Index by author
June 01, 2006; Volume 34,Issue 6
A
Afzelius, Lovisa
- You have accessCOMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONSDiansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael ZamoraDrug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
Agrawal, Nancy G. B.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Akimoto, Kei
- You have accessAUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMESToshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
Amidon, Gordon L.
- You have accessN-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLEPhilip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. AmidonDrug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
Andersson, Tommy B.
- You have accessCOMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONSDiansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael ZamoraDrug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
Api, Anne Marie
- You have accessCOMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTESRaymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie ApiDrug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
Arison, Byron H.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Arya, Vikram
- You have accessCONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDSVikram Arya, Vincent G. Demarco, Manish Issar and Günther HochhausDrug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
Ashby, Charlotte A.
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
Au-Yeung, Sam C. S.
- You have accessA PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISMSam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne RiggsDrug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898
Ayrton, Andrew D.
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
B
Bachmeier, Corbin J.
- You have accessCOMPARISON OF DRUG EFFLUX TRANSPORT KINETICS IN VARIOUS BLOOD-BRAIN BARRIER MODELSCorbin J. Bachmeier, William J. Trickler and Donald W. MillerDrug Metabolism and Disposition June 2006, 34 (6) 998-1003; DOI: https://doi.org/10.1124/dmd.105.006999
Baldwin, Sandra J.
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
Beijnen, Jos H.
- You have accessSATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTESAnthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. HuitemaDrug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
Black, Gordon P.
- You have accessFORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVERGordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek ForkertDrug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
Blacquiere, Dylan P.
- You have accessFORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVERGordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek ForkertDrug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
Bonacorsi, Samuel J.
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
Bondesson, Ulf
- You have accessFLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRYAnnica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael HedelandDrug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
Bramhall, Jo L.
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
Brancale, Andrea
- You have accessN-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLEPhilip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. AmidonDrug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
C
Cai, Shaoqing
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Camenisch, Gian P.
- You have accessIN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMANH. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard GrossDrug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
Catania, Viviana A.
- You have accessETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. CataniaDrug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
- You have accessGALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASISFernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
Chen, Gang
- You have accessIMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORMRyan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip LazarusDrug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
Chiba, Kan
- You have accessINVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVERSachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
- You have accessAUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMESToshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
Chow, David
- You have accessIDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONSChun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi KumarDrug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
Clarke, Stephen E.
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
Collins, Kathy S.
- You have accessFORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVERGordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek ForkertDrug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
Copalu, William
- You have accessSATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTESAnthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. HuitemaDrug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
Crocenzi, Fernando A.
- You have accessGALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASISFernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
Cui, Donghui
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
D
de Kanter, Ruben
- You have accessCOMPARISON OF MOUSE AND RAT CYTOCHROME P450-MEDIATED METABOLISM IN LIVER AND INTESTINEMarcella Martignoni, Geny Groothuis and Ruben de KanterDrug Metabolism and Disposition June 2006, 34 (6) 1047-1054; DOI: https://doi.org/10.1124/dmd.105.009035
Dellinger, Ryan W.
- You have accessIMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORMRyan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip LazarusDrug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
Demarco, Vincent G.
- You have accessCONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDSVikram Arya, Vincent G. Demarco, Manish Issar and Günther HochhausDrug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
Dickinson, Ronald G.
- You have accessIN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTIONAndrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. MinersDrug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
Drach, John C.
- You have accessN-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLEPhilip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. AmidonDrug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
E
Elliot, David J.
- You have accessIN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTIONAndrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. MinersDrug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
F
Fang, Jia-Long
- You have accessIMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORMRyan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip LazarusDrug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
Forkert, Poh-Gek
- You have accessFORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVERGordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek ForkertDrug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
Fresneau, Marcel
- You have accessIN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMANH. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard GrossDrug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
Furihata, Tomomi
- You have accessINVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVERSachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
G
Gannon, Shawn A.
- You have accessCOMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTESRaymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie ApiDrug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
Gentry, W. Brooks
- You have accessANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTEDGrzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks GentryDrug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
Gillespie, Todd A.
- You have accessAPPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensisMilton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan KulanthaivelDrug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
Goel, Thanh V.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Grimm, Scott W.
