Index by author
October 01, 2007; Volume 35,Issue 10
A
Abraham, Trent
- You have accessPharmacokinetics, Metabolism, and Excretion of the Intestinal Peptide Transporter 1 (SLC15A1)-Targeted Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2-Amino)propionyl]aminobicyclo[3.1.0.]hexen-2,6-dicarboxylic acid (LY544344) in Rats and Dogs: Assessment of First-Pass Bioactivation and Dose LinearityEverett J. Perkins and Trent AbrahamDrug Metabolism and Disposition October 2007, 35 (10) 1903-1909; DOI: https://doi.org/10.1124/dmd.107.016154
Adachi, Mayuko
- You have accessLack of Formation of Aldehyde Oxidase Dimer Possibly Due to 377G>A Nucleotide SubstitutionKunio Itoh, Hiroaki Maruyama, Mayuko Adachi, Kouichi Hoshino, Nobuaki Watanabe and Yorihisa TanakaDrug Metabolism and Disposition October 2007, 35 (10) 1860-1864; DOI: https://doi.org/10.1124/dmd.107.015503
Aimová, Dagmar
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Akao, Teruaki
- You have accessIn Vitro Metabolism of Isoline, a Pyrrolizidine Alkaloid from Ligularia duciformis, by Rodent Liver Microsomal Esterase and Enhanced Hepatotoxicity by Esterase InhibitorsJun Tang, Teruaki Akao, Norio Nakamura, Zheng-Tao Wang, Kiyoshi Takagawa, Masakiyo Sasahara and Masao HattoriDrug Metabolism and Disposition October 2007, 35 (10) 1832-1839; DOI: https://doi.org/10.1124/dmd.107.016311
Akasawa, Akira
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Aleksunes, Lauren M.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Alvarez, Ana I.
- You have accessInvolvement of Breast Cancer Resistance Protein (ABCG2) in the Biliary Excretion Mechanism of FluoroquinolonesTomohiro Ando, Hiroyuki Kusuhara, Gracia Merino, Ana I. Alvarez, Alfred H. Schinkel and Yuichi SugiyamaDrug Metabolism and Disposition October 2007, 35 (10) 1873-1879; DOI: https://doi.org/10.1124/dmd.107.014969
Amin, Shantu
- You have accessElimination of Antiestrogenic Effects of Active Tamoxifen Metabolites by GlucuronidationYan Zheng, Dongxiao Sun, Arun K. Sharma, Gang Chen, Shantu Amin and Philip LazarusDrug Metabolism and Disposition October 2007, 35 (10) 1942-1948; DOI: https://doi.org/10.1124/dmd.107.016279
Ando, Tomohiro
- You have accessInvolvement of Breast Cancer Resistance Protein (ABCG2) in the Biliary Excretion Mechanism of FluoroquinolonesTomohiro Ando, Hiroyuki Kusuhara, Gracia Merino, Ana I. Alvarez, Alfred H. Schinkel and Yuichi SugiyamaDrug Metabolism and Disposition October 2007, 35 (10) 1873-1879; DOI: https://doi.org/10.1124/dmd.107.014969
Augustine, Lisa
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
Augustine, Lisa M.
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Axelsson, Bengt-Olof
- You have accessDifferences in Endogenous Esterification and Retention in the Rat Trachea between Budesonide and Ciclesonide Active MetaboliteKristina Lexmüller, Helena Gullstrand, Bengt-Olof Axelsson, Petter Sjölin, Solange H. Korn, David S. Silberstein and Anna Miller-LarssonDrug Metabolism and Disposition October 2007, 35 (10) 1788-1796; DOI: https://doi.org/10.1124/dmd.107.015297
B
Bai, Stephen A.
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Bakhiya, Nadiya
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
Banks, Matthew L.
- You have accessAmbient Temperature Effects on 3,4-Methylenedioxymethamphetamine-Induced Thermodysregulation and Pharmacokinetics in Male MonkeysMatthew L. Banks, Jon E. Sprague, David F. Kisor, Paul W. Czoty, David E. Nichols and Michael A. NaderDrug Metabolism and Disposition October 2007, 35 (10) 1840-1845; DOI: https://doi.org/10.1124/dmd.107.016261
Barnes, Sarah N.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
Barter, Z. E.
- You have accessDisparity in Holoprotein/Apoprotein Ratios of Different Standards Used for Immunoquantification of Hepatic Cytochrome P450 EnzymesH. F. Perrett, Z. E. Barter, B. C. Jones, H. Yamazaki, G. T. Tucker and A. Rostami-HodjeganDrug Metabolism and Disposition October 2007, 35 (10) 1733-1736; DOI: https://doi.org/10.1124/dmd.107.015743
Batke, Monika
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
Bayliss, M. K.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Besselsen, David G.
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Bhadhprasit, Wattanaporn
- You have accessInvolvement of Glucocorticoid Receptor and Pregnane X Receptor in the Regulation of Mouse CYP3A44 Female-Predominant Expression by Glucocorticoid HormoneWattanaporn Bhadhprasit, Tsutomu Sakuma, Nobuyuki Hatakeyama, Masahiro Fuwa, Kaori Kitajima and Nobuo NemotoDrug Metabolism and Disposition October 2007, 35 (10) 1880-1885; DOI: https://doi.org/10.1124/dmd.107.016832
Black, Christopher B.
- You have accessIn Vitro Prediction and in Vivo Verification of Enantioselective Human Tofisopam Metabolite ProfilesMichael D. Cameron, Jason Wright, Christopher B. Black and Naidong YeDrug Metabolism and Disposition October 2007, 35 (10) 1894-1902; DOI: https://doi.org/10.1124/dmd.107.015875
Brogdon, Bernice
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Brüggemann, Svenja Kristin
- You have accessInfluence of Short-Term Use of Dexamethasone on the Pharmacokinetics of Ifosfamide in PatientsSvenja Kristin Brüggemann, Sonja Pfäffle, Stefan Oliver Peters and Thomas WagnerDrug Metabolism and Disposition October 2007, 35 (10) 1721-1724; DOI: https://doi.org/10.1124/dmd.106.014043
Buerger, C.
- You have accessDoes Linezolid Inhibit Its Own Metabolism?—Population Pharmacokinetics As a Tool to Explain the Observed Nonlinearity in Both Healthy Volunteers and Septic PatientsN. Plock, C. Buerger, C. Joukhadar, S. Kljucar and C. KloftDrug Metabolism and Disposition October 2007, 35 (10) 1816-1823; DOI: https://doi.org/10.1124/dmd.106.013755
C
Cameron, Michael D.
- You have accessIn Vitro Prediction and in Vivo Verification of Enantioselective Human Tofisopam Metabolite ProfilesMichael D. Cameron, Jason Wright, Christopher B. Black and Naidong YeDrug Metabolism and Disposition October 2007, 35 (10) 1894-1902; DOI: https://doi.org/10.1124/dmd.107.015875
Cellucci, Antonella
- You have accessHigh-Throughput Radiometric CYP2C19 Inhibition Assay Using Tritiated (S)-MephenytoinAnnalise Di Marco, Antonella Cellucci, Ashok Chaudhary, Massimiliano Fonsi and Ralph LauferDrug Metabolism and Disposition October 2007, 35 (10) 1737-1743; DOI: https://doi.org/10.1124/dmd.107.016345
Chaudhary, Ashok
- You have accessHigh-Throughput Radiometric CYP2C19 Inhibition Assay Using Tritiated (S)-MephenytoinAnnalise Di Marco, Antonella Cellucci, Ashok Chaudhary, Massimiliano Fonsi and Ralph LauferDrug Metabolism and Disposition October 2007, 35 (10) 1737-1743; DOI: https://doi.org/10.1124/dmd.107.016345
Chen, Cuiping
- You have accessP-glycoprotein Has Differential Effects on the Disposition of Statin Acid and Lactone Forms in mdr1a/b Knockout and Wild-Type MiceCuiping Chen, Jian Lin, Teresa Smolarek and Larry TremaineDrug Metabolism and Disposition October 2007, 35 (10) 1725-1729; DOI: https://doi.org/10.1124/dmd.107.015677
Chen, Gang
- You have accessElimination of Antiestrogenic Effects of Active Tamoxifen Metabolites by GlucuronidationYan Zheng, Dongxiao Sun, Arun K. Sharma, Gang Chen, Shantu Amin and Philip LazarusDrug Metabolism and Disposition October 2007, 35 (10) 1942-1948; DOI: https://doi.org/10.1124/dmd.107.016279
Cherrington, Nathan J.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Chovan, James P.
