Index by author
January 01, 2008; Volume 36,Issue 1
A
Adjei, Araba A.
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
Andersson, Tommy B.
- You have accessHepaRG Cells as an in Vitro Model for Evaluation of Cytochrome P450 Induction in HumansKajsa P. Kanebratt and Tommy B. AnderssonDrug Metabolism and Disposition January 2008, 36 (1) 137-145; DOI: https://doi.org/10.1124/dmd.107.017418
B
Backman, Janne T.
- You have accessTrimethoprim and the CYP2C8*3 Allele Have Opposite Effects on the Pharmacokinetics of PioglitazoneAleksi Tornio, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2008, 36 (1) 73-80; DOI: https://doi.org/10.1124/dmd.107.018010
Bennett, J.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Blough, David K.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Bonnardeaux, Alain
- You have accessEffects of Chronic Renal Failure on Liver Drug TransportersJudith Naud, Josée Michaud, Francois A. Leblond, Stéphane Lefrancois, Alain Bonnardeaux and Vincent PichetteDrug Metabolism and Disposition January 2008, 36 (1) 124-128; DOI: https://doi.org/10.1124/dmd.107.018192
Bow, Daniel A. J.
- You have accessLocalization of P-gp (Abcb1) and Mrp2 (Abcc2) in Freshly Isolated Rat HepatocytesDaniel A. J. Bow, Jennifer L. Perry, David S. Miller, John B. Pritchard and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 198-202; DOI: https://doi.org/10.1124/dmd.107.018200
Bridges, Arlene S.
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
Brouwer, Kim L. R.
- You have accessLocalization of P-gp (Abcb1) and Mrp2 (Abcc2) in Freshly Isolated Rat HepatocytesDaniel A. J. Bow, Jennifer L. Perry, David S. Miller, John B. Pritchard and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 198-202; DOI: https://doi.org/10.1124/dmd.107.018200
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
C
Carlson, G. L.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Catz, Paul
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
Chang, Shu Y.
- You have accessDisposition and Metabolism of [14C]Brasofensine in Rats, Monkeys, and HumansMingshe Zhu, Daisy B. Whigan, Shu Y. Chang and Randy C. DockensDrug Metabolism and Disposition January 2008, 36 (1) 24-35; DOI: https://doi.org/10.1124/dmd.107.016139
Chen, Gang
- You have accessRegulation of CYP2A6 Protein Expression by Skatole, Indole, and Testicular Steroids in Primary Cultured Pig HepatocytesGang Chen, Rebecca-Ayme Cue, Kerstin Lundstrom, Jeffrey D. Wood and Olena DoranDrug Metabolism and Disposition January 2008, 36 (1) 56-60; DOI: https://doi.org/10.1124/dmd.107.017285
Chinn, Leslie W.
- You have accessThe Effects of ABCB1 3′-Untranslated Region Variants on mRNA StabilityJason M. Gow, Leslie W. Chinn and Deanna L. KroetzDrug Metabolism and Disposition January 2008, 36 (1) 10-15; DOI: https://doi.org/10.1124/dmd.107.017087
Chuang, Victor Tuan Giam
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Clifford, Michael N.
- You have accessTransport and Metabolism of Ferulic Acid through the Colonic EpitheliumLaure Poquet, Michael N. Clifford and Gary WilliamsonDrug Metabolism and Disposition January 2008, 36 (1) 190-197; DOI: https://doi.org/10.1124/dmd.107.017558
Collett, A.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Coquette, Alain
- You have accessPharmacokinetics and Metabolism of 14C-Brivaracetam, a Novel SV2A Ligand, in Healthy SubjectsMaria Laura Sargentini-Maier, Pascal Espié, Alain Coquette and Armel StockisDrug Metabolism and Disposition January 2008, 36 (1) 36-45; DOI: https://doi.org/10.1124/dmd.107.017129
Cue, Rebecca-Ayme
- You have accessRegulation of CYP2A6 Protein Expression by Skatole, Indole, and Testicular Steroids in Primary Cultured Pig HepatocytesGang Chen, Rebecca-Ayme Cue, Kerstin Lundstrom, Jeffrey D. Wood and Olena DoranDrug Metabolism and Disposition January 2008, 36 (1) 56-60; DOI: https://doi.org/10.1124/dmd.107.017285
D
Dallman, L.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Davis, J.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Dees, E. Claire
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Degawa, Masakuni
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
Dockens, Randy C.
