Index by author
July 01, 2008; Volume 36,Issue 7
A
A, Jiye
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Adachi, Isao
- You have accessInhibitory Effects of Terpenoids on Multidrug Resistance-Associated Protein 2- and Breast Cancer Resistance Protein-Mediated TransportNaoko Yoshida, Tappei Takada, Yoshikazu Yamamura, Isao Adachi, Hiroshi Suzuki and Junichi KawakamiDrug Metabolism and Disposition July 2008, 36 (7) 1206-1211; DOI: https://doi.org/10.1124/dmd.107.019513
Ahn, Choong Y.
- You have accessPharmacokinetic Parameters of Chlorzoxazone and Its Main Metabolite, 6-Hydroxychlorzoxazone, after Intravenous and Oral Administration of Chlorzoxazone to Liver Cirrhotic Rats with Diabetes MellitusChoong Y. Ahn, Soo K. Bae, Young S. Jung, Inchul Lee, Young C. Kim, Myung G. Lee and Wan G. ShinDrug Metabolism and Disposition July 2008, 36 (7) 1233-1241; DOI: https://doi.org/10.1124/dmd.107.017442
Ai, Hua
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Allentoff, Alban
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Andersson, Tommy B.
- You have accessEvaluation of HepaRG Cells as an in Vitro Model for Human Drug Metabolism StudiesKajsa P. Kanebratt and Tommy B. AnderssonDrug Metabolism and Disposition July 2008, 36 (7) 1444-1452; DOI: https://doi.org/10.1124/dmd.107.020016
Annaert, Pieter
- You have accessCellular Accumulation of Cholyl-Glycylamido-Fluorescein in Sandwich-Cultured Rat Hepatocytes: Kinetic Characterization, Transport Mechanisms, and Effect of Human Immunodeficiency Virus Protease InhibitorsZhi-wei Ye, Patrick Augustijns and Pieter AnnaertDrug Metabolism and Disposition July 2008, 36 (7) 1315-1321; DOI: https://doi.org/10.1124/dmd.107.019398
Aparicio-Fabre, Rosaura
- You have accessOsmotic Regulation of a Novel Flavin-Containing Monooxygenase in Primary Cultured Cells from Rainbow Trout (Oncorhynchus mykiss)Gabriela Rodríguez-Fuentes, Rosaura Aparicio-Fabre, Qi Li and Daniel SchlenkDrug Metabolism and Disposition July 2008, 36 (7) 1212-1217; DOI: https://doi.org/10.1124/dmd.107.019968
Arora, Vinod K.
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
Augustijns, Patrick
- You have accessCellular Accumulation of Cholyl-Glycylamido-Fluorescein in Sandwich-Cultured Rat Hepatocytes: Kinetic Characterization, Transport Mechanisms, and Effect of Human Immunodeficiency Virus Protease InhibitorsZhi-wei Ye, Patrick Augustijns and Pieter AnnaertDrug Metabolism and Disposition July 2008, 36 (7) 1315-1321; DOI: https://doi.org/10.1124/dmd.107.019398
B
Bae, Soo K.
- You have accessPharmacokinetic Parameters of Chlorzoxazone and Its Main Metabolite, 6-Hydroxychlorzoxazone, after Intravenous and Oral Administration of Chlorzoxazone to Liver Cirrhotic Rats with Diabetes MellitusChoong Y. Ahn, Soo K. Bae, Young S. Jung, Inchul Lee, Young C. Kim, Myung G. Lee and Wan G. ShinDrug Metabolism and Disposition July 2008, 36 (7) 1233-1241; DOI: https://doi.org/10.1124/dmd.107.017442
Balani, Suresh K.
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. II. In Vitro-in Vivo Correlation with KetoconazoleChuang Lu, Panos Hatsis, Cicely Berg, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1255-1260; DOI: https://doi.org/10.1124/dmd.107.018796
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. III. In Vitro-in Vivo Correlation with FluconazoleChuang Lu, Cicely Berg, Shimoga R. Prakash, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1261-1266; DOI: https://doi.org/10.1124/dmd.107.019000
Barros, Anthony
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Berg, Cicely
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. II. In Vitro-in Vivo Correlation with KetoconazoleChuang Lu, Panos Hatsis, Cicely Berg, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1255-1260; DOI: https://doi.org/10.1124/dmd.107.018796
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. III. In Vitro-in Vivo Correlation with FluconazoleChuang Lu, Cicely Berg, Shimoga R. Prakash, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1261-1266; DOI: https://doi.org/10.1124/dmd.107.019000
Blackwood-Chirchir, Anne
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Bonacorsi, Samuel J.
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Brundage, Richard C.