- You have accessMetabolic Profile of [14C]Bendamustine in Rat Urine and Bile: Preliminary Structural Identification of MetabolitesJames P. Chovan, Feng Li, Erya Yu and Steven C. RingDrug Metabolism and Disposition October 2007, 35 (10) 1744-1753; DOI: https://doi.org/10.1124/dmd.107.015958
Christ, David D.
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Covington, Maryanne B.
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Czoty, Paul W.
- You have accessAmbient Temperature Effects on 3,4-Methylenedioxymethamphetamine-Induced Thermodysregulation and Pharmacokinetics in Male MonkeysMatthew L. Banks, Jon E. Sprague, David F. Kisor, Paul W. Czoty, David E. Nichols and Michael A. NaderDrug Metabolism and Disposition October 2007, 35 (10) 1840-1845; DOI: https://doi.org/10.1124/dmd.107.016261
D
De Buck, Stefan S.
- You have accessPrediction of Human Pharmacokinetics Using Physiologically Based Modeling: A Retrospective Analysis of 26 Clinically Tested DrugsStefan S. De Buck, Vikash K. Sinha, Luca A. Fenu, Marjoleen J. Nijsen, Claire E. Mackie and Ron A. H. J. GilissenDrug Metabolism and Disposition October 2007, 35 (10) 1766-1780; DOI: https://doi.org/10.1124/dmd.107.015644
Decicco, Carl P.
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Degawa, Masakuni
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Deng, Yuzhong
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Desai, Pankaj
- You have accessCytochrome P450 Enzymes and Transporters Induced by Anti-Human Immunodeficiency Virus Protease Inhibitors in Human Hepatocytes: Implications for Predicting Clinical Drug InteractionsVaishali Dixit, Niresh Hariparsad, Fang Li, Pankaj Desai, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition October 2007, 35 (10) 1853-1859; DOI: https://doi.org/10.1124/dmd.107.016089
Di Marco, Annalise
- You have accessHigh-Throughput Radiometric CYP2C19 Inhibition Assay Using Tritiated (S)-MephenytoinAnnalise Di Marco, Antonella Cellucci, Ashok Chaudhary, Massimiliano Fonsi and Ralph LauferDrug Metabolism and Disposition October 2007, 35 (10) 1737-1743; DOI: https://doi.org/10.1124/dmd.107.016345
Dixit, Vaishali
- You have accessCytochrome P450 Enzymes and Transporters Induced by Anti-Human Immunodeficiency Virus Protease Inhibitors in Human Hepatocytes: Implications for Predicting Clinical Drug InteractionsVaishali Dixit, Niresh Hariparsad, Fang Li, Pankaj Desai, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition October 2007, 35 (10) 1853-1859; DOI: https://doi.org/10.1124/dmd.107.016089
Duan, James J.-W.
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
E
Engst, Wolfram
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
F
Fenu, Luca A.
- You have accessPrediction of Human Pharmacokinetics Using Physiologically Based Modeling: A Retrospective Analysis of 26 Clinically Tested DrugsStefan S. De Buck, Vikash K. Sinha, Luca A. Fenu, Marjoleen J. Nijsen, Claire E. Mackie and Ron A. H. J. GilissenDrug Metabolism and Disposition October 2007, 35 (10) 1766-1780; DOI: https://doi.org/10.1124/dmd.107.015644
Fisher, Craig D.
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Fluhler, Eric
- You have accessInterspecies Prediction of Human Drug Clearance Based on Scaling Data from One or Two Animal SpeciesHuadong Tang, Azher Hussain, Mauricio Leal, Michael Mayersohn and Eric FluhlerDrug Metabolism and Disposition October 2007, 35 (10) 1886-1893; DOI: https://doi.org/10.1124/dmd.107.016188
Fonsi, Massimiliano
- You have accessHigh-Throughput Radiometric CYP2C19 Inhibition Assay Using Tritiated (S)-MephenytoinAnnalise Di Marco, Antonella Cellucci, Ashok Chaudhary, Massimiliano Fonsi and Ralph LauferDrug Metabolism and Disposition October 2007, 35 (10) 1737-1743; DOI: https://doi.org/10.1124/dmd.107.016345
Fossler, Michael J.
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Frank, Heinz
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
Freathy, C.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Frei, Eva
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Fujiwara, Ryoichi
- You have accessInteractions between Human UGT1A1, UGT1A4, and UGT1A6 Affect Their Enzymatic ActivitiesRyoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka, Miki Katoh and Tsuyoshi YokoiDrug Metabolism and Disposition October 2007, 35 (10) 1781-1787; DOI: https://doi.org/10.1124/dmd.107.016402
Fukami, Tatsuki
- You have accessHuman CYP2A6 Is Induced by Estrogen via Estrogen ReceptorEriko Higashi, Tatsuki Fukami, Masahiro Itoh, Satoru Kyo, Masaki Inoue, Tsuyoshi Yokoi and Miki NakajimaDrug Metabolism and Disposition October 2007, 35 (10) 1935-1941; DOI: https://doi.org/10.1124/dmd.107.016568
Fuwa, Masahiro
- You have accessInvolvement of Glucocorticoid Receptor and Pregnane X Receptor in the Regulation of Mouse CYP3A44 Female-Predominant Expression by Glucocorticoid HormoneWattanaporn Bhadhprasit, Tsutomu Sakuma, Nobuyuki Hatakeyama, Masahiro Fuwa, Kaori Kitajima and Nobuo NemotoDrug Metabolism and Disposition October 2007, 35 (10) 1880-1885; DOI: https://doi.org/10.1124/dmd.107.016832
G
Garner, C. Edwin
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Gilissen, Ron A. H. J.
- You have accessPrediction of Human Pharmacokinetics Using Physiologically Based Modeling: A Retrospective Analysis of 26 Clinically Tested DrugsStefan S. De Buck, Vikash K. Sinha, Luca A. Fenu, Marjoleen J. Nijsen, Claire E. Mackie and Ron A. H. J. GilissenDrug Metabolism and Disposition October 2007, 35 (10) 1766-1780; DOI: https://doi.org/10.1124/dmd.107.015644
Glatt, Hansruedi
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
Goedken, Michael J.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
Gullstrand, Helena
- You have accessDifferences in Endogenous Esterification and Retention in the Rat Trachea between Budesonide and Ciclesonide Active MetaboliteKristina Lexmüller, Helena Gullstrand, Bengt-Olof Axelsson, Petter Sjölin, Solange H. Korn, David S. Silberstein and Anna Miller-LarssonDrug Metabolism and Disposition October 2007, 35 (10) 1788-1796; DOI: https://doi.org/10.1124/dmd.107.015297
H
Haraguchi, Koichi
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Hariparsad, Niresh
- You have accessCytochrome P450 Enzymes and Transporters Induced by Anti-Human Immunodeficiency Virus Protease Inhibitors in Human Hepatocytes: Implications for Predicting Clinical Drug InteractionsVaishali Dixit, Niresh Hariparsad, Fang Li, Pankaj Desai, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition October 2007, 35 (10) 1853-1859; DOI: https://doi.org/10.1124/dmd.107.016089
Hatakeyama, Nobuyuki
- You have accessInvolvement of Glucocorticoid Receptor and Pregnane X Receptor in the Regulation of Mouse CYP3A44 Female-Predominant Expression by Glucocorticoid HormoneWattanaporn Bhadhprasit, Tsutomu Sakuma, Nobuyuki Hatakeyama, Masahiro Fuwa, Kaori Kitajima and Nobuo NemotoDrug Metabolism and Disposition October 2007, 35 (10) 1880-1885; DOI: https://doi.org/10.1124/dmd.107.016832
Hattori, Masao
- You have accessIn Vitro Metabolism of Isoline, a Pyrrolizidine Alkaloid from Ligularia duciformis, by Rodent Liver Microsomal Esterase and Enhanced Hepatotoxicity by Esterase InhibitorsJun Tang, Teruaki Akao, Norio Nakamura, Zheng-Tao Wang, Kiyoshi Takagawa, Masakiyo Sasahara and Masao HattoriDrug Metabolism and Disposition October 2007, 35 (10) 1832-1839; DOI: https://doi.org/10.1124/dmd.107.016311