- You have accessDisposition and Metabolism of [14C]Brasofensine in Rats, Monkeys, and HumansMingshe Zhu, Daisy B. Whigan, Shu Y. Chang and Randy C. DockensDrug Metabolism and Disposition January 2008, 36 (1) 24-35; DOI: https://doi.org/10.1124/dmd.107.016139
Doran, Olena
- You have accessRegulation of CYP2A6 Protein Expression by Skatole, Indole, and Testicular Steroids in Primary Cultured Pig HepatocytesGang Chen, Rebecca-Ayme Cue, Kerstin Lundstrom, Jeffrey D. Wood and Olena DoranDrug Metabolism and Disposition January 2008, 36 (1) 56-60; DOI: https://doi.org/10.1124/dmd.107.017285
Dumas, Todd E.
- You have accessPharmacokinetics and Metabolic Profile of Free, Conjugated, and Total Silymarin Flavonolignans in Human Plasma after Oral Administration of Milk Thistle ExtractZhiming Wen, Todd E. Dumas, Sarah J. Schrieber, Roy L. Hawke, Michael W. Fried and Philip C. SmithDrug Metabolism and Disposition January 2008, 36 (1) 65-72; DOI: https://doi.org/10.1124/dmd.107.017566
E
Emi, Yoshikazu
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
Espié, Pascal
- You have accessPharmacokinetics and Metabolism of 14C-Brivaracetam, a Novel SV2A Ligand, in Healthy SubjectsMaria Laura Sargentini-Maier, Pascal Espié, Alain Coquette and Armel StockisDrug Metabolism and Disposition January 2008, 36 (1) 36-45; DOI: https://doi.org/10.1124/dmd.107.017129
Evans, Allan M.
- You have accessGlucuronidation of Mycophenolic Acid by Wistar and Mrp2-Deficient TR- Rat Liver MicrosomesIan S. Westley, Raymond G. Morris, Allan M. Evans and Benedetta C. SallustioDrug Metabolism and Disposition January 2008, 36 (1) 46-50; DOI: https://doi.org/10.1124/dmd.107.017210
F
Fried, Michael W.
- You have accessPharmacokinetics and Metabolic Profile of Free, Conjugated, and Total Silymarin Flavonolignans in Human Plasma after Oral Administration of Milk Thistle ExtractZhiming Wen, Todd E. Dumas, Sarah J. Schrieber, Roy L. Hawke, Michael W. Fried and Philip C. SmithDrug Metabolism and Disposition January 2008, 36 (1) 65-72; DOI: https://doi.org/10.1124/dmd.107.017566
Fujita, Takuya
- You have accessOseltamivir (Tamiflu) Efflux Transport at the Blood-Brain Barrier via P-GlycoproteinKaori Morimoto, Masanori Nakakariya, Yoshiyuki Shirasaka, Chihaya Kakinuma, Takuya Fujita, Ikumi Tamai and Takuo OgiharaDrug Metabolism and Disposition January 2008, 36 (1) 6-9; DOI: https://doi.org/10.1124/dmd.107.017699
Fukuda, Hikaru
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Furimsky, Anna M.
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
G
Ghose, Romi
- You have accessRegulation of Hepatic Drug-Metabolizing Enzyme Genes by Toll-Like Receptor 4 Signaling Is Independent of Toll-Interleukin 1 Receptor Domain-Containing Adaptor ProteinRomi Ghose, Damara White, Tao Guo, Jesus Vallejo and Saul J. KarpenDrug Metabolism and Disposition January 2008, 36 (1) 95-101; DOI: https://doi.org/10.1124/dmd.107.018051
Givens, Raymond C.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Gow, Jason M.
- You have accessThe Effects of ABCB1 3′-Untranslated Region Variants on mRNA StabilityJason M. Gow, Leslie W. Chinn and Deanna L. KroetzDrug Metabolism and Disposition January 2008, 36 (1) 10-15; DOI: https://doi.org/10.1124/dmd.107.017087
Green, Carol E.
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
Guo, Tao
- You have accessRegulation of Hepatic Drug-Metabolizing Enzyme Genes by Toll-Like Receptor 4 Signaling Is Independent of Toll-Interleukin 1 Receptor Domain-Containing Adaptor ProteinRomi Ghose, Damara White, Tao Guo, Jesus Vallejo and Saul J. KarpenDrug Metabolism and Disposition January 2008, 36 (1) 95-101; DOI: https://doi.org/10.1124/dmd.107.018051
H
Harwood, M. D.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Hawke, Roy L.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
- You have accessPharmacokinetics and Metabolic Profile of Free, Conjugated, and Total Silymarin Flavonolignans in Human Plasma after Oral Administration of Milk Thistle ExtractZhiming Wen, Todd E. Dumas, Sarah J. Schrieber, Roy L. Hawke, Michael W. Fried and Philip C. SmithDrug Metabolism and Disposition January 2008, 36 (1) 65-72; DOI: https://doi.org/10.1124/dmd.107.017566
Humphrey, M.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
I
Ikushiro, Shin-ichi
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
Isoherranen, Nina
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Iwanaga, Kazunori
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Iyer, Lalitha V.
