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Drug Metabolism & Disposition

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Index by author

June 01, 2006; Volume 34,Issue 6
  • A
  • B
  • C
  • D
  • E
  • F
  • G
  • H
  • I
  • J
  • K
  • L
  • M
  • N
  • O
  • P
  • Q
  • R
  • S
  • T
  • U
  • V
  • W
  • X
  • Y
  • Z

A

  1. Afzelius, Lovisa

    1. You have access
      COMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONS
      Diansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael Zamora
      Drug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
  2. Agrawal, Nancy G. B.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  3. Akimoto, Kei

    1. You have access
      AUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMES
      Toshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
  4. Amidon, Gordon L.

    1. You have access
      N-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLE
      Philip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. Amidon
      Drug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
  5. Andersson, Tommy B.

    1. You have access
      COMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONS
      Diansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael Zamora
      Drug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
  6. Api, Anne Marie

    1. You have access
      COMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTES
      Raymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie Api
      Drug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
  7. Arison, Byron H.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  8. Arya, Vikram

    1. You have access
      CONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDS
      Vikram Arya, Vincent G. Demarco, Manish Issar and Günther Hochhaus
      Drug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
  9. Ashby, Charlotte A.

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
  10. Au-Yeung, Sam C. S.

    1. You have access
      A PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISM
      Sam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne Riggs
      Drug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898
  11. Ayrton, Andrew D.

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185

B

  1. Bachmeier, Corbin J.

    1. You have access
      COMPARISON OF DRUG EFFLUX TRANSPORT KINETICS IN VARIOUS BLOOD-BRAIN BARRIER MODELS
      Corbin J. Bachmeier, William J. Trickler and Donald W. Miller
      Drug Metabolism and Disposition June 2006, 34 (6) 998-1003; DOI: https://doi.org/10.1124/dmd.105.006999
  2. Baldwin, Sandra J.

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
  3. Beijnen, Jos H.

    1. You have access
      SATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTES
      Anthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. Huitema
      Drug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
  4. Black, Gordon P.

    1. You have access
      FORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVER
      Gordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek Forkert
      Drug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
  5. Blacquiere, Dylan P.

    1. You have access
      FORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVER
      Gordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek Forkert
      Drug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
  6. Bonacorsi, Samuel J.

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
  7. Bondesson, Ulf

    1. You have access
      FLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRY
      Annica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael Hedeland
      Drug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
  8. Bramhall, Jo L.

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
  9. Brancale, Andrea

    1. You have access
      N-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLE
      Philip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. Amidon
      Drug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209

C

  1. Cai, Shaoqing

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  2. Camenisch, Gian P.

    1. You have access
      IN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMAN
      H. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard Gross
      Drug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
  3. Catania, Viviana A.

    1. You have access
      ETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3
      María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. Catania
      Drug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
    2. You have access
      GALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASIS
      Fernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez Pozzi
      Drug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
  4. Chen, Gang

    1. You have access
      IMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORM
      Ryan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip Lazarus
      Drug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
  5. Chiba, Kan

    1. You have access
      INVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVER
      Sachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
    2. You have access
      AUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMES
      Toshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
  6. Chow, David

    1. You have access
      IDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONS
      Chun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi Kumar
      Drug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
  7. Clarke, Stephen E.

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
  8. Collins, Kathy S.

    1. You have access
      FORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVER
      Gordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek Forkert
      Drug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
  9. Copalu, William

    1. You have access
      SATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTES
      Anthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. Huitema
      Drug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
  10. Crocenzi, Fernando A.

    1. You have access
      GALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASIS
      Fernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez Pozzi
      Drug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
  11. Cui, Donghui

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193

D

  1. de Kanter, Ruben

    1. You have access
      COMPARISON OF MOUSE AND RAT CYTOCHROME P450-MEDIATED METABOLISM IN LIVER AND INTESTINE
      Marcella Martignoni, Geny Groothuis and Ruben de Kanter
      Drug Metabolism and Disposition June 2006, 34 (6) 1047-1054; DOI: https://doi.org/10.1124/dmd.105.009035
  2. Dellinger, Ryan W.