Higashi, Eriko
- You have accessHuman CYP2A6 Is Induced by Estrogen via Estrogen ReceptorEriko Higashi, Tatsuki Fukami, Masahiro Itoh, Satoru Kyo, Masaki Inoue, Tsuyoshi Yokoi and Miki NakajimaDrug Metabolism and Disposition October 2007, 35 (10) 1935-1941; DOI: https://doi.org/10.1124/dmd.107.016568
Hinai, Yudai
- You have accessCharacterization of Human Cytochrome P450 Enzymes Involved in the Metabolism of CilostazolMasahiro Hiratsuka, Yudai Hinai, Takamitsu Sasaki, Yumiko Konno, Kenichi Imagawa, Masaaki Ishikawa and Michinao MizugakiDrug Metabolism and Disposition October 2007, 35 (10) 1730-1732; DOI: https://doi.org/10.1124/dmd.107.016758
Hiratsuka, Masahiro
- You have accessCharacterization of Human Cytochrome P450 Enzymes Involved in the Metabolism of CilostazolMasahiro Hiratsuka, Yudai Hinai, Takamitsu Sasaki, Yumiko Konno, Kenichi Imagawa, Masaaki Ishikawa and Michinao MizugakiDrug Metabolism and Disposition October 2007, 35 (10) 1730-1732; DOI: https://doi.org/10.1124/dmd.107.016758
Hirota, Takashi
- You have accessCovalent Binding of Rofecoxib, but Not Other Cyclooxygenase-2 Inhibitors, to Allysine Aldehyde in Elastin of Human AortaMasataka Oitate, Takashi Hirota, Takahiro Murai, Shin-ichi Miura and Toshihiko IkedaDrug Metabolism and Disposition October 2007, 35 (10) 1846-1852; DOI: https://doi.org/10.1124/dmd.107.016121
Ho, S.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Hodek, Petr
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Hoshino, Kouichi
- You have accessLack of Formation of Aldehyde Oxidase Dimer Possibly Due to 377G>A Nucleotide SubstitutionKunio Itoh, Hiroaki Maruyama, Mayuko Adachi, Kouichi Hoshino, Nobuaki Watanabe and Yorihisa TanakaDrug Metabolism and Disposition October 2007, 35 (10) 1860-1864; DOI: https://doi.org/10.1124/dmd.107.015503
Hudeček, Jiří
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Hussain, Azher
- You have accessInterspecies Prediction of Human Drug Clearance Based on Scaling Data from One or Two Animal SpeciesHuadong Tang, Azher Hussain, Mauricio Leal, Michael Mayersohn and Eric FluhlerDrug Metabolism and Disposition October 2007, 35 (10) 1886-1893; DOI: https://doi.org/10.1124/dmd.107.016188
I
Ikeda, Toshihiko
- You have accessCovalent Binding of Rofecoxib, but Not Other Cyclooxygenase-2 Inhibitors, to Allysine Aldehyde in Elastin of Human AortaMasataka Oitate, Takashi Hirota, Takahiro Murai, Shin-ichi Miura and Toshihiko IkedaDrug Metabolism and Disposition October 2007, 35 (10) 1846-1852; DOI: https://doi.org/10.1124/dmd.107.016121
Ikushiro, Shin-ichi
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Imagawa, Kenichi
- You have accessCharacterization of Human Cytochrome P450 Enzymes Involved in the Metabolism of CilostazolMasahiro Hiratsuka, Yudai Hinai, Takamitsu Sasaki, Yumiko Konno, Kenichi Imagawa, Masaaki Ishikawa and Michinao MizugakiDrug Metabolism and Disposition October 2007, 35 (10) 1730-1732; DOI: https://doi.org/10.1124/dmd.107.016758
Inoue, Masaki
- You have accessHuman CYP2A6 Is Induced by Estrogen via Estrogen ReceptorEriko Higashi, Tatsuki Fukami, Masahiro Itoh, Satoru Kyo, Masaki Inoue, Tsuyoshi Yokoi and Miki NakajimaDrug Metabolism and Disposition October 2007, 35 (10) 1935-1941; DOI: https://doi.org/10.1124/dmd.107.016568
Ishikawa, Masaaki
- You have accessCharacterization of Human Cytochrome P450 Enzymes Involved in the Metabolism of CilostazolMasahiro Hiratsuka, Yudai Hinai, Takamitsu Sasaki, Yumiko Konno, Kenichi Imagawa, Masaaki Ishikawa and Michinao MizugakiDrug Metabolism and Disposition October 2007, 35 (10) 1730-1732; DOI: https://doi.org/10.1124/dmd.107.016758
Itoh, Kunio
- You have accessLack of Formation of Aldehyde Oxidase Dimer Possibly Due to 377G>A Nucleotide SubstitutionKunio Itoh, Hiroaki Maruyama, Mayuko Adachi, Kouichi Hoshino, Nobuaki Watanabe and Yorihisa TanakaDrug Metabolism and Disposition October 2007, 35 (10) 1860-1864; DOI: https://doi.org/10.1124/dmd.107.015503
Itoh, Masahiro
- You have accessHuman CYP2A6 Is Induced by Estrogen via Estrogen ReceptorEriko Higashi, Tatsuki Fukami, Masahiro Itoh, Satoru Kyo, Masaki Inoue, Tsuyoshi Yokoi and Miki NakajimaDrug Metabolism and Disposition October 2007, 35 (10) 1935-1941; DOI: https://doi.org/10.1124/dmd.107.016568
J
Jakowski, Amy B.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
Jinno, Hideto
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Jones, A. E.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Jones, B. C.
- You have accessDisparity in Holoprotein/Apoprotein Ratios of Different Standards Used for Immunoquantification of Hepatic Cytochrome P450 EnzymesH. F. Perrett, Z. E. Barter, B. C. Jones, H. Yamazaki, G. T. Tucker and A. Rostami-HodjeganDrug Metabolism and Disposition October 2007, 35 (10) 1733-1736; DOI: https://doi.org/10.1124/dmd.107.015743
Joukhadar, C.
- You have accessDoes Linezolid Inhibit Its Own Metabolism?—Population Pharmacokinetics As a Tool to Explain the Observed Nonlinearity in Both Healthy Volunteers and Septic PatientsN. Plock, C. Buerger, C. Joukhadar, S. Kljucar and C. KloftDrug Metabolism and Disposition October 2007, 35 (10) 1816-1823; DOI: https://doi.org/10.1124/dmd.106.013755
Jung, Da W.
- You have accessInduction of Hepatic CYP2E1 by a Subtoxic Dose of Acetaminophen in Rats: Increase in Dichloromethane Metabolism and Carboxyhemoglobin ElevationSu N. Kim, Ji Y. Seo, Da W. Jung, Min Y. Lee, Young S. Jung and Young C. KimDrug Metabolism and Disposition October 2007, 35 (10) 1754-1758; DOI: https://doi.org/10.1124/dmd.107.015545
Jung, Young S.
- You have accessInduction of Hepatic CYP2E1 by a Subtoxic Dose of Acetaminophen in Rats: Increase in Dichloromethane Metabolism and Carboxyhemoglobin ElevationSu N. Kim, Ji Y. Seo, Da W. Jung, Min Y. Lee, Young S. Jung and Young C. KimDrug Metabolism and Disposition October 2007, 35 (10) 1754-1758; DOI: https://doi.org/10.1124/dmd.107.015545
K
Kamatani, Naoyuki
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Kaniwa, Nahoko
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Kanno, Jun
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Kato, Yoshihisa
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Katoh, Miki
- You have accessInteractions between Human UGT1A1, UGT1A4, and UGT1A6 Affect Their Enzymatic ActivitiesRyoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka, Miki Katoh and Tsuyoshi YokoiDrug Metabolism and Disposition October 2007, 35 (10) 1781-1787; DOI: https://doi.org/10.1124/dmd.107.016402
Kim, Dong-Hyun
- You have accessMechanism-Based Inactivation of Cytochrome P450 2A6 by Decursinol Angelate Isolated from Angelica GigasHye Hyun Yoo, Min Woo Lee, Young Choong Kim, Chul-Ho Yun and Dong-Hyun KimDrug Metabolism and Disposition October 2007, 35 (10) 1759-1765; DOI: https://doi.org/10.1124/dmd.107.016584
Kim, Su-Ryang
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Kim, Su N.
- You have accessInduction of Hepatic CYP2E1 by a Subtoxic Dose of Acetaminophen in Rats: Increase in Dichloromethane Metabolism and Carboxyhemoglobin ElevationSu N. Kim, Ji Y. Seo, Da W. Jung, Min Y. Lee, Young S. Jung and Young C. KimDrug Metabolism and Disposition October 2007, 35 (10) 1754-1758; DOI: https://doi.org/10.1124/dmd.107.015545
Kim, Young C.