- You have accessDifferential Genotype Dependent Inhibition of CYP2C9 in HumansVikas Kumar, Richard C. Brundage, William S. Oetting, Ilo E. Leppik and Timothy S. TracyDrug Metabolism and Disposition July 2008, 36 (7) 1242-1248; DOI: https://doi.org/10.1124/dmd.108.020396
Bui, Peter H.
- You have accessThe Mibefradil Derivative NNC55-0396, a Specific T-Type Calcium Channel Antagonist, Exhibits Less CYP3A4 Inhibition than MibefradilPeter H. Bui, Arnulfo Quesada, Adrian Handforth and Oliver HankinsonDrug Metabolism and Disposition July 2008, 36 (7) 1291-1299; DOI: https://doi.org/10.1124/dmd.107.020115
C
Carreiro, Samantha
- You have accessDrug Transporter and Cytochrome P450 mRNA Expression in Human Ocular Barriers: Implications for Ocular Drug DispositionTao Zhang, Cathie D. Xiang, David Gale, Samantha Carreiro, Ellen Y. Wu and Eric Y. ZhangDrug Metabolism and Disposition July 2008, 36 (7) 1300-1307; DOI: https://doi.org/10.1124/dmd.108.021121
Christensen, James G.
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Christopher, Lisa J.
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Cui, Donghui
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
D
Dalvie, Deepak
- You have accessBioactivation of Flutamide Metabolites by Human Liver MicrosomesPing Kang, Deepak Dalvie, Evan Smith, Sue Zhou, Alan Deese and James A. NiemanDrug Metabolism and Disposition July 2008, 36 (7) 1425-1437; DOI: https://doi.org/10.1124/dmd.108.020370
Deese, Alan
- You have accessBioactivation of Flutamide Metabolites by Human Liver MicrosomesPing Kang, Deepak Dalvie, Evan Smith, Sue Zhou, Alan Deese and James A. NiemanDrug Metabolism and Disposition July 2008, 36 (7) 1425-1437; DOI: https://doi.org/10.1124/dmd.108.020370
Dickmann, Leslie J.
- You have accessFunctional Expression and Comparative Characterization of Nine Murine Cytochromes P450 by Fluorescent Inhibition ScreeningLesley A. McLaughlin, Leslie J. Dickmann, C. Roland Wolf and Colin J. HendersonDrug Metabolism and Disposition July 2008, 36 (7) 1322-1331; DOI: https://doi.org/10.1124/dmd.108.021261
F
Farid, Nagy A.
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Fitzsimmons, Patrick N.
- You have accessUse of Online Microdialysis Sampling to Determine the in Vivo Rate of Phenol Glucuronidation in Rainbow TroutJohn W. Nichols, Alex D. Hoffman, Patrick N. Fitzsimmons, Gregory J. Lien and Correne T. JensonDrug Metabolism and Disposition July 2008, 36 (7) 1406-1413; DOI: https://doi.org/10.1124/dmd.107.020123
Fletcher, Anthony M.
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
Fricker, Gert
- You have accessClosing the Gaps: A Full Scan of the Intestinal Expression of P-Glycoprotein, Breast Cancer Resistance Protein, and Multidrug Resistance-Associated Protein 2 in Male and Female RatsCaroline MacLean, Ulla Moenning, Andreas Reichel and Gert FrickerDrug Metabolism and Disposition July 2008, 36 (7) 1249-1254; DOI: https://doi.org/10.1124/dmd.108.020859
Fukuda, Hajime
- You have accessEffect of Plasma Protein Binding on in Vitro-in Vivo Correlation of Biliary Excretion of Drugs Evaluated by Sandwich-Cultured Rat HepatocytesHajime Fukuda, Rikiya Ohashi, Minoru Tsuda-Tsukimoto and Ikumi TamaiDrug Metabolism and Disposition July 2008, 36 (7) 1275-1282; DOI: https://doi.org/10.1124/dmd.107.019026
G
Galbraith, Susan
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Gale, David
- You have accessDrug Transporter and Cytochrome P450 mRNA Expression in Human Ocular Barriers: Implications for Ocular Drug DispositionTao Zhang, Cathie D. Xiang, David Gale, Samantha Carreiro, Ellen Y. Wu and Eric Y. ZhangDrug Metabolism and Disposition July 2008, 36 (7) 1300-1307; DOI: https://doi.org/10.1124/dmd.108.021121
Galetin, Aleksandra
- You have accessHepatocellular Binding of Drugs: Correction for Unbound Fraction in Hepatocyte Incubations Using Microsomal Binding or Drug Lipophilicity DataPeter J. Kilford, Michael Gertz, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition July 2008, 36 (7) 1194-1197; DOI: https://doi.org/10.1124/dmd.108.020834
- You have accessComparative Analysis of CYP3A Heteroactivation by Steroid Hormones and Flavonoids in Different in Vitro Systems and Potential in Vivo ImplicationsJamie Henshall, Aleksandra Galetin, Anthony Harrison and J. Brian HoustonDrug Metabolism and Disposition July 2008, 36 (7) 1332-1340; DOI: https://doi.org/10.1124/dmd.108.021279
Gardiner, Philip
- You have accessPrediction of the Pharmacokinetics of Atorvastatin, Cerivastatin, and Indomethacin Using Kinetic Models Applied to Isolated Rat HepatocytesStuart W. Paine, Alison J. Parker, Philip Gardiner, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition July 2008, 36 (7) 1365-1374; DOI: https://doi.org/10.1124/dmd.107.019455
Gardner, Mark J.