    1. You have access
      IMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORM
      Ryan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip Lazarus
      Drug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
  3. Demarco, Vincent G.

    1. You have access
      CONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDS
      Vikram Arya, Vincent G. Demarco, Manish Issar and Günther Hochhaus
      Drug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
  4. Dickinson, Ronald G.

    1. You have access
      IN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTION
      Andrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. Miners
      Drug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
  5. Drach, John C.

    1. You have access
      N-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLE
      Philip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. Amidon
      Drug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209

E

  1. Elliot, David J.

    1. You have access
      IN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTION
      Andrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. Miners
      Drug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340

F

  1. Fang, Jia-Long

    1. You have access
      IMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORM
      Ryan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip Lazarus
      Drug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
  2. Forkert, Poh-Gek

    1. You have access
      FORMATION OF N-ALKYLPROTOPORPHYRIN IX FROM METABOLISM OF DIALLYL SULFONE IN LUNG AND LIVER
      Gordon P. Black, Kathy S. Collins, Dylan P. Blacquiere and Poh-Gek Forkert
      Drug Metabolism and Disposition June 2006, 34 (6) 895-900; DOI: https://doi.org/10.1124/dmd.106.009928
  3. Fresneau, Marcel

    1. You have access
      IN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMAN
      H. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard Gross
      Drug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
  4. Furihata, Tomomi

    1. You have access
      INVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVER
      Sachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365

G

  1. Gannon, Shawn A.

    1. You have access
      COMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTES
      Raymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie Api
      Drug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
  2. Gentry, W. Brooks

    1. You have access
      ANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTED
      Grzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks Gentry
      Drug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
  3. Gillespie, Todd A.

    1. You have access
      APPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensis
      Milton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan Kulanthaivel
      Drug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
  4. Goel, Thanh V.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  5. Grimm, Scott W.

    1. You have access
      COMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONS
      Diansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael Zamora
      Drug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
  6. Groothuis, Geny

    1. You have access
      COMPARISON OF MOUSE AND RAT CYTOCHROME P450-MEDIATED METABOLISM IN LIVER AND INTESTINE
      Marcella Martignoni, Geny Groothuis and Ruben de Kanter
      Drug Metabolism and Disposition June 2006, 34 (6) 1047-1054; DOI: https://doi.org/10.1124/dmd.105.009035
  7. Gross, Gerhard

    1. You have access
      IN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMAN
      H. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard Gross
      Drug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
  8. Gruber, Nancy

    1. You have access
      A PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISM
      Sam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne Riggs
      Drug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898

H

  1. Hedeland, Mikael

    1. You have access
      FLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRY
      Annica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael Hedeland
      Drug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
  2. Higuchi, Tomoaki

    1. You have access
      INVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVER
      Sachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
  3. Hochhaus, Günther

    1. You have access
      CONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDS
      Vikram Arya, Vincent G. Demarco, Manish Issar and Günther Hochhaus
      Drug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
  4. Hood, Steven R.

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
  5. Hosokawa, Masakiyo

    1. You have access
      INVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVER
      Sachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
  6. Huitema, Alwin D. R.

    1. You have access
      SATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTES
      Anthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. Huitema
      Drug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326

I

  1. Issar, Manish

    1. You have access
      CONTRARY TO ADULT, NEONATAL RATS SHOW PRONOUNCED BRAIN UPTAKE OF CORTICOSTEROIDS
      Vikram Arya, Vincent G. Demarco, Manish Issar and Günther Hochhaus
      Drug Metabolism and Disposition June 2006, 34 (6) 939-942; DOI: https://doi.org/10.1124/dmd.105.007419
  2. Iyer, Ramaswamy A.

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500

J

  1. Jackson, David A.

    1. You have access
      APPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensis
      Milton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan Kulanthaivel
      Drug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
  2. James, Margaret O.

    1. You have access
      DEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMES
      Leah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. James
      Drug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
  3. Jemal, Mohammed

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
  4. Jönsson, Mats

    1. You have access
      FLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRY
      Annica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael Hedeland
      Drug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516

K

  1. Kawashima, Sachiyo

    1. You have access
      INVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVER
      Sachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
  2. Kearns, Gregory L.