- You have accessInduction of Hepatic CYP2E1 by a Subtoxic Dose of Acetaminophen in Rats: Increase in Dichloromethane Metabolism and Carboxyhemoglobin ElevationSu N. Kim, Ji Y. Seo, Da W. Jung, Min Y. Lee, Young S. Jung and Young C. KimDrug Metabolism and Disposition October 2007, 35 (10) 1754-1758; DOI: https://doi.org/10.1124/dmd.107.015545
Kim, Young Choong
- You have accessMechanism-Based Inactivation of Cytochrome P450 2A6 by Decursinol Angelate Isolated from Angelica GigasHye Hyun Yoo, Min Woo Lee, Young Choong Kim, Chul-Ho Yun and Dong-Hyun KimDrug Metabolism and Disposition October 2007, 35 (10) 1759-1765; DOI: https://doi.org/10.1124/dmd.107.016584
Kisor, David F.
- You have accessAmbient Temperature Effects on 3,4-Methylenedioxymethamphetamine-Induced Thermodysregulation and Pharmacokinetics in Male MonkeysMatthew L. Banks, Jon E. Sprague, David F. Kisor, Paul W. Czoty, David E. Nichols and Michael A. NaderDrug Metabolism and Disposition October 2007, 35 (10) 1840-1845; DOI: https://doi.org/10.1124/dmd.107.016261
Kitajima, Kaori
- You have accessInvolvement of Glucocorticoid Receptor and Pregnane X Receptor in the Regulation of Mouse CYP3A44 Female-Predominant Expression by Glucocorticoid HormoneWattanaporn Bhadhprasit, Tsutomu Sakuma, Nobuyuki Hatakeyama, Masahiro Fuwa, Kaori Kitajima and Nobuo NemotoDrug Metabolism and Disposition October 2007, 35 (10) 1880-1885; DOI: https://doi.org/10.1124/dmd.107.016832
Klaassen, Curtis D.
- You have accessImportance of Hepatic Induction of Constitutive Androstane Receptor and Other Transcription Factors That Regulate Xenobiotic Metabolism and TransportJay S. Petrick and Curtis D. KlaassenDrug Metabolism and Disposition October 2007, 35 (10) 1806-1815; DOI: https://doi.org/10.1124/dmd.107.015974
Kljucar, S.
- You have accessDoes Linezolid Inhibit Its Own Metabolism?—Population Pharmacokinetics As a Tool to Explain the Observed Nonlinearity in Both Healthy Volunteers and Septic PatientsN. Plock, C. Buerger, C. Joukhadar, S. Kljucar and C. KloftDrug Metabolism and Disposition October 2007, 35 (10) 1816-1823; DOI: https://doi.org/10.1124/dmd.106.013755
Kloft, C.
- You have accessDoes Linezolid Inhibit Its Own Metabolism?—Population Pharmacokinetics As a Tool to Explain the Observed Nonlinearity in Both Healthy Volunteers and Septic PatientsN. Plock, C. Buerger, C. Joukhadar, S. Kljucar and C. KloftDrug Metabolism and Disposition October 2007, 35 (10) 1816-1823; DOI: https://doi.org/10.1124/dmd.106.013755
Koga, Nobuyuki
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Konno, Yumiko
- You have accessCharacterization of Human Cytochrome P450 Enzymes Involved in the Metabolism of CilostazolMasahiro Hiratsuka, Yudai Hinai, Takamitsu Sasaki, Yumiko Konno, Kenichi Imagawa, Masaaki Ishikawa and Michinao MizugakiDrug Metabolism and Disposition October 2007, 35 (10) 1730-1732; DOI: https://doi.org/10.1124/dmd.107.016758
Korn, Solange H.
- You have accessDifferences in Endogenous Esterification and Retention in the Rat Trachea between Budesonide and Ciclesonide Active MetaboliteKristina Lexmüller, Helena Gullstrand, Bengt-Olof Axelsson, Petter Sjölin, Solange H. Korn, David S. Silberstein and Anna Miller-LarssonDrug Metabolism and Disposition October 2007, 35 (10) 1788-1796; DOI: https://doi.org/10.1124/dmd.107.015297
Kotrbová, Věra
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Kuester, R. K.
- You have accessPrediction of Metabolic Clearance of Bisphenol A (4,4 ′-Dihydroxy-2,2-diphenylpropane) using Cryopreserved Human HepatocytesR. K. Kuester and I. G. SipesDrug Metabolism and Disposition October 2007, 35 (10) 1910-1915; DOI: https://doi.org/10.1124/dmd.107.014787
Kusuhara, Hiroyuki
- You have accessInvolvement of Breast Cancer Resistance Protein (ABCG2) in the Biliary Excretion Mechanism of FluoroquinolonesTomohiro Ando, Hiroyuki Kusuhara, Gracia Merino, Ana I. Alvarez, Alfred H. Schinkel and Yuichi SugiyamaDrug Metabolism and Disposition October 2007, 35 (10) 1873-1879; DOI: https://doi.org/10.1124/dmd.107.014969
Kyo, Satoru
- You have accessHuman CYP2A6 Is Induced by Estrogen via Estrogen ReceptorEriko Higashi, Tatsuki Fukami, Masahiro Itoh, Satoru Kyo, Masaki Inoue, Tsuyoshi Yokoi and Miki NakajimaDrug Metabolism and Disposition October 2007, 35 (10) 1935-1941; DOI: https://doi.org/10.1124/dmd.107.016568
L
Laake, Janet
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
Laufer, Ralph
- You have accessHigh-Throughput Radiometric CYP2C19 Inhibition Assay Using Tritiated (S)-MephenytoinAnnalise Di Marco, Antonella Cellucci, Ashok Chaudhary, Massimiliano Fonsi and Ralph LauferDrug Metabolism and Disposition October 2007, 35 (10) 1737-1743; DOI: https://doi.org/10.1124/dmd.107.016345
Lazarus, Philip
- You have accessElimination of Antiestrogenic Effects of Active Tamoxifen Metabolites by GlucuronidationYan Zheng, Dongxiao Sun, Arun K. Sharma, Gang Chen, Shantu Amin and Philip LazarusDrug Metabolism and Disposition October 2007, 35 (10) 1942-1948; DOI: https://doi.org/10.1124/dmd.107.016279
Leal, Mauricio
- You have accessInterspecies Prediction of Human Drug Clearance Based on Scaling Data from One or Two Animal SpeciesHuadong Tang, Azher Hussain, Mauricio Leal, Michael Mayersohn and Eric FluhlerDrug Metabolism and Disposition October 2007, 35 (10) 1886-1893; DOI: https://doi.org/10.1124/dmd.107.016188
Lee, Min Woo
- You have accessMechanism-Based Inactivation of Cytochrome P450 2A6 by Decursinol Angelate Isolated from Angelica GigasHye Hyun Yoo, Min Woo Lee, Young Choong Kim, Chul-Ho Yun and Dong-Hyun KimDrug Metabolism and Disposition October 2007, 35 (10) 1759-1765; DOI: https://doi.org/10.1124/dmd.107.016584
Lee, Min Y.
- You have accessInduction of Hepatic CYP2E1 by a Subtoxic Dose of Acetaminophen in Rats: Increase in Dichloromethane Metabolism and Carboxyhemoglobin ElevationSu N. Kim, Ji Y. Seo, Da W. Jung, Min Y. Lee, Young S. Jung and Young C. KimDrug Metabolism and Disposition October 2007, 35 (10) 1754-1758; DOI: https://doi.org/10.1124/dmd.107.015545
Lexmüller, Kristina
- You have accessDifferences in Endogenous Esterification and Retention in the Rat Trachea between Budesonide and Ciclesonide Active MetaboliteKristina Lexmüller, Helena Gullstrand, Bengt-Olof Axelsson, Petter Sjölin, Solange H. Korn, David S. Silberstein and Anna Miller-LarssonDrug Metabolism and Disposition October 2007, 35 (10) 1788-1796; DOI: https://doi.org/10.1124/dmd.107.015297
Li, Fang
- You have accessCytochrome P450 Enzymes and Transporters Induced by Anti-Human Immunodeficiency Virus Protease Inhibitors in Human Hepatocytes: Implications for Predicting Clinical Drug InteractionsVaishali Dixit, Niresh Hariparsad, Fang Li, Pankaj Desai, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition October 2007, 35 (10) 1853-1859; DOI: https://doi.org/10.1124/dmd.107.016089
Li, Feng
- You have accessMetabolic Profile of [14C]Bendamustine in Rat Urine and Bile: Preliminary Structural Identification of MetabolitesJames P. Chovan, Feng Li, Erya Yu and Steven C. RingDrug Metabolism and Disposition October 2007, 35 (10) 1744-1753; DOI: https://doi.org/10.1124/dmd.107.015958
Lickteig, Andrew J.