- You have accessDisposition of Lasofoxifene, a Next-Generation Selective Estrogen Receptor Modulator, in Healthy Male SubjectsChandra Prakash, Kim A. Johnson and Mark J. GardnerDrug Metabolism and Disposition July 2008, 36 (7) 1218-1226; DOI: https://doi.org/10.1124/dmd.108.020404
Garmire, Lana X.
- You have accessIn Silico Methods for Unraveling the Mechanistic Complexities of Intestinal Absorption: Metabolism-Efflux Transport InteractionsLana X. Garmire and C. Anthony HuntDrug Metabolism and Disposition July 2008, 36 (7) 1414-1424; DOI: https://doi.org/10.1124/dmd.107.020164
Generaux, Grant T.
- You have accessAn in Vitro Mechanistic Study to Elucidate the Desipramine/Bupropion Clinical Drug-Drug InteractionMelinda J. Reese, Robert M. Wurm, Keith T. Muir, Grant T. Generaux, Lisa St. John-Williams and Donavon J. McconnDrug Metabolism and Disposition July 2008, 36 (7) 1198-1201; DOI: https://doi.org/10.1124/dmd.107.020198
Gertz, Michael
- You have accessHepatocellular Binding of Drugs: Correction for Unbound Fraction in Hepatocyte Incubations Using Microsomal Binding or Drug Lipophilicity DataPeter J. Kilford, Michael Gertz, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition July 2008, 36 (7) 1194-1197; DOI: https://doi.org/10.1124/dmd.108.020834
H
Handforth, Adrian
- You have accessThe Mibefradil Derivative NNC55-0396, a Specific T-Type Calcium Channel Antagonist, Exhibits Less CYP3A4 Inhibition than MibefradilPeter H. Bui, Arnulfo Quesada, Adrian Handforth and Oliver HankinsonDrug Metabolism and Disposition July 2008, 36 (7) 1291-1299; DOI: https://doi.org/10.1124/dmd.107.020115
Hankinson, Oliver
- You have accessThe Mibefradil Derivative NNC55-0396, a Specific T-Type Calcium Channel Antagonist, Exhibits Less CYP3A4 Inhibition than MibefradilPeter H. Bui, Arnulfo Quesada, Adrian Handforth and Oliver HankinsonDrug Metabolism and Disposition July 2008, 36 (7) 1291-1299; DOI: https://doi.org/10.1124/dmd.107.020115
Hao, Haiping
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Harrison, Anthony
- You have accessComparative Analysis of CYP3A Heteroactivation by Steroid Hormones and Flavonoids in Different in Vitro Systems and Potential in Vivo ImplicationsJamie Henshall, Aleksandra Galetin, Anthony Harrison and J. Brian HoustonDrug Metabolism and Disposition July 2008, 36 (7) 1332-1340; DOI: https://doi.org/10.1124/dmd.108.021279
Hatsis, Panos
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. II. In Vitro-in Vivo Correlation with KetoconazoleChuang Lu, Panos Hatsis, Cicely Berg, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1255-1260; DOI: https://doi.org/10.1124/dmd.107.018796
He, Kan
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Henderson, Colin J.
- You have accessFunctional Expression and Comparative Characterization of Nine Murine Cytochromes P450 by Fluorescent Inhibition ScreeningLesley A. McLaughlin, Leslie J. Dickmann, C. Roland Wolf and Colin J. HendersonDrug Metabolism and Disposition July 2008, 36 (7) 1322-1331; DOI: https://doi.org/10.1124/dmd.108.021261
Henshall, Jamie
- You have accessComparative Analysis of CYP3A Heteroactivation by Steroid Hormones and Flavonoids in Different in Vitro Systems and Potential in Vivo ImplicationsJamie Henshall, Aleksandra Galetin, Anthony Harrison and J. Brian HoustonDrug Metabolism and Disposition July 2008, 36 (7) 1332-1340; DOI: https://doi.org/10.1124/dmd.108.021279
Hoffman, Alex D.