    1. You have access
      BIOTRANSFORMATION OF FLUTICASONE: IN VITRO CHARACTERIZATION
      Robin E. Pearce, J. Steven Leeder and Gregory L. Kearns
      Drug Metabolism and Disposition June 2006, 34 (6) 1035-1040; DOI: https://doi.org/10.1124/dmd.105.009043
  3. Kemper, Raymond A.

    1. You have access
      COMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTES
      Raymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie Api
      Drug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
  4. Khan, Sanaullah

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
  5. Kleinow, Kevin M.

    1. You have access
      DEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMES
      Leah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. James
      Drug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
  6. Kobayashi, Kaoru

    1. You have access
      INVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVER
      Sachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
    2. You have access
      AUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMES
      Toshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
  7. Kretz, Olivier

    1. You have access
      IN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMAN
      H. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard Gross
      Drug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
  8. Kulanthaivel, Palaniappan

    1. You have access
      APPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensis
      Milton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan Kulanthaivel
      Drug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
  9. Kumar, Gondi

    1. You have access
      IDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONS
      Chun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi Kumar
      Drug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367

L

  1. Landowski, Christopher P.

    1. You have access
      N-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLE
      Philip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. Amidon
      Drug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
  2. Lasseter, Kenneth C.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  3. Laurenzana, Elizabeth M.

    1. You have access
      ANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTED
      Grzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks Gentry
      Drug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
  4. Lazarus, Philip

    1. You have access
      IMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORM
      Ryan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip Lazarus
      Drug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
  5. Leeder, J. Steven

    1. You have access
      BIOTRANSFORMATION OF FLUTICASONE: IN VITRO CHARACTERIZATION
      Robin E. Pearce, J. Steven Leeder and Gregory L. Kearns
      Drug Metabolism and Disposition June 2006, 34 (6) 1035-1040; DOI: https://doi.org/10.1124/dmd.105.009043
  6. Lennernäs, Bo

    1. You have access
      FLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRY
      Annica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael Hedeland
      Drug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
  7. Lennernäs, Hans

    1. You have access
      FLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRY
      Annica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael Hedeland
      Drug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
  8. Li, Changling

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  9. Li, Chun

    1. You have access
      IDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONS
      Chun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi Kumar
      Drug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
  10. Lorenzi, Philip L.

    1. You have access
      N-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLE
      Philip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. Amidon
      Drug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
  11. Lu, Xiaowei

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  12. Luquita, Marcelo G.

    1. You have access
      ETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3
      María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. Catania
      Drug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
    2. You have access
      GALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASIS
      Fernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez Pozzi
      Drug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308

M

  1. Mackenzie, Peter I.

    1. You have access
      IN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTION
      Andrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. Miners
      Drug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
  2. Marquez, Brian

    1. You have access
      IDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONS
      Chun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi Kumar
      Drug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
  3. Martignoni, Marcella

    1. You have access
      COMPARISON OF MOUSE AND RAT CYTOCHROME P450-MEDIATED METABOLISM IN LIVER AND INTESTINE
      Marcella Martignoni, Geny Groothuis and Ruben de Kanter
      Drug Metabolism and Disposition June 2006, 34 (6) 1047-1054; DOI: https://doi.org/10.1124/dmd.105.009035
  4. Miller, Donald W.

    1. You have access
      COMPARISON OF DRUG EFFLUX TRANSPORT KINETICS IN VARIOUS BLOOD-BRAIN BARRIER MODELS
      Corbin J. Bachmeier, William J. Trickler and Donald W. Miller
      Drug Metabolism and Disposition June 2006, 34 (6) 998-1003; DOI: https://doi.org/10.1124/dmd.105.006999
  5. Miners, John O.

    1. You have access
      IN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTION
      Andrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. Miners
      Drug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
  6. Mitroka, James

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
  7. Mottino, Aldo D.

    1. You have access
      ETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3
      María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. Catania
      Drug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
    2. You have access
      GALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASIS
      Fernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez Pozzi
      Drug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
  8. Murdock, Paul R.