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
J
Jeannesson, Elise
- You have accessTranscription Factor and Drug-Metabolizing Enzyme Gene Expression in Lymphocytes from Healthy Human SubjectsGérard Siest, Elise Jeannesson, Jean-Brice Marteau, Anastasia Samara, Bérangère Marie, Michèle Pfister and Sophie Visvikis-SiestDrug Metabolism and Disposition January 2008, 36 (1) 182-189; DOI: https://doi.org/10.1124/dmd.107.017228
K
Kakinuma, Chihaya
- You have accessOseltamivir (Tamiflu) Efflux Transport at the Blood-Brain Barrier via P-GlycoproteinKaori Morimoto, Masanori Nakakariya, Yoshiyuki Shirasaka, Chihaya Kakinuma, Takuya Fujita, Ikumi Tamai and Takuo OgiharaDrug Metabolism and Disposition January 2008, 36 (1) 6-9; DOI: https://doi.org/10.1124/dmd.107.017699
Kanebratt, Kajsa P.
- You have accessHepaRG Cells as an in Vitro Model for Evaluation of Cytochrome P450 Induction in HumansKajsa P. Kanebratt and Tommy B. AnderssonDrug Metabolism and Disposition January 2008, 36 (1) 137-145; DOI: https://doi.org/10.1124/dmd.107.017418
Kaneko, Ken-ichi
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Kapetanovic, Izet M.
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
Karpen, Saul J.
- You have accessRegulation of Hepatic Drug-Metabolizing Enzyme Genes by Toll-Like Receptor 4 Signaling Is Independent of Toll-Interleukin 1 Receptor Domain-Containing Adaptor ProteinRomi Ghose, Damara White, Tao Guo, Jesus Vallejo and Saul J. KarpenDrug Metabolism and Disposition January 2008, 36 (1) 95-101; DOI: https://doi.org/10.1124/dmd.107.018051
Kartha, Jaya S.
- You have accessMechanism-Based Inactivation of Lung-Selective Cytochrome P450 CYP2F EnzymesJaya S. Kartha and Garold S. YostDrug Metabolism and Disposition January 2008, 36 (1) 155-162; DOI: https://doi.org/10.1124/dmd.107.017897
Kato, Yoshihisa
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
Kawahara, Kohichi
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Klaassen, Curtis
- You have accessGender Differences in mRNA Expression of ATP-Binding Cassette Efflux and Bile Acid Transporters in Kidney, Liver, and Intestine of 5/6 Nephrectomized RatsHong Lu and Curtis KlaassenDrug Metabolism and Disposition January 2008, 36 (1) 16-23; DOI: https://doi.org/10.1124/dmd.107.014845
Kroetz, Deanna L.
- You have accessThe Effects of ABCB1 3′-Untranslated Region Variants on mRNA StabilityJason M. Gow, Leslie W. Chinn and Deanna L. KroetzDrug Metabolism and Disposition January 2008, 36 (1) 10-15; DOI: https://doi.org/10.1124/dmd.107.017087
L
Lamba, Jatinder
- You have accessNovel Single Nucleotide Polymorphisms in the Promoter and Intron 1 of Human Pregnane X Receptor/NR1I2 and Their Association with CYP3A4 ExpressionJatinder Lamba, Vishal Lamba, Stephen Strom, Raman Venkataramanan and Erin SchuetzDrug Metabolism and Disposition January 2008, 36 (1) 169-181; DOI: https://doi.org/10.1124/dmd.107.016600
Lamba, Jatinder K.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Lamba, Vishal
- You have accessNovel Single Nucleotide Polymorphisms in the Promoter and Intron 1 of Human Pregnane X Receptor/NR1I2 and Their Association with CYP3A4 ExpressionJatinder Lamba, Vishal Lamba, Stephen Strom, Raman Venkataramanan and Erin SchuetzDrug Metabolism and Disposition January 2008, 36 (1) 169-181; DOI: https://doi.org/10.1124/dmd.107.016600
Leblond, Francois A.
