALCIPARUMWassim Daher, Lydie Pelinski, Sylvie Klieber, Freddy Sadoun, Viviane Meunier, Martine Bourrié, Christophe Biot, François Guillou, Gérard Fabre, Jacques Brocard, Laurent Fraisse, Jean-Pierre Maffrand, Jamal Khalife and Daniel DiveDrug Metabolism and Disposition April 2006, 34 (4) 667-682; DOI: https://doi.org/10.1124/dmd.104.003202
Sarkar, Mohamadi A.
- You have accessEFFECT OF CHRONIC RENAL INSUFFICIENCY ON HEPATIC AND RENAL UDP-GLUCURONYLTRANSFERASES IN RATSChuanhui Yu, Joseph K. Ritter, Richard J. Krieg, Bhaskar Rege, Thomas H. Karnes and Mohamadi A. SarkarDrug Metabolism and Disposition April 2006, 34 (4) 621-627; DOI: https://doi.org/10.1124/dmd.105.006601
Satoh, Fumiyasu
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Satoh, Hiroki
- You have accessEFFECTS OF HERBAL EXTRACTS ON THE FUNCTION OF HUMAN ORGANIC ANION-TRANSPORTING POLYPEPTIDE OATP-BHiromi Fuchikami, Hiroki Satoh, Masayuki Tsujimoto, Shigehiro Ohdo, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition April 2006, 34 (4) 577-582; DOI: https://doi.org/10.1124/dmd.105.007872
Sawada, Yasufumi
- You have accessEFFECTS OF HERBAL EXTRACTS ON THE FUNCTION OF HUMAN ORGANIC ANION-TRANSPORTING POLYPEPTIDE OATP-BHiromi Fuchikami, Hiroki Satoh, Masayuki Tsujimoto, Shigehiro Ohdo, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition April 2006, 34 (4) 577-582; DOI: https://doi.org/10.1124/dmd.105.007872
Schinkel, Alfred H.
- You have accessBREAST CANCER RESISTANCE PROTEIN (BCRP/ABCG2) TRANSPORTS FLUOROQUINOLONE ANTIBIOTICS AND AFFECTS THEIR ORAL AVAILABILITY, PHARMACOKINETICS, AND MILK SECRETIONGracia Merino, Ana I. Álvarez, Mivis M. Pulido, Antonio J. Molina, Alfred H. Schinkel and Julio G. PrietoDrug Metabolism and Disposition April 2006, 34 (4) 690-695; DOI: https://doi.org/10.1124/dmd.105.008219
Schuetz, John D.
- You have accessCHARACTERIZATION OF TRANSPORT PROTEIN EXPRESSION IN MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) 2-DEFICIENT RATSBrendan M. Johnson, Peijin Zhang, John D. Schuetz and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 556-562; DOI: https://doi.org/10.1124/dmd.105.005793
Shen, Danny D.