- You have accessUse of Online Microdialysis Sampling to Determine the in Vivo Rate of Phenol Glucuronidation in Rainbow TroutJohn W. Nichols, Alex D. Hoffman, Patrick N. Fitzsimmons, Gregory J. Lien and Correne T. JensonDrug Metabolism and Disposition July 2008, 36 (7) 1406-1413; DOI: https://doi.org/10.1124/dmd.107.020123
Horie, Toru
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
Houston, J. Brian
- You have accessHepatocellular Binding of Drugs: Correction for Unbound Fraction in Hepatocyte Incubations Using Microsomal Binding or Drug Lipophilicity DataPeter J. Kilford, Michael Gertz, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition July 2008, 36 (7) 1194-1197; DOI: https://doi.org/10.1124/dmd.108.020834
- You have accessComparative Analysis of CYP3A Heteroactivation by Steroid Hormones and Flavonoids in Different in Vitro Systems and Potential in Vivo ImplicationsJamie Henshall, Aleksandra Galetin, Anthony Harrison and J. Brian HoustonDrug Metabolism and Disposition July 2008, 36 (7) 1332-1340; DOI: https://doi.org/10.1124/dmd.108.021279
- You have accessRate-Limiting Steps in Hepatic Drug Clearance: Comparison of Hepatocellular Uptake and Metabolism with Microsomal Metabolism of Saquinavir, Nelfinavir, and RitonavirAlison J. Parker and J. Brian HoustonDrug Metabolism and Disposition July 2008, 36 (7) 1375-1384; DOI: https://doi.org/10.1124/dmd.108.020917
Humphreys, W. Griffith
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Hunt, C. Anthony
- You have accessIn Silico Methods for Unraveling the Mechanistic Complexities of Intestinal Absorption: Metabolism-Efflux Transport InteractionsLana X. Garmire and C. Anthony HuntDrug Metabolism and Disposition July 2008, 36 (7) 1414-1424; DOI: https://doi.org/10.1124/dmd.107.020164
I
Iizuka, Seiichi
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
Imamura, Sachiko
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
Inoue, Makoto
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
Inoue, Tae
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
Iyer, Ramaswamy A.
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
J
Jenson, Correne T.
- You have accessUse of Online Microdialysis Sampling to Determine the in Vivo Rate of Phenol Glucuronidation in Rainbow TroutJohn W. Nichols, Alex D. Hoffman, Patrick N. Fitzsimmons, Gregory J. Lien and Correne T. JensonDrug Metabolism and Disposition July 2008, 36 (7) 1406-1413; DOI: https://doi.org/10.1124/dmd.107.020123
Johnson, Kim A.
- You have accessDisposition of Lasofoxifene, a Next-Generation Selective Estrogen Receptor Modulator, in Healthy Male SubjectsChandra Prakash, Kim A. Johnson and Mark J. GardnerDrug Metabolism and Disposition July 2008, 36 (7) 1218-1226; DOI: https://doi.org/10.1124/dmd.108.020404
Jones, Karen O.
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Jung, Young S.
- You have accessPharmacokinetic Parameters of Chlorzoxazone and Its Main Metabolite, 6-Hydroxychlorzoxazone, after Intravenous and Oral Administration of Chlorzoxazone to Liver Cirrhotic Rats with Diabetes MellitusChoong Y. Ahn, Soo K. Bae, Young S. Jung, Inchul Lee, Young C. Kim, Myung G. Lee and Wan G. ShinDrug Metabolism and Disposition July 2008, 36 (7) 1233-1241; DOI: https://doi.org/10.1124/dmd.107.017442
K
Kanebratt, Kajsa P.
- You have accessEvaluation of HepaRG Cells as an in Vitro Model for Human Drug Metabolism StudiesKajsa P. Kanebratt and Tommy B. AnderssonDrug Metabolism and Disposition July 2008, 36 (7) 1444-1452; DOI: https://doi.org/10.1124/dmd.107.020016
Kang, Ping
- You have accessBioactivation of Flutamide Metabolites by Human Liver MicrosomesPing Kang, Deepak Dalvie, Evan Smith, Sue Zhou, Alan Deese and James A. NiemanDrug Metabolism and Disposition July 2008, 36 (7) 1425-1437; DOI: https://doi.org/10.1124/dmd.108.020370
Kawakami, Junichi
- You have accessInhibitory Effects of Terpenoids on Multidrug Resistance-Associated Protein 2- and Breast Cancer Resistance Protein-Mediated TransportNaoko Yoshida, Tappei Takada, Yoshikazu Yamamura, Isao Adachi, Hiroshi Suzuki and Junichi KawakamiDrug Metabolism and Disposition July 2008, 36 (7) 1206-1211; DOI: https://doi.org/10.1124/dmd.107.019513
Kazui, Miho
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Kilford, Peter J.