- You have accessEffects of Chronic Renal Failure on Liver Drug TransportersJudith Naud, Josée Michaud, Francois A. Leblond, Stéphane Lefrancois, Alain Bonnardeaux and Vincent PichetteDrug Metabolism and Disposition January 2008, 36 (1) 124-128; DOI: https://doi.org/10.1124/dmd.107.018192
Lefrancois, Stéphane
- You have accessEffects of Chronic Renal Failure on Liver Drug TransportersJudith Naud, Josée Michaud, Francois A. Leblond, Stéphane Lefrancois, Alain Bonnardeaux and Vincent PichetteDrug Metabolism and Disposition January 2008, 36 (1) 124-128; DOI: https://doi.org/10.1124/dmd.107.018192
Li, Jun
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
Lu, Hong
- You have accessGender Differences in mRNA Expression of ATP-Binding Cassette Efflux and Bile Acid Transporters in Kidney, Liver, and Intestine of 5/6 Nephrectomized RatsHong Lu and Curtis KlaassenDrug Metabolism and Disposition January 2008, 36 (1) 16-23; DOI: https://doi.org/10.1124/dmd.107.014845
Ludington, Shana R.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Lundstrom, Kerstin
- You have accessRegulation of CYP2A6 Protein Expression by Skatole, Indole, and Testicular Steroids in Primary Cultured Pig HepatocytesGang Chen, Rebecca-Ayme Cue, Kerstin Lundstrom, Jeffrey D. Wood and Olena DoranDrug Metabolism and Disposition January 2008, 36 (1) 56-60; DOI: https://doi.org/10.1124/dmd.107.017285
M
Marie, Bérangère
- You have accessTranscription Factor and Drug-Metabolizing Enzyme Gene Expression in Lymphocytes from Healthy Human SubjectsGérard Siest, Elise Jeannesson, Jean-Brice Marteau, Anastasia Samara, Bérangère Marie, Michèle Pfister and Sophie Visvikis-SiestDrug Metabolism and Disposition January 2008, 36 (1) 182-189; DOI: https://doi.org/10.1124/dmd.107.017228
Marteau, Jean-Brice
- You have accessTranscription Factor and Drug-Metabolizing Enzyme Gene Expression in Lymphocytes from Healthy Human SubjectsGérard Siest, Elise Jeannesson, Jean-Brice Marteau, Anastasia Samara, Bérangère Marie, Michèle Pfister and Sophie Visvikis-SiestDrug Metabolism and Disposition January 2008, 36 (1) 182-189; DOI: https://doi.org/10.1124/dmd.107.017228
Maruyama, Toru
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Maurer, Hans H.
- You have accessIdentification of Cytochrome P450 Enzymes Involved in the Metabolism of the New Designer Drug 4′-Methyl-α-pyrrolidinobutyrophenoneFrank T. Peters, Markus R. Meyer, Denis S. Theobald and Hans H. MaurerDrug Metabolism and Disposition January 2008, 36 (1) 163-168; DOI: https://doi.org/10.1124/dmd.107.017293
Meyer, Markus R.
- You have accessIdentification of Cytochrome P450 Enzymes Involved in the Metabolism of the New Designer Drug 4′-Methyl-α-pyrrolidinobutyrophenoneFrank T. Peters, Markus R. Meyer, Denis S. Theobald and Hans H. MaurerDrug Metabolism and Disposition January 2008, 36 (1) 163-168; DOI: https://doi.org/10.1124/dmd.107.017293
Michaud, Josée
- You have accessEffects of Chronic Renal Failure on Liver Drug TransportersJudith Naud, Josée Michaud, Francois A. Leblond, Stéphane Lefrancois, Alain Bonnardeaux and Vincent PichetteDrug Metabolism and Disposition January 2008, 36 (1) 124-128; DOI: https://doi.org/10.1124/dmd.107.018192
Miller, David S.
- You have accessLocalization of P-gp (Abcb1) and Mrp2 (Abcc2) in Freshly Isolated Rat HepatocytesDaniel A. J. Bow, Jennifer L. Perry, David S. Miller, John B. Pritchard and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 198-202; DOI: https://doi.org/10.1124/dmd.107.018200
Morimoto, Kaori
- You have accessOseltamivir (Tamiflu) Efflux Transport at the Blood-Brain Barrier via P-GlycoproteinKaori Morimoto, Masanori Nakakariya, Yoshiyuki Shirasaka, Chihaya Kakinuma, Takuya Fujita, Ikumi Tamai and Takuo OgiharaDrug Metabolism and Disposition January 2008, 36 (1) 6-9; DOI: https://doi.org/10.1124/dmd.107.017699
Morris, Raymond G.
- You have accessGlucuronidation of Mycophenolic Acid by Wistar and Mrp2-Deficient TR- Rat Liver MicrosomesIan S. Westley, Raymond G. Morris, Allan M. Evans and Benedetta C. SallustioDrug Metabolism and Disposition January 2008, 36 (1) 46-50; DOI: https://doi.org/10.1124/dmd.107.017210
Murphy, Patrick J.