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185
  9. Murphy, M. Gail

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193

N

  1. Nabb, Diane L.

    1. You have access
      COMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTES
      Raymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie Api
      Drug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
  2. Niwa, Takuro

    1. You have access
      AUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMES
      Toshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
  3. Norlin, Maria

    1. You have access
      FLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRY
      Annica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael Hedeland
      Drug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516

O

  1. Owens, S. Michael

    1. You have access
      ANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTED
      Grzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks Gentry
      Drug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934

P

  1. Pearce, Robin E.

    1. You have access
      BIOTRANSFORMATION OF FLUTICASONE: IN VITRO CHARACTERIZATION
      Robin E. Pearce, J. Steven Leeder and Gregory L. Kearns
      Drug Metabolism and Disposition June 2006, 34 (6) 1035-1040; DOI: https://doi.org/10.1124/dmd.105.009043
  2. Pellegrino, José M.

    1. You have access
      GALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASIS
      Fernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez Pozzi
      Drug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
  3. Pitas, Grzegorz

    1. You have access
      ANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTED
      Grzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks Gentry
      Drug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
  4. Polsky-Fisher, Stacey L.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  5. Pozzi, Enrique J. Sánchez

    1. You have access
      GALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASIS
      Fernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez Pozzi
      Drug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308

R

  1. Riggs, K. Wayne

    1. You have access
      A PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISM
      Sam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne Riggs
      Drug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898
  2. Rinehart, J. Kent

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
  3. Rodrigues, A. David

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  4. Roma, Marcelo G.

    1. You have access
      GALACTOSAMINE PREVENTS ETHINYLESTRADIOL-INDUCED CHOLESTASIS
      Fernando A. Crocenzi, José M. Pellegrino, Viviana A. Catania, Marcelo G. Luquita, Marcelo G. Roma, Aldo D. Mottino and Enrique J. Sánchez Pozzi
      Drug Metabolism and Disposition June 2006, 34 (6) 993-997; DOI: https://doi.org/10.1124/dmd.106.009308
  5. Rowland, Andrew

    1. You have access
      IN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTION
      Andrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. Miners
      Drug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340
  6. Ruiz, María L.

    1. You have access
      ETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3
      María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. Catania
      Drug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
  7. Rurak, Dan W.

    1. You have access
      A PHARMACOKINETIC STUDY OF DIPHENHYDRAMINE TRANSPORT ACROSS THE BLOOD-BRAIN BARRIER IN ADULT SHEEP: POTENTIAL INVOLVEMENT OF A CARRIER-MEDIATED MECHANISM
      Sam C. S. Au-Yeung, Dan W. Rurak, Nancy Gruber and K. Wayne Riggs
      Drug Metabolism and Disposition June 2006, 34 (6) 955-960; DOI: https://doi.org/10.1124/dmd.105.007898

S

  1. Schellens, Jan H. M.

    1. You have access
      SATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTES
      Anthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. Huitema
      Drug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
  2. Schmidt, Douglas F.

    1. You have access
      APPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensis
      Milton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan Kulanthaivel
      Drug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
  3. Shang, Mingying

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  4. Shimizu, Toshiyuki

    1. You have access
      AUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMES
      Toshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
  5. Simpson, Richard C.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  6. Snow, Timothy A.

    1. You have access
      COMPARATIVE METABOLISM OF GERANYL NITRILE AND CITRONELLYL NITRILE IN MOUSE, RAT, AND HUMAN HEPATOCYTES
      Raymond A. Kemper, Diane L. Nabb, Shawn A. Gannon, Timothy A. Snow and Anne Marie Api
      Drug Metabolism and Disposition June 2006, 34 (6) 1019-1029; DOI: https://doi.org/10.1124/dmd.105.005496
  7. Song, Xueqin

    1. You have access
      N-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLE
      Philip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. Amidon
      Drug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
  8. Stegeman, John J.

    1. You have access
      DEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMES
      Leah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. James
      Drug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
  9. Stuchal, Leah D.