- You have accessINTERACTIONS OF AMOXICILLIN AND CEFACLOR WITH HUMAN RENAL ORGANIC ANION AND PEPTIDE TRANSPORTERSMeng Li, Gail D. Anderson, Brian R. Phillips, Wei Kong, Danny D. Shen and Joanne WangDrug Metabolism and Disposition April 2006, 34 (4) 547-555; DOI: https://doi.org/10.1124/dmd.105.006791
Shibata, Nobuo
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Shin, Jae-Gook
- You have accessINHIBITORY EFFECTS OF FRUIT JUICES ON CYP3A ACTIVITYHyunmi Kim, Yune-Jung Yoon, Ji-Hong Shon, In-June Cha, Jae-Gook Shin and Kwang-Hyeon LiuDrug Metabolism and Disposition April 2006, 34 (4) 521-523; DOI: https://doi.org/10.1124/dmd.105.007930
Shon, Ji-Hong
- You have accessINHIBITORY EFFECTS OF FRUIT JUICES ON CYP3A ACTIVITYHyunmi Kim, Yune-Jung Yoon, Ji-Hong Shon, In-June Cha, Jae-Gook Shin and Kwang-Hyeon LiuDrug Metabolism and Disposition April 2006, 34 (4) 521-523; DOI: https://doi.org/10.1124/dmd.105.007930
Smith, Evan
- You have accessIN VITRO METABOLIC ACTIVATION OF THIABENDAZOLE VIA 5-HYDROXYTHIABENDAZOLE: IDENTIFICATION OF A GLUTATHIONE CONJUGATE OF 5-HYDROXYTHIABENDAZOLEDeepak Dalvie, Evan Smith, Alan Deese and Stephen BowlinDrug Metabolism and Disposition April 2006, 34 (4) 709-717; DOI: https://doi.org/10.1124/dmd.105.008094
Song, Lin
- You have accessDEPENDENCE OF NELFINAVIR BRAIN UPTAKE ON DOSE AND TISSUE CONCENTRATIONS OF THE SELECTIVE P-GLYCOPROTEIN INHIBITOR ZOSUQUIDAR IN RATSBradley D. Anderson, Melissa J. May, Sherri Jordan, Lin Song, Michael J. Roberts and Markos LeggasDrug Metabolism and Disposition April 2006, 34 (4) 653-659; DOI: https://doi.org/10.1124/dmd.105.006536
Stark, Raymond I.
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Su, Ai-Duen
- You have accessIDENTIFICATION OF HUMAN LIVER CYTOCHROME P450 ENZYMES RESPONSIBLE FOR THE METABOLISM OF LONAFARNIB (SARASAR)Anima Ghosal, Swapan K. Chowdhury, Wei Tong, Neil Hapangama, Yuan Yuan, Ai-Duen Su and Shmuel ZbaidaDrug Metabolism and Disposition April 2006, 34 (4) 628-635; DOI: https://doi.org/10.1124/dmd.105.007906
Sutcliffe, Michael J.
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
T
Tagawa, Yoh-ichi
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Tanaka, Satoru
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Taylor, Samantha
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Thummel, Kenneth E.
- You have accessSTEREOCHEMICAL ASPECTS OF ITRACONAZOLE METABOLISM IN VITRO AND IN VIVOKent L. Kunze, Wendel L. Nelson, Evan D. Kharasch, Kenneth E. Thummel and Nina IsoherranenDrug Metabolism and Disposition April 2006, 34 (4) 583-590; DOI: https://doi.org/10.1124/dmd.105.008508
Tian, Xianbin
- You have accessALTERED HEPATOBILIARY DISPOSITION OF 5 (AND 6)-CARBOXY-2′,7′-DICHLOROFLUORESCEIN IN Abcg2 (Bcrp1) AND Abcc2 (Mrp2) KNOCKOUT MICEKen-ichi Nezasa, Xianbin Tian, Maciej J. Zamek-Gliszczynski, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 718-723; DOI: https://doi.org/10.1124/dmd.105.007922
Tomioka, Eisuke
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Tong, Wei
- You have accessIDENTIFICATION OF HUMAN LIVER CYTOCHROME P450 ENZYMES RESPONSIBLE FOR THE METABOLISM OF LONAFARNIB (SARASAR)Anima Ghosal, Swapan K. Chowdhury, Wei Tong, Neil Hapangama, Yuan Yuan, Ai-Duen Su and Shmuel ZbaidaDrug Metabolism and Disposition April 2006, 34 (4) 628-635; DOI: https://doi.org/10.1124/dmd.105.007906
Tran, Agnès
- You have accessIN VITRO AND IN VIVO INHIBITORY EFFECT OF STIRIPENTOL ON CLOBAZAM METABOLISMCarole Giraud, Jean-Marc Treluyer, Elisabeth Rey, Catherine Chiron, Jean Vincent, Gérard Pons and Agnès TranDrug Metabolism and Disposition April 2006, 34 (4) 608-611; DOI: https://doi.org/10.1124/dmd.105.007237