- You have accessHepatocellular Binding of Drugs: Correction for Unbound Fraction in Hepatocyte Incubations Using Microsomal Binding or Drug Lipophilicity DataPeter J. Kilford, Michael Gertz, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition July 2008, 36 (7) 1194-1197; DOI: https://doi.org/10.1124/dmd.108.020834
Kim, Young C.
- You have accessPharmacokinetic Parameters of Chlorzoxazone and Its Main Metabolite, 6-Hydroxychlorzoxazone, after Intravenous and Oral Administration of Chlorzoxazone to Liver Cirrhotic Rats with Diabetes MellitusChoong Y. Ahn, Soo K. Bae, Young S. Jung, Inchul Lee, Young C. Kim, Myung G. Lee and Wan G. ShinDrug Metabolism and Disposition July 2008, 36 (7) 1233-1241; DOI: https://doi.org/10.1124/dmd.107.017442
Kitamura, Shigeyuki
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
Koudriakova, Tatiana
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Koup, Jeffrey R.
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Kumar, Vikas
- You have accessDifferential Genotype Dependent Inhibition of CYP2C9 in HumansVikas Kumar, Richard C. Brundage, William S. Oetting, Ilo E. Leppik and Timothy S. TracyDrug Metabolism and Disposition July 2008, 36 (7) 1242-1248; DOI: https://doi.org/10.1124/dmd.108.020396
L
Lago, Michael
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Lee, Francis Y. F.
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Lee, Frank W.
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. II. In Vitro-in Vivo Correlation with KetoconazoleChuang Lu, Panos Hatsis, Cicely Berg, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1255-1260; DOI: https://doi.org/10.1124/dmd.107.018796
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. III. In Vitro-in Vivo Correlation with FluconazoleChuang Lu, Cicely Berg, Shimoga R. Prakash, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1261-1266; DOI: https://doi.org/10.1124/dmd.107.019000
Lee, Inchul
- You have accessPharmacokinetic Parameters of Chlorzoxazone and Its Main Metabolite, 6-Hydroxychlorzoxazone, after Intravenous and Oral Administration of Chlorzoxazone to Liver Cirrhotic Rats with Diabetes MellitusChoong Y. Ahn, Soo K. Bae, Young S. Jung, Inchul Lee, Young C. Kim, Myung G. Lee and Wan G. ShinDrug Metabolism and Disposition July 2008, 36 (7) 1233-1241; DOI: https://doi.org/10.1124/dmd.107.017442
Lee, Joseph H.
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Lee, Myung G.
- You have accessPharmacokinetic Parameters of Chlorzoxazone and Its Main Metabolite, 6-Hydroxychlorzoxazone, after Intravenous and Oral Administration of Chlorzoxazone to Liver Cirrhotic Rats with Diabetes MellitusChoong Y. Ahn, Soo K. Bae, Young S. Jung, Inchul Lee, Young C. Kim, Myung G. Lee and Wan G. ShinDrug Metabolism and Disposition July 2008, 36 (7) 1233-1241; DOI: https://doi.org/10.1124/dmd.107.017442
Leppik, Ilo E.
- You have accessDifferential Genotype Dependent Inhibition of CYP2C9 in HumansVikas Kumar, Richard C. Brundage, William S. Oetting, Ilo E. Leppik and Timothy S. TracyDrug Metabolism and Disposition July 2008, 36 (7) 1242-1248; DOI: https://doi.org/10.1124/dmd.108.020396
Li, Qi
- You have accessOsmotic Regulation of a Novel Flavin-Containing Monooxygenase in Primary Cultured Cells from Rainbow Trout (Oncorhynchus mykiss)Gabriela Rodríguez-Fuentes, Rosaura Aparicio-Fabre, Qi Li and Daniel SchlenkDrug Metabolism and Disposition July 2008, 36 (7) 1212-1217; DOI: https://doi.org/10.1124/dmd.107.019968
Li, Wenying
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
Lien, Gregory J.
- You have accessUse of Online Microdialysis Sampling to Determine the in Vivo Rate of Phenol Glucuronidation in Rainbow TroutJohn W. Nichols, Alex D. Hoffman, Patrick N. Fitzsimmons, Gregory J. Lien and Correne T. JensonDrug Metabolism and Disposition July 2008, 36 (7) 1406-1413; DOI: https://doi.org/10.1124/dmd.107.020123
Lim, Lee-Yong
- You have accessEffects of Spice Constituents on P-Glycoprotein-Mediated Transport and CYP3A4-Mediated Metabolism in VitroWenxia Zhang and Lee-Yong LimDrug Metabolism and Disposition July 2008, 36 (7) 1283-1290; DOI: https://doi.org/10.1124/dmd.107.019737
Lombardo, Franco
- You have accessTrend Analysis of a Database of Intravenous Pharmacokinetic Parameters in Humans for 670 Drug CompoundsR. Scott Obach, Franco Lombardo and Nigel J. WatersDrug Metabolism and Disposition July 2008, 36 (7) 1385-1405; DOI: https://doi.org/10.1124/dmd.108.020479
Lowery, Shane M.