    1. You have access
      DEMETHYLATION OF THE PESTICIDE METHOXYCHLOR IN LIVER AND INTESTINE FROM UNTREATED, METHOXYCHLOR-TREATED, AND 3-METHYLCHOLANTHRENE-TREATED CHANNEL CATFISH (ICTALURUS PUNCTATUS): EVIDENCE FOR ROLES OF CYP1 AND CYP3A FAMILY ISOZYMES
      Leah D. Stuchal, Kevin M. Kleinow, John J. Stegeman and Margaret O. James
      Drug Metabolism and Disposition June 2006, 34 (6) 932-938; DOI: https://doi.org/10.1124/dmd.105.009068
  10. Subramanian, Raju

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  11. Surapaneni, Sekhar

    1. You have access
      IDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONS
      Chun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi Kumar
      Drug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367

T

  1. Takama, Kaori

    1. You have access
      INVOLVEMENT OF HEPATOCYTE NUCLEAR FACTOR 4α IN THE DIFFERENT EXPRESSION LEVEL BETWEEN CYP2C9 AND CYP2C19 IN THE HUMAN LIVER
      Sachiyo Kawashima, Kaoru Kobayashi, Kaori Takama, Tomoaki Higuchi, Tomomi Furihata, Masakiyo Hosokawa and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 1012-1018; DOI: https://doi.org/10.1124/dmd.106.009365
  2. Tevell, Annica

    1. You have access
      FLUTAMIDE METABOLISM IN FOUR DIFFERENT SPECIES IN VITRO AND IDENTIFICATION OF FLUTAMIDE METABOLITES IN HUMAN PATIENT URINE BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHY/TANDEM MASS SPECTROMETRY
      Annica Tevell, Hans Lennernäs, Mats Jönsson, Maria Norlin, Bo Lennernäs, Ulf Bondesson and Mikael Hedeland
      Drug Metabolism and Disposition June 2006, 34 (6) 984-992; DOI: https://doi.org/10.1124/dmd.105.008516
  3. Townsend, Leroy B.

    1. You have access
      N-METHYLPURINE DNA GLYCOSYLASE AND 8-OXOGUANINE DNA GLYCOSYLASE METABOLIZE THE ANTIVIRAL NUCLEOSIDE 2-BROMO-5,6-DICHLORO-1-(β-D-RIBOFURANOSYL)BENZIMIDAZOLE
      Philip L. Lorenzi, Christopher P. Landowski, Andrea Brancale, Xueqin Song, Leroy B. Townsend, John C. Drach and Gordon L. Amidon
      Drug Metabolism and Disposition June 2006, 34 (6) 1070-1077; DOI: https://doi.org/10.1124/dmd.105.009209
  4. Trickler, William J.

    1. You have access
      COMPARISON OF DRUG EFFLUX TRANSPORT KINETICS IN VARIOUS BLOOD-BRAIN BARRIER MODELS
      Corbin J. Bachmeier, William J. Trickler and Donald W. Miller
      Drug Metabolism and Disposition June 2006, 34 (6) 998-1003; DOI: https://doi.org/10.1124/dmd.105.006999
  5. Tsunoo, Michio

    1. You have access
      AUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMES
      Toshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
  6. Tu, Pengfei

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300

V

  1. Vaccharajani, Nimish

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
  2. Vega, Jose M.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  3. Vessey, Laura K.

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  4. Vickers, Stanley

    1. You have access
      METABOLISM AND DISPOSITION OF A POTENT AND SELECTIVE GABA-Aα2/3 RECEPTOR AGONIST IN HEALTHY MALE VOLUNTEERS
      Stacey L. Polsky-Fisher, Stanley Vickers, Donghui Cui, Raju Subramanian, Byron H. Arison, Nancy G. B. Agrawal, Thanh V. Goel, Laura K. Vessey, M. Gail Murphy, Kenneth C. Lasseter, Richard C. Simpson, Jose M. Vega and A. David Rodrigues
      Drug Metabolism and Disposition June 2006, 34 (6) 1004-1011; DOI: https://doi.org/10.1124/dmd.105.008193
  5. Villanueva, Silvina S. M.