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Lin, Jian
- You have accessP-glycoprotein Has Differential Effects on the Disposition of Statin Acid and Lactone Forms in mdr1a/b Knockout and Wild-Type MiceCuiping Chen, Jian Lin, Teresa Smolarek and Larry TremaineDrug Metabolism and Disposition October 2007, 35 (10) 1725-1729; DOI: https://doi.org/10.1124/dmd.107.015677
Lindsay, N.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Liu, Rui-Qin
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Lowdon, B. M.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
M
Mackie, Claire E.
- You have accessPrediction of Human Pharmacokinetics Using Physiologically Based Modeling: A Retrospective Analysis of 26 Clinically Tested DrugsStefan S. De Buck, Vikash K. Sinha, Luca A. Fenu, Marjoleen J. Nijsen, Claire E. Mackie and Ron A. H. J. GilissenDrug Metabolism and Disposition October 2007, 35 (10) 1766-1780; DOI: https://doi.org/10.1124/dmd.107.015644
Maduskuie, Thomas
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Manautou, Jose E.
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Manautou, José E.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
Manchee, G. R.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Maruyama, Hiroaki
- You have accessLack of Formation of Aldehyde Oxidase Dimer Possibly Due to 377G>A Nucleotide SubstitutionKunio Itoh, Hiroaki Maruyama, Mayuko Adachi, Kouichi Hoshino, Nobuaki Watanabe and Yorihisa TanakaDrug Metabolism and Disposition October 2007, 35 (10) 1860-1864; DOI: https://doi.org/10.1124/dmd.107.015503
Matsumoto, Kenji
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Mayersohn, Michael
- You have accessInterspecies Prediction of Human Drug Clearance Based on Scaling Data from One or Two Animal SpeciesHuadong Tang, Azher Hussain, Mauricio Leal, Michael Mayersohn and Eric FluhlerDrug Metabolism and Disposition October 2007, 35 (10) 1886-1893; DOI: https://doi.org/10.1124/dmd.107.016188
Merino, Gracia
- You have accessInvolvement of Breast Cancer Resistance Protein (ABCG2) in the Biliary Excretion Mechanism of FluoroquinolonesTomohiro Ando, Hiroyuki Kusuhara, Gracia Merino, Ana I. Alvarez, Alfred H. Schinkel and Yuichi SugiyamaDrug Metabolism and Disposition October 2007, 35 (10) 1873-1879; DOI: https://doi.org/10.1124/dmd.107.014969
Miller-Larsson, Anna
- You have accessDifferences in Endogenous Esterification and Retention in the Rat Trachea between Budesonide and Ciclesonide Active MetaboliteKristina Lexmüller, Helena Gullstrand, Bengt-Olof Axelsson, Petter Sjölin, Solange H. Korn, David S. Silberstein and Anna Miller-LarssonDrug Metabolism and Disposition October 2007, 35 (10) 1788-1796; DOI: https://doi.org/10.1124/dmd.107.015297
Minami, Hironobu
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Miura, Shin-ichi
- You have accessCovalent Binding of Rofecoxib, but Not Other Cyclooxygenase-2 Inhibitors, to Allysine Aldehyde in Elastin of Human AortaMasataka Oitate, Takashi Hirota, Takahiro Murai, Shin-ichi Miura and Toshihiko IkedaDrug Metabolism and Disposition October 2007, 35 (10) 1846-1852; DOI: https://doi.org/10.1124/dmd.107.016121
Mizugaki, Michinao
- You have accessCharacterization of Human Cytochrome P450 Enzymes Involved in the Metabolism of CilostazolMasahiro Hiratsuka, Yudai Hinai, Takamitsu Sasaki, Yumiko Konno, Kenichi Imagawa, Masaaki Ishikawa and Michinao MizugakiDrug Metabolism and Disposition October 2007, 35 (10) 1730-1732; DOI: https://doi.org/10.1124/dmd.107.016758
Monien, Bernhard H.
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
Mrázová, Barbora
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Murai, Takahiro
- You have accessCovalent Binding of Rofecoxib, but Not Other Cyclooxygenase-2 Inhibitors, to Allysine Aldehyde in Elastin of Human AortaMasataka Oitate, Takashi Hirota, Takahiro Murai, Shin-ichi Miura and Toshihiko IkedaDrug Metabolism and Disposition October 2007, 35 (10) 1846-1852; DOI: https://doi.org/10.1124/dmd.107.016121
N
Nader, Michael A.
- You have accessAmbient Temperature Effects on 3,4-Methylenedioxymethamphetamine-Induced Thermodysregulation and Pharmacokinetics in Male MonkeysMatthew L. Banks, Jon E. Sprague, David F. Kisor, Paul W. Czoty, David E. Nichols and Michael A. NaderDrug Metabolism and Disposition October 2007, 35 (10) 1840-1845; DOI: https://doi.org/10.1124/dmd.107.016261
Nakajima, Miki
- You have accessHuman CYP2A6 Is Induced by Estrogen via Estrogen ReceptorEriko Higashi, Tatsuki Fukami, Masahiro Itoh, Satoru Kyo, Masaki Inoue, Tsuyoshi Yokoi and Miki NakajimaDrug Metabolism and Disposition October 2007, 35 (10) 1935-1941; DOI: https://doi.org/10.1124/dmd.107.016568
- You have accessInteractions between Human UGT1A1, UGT1A4, and UGT1A6 Affect Their Enzymatic ActivitiesRyoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka, Miki Katoh and Tsuyoshi YokoiDrug Metabolism and Disposition October 2007, 35 (10) 1781-1787; DOI: https://doi.org/10.1124/dmd.107.016402
Nakamura, Norio
- You have accessIn Vitro Metabolism of Isoline, a Pyrrolizidine Alkaloid from Ligularia duciformis, by Rodent Liver Microsomal Esterase and Enhanced Hepatotoxicity by Esterase InhibitorsJun Tang, Teruaki Akao, Norio Nakamura, Zheng-Tao Wang, Kiyoshi Takagawa, Masakiyo Sasahara and Masao HattoriDrug Metabolism and Disposition October 2007, 35 (10) 1832-1839; DOI: https://doi.org/10.1124/dmd.107.016311
Nemoto, Nobuo
- You have accessInvolvement of Glucocorticoid Receptor and Pregnane X Receptor in the Regulation of Mouse CYP3A44 Female-Predominant Expression by Glucocorticoid HormoneWattanaporn Bhadhprasit, Tsutomu Sakuma, Nobuyuki Hatakeyama, Masahiro Fuwa, Kaori Kitajima and Nobuo NemotoDrug Metabolism and Disposition October 2007, 35 (10) 1880-1885; DOI: https://doi.org/10.1124/dmd.107.016832
Newton, Robert C.
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Nichols, David E.
- You have accessAmbient Temperature Effects on 3,4-Methylenedioxymethamphetamine-Induced Thermodysregulation and Pharmacokinetics in Male MonkeysMatthew L. Banks, Jon E. Sprague, David F. Kisor, Paul W. Czoty, David E. Nichols and Michael A. NaderDrug Metabolism and Disposition October 2007, 35 (10) 1840-1845; DOI: https://doi.org/10.1124/dmd.107.016261
Nijsen, Marjoleen J.
- You have accessPrediction of Human Pharmacokinetics Using Physiologically Based Modeling: A Retrospective Analysis of 26 Clinically Tested DrugsStefan S. De Buck, Vikash K. Sinha, Luca A. Fenu, Marjoleen J. Nijsen, Claire E. Mackie and Ron A. H. J. GilissenDrug Metabolism and Disposition October 2007, 35 (10) 1766-1780; DOI: https://doi.org/10.1124/dmd.107.015644
O
Ohtsu, Atsushi
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Oitate, Masataka
- You have accessCovalent Binding of Rofecoxib, but Not Other Cyclooxygenase-2 Inhibitors, to Allysine Aldehyde in Elastin of Human AortaMasataka Oitate, Takashi Hirota, Takahiro Murai, Shin-ichi Miura and Toshihiko IkedaDrug Metabolism and Disposition October 2007, 35 (10) 1846-1852; DOI: https://doi.org/10.1124/dmd.107.016121
Ozawa, Shogo
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
P
Perkins, Everett J.