Treluyer, Jean-Marc
- You have accessIN VITRO AND IN VIVO INHIBITORY EFFECT OF STIRIPENTOL ON CLOBAZAM METABOLISMCarole Giraud, Jean-Marc Treluyer, Elisabeth Rey, Catherine Chiron, Jean Vincent, Gérard Pons and Agnès TranDrug Metabolism and Disposition April 2006, 34 (4) 608-611; DOI: https://doi.org/10.1124/dmd.105.007237
Tsujimoto, Masayuki
- You have accessEFFECTS OF HERBAL EXTRACTS ON THE FUNCTION OF HUMAN ORGANIC ANION-TRANSPORTING POLYPEPTIDE OATP-BHiromi Fuchikami, Hiroki Satoh, Masayuki Tsujimoto, Shigehiro Ohdo, Hisakazu Ohtani and Yasufumi SawadaDrug Metabolism and Disposition April 2006, 34 (4) 577-582; DOI: https://doi.org/10.1124/dmd.105.007872
Tsutsui, Masaru
- You have accessCHARACTERIZATION OF CYTOCHROME P450 EXPRESSION IN MURINE EMBRYONIC STEM CELL-DERIVED HEPATIC TISSUE SYSTEMMasaru Tsutsui, Shinichiro Ogawa, Yoichi Inada, Eisuke Tomioka, Akiko Kamiyoshi, Satoru Tanaka, Tomoyuki Kishida, Masahiko Nishiyama, Makoto Murakami, Junji Kuroda, Yasuhiko Hashikura, Shinichi Miyagawa, Fumiyasu Satoh, Nobuo Shibata and Yoh-ichi TagawaDrug Metabolism and Disposition April 2006, 34 (4) 696-701; DOI: https://doi.org/10.1124/dmd.105.007674
Tyndale, Rachel F.
- You have accessINDUCTION AND RECOVERY TIME COURSE OF RAT BRAIN CYP2E1 AFTER NICOTINE TREATMENTMeenal Joshi and Rachel F. TyndaleDrug Metabolism and Disposition April 2006, 34 (4) 647-652; DOI: https://doi.org/10.1124/dmd.105.008029
U
Uttamsingh, Vinita
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
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van de Kerkhof, Esther G.
- You have accessEMPIRICAL VALIDATION OF A RAT IN VITRO ORGAN SLICE MODEL AS A TOOL FOR IN VIVO CLEARANCE PREDICTIONInge A. M. de Graaf, Ruben de Kanter, Marina H. de Jager, Raquel Camacho, Elise Langenkamp, Esther G. van de Kerkhof and Geny M. M. GroothuisDrug Metabolism and Disposition April 2006, 34 (4) 591-599; DOI: https://doi.org/10.1124/dmd.105.006726
Vasa, Monika
- You have accessMUTATIONAL ANALYSIS OF POLAR AMINO ACID RESIDUES WITHIN PREDICTED TRANSMEMBRANE HELICES 10 AND 16 OF MULTIDRUG RESISTANCE PROTEIN 1 (ABCC1): EFFECT ON SUBSTRATE SPECIFICITYDa-Wei Zhang, Kenichi Nunoya, Monika Vasa, Hong-Mei Gu, Susan P. C. Cole and Roger G. DeeleyDrug Metabolism and Disposition April 2006, 34 (4) 539-546; DOI: https://doi.org/10.1124/dmd.105.007740
Vincent, Jean
- You have accessIN VITRO AND IN VIVO INHIBITORY EFFECT OF STIRIPENTOL ON CLOBAZAM METABOLISMCarole Giraud, Jean-Marc Treluyer, Elisabeth Rey, Catherine Chiron, Jean Vincent, Gérard Pons and Agnès TranDrug Metabolism and Disposition April 2006, 34 (4) 608-611; DOI: https://doi.org/10.1124/dmd.105.007237
Völker, Uwe
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
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Wang, Joanne
- You have accessINTERACTIONS OF AMOXICILLIN AND CEFACLOR WITH HUMAN RENAL ORGANIC ANION AND PEPTIDE TRANSPORTERSMeng Li, Gail D. Anderson, Brian R. Phillips, Wei Kong, Danny D. Shen and Joanne WangDrug Metabolism and Disposition April 2006, 34 (4) 547-555; DOI: https://doi.org/10.1124/dmd.105.006791
Weldy, Piper
- You have accessFETAL MORPHINE METABOLISM AND CLEARANCE ARE CONSTANT DURING LATE GESTATIONMarianne Garland, Kirsten M. Abildskov, Samantha Taylor, Kenza Benzeroual, Casper S. Caspersen, Sylvia E. Arroyo, Tung-wah Kiu, Boris Reznik, Piper Weldy, Salha S. Daniel and Raymond I. StarkDrug Metabolism and Disposition April 2006, 34 (4) 636-646; DOI: https://doi.org/10.1124/dmd.105.007567
Wolf, C. Roland
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
Wrighton, Steven A.