    1. You have access
      ETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3
      María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. Catania
      Drug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316
  6. Vore, Mary

    1. You have access
      ETHYNYLESTRADIOL INCREASES EXPRESSION AND ACTIVITY OF RAT LIVER MRP3
      María L. Ruiz, Silvina S. M. Villanueva, Marcelo G. Luquita, Mary Vore, Aldo D. Mottino and Viviana A. Catania
      Drug Metabolism and Disposition June 2006, 34 (6) 1030-1034; DOI: https://doi.org/10.1124/dmd.106.009316

W

  1. Wait, Jill C. M.

    1. You have access
      METABOLISM OF [14C]GEMOPATRILAT AFTER ORAL ADMINISTRATION TO RATS, DOGS, AND HUMANS
      Jill C. M. Wait, Nimish Vaccharajani, James Mitroka, Mohammed Jemal, Sanaullah Khan, Samuel J. Bonacorsi, J. Kent Rinehart and Ramaswamy A. Iyer
      Drug Metabolism and Disposition June 2006, 34 (6) 961-970; DOI: https://doi.org/10.1124/dmd.105.007500
  2. Weinberg, Rebecca

    1. You have access
      IMPORTANCE OF UDP-GLUCURONOSYLTRANSFERASE 1A10 (UGT1A10) IN THE DETOXIFICATION OF POLYCYCLIC AROMATIC HYDROCARBONS: DECREASED GLUCURONIDATIVE ACTIVITY OF THE UGT1A10139LYS ISOFORM
      Ryan W. Dellinger, Jia-Long Fang, Gang Chen, Rebecca Weinberg and Philip Lazarus
      Drug Metabolism and Disposition June 2006, 34 (6) 943-949; DOI: https://doi.org/10.1124/dmd.105.009100
  3. Weiss, H. Markus

    1. You have access
      IN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMAN
      H. Markus Weiss, Marcel Fresneau, Gian P. Camenisch, Olivier Kretz and Gerhard Gross
      Drug Metabolism and Disposition June 2006, 34 (6) 971-975; DOI: https://doi.org/10.1124/dmd.105.006429
  4. Williams, D. Keith

    1. You have access
      ANTI-PHENCYCLIDINE MONOCLONAL ANTIBODY BINDING CAPACITY IS NOT THE ONLY DETERMINANT OF EFFECTIVENESS, DISPROVING THE CONCEPT THAT ANTIBODY CAPACITY IS EASILY SURMOUNTED
      Grzegorz Pitas, Elizabeth M. Laurenzana, D. Keith Williams, S. Michael Owens and W. Brooks Gentry
      Drug Metabolism and Disposition June 2006, 34 (6) 906-912; DOI: https://doi.org/10.1124/dmd.105.005934
  5. Williams, J. Andrew

    1. You have access
      IN VITRO CHARACTERIZATION OF LAMOTRIGINE N2-GLUCURONIDATION AND THE LAMOTRIGINE-VALPROIC ACID INTERACTION
      Andrew Rowland, David J. Elliot, J. Andrew Williams, Peter I. Mackenzie, Ronald G. Dickinson and John O. Miners
      Drug Metabolism and Disposition June 2006, 34 (6) 1055-1062; DOI: https://doi.org/10.1124/dmd.106.009340

X

  1. Xiao, Shengyuan

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  2. Xu, Feng

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300

Y

  1. Yang, Donghui

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  2. Yang, Xiaoda

    1. You have access
      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  3. Yi, Ping

    1. You have access
      APPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensis
      Milton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan Kulanthaivel
      Drug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
  4. Yoshimura, Takuya

    1. You have access
      AUTOINDUCTION OF MKC-963 [(R)-1-(1-CYCLOHEXYLETHYLAMINO)-4-PHENYLPHTHALAZINE] METABOLISM IN HEALTHY VOLUNTEERS AND ITS RETROSPECTIVE EVALUATION USING PRIMARY HUMAN HEPATOCYTES AND CDNA-EXPRESSED ENZYMES
      Toshiyuki Shimizu, Kei Akimoto, Takuya Yoshimura, Takuro Niwa, Kaoru Kobayashi, Michio Tsunoo and Kan Chiba
      Drug Metabolism and Disposition June 2006, 34 (6) 950-954; DOI: https://doi.org/10.1124/dmd.105.007997
  5. Yue, Lin

    1. You have access
      CYTOCHROME P450 GENE INDUCTION IN RATS EX VIVO ASSESSED BY QUANTITATIVE REAL-TIME REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTION (TAQMAN)
      Sandra J. Baldwin, Jo L. Bramhall, Charlotte A. Ashby, Lin Yue, Paul R. Murdock, Steven R. Hood, Andrew D. Ayrton and Stephen E. Clarke
      Drug Metabolism and Disposition June 2006, 34 (6) 1063-1069; DOI: https://doi.org/10.1124/dmd.105.008185

Z

  1. Zamora, Ismael

    1. You have access
      COMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONS
      Diansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael Zamora
      Drug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
  2. Zandvliet, Anthe S.