- You have accessPharmacokinetics, Metabolism, and Excretion of the Intestinal Peptide Transporter 1 (SLC15A1)-Targeted Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2-Amino)propionyl]aminobicyclo[3.1.0.]hexen-2,6-dicarboxylic acid (LY544344) in Rats and Dogs: Assessment of First-Pass Bioactivation and Dose LinearityEverett J. Perkins and Trent AbrahamDrug Metabolism and Disposition October 2007, 35 (10) 1903-1909; DOI: https://doi.org/10.1124/dmd.107.016154
Perrett, H. F.
- You have accessDisparity in Holoprotein/Apoprotein Ratios of Different Standards Used for Immunoquantification of Hepatic Cytochrome P450 EnzymesH. F. Perrett, Z. E. Barter, B. C. Jones, H. Yamazaki, G. T. Tucker and A. Rostami-HodjeganDrug Metabolism and Disposition October 2007, 35 (10) 1733-1736; DOI: https://doi.org/10.1124/dmd.107.015743
Peters, Stefan Oliver
- You have accessInfluence of Short-Term Use of Dexamethasone on the Pharmacokinetics of Ifosfamide in PatientsSvenja Kristin Brüggemann, Sonja Pfäffle, Stefan Oliver Peters and Thomas WagnerDrug Metabolism and Disposition October 2007, 35 (10) 1721-1724; DOI: https://doi.org/10.1124/dmd.106.014043
Petrick, Jay S.
- You have accessImportance of Hepatic Induction of Constitutive Androstane Receptor and Other Transcription Factors That Regulate Xenobiotic Metabolism and TransportJay S. Petrick and Curtis D. KlaassenDrug Metabolism and Disposition October 2007, 35 (10) 1806-1815; DOI: https://doi.org/10.1124/dmd.107.015974
Pfäffle, Sonja
- You have accessInfluence of Short-Term Use of Dexamethasone on the Pharmacokinetics of Ifosfamide in PatientsSvenja Kristin Brüggemann, Sonja Pfäffle, Stefan Oliver Peters and Thomas WagnerDrug Metabolism and Disposition October 2007, 35 (10) 1721-1724; DOI: https://doi.org/10.1124/dmd.106.014043
Plock, N.
- You have accessDoes Linezolid Inhibit Its Own Metabolism?—Population Pharmacokinetics As a Tool to Explain the Observed Nonlinearity in Both Healthy Volunteers and Septic PatientsN. Plock, C. Buerger, C. Joukhadar, S. Kljucar and C. KloftDrug Metabolism and Disposition October 2007, 35 (10) 1816-1823; DOI: https://doi.org/10.1124/dmd.106.013755
Pruimboom-Brees, Ingrid M.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
Q
Qian, Mingxin
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
R
Ring, Steven C.
- You have accessMetabolic Profile of [14C]Bendamustine in Rat Urine and Bile: Preliminary Structural Identification of MetabolitesJames P. Chovan, Feng Li, Erya Yu and Steven C. RingDrug Metabolism and Disposition October 2007, 35 (10) 1744-1753; DOI: https://doi.org/10.1124/dmd.107.015958
Rostami-Hodjegan, A.
- You have accessDisparity in Holoprotein/Apoprotein Ratios of Different Standards Used for Immunoquantification of Hepatic Cytochrome P450 EnzymesH. F. Perrett, Z. E. Barter, B. C. Jones, H. Yamazaki, G. T. Tucker and A. Rostami-HodjeganDrug Metabolism and Disposition October 2007, 35 (10) 1733-1736; DOI: https://doi.org/10.1124/dmd.107.015743
S
Sai, Kimie
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Saijo, Nagahiro
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Saito, Hirohisa
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Saito, Yoshiro
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Sakaki, Toshiyuki
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Sakuma, Tsutomu
- You have accessInvolvement of Glucocorticoid Receptor and Pregnane X Receptor in the Regulation of Mouse CYP3A44 Female-Predominant Expression by Glucocorticoid HormoneWattanaporn Bhadhprasit, Tsutomu Sakuma, Nobuyuki Hatakeyama, Masahiro Fuwa, Kaori Kitajima and Nobuo NemotoDrug Metabolism and Disposition October 2007, 35 (10) 1880-1885; DOI: https://doi.org/10.1124/dmd.107.016832
Sasahara, Masakiyo
- You have accessIn Vitro Metabolism of Isoline, a Pyrrolizidine Alkaloid from Ligularia duciformis, by Rodent Liver Microsomal Esterase and Enhanced Hepatotoxicity by Esterase InhibitorsJun Tang, Teruaki Akao, Norio Nakamura, Zheng-Tao Wang, Kiyoshi Takagawa, Masakiyo Sasahara and Masao HattoriDrug Metabolism and Disposition October 2007, 35 (10) 1832-1839; DOI: https://doi.org/10.1124/dmd.107.016311
Sasaki, Takamitsu
- You have accessCharacterization of Human Cytochrome P450 Enzymes Involved in the Metabolism of CilostazolMasahiro Hiratsuka, Yudai Hinai, Takamitsu Sasaki, Yumiko Konno, Kenichi Imagawa, Masaaki Ishikawa and Michinao MizugakiDrug Metabolism and Disposition October 2007, 35 (10) 1730-1732; DOI: https://doi.org/10.1124/dmd.107.016758
Sawada, Jun-ichi
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Scheffer, George L.
- You have accessInduction of Hepatobiliary Efflux Transporters in Acetaminophen-Induced Acute Liver Failure CasesSarah N. Barnes, Lauren M. Aleksunes, Lisa Augustine, George L. Scheffer, Michael J. Goedken, Amy B. Jakowski, Ingrid M. Pruimboom-Brees, Nathan J. Cherrington and José E. ManautouDrug Metabolism and Disposition October 2007, 35 (10) 1963-1969; DOI: https://doi.org/10.1124/dmd.107.016170
Schinkel, Alfred H.
- You have accessInvolvement of Breast Cancer Resistance Protein (ABCG2) in the Biliary Excretion Mechanism of FluoroquinolonesTomohiro Ando, Hiroyuki Kusuhara, Gracia Merino, Ana I. Alvarez, Alfred H. Schinkel and Yuichi SugiyamaDrug Metabolism and Disposition October 2007, 35 (10) 1873-1879; DOI: https://doi.org/10.1124/dmd.107.014969
Seidel, Albrecht
- You have accessDirecting Role of Organic Anion Transporters in the Excretion of Mercapturic Acids of Alkylated Polycyclic Aromatic HydrocarbonsNadiya Bakhiya, Monika Batke, Janet Laake, Bernhard H. Monien, Heinz Frank, Albrecht Seidel, Wolfram Engst and Hansruedi GlattDrug Metabolism and Disposition October 2007, 35 (10) 1824-1831; DOI: https://doi.org/10.1124/dmd.107.016964
Seo, Ji Y.
- You have accessInduction of Hepatic CYP2E1 by a Subtoxic Dose of Acetaminophen in Rats: Increase in Dichloromethane Metabolism and Carboxyhemoglobin ElevationSu N. Kim, Ji Y. Seo, Da W. Jung, Min Y. Lee, Young S. Jung and Young C. KimDrug Metabolism and Disposition October 2007, 35 (10) 1754-1758; DOI: https://doi.org/10.1124/dmd.107.015545
Sharma, Arun K.
- You have accessElimination of Antiestrogenic Effects of Active Tamoxifen Metabolites by GlucuronidationYan Zheng, Dongxiao Sun, Arun K. Sharma, Gang Chen, Shantu Amin and Philip LazarusDrug Metabolism and Disposition October 2007, 35 (10) 1942-1948; DOI: https://doi.org/10.1124/dmd.107.016279
Shirao, Kuniaki
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Silberstein, David S.
- You have accessDifferences in Endogenous Esterification and Retention in the Rat Trachea between Budesonide and Ciclesonide Active MetaboliteKristina Lexmüller, Helena Gullstrand, Bengt-Olof Axelsson, Petter Sjölin, Solange H. Korn, David S. Silberstein and Anna Miller-LarssonDrug Metabolism and Disposition October 2007, 35 (10) 1788-1796; DOI: https://doi.org/10.1124/dmd.107.015297
Sinha, Vikash K.
- You have accessPrediction of Human Pharmacokinetics Using Physiologically Based Modeling: A Retrospective Analysis of 26 Clinically Tested DrugsStefan S. De Buck, Vikash K. Sinha, Luca A. Fenu, Marjoleen J. Nijsen, Claire E. Mackie and Ron A. H. J. GilissenDrug Metabolism and Disposition October 2007, 35 (10) 1766-1780; DOI: https://doi.org/10.1124/dmd.107.015644
Sipes, I. G.