- You have accessThe Development of Drug Metabolism Research as Expressed in the Publications of ASPET: Part 1, 1909–1958Patrick J. MurphyDrug Metabolism and Disposition January 2008, 36 (1) 1-5; DOI: https://doi.org/10.1124/dmd.107.017079
N
Nakakariya, Masanori
- You have accessOseltamivir (Tamiflu) Efflux Transport at the Blood-Brain Barrier via P-GlycoproteinKaori Morimoto, Masanori Nakakariya, Yoshiyuki Shirasaka, Chihaya Kakinuma, Takuya Fujita, Ikumi Tamai and Takuo OgiharaDrug Metabolism and Disposition January 2008, 36 (1) 6-9; DOI: https://doi.org/10.1124/dmd.107.017699
Nakayama, Hitoshi
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Naud, Judith
- You have accessEffects of Chronic Renal Failure on Liver Drug TransportersJudith Naud, Josée Michaud, Francois A. Leblond, Stéphane Lefrancois, Alain Bonnardeaux and Vincent PichetteDrug Metabolism and Disposition January 2008, 36 (1) 124-128; DOI: https://doi.org/10.1124/dmd.107.018192
Neuvonen, Pertti J.
- You have accessTrimethoprim and the CYP2C8*3 Allele Have Opposite Effects on the Pharmacokinetics of PioglitazoneAleksi Tornio, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2008, 36 (1) 73-80; DOI: https://doi.org/10.1124/dmd.107.018010
Nezasa, Ken-ichi
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
Niemi, Mikko
- You have accessTrimethoprim and the CYP2C8*3 Allele Have Opposite Effects on the Pharmacokinetics of PioglitazoneAleksi Tornio, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2008, 36 (1) 73-80; DOI: https://doi.org/10.1124/dmd.107.018010
O
Ogihara, Takuo
- You have accessOseltamivir (Tamiflu) Efflux Transport at the Blood-Brain Barrier via P-GlycoproteinKaori Morimoto, Masanori Nakakariya, Yoshiyuki Shirasaka, Chihaya Kakinuma, Takuya Fujita, Ikumi Tamai and Takuo OgiharaDrug Metabolism and Disposition January 2008, 36 (1) 6-9; DOI: https://doi.org/10.1124/dmd.107.017699
Otagiri, Masaki
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
P
Paine, Mary F.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Pang, K. Sandy
- You have accessPermeability, Transport, and Metabolism of Solutes in Caco-2 Cell Monolayers: A Theoretical StudyHuadong Sun and K. Sandy PangDrug Metabolism and Disposition January 2008, 36 (1) 102-123; DOI: https://doi.org/10.1124/dmd.107.015321
Parman, Toufan
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
Patel, Nita J.
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
Perry, Jennifer L.
- You have accessLocalization of P-gp (Abcb1) and Mrp2 (Abcc2) in Freshly Isolated Rat HepatocytesDaniel A. J. Bow, Jennifer L. Perry, David S. Miller, John B. Pritchard and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 198-202; DOI: https://doi.org/10.1124/dmd.107.018200
Peters, Frank T.
- You have accessIdentification of Cytochrome P450 Enzymes Involved in the Metabolism of the New Designer Drug 4′-Methyl-α-pyrrolidinobutyrophenoneFrank T. Peters, Markus R. Meyer, Denis S. Theobald and Hans H. MaurerDrug Metabolism and Disposition January 2008, 36 (1) 163-168; DOI: https://doi.org/10.1124/dmd.107.017293
Pfister, Michèle
- You have accessTranscription Factor and Drug-Metabolizing Enzyme Gene Expression in Lymphocytes from Healthy Human SubjectsGérard Siest, Elise Jeannesson, Jean-Brice Marteau, Anastasia Samara, Bérangère Marie, Michèle Pfister and Sophie Visvikis-SiestDrug Metabolism and Disposition January 2008, 36 (1) 182-189; DOI: https://doi.org/10.1124/dmd.107.017228
Pichette, Vincent
- You have accessEffects of Chronic Renal Failure on Liver Drug TransportersJudith Naud, Josée Michaud, Francois A. Leblond, Stéphane Lefrancois, Alain Bonnardeaux and Vincent PichetteDrug Metabolism and Disposition January 2008, 36 (1) 124-128; DOI: https://doi.org/10.1124/dmd.107.018192
Poquet, Laure
- You have accessTransport and Metabolism of Ferulic Acid through the Colonic EpitheliumLaure Poquet, Michael N. Clifford and Gary WilliamsonDrug Metabolism and Disposition January 2008, 36 (1) 190-197; DOI: https://doi.org/10.1124/dmd.107.017558
Pritchard, John B.
- You have accessLocalization of P-gp (Abcb1) and Mrp2 (Abcc2) in Freshly Isolated Rat HepatocytesDaniel A. J. Bow, Jennifer L. Perry, David S. Miller, John B. Pritchard and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 198-202; DOI: https://doi.org/10.1124/dmd.107.018200
Pusek, Susan N.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
R
Raub, Thomas J.
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
S
Sakaki, Toshiyuki
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
Sallustio, Benedetta C.