- You have accessCOMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONSDiansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael ZamoraDrug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
Groothuis, Geny
- You have accessCOMPARISON OF MOUSE AND RAT CYTOCHROME P450-MEDIATED METABOLISM IN LIVER AND INTESTINEMarcella Martignoni, Geny Groothuis and Ruben de KanterDrug Metabolism and Disposition June 2006, 34 (6) 1047-1054; DOI: https://doi.org/10.1124/dmd.105.009035
Gross, Gerhard
- You have accessIN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMANH. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard GrossDrug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
Gruber, Nancy
- You have accessA PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISMSam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne RiggsDrug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898
H
Hedeland, Mikael
- You have accessFLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRYAnnica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael HedelandDrug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
Higuchi, Tomoaki
- You have accessINVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVERSachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
Hochhaus, Günther
- You have accessCONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDSVikram Arya, Vincent G. Demarco, Manish Issar and Günther HochhausDrug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
Hood, Steven R.
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
Hosokawa, Masakiyo
- You have accessINVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVERSachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
Huitema, Alwin D. R.
- You have accessSATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTESAnthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. HuitemaDrug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
I
Issar, Manish
- You have accessCONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDSVikram Arya, Vincent G. Demarco, Manish Issar and Günther HochhausDrug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
Iyer, Ramaswamy A.
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
J
Jackson, David A.
- You have accessAPPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensisMilton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan KulanthaivelDrug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
James, Margaret O.
- You have accessDEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMESLeah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. JamesDrug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
Jemal, Mohammed
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
Jönsson, Mats
- You have accessFLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRYAnnica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael HedelandDrug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
K
Kawashima, Sachiyo
- You have accessINVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVERSachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
Kearns, Gregory L.
- You have accessBIOTRANSFORMATION OF FLUTICASONE: IN VITRO CHARACTERIZATIONRobin E. Pearce, J. Steven Leeder and Gregory L. KearnsDrug Metabolism and Disposition June 2006, 34 (6) 1035-1040; DOI: https://doi.org/10.1124/dmd.105.009043
Kemper, Raymond A.
- You have accessCOMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTESRaymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie ApiDrug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
Khan, Sanaullah
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
Kleinow, Kevin M.
- You have accessDEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMESLeah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. JamesDrug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
Kobayashi, Kaoru
- You have accessINVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVERSachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
- You have accessAUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMESToshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
Kretz, Olivier
- You have accessIN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMANH. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard GrossDrug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
Kulanthaivel, Palaniappan
- You have accessAPPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensisMilton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan KulanthaivelDrug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
Kumar, Gondi
- You have accessIDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONSChun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi KumarDrug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
L
Landowski, Christopher P.
- You have accessN-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLEPhilip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. AmidonDrug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
Lasseter, Kenneth C.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Laurenzana, Elizabeth M.
- You have accessANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTEDGrzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks GentryDrug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
Lazarus, Philip
- You have accessIMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORMRyan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip LazarusDrug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
Leeder, J. Steven
- You have accessBIOTRANSFORMATION OF FLUTICASONE: IN VITRO CHARACTERIZATIONRobin E. Pearce, J. Steven Leeder and Gregory L. KearnsDrug Metabolism and Disposition June 2006, 34 (6) 1035-1040; DOI: https://doi.org/10.1124/dmd.105.009043
Lennernäs, Bo
- You have accessFLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRYAnnica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael HedelandDrug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
Lennernäs, Hans
- You have accessFLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRYAnnica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael HedelandDrug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
Li, Changling
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Li, Chun
- You have accessIDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONSChun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi KumarDrug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
Lorenzi, Philip L.
- You have accessN-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLEPhilip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. AmidonDrug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
Lu, Xiaowei
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Luquita, Marcelo G.
- You have accessETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. CataniaDrug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
- You have accessGALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASISFernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
M
Mackenzie, Peter I.
- You have accessIN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTIONAndrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. MinersDrug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
Marquez, Brian
- You have accessIDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONSChun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi KumarDrug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
Martignoni, Marcella
- You have accessCOMPARISON OF MOUSE AND RAT CYTOCHROME P450-MEDIATED METABOLISM IN LIVER AND INTESTINEMarcella Martignoni, Geny Groothuis and Ruben de KanterDrug Metabolism and Disposition June 2006, 34 (6) 1047-1054; DOI: https://doi.org/10.1124/dmd.105.009035
Miller, Donald W.
- You have accessCOMPARISON OF DRUG EFFLUX TRANSPORT KINETICS IN VARIOUS BLOOD-BRAIN BARRIER MODELSCorbin J. Bachmeier, William J. Trickler and Donald W. MillerDrug Metabolism and Disposition June 2006, 34 (6) 998-1003; DOI: https://doi.org/10.1124/dmd.105.006999
Miners, John O.
- You have accessIN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTIONAndrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. MinersDrug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
Mitroka, James
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
Mottino, Aldo D.
- You have accessETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. CataniaDrug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
- You have accessGALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASISFernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
Murdock, Paul R.
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
Murphy, M. Gail
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
N
Nabb, Diane L.