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Lu, Chuang
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. II. In Vitro-in Vivo Correlation with KetoconazoleChuang Lu, Panos Hatsis, Cicely Berg, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1255-1260; DOI: https://doi.org/10.1124/dmd.107.018796
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. III. In Vitro-in Vivo Correlation with FluconazoleChuang Lu, Cicely Berg, Shimoga R. Prakash, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1261-1266; DOI: https://doi.org/10.1124/dmd.107.019000
Luo, Roger
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
M
MacLean, Caroline
- You have accessClosing the Gaps: A Full Scan of the Intestinal Expression of P-Glycoprotein, Breast Cancer Resistance Protein, and Multidrug Resistance-Associated Protein 2 in Male and Female RatsCaroline MacLean, Ulla Moenning, Andreas Reichel and Gert FrickerDrug Metabolism and Disposition July 2008, 36 (7) 1249-1254; DOI: https://doi.org/10.1124/dmd.108.020859
Makino, Toshiaki
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
Manning, James A.
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
McCann, Betty
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Mcconn, Donavon J.
- You have accessAn in Vitro Mechanistic Study to Elucidate the Desipramine/Bupropion Clinical Drug-Drug InteractionMelinda J. Reese, Robert M. Wurm, Keith T. Muir, Grant T. Generaux, Lisa St. John-Williams and Donavon J. McconnDrug Metabolism and Disposition July 2008, 36 (7) 1198-1201; DOI: https://doi.org/10.1124/dmd.107.020198
McLaughlin, Lesley A.
- You have accessFunctional Expression and Comparative Characterization of Nine Murine Cytochromes P450 by Fluorescent Inhibition ScreeningLesley A. McLaughlin, Leslie J. Dickmann, C. Roland Wolf and Colin J. HendersonDrug Metabolism and Disposition July 2008, 36 (7) 1322-1331; DOI: https://doi.org/10.1124/dmd.108.021261
Mizukami, Hajime
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
Moenning, Ulla
- You have accessClosing the Gaps: A Full Scan of the Intestinal Expression of P-Glycoprotein, Breast Cancer Resistance Protein, and Multidrug Resistance-Associated Protein 2 in Male and Female RatsCaroline MacLean, Ulla Moenning, Andreas Reichel and Gert FrickerDrug Metabolism and Disposition July 2008, 36 (7) 1249-1254; DOI: https://doi.org/10.1124/dmd.108.020859
Muir, Keith T.
- You have accessAn in Vitro Mechanistic Study to Elucidate the Desipramine/Bupropion Clinical Drug-Drug InteractionMelinda J. Reese, Robert M. Wurm, Keith T. Muir, Grant T. Generaux, Lisa St. John-Williams and Donavon J. McconnDrug Metabolism and Disposition July 2008, 36 (7) 1198-1201; DOI: https://doi.org/10.1124/dmd.107.020198
N
Negishi, Masahiko
- You have accessThe Antiapoptotic Factor Growth Arrest and DNA-Damage-Inducible 45 β Regulates the Nuclear Receptor Constitutive Active/Androstane Receptor-Mediated TranscriptionYukio Yamamoto and Masahiko NegishiDrug Metabolism and Disposition July 2008, 36 (7) 1189-1193; DOI: https://doi.org/10.1124/dmd.108.020628
Nichols, John W.
- You have accessUse of Online Microdialysis Sampling to Determine the in Vivo Rate of Phenol Glucuronidation in Rainbow TroutJohn W. Nichols, Alex D. Hoffman, Patrick N. Fitzsimmons, Gregory J. Lien and Correne T. JensonDrug Metabolism and Disposition July 2008, 36 (7) 1406-1413; DOI: https://doi.org/10.1124/dmd.107.020123
Nieman, James A.
- You have accessBioactivation of Flutamide Metabolites by Human Liver MicrosomesPing Kang, Deepak Dalvie, Evan Smith, Sue Zhou, Alan Deese and James A. NiemanDrug Metabolism and Disposition July 2008, 36 (7) 1425-1437; DOI: https://doi.org/10.1124/dmd.108.020370
Nitta, Kayoko
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
O
Obach, R. Scott
- You have accessTrend Analysis of a Database of Intravenous Pharmacokinetic Parameters in Humans for 670 Drug CompoundsR. Scott Obach, Franco Lombardo and Nigel J. WatersDrug Metabolism and Disposition July 2008, 36 (7) 1385-1405; DOI: https://doi.org/10.1124/dmd.108.020479
Oetting, William S.