- You have accessGlucuronidation of Mycophenolic Acid by Wistar and Mrp2-Deficient TR- Rat Liver MicrosomesIan S. Westley, Raymond G. Morris, Allan M. Evans and Benedetta C. SallustioDrug Metabolism and Disposition January 2008, 36 (1) 46-50; DOI: https://doi.org/10.1124/dmd.107.017210
Samara, Anastasia
- You have accessTranscription Factor and Drug-Metabolizing Enzyme Gene Expression in Lymphocytes from Healthy Human SubjectsGérard Siest, Elise Jeannesson, Jean-Brice Marteau, Anastasia Samara, Bérangère Marie, Michèle Pfister and Sophie Visvikis-SiestDrug Metabolism and Disposition January 2008, 36 (1) 182-189; DOI: https://doi.org/10.1124/dmd.107.017228
Sargentini-Maier, Maria Laura
- You have accessPharmacokinetics and Metabolism of 14C-Brivaracetam, a Novel SV2A Ligand, in Healthy SubjectsMaria Laura Sargentini-Maier, Pascal Espié, Alain Coquette and Armel StockisDrug Metabolism and Disposition January 2008, 36 (1) 36-45; DOI: https://doi.org/10.1124/dmd.107.017129
Schrieber, Sarah J.
- You have accessPharmacokinetics and Metabolic Profile of Free, Conjugated, and Total Silymarin Flavonolignans in Human Plasma after Oral Administration of Milk Thistle ExtractZhiming Wen, Todd E. Dumas, Sarah J. Schrieber, Roy L. Hawke, Michael W. Fried and Philip C. SmithDrug Metabolism and Disposition January 2008, 36 (1) 65-72; DOI: https://doi.org/10.1124/dmd.107.017566
Schuetz, Erin
- You have accessNovel Single Nucleotide Polymorphisms in the Promoter and Intron 1 of Human Pregnane X Receptor/NR1I2 and Their Association with CYP3A4 ExpressionJatinder Lamba, Vishal Lamba, Stephen Strom, Raman Venkataramanan and Erin SchuetzDrug Metabolism and Disposition January 2008, 36 (1) 169-181; DOI: https://doi.org/10.1124/dmd.107.016600
Schuetz, Erin G.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Sharp, Lewanne E. Hunt
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
Shirasaka, Yoshiyuki
- You have accessOseltamivir (Tamiflu) Efflux Transport at the Blood-Brain Barrier via P-GlycoproteinKaori Morimoto, Masanori Nakakariya, Yoshiyuki Shirasaka, Chihaya Kakinuma, Takuya Fujita, Ikumi Tamai and Takuo OgiharaDrug Metabolism and Disposition January 2008, 36 (1) 6-9; DOI: https://doi.org/10.1124/dmd.107.017699
Siest, Gérard
- You have accessTranscription Factor and Drug-Metabolizing Enzyme Gene Expression in Lymphocytes from Healthy Human SubjectsGérard Siest, Elise Jeannesson, Jean-Brice Marteau, Anastasia Samara, Bérangère Marie, Michèle Pfister and Sophie Visvikis-SiestDrug Metabolism and Disposition January 2008, 36 (1) 182-189; DOI: https://doi.org/10.1124/dmd.107.017228
Smith, Philip C.
- You have accessPharmacokinetics and Metabolic Profile of Free, Conjugated, and Total Silymarin Flavonolignans in Human Plasma after Oral Administration of Milk Thistle ExtractZhiming Wen, Todd E. Dumas, Sarah J. Schrieber, Roy L. Hawke, Michael W. Fried and Philip C. SmithDrug Metabolism and Disposition January 2008, 36 (1) 65-72; DOI: https://doi.org/10.1124/dmd.107.017566
Stephens, R. H.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Stockis, Armel
- You have accessPharmacokinetics and Metabolism of 14C-Brivaracetam, a Novel SV2A Ligand, in Healthy SubjectsMaria Laura Sargentini-Maier, Pascal Espié, Alain Coquette and Armel StockisDrug Metabolism and Disposition January 2008, 36 (1) 36-45; DOI: https://doi.org/10.1124/dmd.107.017129
Strom, Stephen
- You have accessNovel Single Nucleotide Polymorphisms in the Promoter and Intron 1 of Human Pregnane X Receptor/NR1I2 and Their Association with CYP3A4 ExpressionJatinder Lamba, Vishal Lamba, Stephen Strom, Raman Venkataramanan and Erin SchuetzDrug Metabolism and Disposition January 2008, 36 (1) 169-181; DOI: https://doi.org/10.1124/dmd.107.016600
Suenaga, Ayaka
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Sun, Huadong
- You have accessPermeability, Transport, and Metabolism of Solutes in Caco-2 Cell Monolayers: A Theoretical StudyHuadong Sun and K. Sandy PangDrug Metabolism and Disposition January 2008, 36 (1) 102-123; DOI: https://doi.org/10.1124/dmd.107.015321
Suzuki, Hiroshi
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
T
Tamai, Ikumi
- You have accessOseltamivir (Tamiflu) Efflux Transport at the Blood-Brain Barrier via P-GlycoproteinKaori Morimoto, Masanori Nakakariya, Yoshiyuki Shirasaka, Chihaya Kakinuma, Takuya Fujita, Ikumi Tamai and Takuo OgiharaDrug Metabolism and Disposition January 2008, 36 (1) 6-9; DOI: https://doi.org/10.1124/dmd.107.017699
Tamaki, Sekihiro
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
Theobald, Denis S.