- You have accessCOMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTESRaymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie ApiDrug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
Niwa, Takuro
- You have accessAUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMESToshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
Norlin, Maria
- You have accessFLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRYAnnica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael HedelandDrug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
O
Owens, S. Michael
- You have accessANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTEDGrzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks GentryDrug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
P
Pearce, Robin E.
- You have accessBIOTRANSFORMATION OF FLUTICASONE: IN VITRO CHARACTERIZATIONRobin E. Pearce, J. Steven Leeder and Gregory L. KearnsDrug Metabolism and Disposition June 2006, 34 (6) 1035-1040; DOI: https://doi.org/10.1124/dmd.105.009043
Pellegrino, José M.
- You have accessGALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASISFernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
Pitas, Grzegorz
- You have accessANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTEDGrzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks GentryDrug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
Polsky-Fisher, Stacey L.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Pozzi, Enrique J. Sánchez
- You have accessGALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASISFernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
R
Riggs, K. Wayne
- You have accessA PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISMSam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne RiggsDrug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898
Rinehart, J. Kent
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
Rodrigues, A. David
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Roma, Marcelo G.
- You have accessGALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASISFernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez PozziDrug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
Rowland, Andrew
- You have accessIN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTIONAndrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. MinersDrug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
Ruiz, María L.
- You have accessETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. CataniaDrug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
Rurak, Dan W.
- You have accessA PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISMSam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne RiggsDrug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898
S
Schellens, Jan H. M.
- You have accessSATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTESAnthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. HuitemaDrug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
Schmidt, Douglas F.
- You have accessAPPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensisMilton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan KulanthaivelDrug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
Shang, Mingying
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Shimizu, Toshiyuki
- You have accessAUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMESToshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
Simpson, Richard C.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Snow, Timothy A.
- You have accessCOMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTESRaymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie ApiDrug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
Song, Xueqin
- You have accessN-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLEPhilip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. AmidonDrug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
Stegeman, John J.
- You have accessDEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMESLeah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. JamesDrug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
Stuchal, Leah D.
- You have accessDEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMESLeah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. JamesDrug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
Subramanian, Raju
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Surapaneni, Sekhar
- You have accessIDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONSChun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi KumarDrug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
T
Takama, Kaori
- You have accessINVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVERSachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
Tevell, Annica
- You have accessFLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRYAnnica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael HedelandDrug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
Townsend, Leroy B.
- You have accessN-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLEPhilip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. AmidonDrug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
Trickler, William J.
- You have accessCOMPARISON OF DRUG EFFLUX TRANSPORT KINETICS IN VARIOUS BLOOD-BRAIN BARRIER MODELSCorbin J. Bachmeier, William J. Trickler and Donald W. MillerDrug Metabolism and Disposition June 2006, 34 (6) 998-1003; DOI: https://doi.org/10.1124/dmd.105.006999
Tsunoo, Michio
- You have accessAUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMESToshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
Tu, Pengfei
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
V
Vaccharajani, Nimish
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
Vega, Jose M.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Vessey, Laura K.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Vickers, Stanley
- You have accessMETABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERSStacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David RodriguesDrug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
Villanueva, Silvina S. M.
- You have accessETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. CataniaDrug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
Vore, Mary
- You have accessETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. CataniaDrug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
W
Wait, Jill C. M.
- You have accessMETABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANSJill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. IyerDrug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
Weinberg, Rebecca
- You have accessIMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORMRyan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip LazarusDrug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
Weiss, H. Markus
- You have accessIN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMANH. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard GrossDrug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
Williams, D. Keith
- You have accessANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTEDGrzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks GentryDrug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
Williams, J. Andrew
- You have accessIN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTIONAndrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. MinersDrug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
X
Xiao, Shengyuan
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Xu, Feng
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Y
Yang, Donghui
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Yang, Xiaoda
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Yi, Ping
- You have accessAPPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensisMilton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan KulanthaivelDrug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
Yoshimura, Takuya
- You have accessAUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMESToshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan ChibaDrug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
Yue, Lin
- You have accessCYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. ClarkeDrug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
Z
Zamora, Ismael
- You have accessCOMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONSDiansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael ZamoraDrug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
Zandvliet, Anthe S.
- You have accessSATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTESAnthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. HuitemaDrug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
Zauhar, Randy J.
- You have accessCOMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONSDiansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael ZamoraDrug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
Zeng, QingPing
- You have accessIDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONSChun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi KumarDrug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
Zhang, Yue
- You have accessABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVOFeng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing CaiDrug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
Zhou, Diansong
- You have accessCOMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONSDiansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael ZamoraDrug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
Zmijewski, Milton
- You have accessAPPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensisMilton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan KulanthaivelDrug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
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