- You have accessDifferential Genotype Dependent Inhibition of CYP2C9 in HumansVikas Kumar, Richard C. Brundage, William S. Oetting, Ilo E. Leppik and Timothy S. TracyDrug Metabolism and Disposition July 2008, 36 (7) 1242-1248; DOI: https://doi.org/10.1124/dmd.108.020396
Ogan, Marc
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
Ohashi, Rikiya
- You have accessEffect of Plasma Protein Binding on in Vitro-in Vivo Correlation of Biliary Excretion of Drugs Evaluated by Sandwich-Cultured Rat HepatocytesHajime Fukuda, Rikiya Ohashi, Minoru Tsuda-Tsukimoto and Ikumi TamaiDrug Metabolism and Disposition July 2008, 36 (7) 1275-1282; DOI: https://doi.org/10.1124/dmd.107.019026
Ohta, Shigeru
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
Ohtake, Nobuhiro
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
P
Paine, Stuart W.
- You have accessPrediction of the Pharmacokinetics of Atorvastatin, Cerivastatin, and Indomethacin Using Kinetic Models Applied to Isolated Rat HepatocytesStuart W. Paine, Alison J. Parker, Philip Gardiner, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition July 2008, 36 (7) 1365-1374; DOI: https://doi.org/10.1124/dmd.107.019455
Parker, Alison J.
- You have accessRate-Limiting Steps in Hepatic Drug Clearance: Comparison of Hepatocellular Uptake and Metabolism with Microsomal Metabolism of Saquinavir, Nelfinavir, and RitonavirAlison J. Parker and J. Brian HoustonDrug Metabolism and Disposition July 2008, 36 (7) 1375-1384; DOI: https://doi.org/10.1124/dmd.108.020917
- You have accessPrediction of the Pharmacokinetics of Atorvastatin, Cerivastatin, and Indomethacin Using Kinetic Models Applied to Isolated Rat HepatocytesStuart W. Paine, Alison J. Parker, Philip Gardiner, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition July 2008, 36 (7) 1365-1374; DOI: https://doi.org/10.1124/dmd.107.019455
Peng, Ying
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Perkins, Everett J.
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Ponsler, G. Douglas
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Prakash, Chandra
- You have accessDisposition of Lasofoxifene, a Next-Generation Selective Estrogen Receptor Modulator, in Healthy Male SubjectsChandra Prakash, Kim A. Johnson and Mark J. GardnerDrug Metabolism and Disposition July 2008, 36 (7) 1218-1226; DOI: https://doi.org/10.1124/dmd.108.020404
Prakash, Shimoga R.
- You have accessPrediction of Pharmacokinetic Drug-Drug Interactions Using Human Hepatocyte Suspension in Plasma and Cytochrome P450 Phenotypic Data. III. In Vitro-in Vivo Correlation with FluconazoleChuang Lu, Cicely Berg, Shimoga R. Prakash, Frank W. Lee and Suresh K. BalaniDrug Metabolism and Disposition July 2008, 36 (7) 1261-1266; DOI: https://doi.org/10.1124/dmd.107.019000
Q
Qiu, Furong
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Quesada, Arnulfo
- You have accessThe Mibefradil Derivative NNC55-0396, a Specific T-Type Calcium Channel Antagonist, Exhibits Less CYP3A4 Inhibition than MibefradilPeter H. Bui, Arnulfo Quesada, Adrian Handforth and Oliver HankinsonDrug Metabolism and Disposition July 2008, 36 (7) 1291-1299; DOI: https://doi.org/10.1124/dmd.107.020115
R
Reese, Melinda J.
- You have accessAn in Vitro Mechanistic Study to Elucidate the Desipramine/Bupropion Clinical Drug-Drug InteractionMelinda J. Reese, Robert M. Wurm, Keith T. Muir, Grant T. Generaux, Lisa St. John-Williams and Donavon J. McconnDrug Metabolism and Disposition July 2008, 36 (7) 1198-1201; DOI: https://doi.org/10.1124/dmd.107.020198
Reichel, Andreas
- You have accessClosing the Gaps: A Full Scan of the Intestinal Expression of P-Glycoprotein, Breast Cancer Resistance Protein, and Multidrug Resistance-Associated Protein 2 in Male and Female RatsCaroline MacLean, Ulla Moenning, Andreas Reichel and Gert FrickerDrug Metabolism and Disposition July 2008, 36 (7) 1249-1254; DOI: https://doi.org/10.1124/dmd.108.020859
Reitberg, Donald P.