- You have accessIdentification of Cytochrome P450 Enzymes Involved in the Metabolism of the New Designer Drug 4′-Methyl-α-pyrrolidinobutyrophenoneFrank T. Peters, Markus R. Meyer, Denis S. Theobald and Hans H. MaurerDrug Metabolism and Disposition January 2008, 36 (1) 163-168; DOI: https://doi.org/10.1124/dmd.107.017293
Thummel, Kenneth E.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Tian, Xianbin
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
Tornio, Aleksi
- You have accessTrimethoprim and the CYP2C8*3 Allele Have Opposite Effects on the Pharmacokinetics of PioglitazoneAleksi Tornio, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2008, 36 (1) 73-80; DOI: https://doi.org/10.1124/dmd.107.018010
V
Vallejo, Jesus
- You have accessRegulation of Hepatic Drug-Metabolizing Enzyme Genes by Toll-Like Receptor 4 Signaling Is Independent of Toll-Interleukin 1 Receptor Domain-Containing Adaptor ProteinRomi Ghose, Damara White, Tao Guo, Jesus Vallejo and Saul J. KarpenDrug Metabolism and Disposition January 2008, 36 (1) 95-101; DOI: https://doi.org/10.1124/dmd.107.018051
Venkataramanan, Raman
- You have accessNovel Single Nucleotide Polymorphisms in the Promoter and Intron 1 of Human Pregnane X Receptor/NR1I2 and Their Association with CYP3A4 ExpressionJatinder Lamba, Vishal Lamba, Stephen Strom, Raman Venkataramanan and Erin SchuetzDrug Metabolism and Disposition January 2008, 36 (1) 169-181; DOI: https://doi.org/10.1124/dmd.107.016600
Visvikis-Siest, Sophie
- You have accessTranscription Factor and Drug-Metabolizing Enzyme Gene Expression in Lymphocytes from Healthy Human SubjectsGérard Siest, Elise Jeannesson, Jean-Brice Marteau, Anastasia Samara, Bérangère Marie, Michèle Pfister and Sophie Visvikis-SiestDrug Metabolism and Disposition January 2008, 36 (1) 182-189; DOI: https://doi.org/10.1124/dmd.107.017228
W
Warhurst, G.
- You have accessInvestigation of Regional Mechanisms Responsible for Poor Oral Absorption in Humans of a Modified Release Preparation of the α-Adrenoreceptor Antagonist, 4-Amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4 tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline (UK-338,003): The Rational Use of ex Vivo Intestine to Predict in Vivo AbsorptionA. Collett, R. H. Stephens, M. D. Harwood, M. Humphrey, L. Dallman, J. Bennett, J. Davis, G. L. Carlson and G. WarhurstDrug Metabolism and Disposition January 2008, 36 (1) 87-94; DOI: https://doi.org/10.1124/dmd.107.016865
Watkins, Paul B.
- You have accessThe Influence of CYP3A5 Expression on the Extent of Hepatic CYP3A Inhibition Is Substrate-Dependent: An in Vitro-in Vivo EvaluationNina Isoherranen, Shana R. Ludington, Raymond C. Givens, Jatinder K. Lamba, Susan N. Pusek, E. Claire Dees, David K. Blough, Kazunori Iwanaga, Roy L. Hawke, Erin G. Schuetz, Paul B. Watkins, Kenneth E. Thummel and Mary F. PaineDrug Metabolism and Disposition January 2008, 36 (1) 146-154; DOI: https://doi.org/10.1124/dmd.107.018382
Weinshilboum, Richard M.