- You have accessINTERACTIONS OF TWO MAJOR METABOLITES OF PRASUGREL, A THIENOPYRIDINE ANTIPLATELET AGENT, WITH THE CYTOCHROMES P450Jessica L. Fayer Rehmel, James A. Eckstein, Nagy A. Farid, John B. Heim, Steve C. Kasper, Atsushi Kurihara, Steven A. Wrighton and Barbara J. RingDrug Metabolism and Disposition April 2006, 34 (4) 600-607; DOI: https://doi.org/10.1124/dmd.105.007989
Wutz, Walter
- You have accessMETABOLISM OF THE A1 ADENOSINE RECEPTOR POSITRON EMISSION TOMOGRAPHY LIGAND [18F]8-CYCLOPENTYL-3-(3-FLUOROPROPYL)-1-PROPYLXANTHINE ([18F]CPFPX) IN RODENTS AND HUMANSDirk Bier, Marcus H. Holschbach, Walter Wutz, Ray A. Olsson and Heinz H. CoenenDrug Metabolism and Disposition April 2006, 34 (4) 570-576; DOI: https://doi.org/10.1124/dmd.105.006411
X
Xia, Cindy Q.
- You have accessINVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMESChuang Lu, Richard Gallegos, Ping Li, Cindy Q. Xia, Sandeepraj Pusalkar, Vinita Uttamsingh, Darrell Nix, Gerald T. Miwa and Liang-Shang GanDrug Metabolism and Disposition April 2006, 34 (4) 702-708; DOI: https://doi.org/10.1124/dmd.105.008060
Y
Yoon, Yune-Jung
- You have accessINHIBITORY EFFECTS OF FRUIT JUICES ON CYP3A ACTIVITYHyunmi Kim, Yune-Jung Yoon, Ji-Hong Shon, In-June Cha, Jae-Gook Shin and Kwang-Hyeon LiuDrug Metabolism and Disposition April 2006, 34 (4) 521-523; DOI: https://doi.org/10.1124/dmd.105.007930
Yu, Chuanhui
- You have accessEFFECT OF CHRONIC RENAL INSUFFICIENCY ON HEPATIC AND RENAL UDP-GLUCURONYLTRANSFERASES IN RATSChuanhui Yu, Joseph K. Ritter, Richard J. Krieg, Bhaskar Rege, Thomas H. Karnes and Mohamadi A. SarkarDrug Metabolism and Disposition April 2006, 34 (4) 621-627; DOI: https://doi.org/10.1124/dmd.105.006601
Yu, Jinglei
- You have accessIN SILICO AND IN VITRO SCREENING FOR INHIBITION OF CYTOCHROME P450 CYP3A4 BY COMEDICATIONS COMMONLY USED BY PATIENTS WITH CANCERJean-Didier Marechal, Jinglei Yu, Simon Brown, Iouri Kapelioukh, Elaine M. Rankin, C. Roland Wolf, Gordon C. K. Roberts, Mark. J. I. Paine and Michael J. SutcliffeDrug Metabolism and Disposition April 2006, 34 (4) 534-538; DOI: https://doi.org/10.1124/dmd.105.007625
Yuan, Yuan
- You have accessIDENTIFICATION OF HUMAN LIVER CYTOCHROME P450 ENZYMES RESPONSIBLE FOR THE METABOLISM OF LONAFARNIB (SARASAR)Anima Ghosal, Swapan K. Chowdhury, Wei Tong, Neil Hapangama, Yuan Yuan, Ai-Duen Su and Shmuel ZbaidaDrug Metabolism and Disposition April 2006, 34 (4) 628-635; DOI: https://doi.org/10.1124/dmd.105.007906
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Zamek-Gliszczynski, Maciej J.