- You have accessPrediction of Metabolic Clearance of Bisphenol A (4,4 ′-Dihydroxy-2,2-diphenylpropane) using Cryopreserved Human HepatocytesR. K. Kuester and I. G. SipesDrug Metabolism and Disposition October 2007, 35 (10) 1910-1915; DOI: https://doi.org/10.1124/dmd.107.014787
Sjölin, Petter
- You have accessDifferences in Endogenous Esterification and Retention in the Rat Trachea between Budesonide and Ciclesonide Active MetaboliteKristina Lexmüller, Helena Gullstrand, Bengt-Olof Axelsson, Petter Sjölin, Solange H. Korn, David S. Silberstein and Anna Miller-LarssonDrug Metabolism and Disposition October 2007, 35 (10) 1788-1796; DOI: https://doi.org/10.1124/dmd.107.015297
Slitt, Angela L.
- You have accessEfflux Transporter Expression and Acetaminophen Metabolite Excretion Are Altered in Rodent Models of Nonalcoholic Fatty Liver DiseaseAndrew J. Lickteig, Craig D. Fisher, Lisa M. Augustine, Lauren M. Aleksunes, David G. Besselsen, Angela L. Slitt, Jose E. Manautou and Nathan J. CherringtonDrug Metabolism and Disposition October 2007, 35 (10) 1970-1978; DOI: https://doi.org/10.1124/dmd.107.015107
Smolarek, Teresa
- You have accessP-glycoprotein Has Differential Effects on the Disposition of Statin Acid and Lactone Forms in mdr1a/b Knockout and Wild-Type MiceCuiping Chen, Jian Lin, Teresa Smolarek and Larry TremaineDrug Metabolism and Disposition October 2007, 35 (10) 1725-1729; DOI: https://doi.org/10.1124/dmd.107.015677
Somers, G. I.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Sprague, Jon E.
- You have accessAmbient Temperature Effects on 3,4-Methylenedioxymethamphetamine-Induced Thermodysregulation and Pharmacokinetics in Male MonkeysMatthew L. Banks, Jon E. Sprague, David F. Kisor, Paul W. Czoty, David E. Nichols and Michael A. NaderDrug Metabolism and Disposition October 2007, 35 (10) 1840-1845; DOI: https://doi.org/10.1124/dmd.107.016261
Stiborová, Marie
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Sugiyama, Yuichi
- You have accessInvolvement of Breast Cancer Resistance Protein (ABCG2) in the Biliary Excretion Mechanism of FluoroquinolonesTomohiro Ando, Hiroyuki Kusuhara, Gracia Merino, Ana I. Alvarez, Alfred H. Schinkel and Yuichi SugiyamaDrug Metabolism and Disposition October 2007, 35 (10) 1873-1879; DOI: https://doi.org/10.1124/dmd.107.014969
Sun, Dongxiao
- You have accessElimination of Antiestrogenic Effects of Active Tamoxifen Metabolites by GlucuronidationYan Zheng, Dongxiao Sun, Arun K. Sharma, Gang Chen, Shantu Amin and Philip LazarusDrug Metabolism and Disposition October 2007, 35 (10) 1942-1948; DOI: https://doi.org/10.1124/dmd.107.016279
Svobodová, Lucie
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
T
Takagawa, Kiyoshi
- You have accessIn Vitro Metabolism of Isoline, a Pyrrolizidine Alkaloid from Ligularia duciformis, by Rodent Liver Microsomal Esterase and Enhanced Hepatotoxicity by Esterase InhibitorsJun Tang, Teruaki Akao, Norio Nakamura, Zheng-Tao Wang, Kiyoshi Takagawa, Masakiyo Sasahara and Masao HattoriDrug Metabolism and Disposition October 2007, 35 (10) 1832-1839; DOI: https://doi.org/10.1124/dmd.107.016311
Takiguchi, Rie
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Tanaka, Yorihisa
- You have accessLack of Formation of Aldehyde Oxidase Dimer Possibly Due to 377G>A Nucleotide SubstitutionKunio Itoh, Hiroaki Maruyama, Mayuko Adachi, Kouichi Hoshino, Nobuaki Watanabe and Yorihisa TanakaDrug Metabolism and Disposition October 2007, 35 (10) 1860-1864; DOI: https://doi.org/10.1124/dmd.107.015503
Tanaka-Kagawa, Toshiko
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Tang, Huadong
- You have accessInterspecies Prediction of Human Drug Clearance Based on Scaling Data from One or Two Animal SpeciesHuadong Tang, Azher Hussain, Mauricio Leal, Michael Mayersohn and Eric FluhlerDrug Metabolism and Disposition October 2007, 35 (10) 1886-1893; DOI: https://doi.org/10.1124/dmd.107.016188
Tang, Jun
- You have accessIn Vitro Metabolism of Isoline, a Pyrrolizidine Alkaloid from Ligularia duciformis, by Rodent Liver Microsomal Esterase and Enhanced Hepatotoxicity by Esterase InhibitorsJun Tang, Teruaki Akao, Norio Nakamura, Zheng-Tao Wang, Kiyoshi Takagawa, Masakiyo Sasahara and Masao HattoriDrug Metabolism and Disposition October 2007, 35 (10) 1832-1839; DOI: https://doi.org/10.1124/dmd.107.016311
Thummel, Kenneth E.
- You have accessCytochrome P450 Enzymes and Transporters Induced by Anti-Human Immunodeficiency Virus Protease Inhibitors in Human Hepatocytes: Implications for Predicting Clinical Drug InteractionsVaishali Dixit, Niresh Hariparsad, Fang Li, Pankaj Desai, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition October 2007, 35 (10) 1853-1859; DOI: https://doi.org/10.1124/dmd.107.016089
Tremaine, Larry
- You have accessP-glycoprotein Has Differential Effects on the Disposition of Statin Acid and Lactone Forms in mdr1a/b Knockout and Wild-Type MiceCuiping Chen, Jian Lin, Teresa Smolarek and Larry TremaineDrug Metabolism and Disposition October 2007, 35 (10) 1725-1729; DOI: https://doi.org/10.1124/dmd.107.015677
Trzaskos, James
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
Tucker, G. T.
- You have accessDisparity in Holoprotein/Apoprotein Ratios of Different Standards Used for Immunoquantification of Hepatic Cytochrome P450 EnzymesH. F. Perrett, Z. E. Barter, B. C. Jones, H. Yamazaki, G. T. Tucker and A. Rostami-HodjeganDrug Metabolism and Disposition October 2007, 35 (10) 1733-1736; DOI: https://doi.org/10.1124/dmd.107.015743
U
Uchida, Shinya
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Unadkat, Jashvant D.
- You have accessCytochrome P450 Enzymes and Transporters Induced by Anti-Human Immunodeficiency Virus Protease Inhibitors in Human Hepatocytes: Implications for Predicting Clinical Drug InteractionsVaishali Dixit, Niresh Hariparsad, Fang Li, Pankaj Desai, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition October 2007, 35 (10) 1853-1859; DOI: https://doi.org/10.1124/dmd.107.016089
V
Václavíková, Radka
- You have accessThe Anticancer Drug Ellipticine Is a Potent Inducer of Rat Cytochromes P450 1A1 and 1A2, Thereby Modulating Its Own MetabolismDagmar Aimová, Lucie Svobodová, Věra Kotrbová, Barbora Mrázová, Petr Hodek, Jiří Hudeček, Radka Václavíková, Eva Frei and Marie StiborováDrug Metabolism and Disposition October 2007, 35 (10) 1926-1934; DOI: https://doi.org/10.1124/dmd.107.016048
Vaddi, Kris
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
W
Wagner, Thomas
- You have accessInfluence of Short-Term Use of Dexamethasone on the Pharmacokinetics of Ifosfamide in PatientsSvenja Kristin Brüggemann, Sonja Pfäffle, Stefan Oliver Peters and Thomas WagnerDrug Metabolism and Disposition October 2007, 35 (10) 1721-1724; DOI: https://doi.org/10.1124/dmd.106.014043
Wang, Joanne
- You have accessMetformin Transport by a Newly Cloned Proton-Stimulated Organic Cation Transporter (Plasma Membrane Monoamine Transporter) Expressed in Human IntestineMingyan Zhou, Li Xia and Joanne WangDrug Metabolism and Disposition October 2007, 35 (10) 1956-1962; DOI: https://doi.org/10.1124/dmd.107.015495
Wang, Zheng-Tao
- You have accessIn Vitro Metabolism of Isoline, a Pyrrolizidine Alkaloid from Ligularia duciformis, by Rodent Liver Microsomal Esterase and Enhanced Hepatotoxicity by Esterase InhibitorsJun Tang, Teruaki Akao, Norio Nakamura, Zheng-Tao Wang, Kiyoshi Takagawa, Masakiyo Sasahara and Masao HattoriDrug Metabolism and Disposition October 2007, 35 (10) 1832-1839; DOI: https://doi.org/10.1124/dmd.107.016311
Watanabe, Nobuaki
- You have accessLack of Formation of Aldehyde Oxidase Dimer Possibly Due to 377G>A Nucleotide SubstitutionKunio Itoh, Hiroaki Maruyama, Mayuko Adachi, Kouichi Hoshino, Nobuaki Watanabe and Yorihisa TanakaDrug Metabolism and Disposition October 2007, 35 (10) 1860-1864; DOI: https://doi.org/10.1124/dmd.107.015503
Woodrooffe, A. J. M.