- You have accessEffect of Resveratrol on 17β-Estradiol Sulfation by Human Hepatic and Jejunal S9 and Recombinant Sulfotransferase 1E1Anna M. Furimsky, Carol E. Green, Lewanne E. Hunt Sharp, Paul Catz, Araba A. Adjei, Toufan Parman, Izet M. Kapetanovic, Richard M. Weinshilboum and Lalitha V. IyerDrug Metabolism and Disposition January 2008, 36 (1) 129-136; DOI: https://doi.org/10.1124/dmd.107.016725
Wen, Zhiming
- You have accessPharmacokinetics and Metabolic Profile of Free, Conjugated, and Total Silymarin Flavonolignans in Human Plasma after Oral Administration of Milk Thistle ExtractZhiming Wen, Todd E. Dumas, Sarah J. Schrieber, Roy L. Hawke, Michael W. Fried and Philip C. SmithDrug Metabolism and Disposition January 2008, 36 (1) 65-72; DOI: https://doi.org/10.1124/dmd.107.017566
Westley, Ian S.
- You have accessGlucuronidation of Mycophenolic Acid by Wistar and Mrp2-Deficient TR- Rat Liver MicrosomesIan S. Westley, Raymond G. Morris, Allan M. Evans and Benedetta C. SallustioDrug Metabolism and Disposition January 2008, 36 (1) 46-50; DOI: https://doi.org/10.1124/dmd.107.017210
Whigan, Daisy B.
- You have accessDisposition and Metabolism of [14C]Brasofensine in Rats, Monkeys, and HumansMingshe Zhu, Daisy B. Whigan, Shu Y. Chang and Randy C. DockensDrug Metabolism and Disposition January 2008, 36 (1) 24-35; DOI: https://doi.org/10.1124/dmd.107.016139
White, Damara
- You have accessRegulation of Hepatic Drug-Metabolizing Enzyme Genes by Toll-Like Receptor 4 Signaling Is Independent of Toll-Interleukin 1 Receptor Domain-Containing Adaptor ProteinRomi Ghose, Damara White, Tao Guo, Jesus Vallejo and Saul J. KarpenDrug Metabolism and Disposition January 2008, 36 (1) 95-101; DOI: https://doi.org/10.1124/dmd.107.018051
Williamson, Gary
- You have accessTransport and Metabolism of Ferulic Acid through the Colonic EpitheliumLaure Poquet, Michael N. Clifford and Gary WilliamsonDrug Metabolism and Disposition January 2008, 36 (1) 190-197; DOI: https://doi.org/10.1124/dmd.107.017558
Wood, Jeffrey D.
- You have accessRegulation of CYP2A6 Protein Expression by Skatole, Indole, and Testicular Steroids in Primary Cultured Pig HepatocytesGang Chen, Rebecca-Ayme Cue, Kerstin Lundstrom, Jeffrey D. Wood and Olena DoranDrug Metabolism and Disposition January 2008, 36 (1) 56-60; DOI: https://doi.org/10.1124/dmd.107.017285
Y
Yamada, Shizuo
- You have accessHepatic UDP-Glucuronosyltransferases Responsible for Glucuronidation of Thyroxine in HumansYoshihisa Kato, Shin-ichi Ikushiro, Yoshikazu Emi, Sekihiro Tamaki, Hiroshi Suzuki, Toshiyuki Sakaki, Shizuo Yamada and Masakuni DegawaDrug Metabolism and Disposition January 2008, 36 (1) 51-55; DOI: https://doi.org/10.1124/dmd.107.018184
Yamasaki, Keishi
- You have accessSubdomain IIIA of Dog Albumin Contains a Binding Site Similar to Site II of Human AlbuminKen-ichi Kaneko, Hikaru Fukuda, Victor Tuan Giam Chuang, Keishi Yamasaki, Kohichi Kawahara, Hitoshi Nakayama, Ayaka Suenaga, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition January 2008, 36 (1) 81-86; DOI: https://doi.org/10.1124/dmd.107.016873
Yost, Garold S.
- You have accessMechanism-Based Inactivation of Lung-Selective Cytochrome P450 CYP2F EnzymesJaya S. Kartha and Garold S. YostDrug Metabolism and Disposition January 2008, 36 (1) 155-162; DOI: https://doi.org/10.1124/dmd.107.017897
Z
Zamek-Gliszczynski, Maciej J.
- You have accessMultidrug Resistance-Associated Protein 2 Is Primarily Responsible for the Biliary Excretion of Fexofenadine in MiceXianbin Tian, Maciej J. Zamek-Gliszczynski, Jun Li, Arlene S. Bridges, Ken-ichi Nezasa, Nita J. Patel, Thomas J. Raub and Kim L. R. BrouwerDrug Metabolism and Disposition January 2008, 36 (1) 61-64; DOI: https://doi.org/10.1124/dmd.107.017319
Zhu, Mingshe
- You have accessDisposition and Metabolism of [14C]Brasofensine in Rats, Monkeys, and HumansMingshe Zhu, Daisy B. Whigan, Shu Y. Chang and Randy C. DockensDrug Metabolism and Disposition January 2008, 36 (1) 24-35; DOI: https://doi.org/10.1124/dmd.107.016139
In this issue

Advertisement