    1. You have access
      SATURABLE BINDING OF INDISULAM TO PLASMA PROTEINS AND DISTRIBUTION TO HUMAN ERYTHROCYTES
      Anthe S. Zandvliet, William Copalu, Jan H. M. Schellens, Jos H. Beijnen and Alwin D. R. Huitema
      Drug Metabolism and Disposition June 2006, 34 (6) 1041-1046; DOI: https://doi.org/10.1124/dmd.105.008326
  3. Zauhar, Randy J.

    1. You have access
      COMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONS
      Diansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael Zamora
      Drug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
  4. Zeng, QingPing

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      IDENTIFICATION OF A NOVEL IN VITRO METABONATE FROM LIVER MICROSOMAL INCUBATIONS
      Chun Li, Sekhar Surapaneni, QingPing Zeng, Brian Marquez, David Chow and Gondi Kumar
      Drug Metabolism and Disposition June 2006, 34 (6) 901-905; DOI: https://doi.org/10.1124/dmd.105.008367
  5. Zhang, Yue

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      ABSORPTION AND METABOLISM OF ASTRAGALI RADIX DECOCTION: IN SILICO, IN VITRO, AND A CASE STUDY IN VIVO
      Feng Xu, Yue Zhang, Shengyuan Xiao, Xiaowei Lu, Donghui Yang, Xiaoda Yang, Changling Li, Mingying Shang, Pengfei Tu and Shaoqing Cai
      Drug Metabolism and Disposition June 2006, 34 (6) 913-924; DOI: https://doi.org/10.1124/dmd.105.008300
  6. Zhou, Diansong

    1. You have access
      COMPARISON OF METHODS FOR THE PREDICTION OF THE METABOLIC SITES FOR CYP3A4-MEDIATED METABOLIC REACTIONS
      Diansong Zhou, Lovisa Afzelius, Scott W. Grimm, Tommy B. Andersson, Randy J. Zauhar and Ismael Zamora
      Drug Metabolism and Disposition June 2006, 34 (6) 976-983; DOI: https://doi.org/10.1124/dmd.105.008631
  7. Zmijewski, Milton

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      APPLICATION OF BIOCATALYSIS TO DRUG METABOLISM: PREPARATION OF MAMMALIAN METABOLITES OF A BIARYL-BIS-SULFONAMIDE AMPA (α-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID) RECEPTOR POTENTIATOR USING Actinoplanes missouriensis
      Milton Zmijewski, Todd A. Gillespie, David A. Jackson, Douglas F. Schmidt, Ping Yi and Palaniappan Kulanthaivel
      Drug Metabolism and Disposition June 2006, 34 (6) 925-931; DOI: https://doi.org/10.1124/dmd.106.009522
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Drug Metabolism and Disposition: 34 (6)
Drug Metabolism and Disposition
Vol. 34, Issue 6
1 Jun 2006
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  • Cytochrome P450 inhibitors. Evaluation of specificities in the in vitrometabolism of therapeutic agents by human liver microsomes.
  • Prediction of Human Clearance of Twenty-Nine Drugs from Hepatic Microsomal Intrinsic Clearance Data: An Examination of In Vitro Half-Life Approach and Nonspecific Binding to Microsomes
  • THE HUMAN INTESTINAL CYTOCHROME P450 “PIE”
  • DRUG-DRUG INTERACTIONS FOR UDP-GLUCURONOSYLTRANSFERASE SUBSTRATES: A PHARMACOKINETIC EXPLANATION FOR TYPICALLY OBSERVED LOW EXPOSURE (AUCI/AUC) RATIOS
  • In Vitro-In Vivo Scaling of CYP Kinetic Data Not Consistent with the Classical Michaelis-Menten Model
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