- You have accessA Comparison of the Expression and Metabolizing Activities of Phase I and II Enzymes in Freshly Isolated Human Lung Parenchymal Cells and Cryopreserved Human HepatocytesG. I. Somers, N. Lindsay, B. M. Lowdon, A. E. Jones, C. Freathy, S. Ho, A. J. M. Woodrooffe, M. K. Bayliss and G. R. MancheeDrug Metabolism and Disposition October 2007, 35 (10) 1797-1805; DOI: https://doi.org/10.1124/dmd.107.015966
Wright, Jason
- You have accessIn Vitro Prediction and in Vivo Verification of Enantioselective Human Tofisopam Metabolite ProfilesMichael D. Cameron, Jason Wright, Christopher B. Black and Naidong YeDrug Metabolism and Disposition October 2007, 35 (10) 1894-1902; DOI: https://doi.org/10.1124/dmd.107.015875
Wu, Jing-Tao
- You have accessPharmacokinetics and Pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-Amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a Potent and Selective Inhibitor of Tumor Necrosis Factor α-Converting Enzyme in Rodents, Dogs, Chimpanzees, and HumansMingxin Qian, Stephen A. Bai, Bernice Brogdon, Jing-Tao Wu, Rui-Qin Liu, Maryanne B. Covington, Kris Vaddi, Robert C. Newton, Michael J. Fossler, C. Edwin Garner, Yuzhong Deng, Thomas Maduskuie, James Trzaskos, James J.-W. Duan, Carl P. Decicco and David D. ChristDrug Metabolism and Disposition October 2007, 35 (10) 1916-1925; DOI: https://doi.org/10.1124/dmd.107.015933
X
Xia, Li
- You have accessMetformin Transport by a Newly Cloned Proton-Stimulated Organic Cation Transporter (Plasma Membrane Monoamine Transporter) Expressed in Human IntestineMingyan Zhou, Li Xia and Joanne WangDrug Metabolism and Disposition October 2007, 35 (10) 1956-1962; DOI: https://doi.org/10.1124/dmd.107.015495
Y
Yamada, Shizuo
- You have accessA Novel Mechanism for Polychlorinated Biphenyl-Induced Decrease in Serum Thyroxine Level in RatsYoshihisa Kato, Shin-ichi Ikushiro, Rie Takiguchi, Koichi Haraguchi, Nobuyuki Koga, Shinya Uchida, Toshiyuki Sakaki, Shizuo Yamada, Jun Kanno and Masakuni DegawaDrug Metabolism and Disposition October 2007, 35 (10) 1949-1955; DOI: https://doi.org/10.1124/dmd.107.017327
Yamamoto, Noboru
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Yamanaka, Hiroyuki
- You have accessInteractions between Human UGT1A1, UGT1A4, and UGT1A6 Affect Their Enzymatic ActivitiesRyoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka, Miki Katoh and Tsuyoshi YokoiDrug Metabolism and Disposition October 2007, 35 (10) 1781-1787; DOI: https://doi.org/10.1124/dmd.107.016402
Yamazaki, H.
- You have accessDisparity in Holoprotein/Apoprotein Ratios of Different Standards Used for Immunoquantification of Hepatic Cytochrome P450 EnzymesH. F. Perrett, Z. E. Barter, B. C. Jones, H. Yamazaki, G. T. Tucker and A. Rostami-HodjeganDrug Metabolism and Disposition October 2007, 35 (10) 1733-1736; DOI: https://doi.org/10.1124/dmd.107.015743
Ye, Naidong
- You have accessIn Vitro Prediction and in Vivo Verification of Enantioselective Human Tofisopam Metabolite ProfilesMichael D. Cameron, Jason Wright, Christopher B. Black and Naidong YeDrug Metabolism and Disposition October 2007, 35 (10) 1894-1902; DOI: https://doi.org/10.1124/dmd.107.015875
Yokoi, Tsuyoshi
- You have accessHuman CYP2A6 Is Induced by Estrogen via Estrogen ReceptorEriko Higashi, Tatsuki Fukami, Masahiro Itoh, Satoru Kyo, Masaki Inoue, Tsuyoshi Yokoi and Miki NakajimaDrug Metabolism and Disposition October 2007, 35 (10) 1935-1941; DOI: https://doi.org/10.1124/dmd.107.016568
- You have accessInteractions between Human UGT1A1, UGT1A4, and UGT1A6 Affect Their Enzymatic ActivitiesRyoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka, Miki Katoh and Tsuyoshi YokoiDrug Metabolism and Disposition October 2007, 35 (10) 1781-1787; DOI: https://doi.org/10.1124/dmd.107.016402
Yoo, Hye Hyun
- You have accessMechanism-Based Inactivation of Cytochrome P450 2A6 by Decursinol Angelate Isolated from Angelica GigasHye Hyun Yoo, Min Woo Lee, Young Choong Kim, Chul-Ho Yun and Dong-Hyun KimDrug Metabolism and Disposition October 2007, 35 (10) 1759-1765; DOI: https://doi.org/10.1124/dmd.107.016584
Yoshida, Teruhiko
- You have accessHaplotypes and a Novel Defective Allele of CES2 Found in a Japanese PopulationSu-Ryang Kim, Kimie Sai, Toshiko Tanaka-Kagawa, Hideto Jinno, Shogo Ozawa, Nahoko Kaniwa, Yoshiro Saito, Akira Akasawa, Kenji Matsumoto, Hirohisa Saito, Naoyuki Kamatani, Kuniaki Shirao, Noboru Yamamoto, Teruhiko Yoshida, Hironobu Minami, Atsushi Ohtsu, Nagahiro Saijo and Jun-ichi SawadaDrug Metabolism and Disposition October 2007, 35 (10) 1865-1872; DOI: https://doi.org/10.1124/dmd.107.015339
Yu, Erya
- You have accessMetabolic Profile of [14C]Bendamustine in Rat Urine and Bile: Preliminary Structural Identification of MetabolitesJames P. Chovan, Feng Li, Erya Yu and Steven C. RingDrug Metabolism and Disposition October 2007, 35 (10) 1744-1753; DOI: https://doi.org/10.1124/dmd.107.015958
Yun, Chul-Ho
- You have accessMechanism-Based Inactivation of Cytochrome P450 2A6 by Decursinol Angelate Isolated from Angelica GigasHye Hyun Yoo, Min Woo Lee, Young Choong Kim, Chul-Ho Yun and Dong-Hyun KimDrug Metabolism and Disposition October 2007, 35 (10) 1759-1765; DOI: https://doi.org/10.1124/dmd.107.016584
Z
Zheng, Yan
- You have accessElimination of Antiestrogenic Effects of Active Tamoxifen Metabolites by GlucuronidationYan Zheng, Dongxiao Sun, Arun K. Sharma, Gang Chen, Shantu Amin and Philip LazarusDrug Metabolism and Disposition October 2007, 35 (10) 1942-1948; DOI: https://doi.org/10.1124/dmd.107.016279
Zhou, Mingyan
- You have accessMetformin Transport by a Newly Cloned Proton-Stimulated Organic Cation Transporter (Plasma Membrane Monoamine Transporter) Expressed in Human IntestineMingyan Zhou, Li Xia and Joanne WangDrug Metabolism and Disposition October 2007, 35 (10) 1956-1962; DOI: https://doi.org/10.1124/dmd.107.015495
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