- You have accessALTERED HEPATOBILIARY DISPOSITION OF 5 (AND 6)-CARBOXY-2′,7′-DICHLOROFLUORESCEIN IN Abcg2 (Bcrp1) AND Abcc2 (Mrp2) KNOCKOUT MICEKen-ichi Nezasa, Xianbin Tian, Maciej J. Zamek-Gliszczynski, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 718-723; DOI: https://doi.org/10.1124/dmd.105.007922
Zbaida, Shmuel
- You have accessIDENTIFICATION OF HUMAN LIVER CYTOCHROME P450 ENZYMES RESPONSIBLE FOR THE METABOLISM OF LONAFARNIB (SARASAR)Anima Ghosal, Swapan K. Chowdhury, Wei Tong, Neil Hapangama, Yuan Yuan, Ai-Duen Su and Shmuel ZbaidaDrug Metabolism and Disposition April 2006, 34 (4) 628-635; DOI: https://doi.org/10.1124/dmd.105.007906
Zhang, Da-Wei
- You have accessMUTATIONAL ANALYSIS OF POLAR AMINO ACID RESIDUES WITHIN PREDICTED TRANSMEMBRANE HELICES 10 AND 16 OF MULTIDRUG RESISTANCE PROTEIN 1 (ABCC1): EFFECT ON SUBSTRATE SPECIFICITYDa-Wei Zhang, Kenichi Nunoya, Monika Vasa, Hong-Mei Gu, Susan P. C. Cole and Roger G. DeeleyDrug Metabolism and Disposition April 2006, 34 (4) 539-546; DOI: https://doi.org/10.1124/dmd.105.007740
Zhang, Peijin
- You have accessCHARACTERIZATION OF TRANSPORT PROTEIN EXPRESSION IN MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN (MRP) 2-DEFICIENT RATSBrendan M. Johnson, Peijin Zhang, John D. Schuetz and Kim L. R. BrouwerDrug Metabolism and Disposition April 2006, 34 (4) 556-562; DOI: https://doi.org/10.1124/dmd.105.005793
Zoll, Karolin
- You have accessS-2-PENTYL-4-PENTYNOIC HYDROXAMIC ACID AND ITS METABOLITE S-2-PENTYL-4-PENTYNOIC ACID IN THE NMRI-EXENCEPHALY-MOUSE MODEL: PHARMACOKINETIC PROFILES, TERATOGENIC EFFECTS, AND HISTONE DEACETYLASE INHIBITION ABILITIES OF FURTHER VALPROIC ACID HYDROXAMATES AND AMIDESDaniel Eikel, Katrin Hoffmann, Karolin Zoll, Alfonso Lampen and Heinz NauDrug Metabolism and Disposition April 2006, 34 (4) 612-620; DOI: https://doi.org/10.1124/dmd.105.008078
zu Schwabedissen, Henriette E. Meyer
- You have accessEPIDERMAL GROWTH FACTOR-MEDIATED ACTIVATION OF THE MAP KINASE CASCADE RESULTS IN ALTERED EXPRESSION AND FUNCTION OF ABCG2 (BCRP)Henriette E. Meyer zu Schwabedissen, Markus Grube, Annette Dreisbach, Gabriele Jedlitschky, Konrad Meissner, Knud Linnemann, Christoph Fusch, Christoph A. Ritter, Uwe Völker and Heyo K. KroemerDrug Metabolism and Disposition April 2006, 34 (4) 524-533; DOI: https://doi.org/10.1124/dmd.105.007591
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