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Riley, Robert J.
- You have accessPrediction of the Pharmacokinetics of Atorvastatin, Cerivastatin, and Indomethacin Using Kinetic Models Applied to Isolated Rat HepatocytesStuart W. Paine, Alison J. Parker, Philip Gardiner, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition July 2008, 36 (7) 1365-1374; DOI: https://doi.org/10.1124/dmd.107.019455
Rodríguez-Fuentes, Gabriela
- You have accessOsmotic Regulation of a Novel Flavin-Containing Monooxygenase in Primary Cultured Cells from Rainbow Trout (Oncorhynchus mykiss)Gabriela Rodríguez-Fuentes, Rosaura Aparicio-Fabre, Qi Li and Daniel SchlenkDrug Metabolism and Disposition July 2008, 36 (7) 1212-1217; DOI: https://doi.org/10.1124/dmd.107.019968
Romero, David
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Ruterbories, Kenneth J.
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
S
Schlenk, Daniel
- You have accessOsmotic Regulation of a Novel Flavin-Containing Monooxygenase in Primary Cultured Cells from Rainbow Trout (Oncorhynchus mykiss)Gabriela Rodríguez-Fuentes, Rosaura Aparicio-Fabre, Qi Li and Daniel SchlenkDrug Metabolism and Disposition July 2008, 36 (7) 1212-1217; DOI: https://doi.org/10.1124/dmd.107.019968
Shin, Wan G.
- You have accessPharmacokinetic Parameters of Chlorzoxazone and Its Main Metabolite, 6-Hydroxychlorzoxazone, after Intravenous and Oral Administration of Chlorzoxazone to Liver Cirrhotic Rats with Diabetes MellitusChoong Y. Ahn, Soo K. Bae, Young S. Jung, Inchul Lee, Young C. Kim, Myung G. Lee and Wan G. ShinDrug Metabolism and Disposition July 2008, 36 (7) 1233-1241; DOI: https://doi.org/10.1124/dmd.107.017442
Skaptason, Judith
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Smith, Bill J.
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Smith, Evan
- You have accessBioactivation of Flutamide Metabolites by Human Liver MicrosomesPing Kang, Deepak Dalvie, Evan Smith, Sue Zhou, Alan Deese and James A. NiemanDrug Metabolism and Disposition July 2008, 36 (7) 1425-1437; DOI: https://doi.org/10.1124/dmd.108.020370
St. John-Williams, Lisa
- You have accessAn in Vitro Mechanistic Study to Elucidate the Desipramine/Bupropion Clinical Drug-Drug InteractionMelinda J. Reese, Robert M. Wurm, Keith T. Muir, Grant T. Generaux, Lisa St. John-Williams and Donavon J. McconnDrug Metabolism and Disposition July 2008, 36 (7) 1198-1201; DOI: https://doi.org/10.1124/dmd.107.020198
Sugihara, Kazumi
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
Sun, Jianguo
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Suzuki, Hiroshi
- You have accessInhibitory Effects of Terpenoids on Multidrug Resistance-Associated Protein 2- and Breast Cancer Resistance Protein-Mediated TransportNaoko Yoshida, Tappei Takada, Yoshikazu Yamamura, Isao Adachi, Hiroshi Suzuki and Junichi KawakamiDrug Metabolism and Disposition July 2008, 36 (7) 1206-1211; DOI: https://doi.org/10.1124/dmd.107.019513
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Takada, Tappei
- You have accessInhibitory Effects of Terpenoids on Multidrug Resistance-Associated Protein 2- and Breast Cancer Resistance Protein-Mediated TransportNaoko Yoshida, Tappei Takada, Yoshikazu Yamamura, Isao Adachi, Hiroshi Suzuki and Junichi KawakamiDrug Metabolism and Disposition July 2008, 36 (7) 1206-1211; DOI: https://doi.org/10.1124/dmd.107.019513
Tamai, Ikumi
- You have accessEffect of Plasma Protein Binding on in Vitro-in Vivo Correlation of Biliary Excretion of Drugs Evaluated by Sandwich-Cultured Rat HepatocytesHajime Fukuda, Rikiya Ohashi, Minoru Tsuda-Tsukimoto and Ikumi TamaiDrug Metabolism and Disposition July 2008, 36 (7) 1275-1282; DOI: https://doi.org/10.1124/dmd.107.019026
Tanoue, Chiaki
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
Tayama, Yoshitaka
- You have accessAldehyde Oxidase-Catalyzed Metabolism of N1-Methylnicotinamide in Vivo and in Vitro in Chimeric Mice with Humanized LiverShigeyuki Kitamura, Kayoko Nitta, Yoshitaka Tayama, Chiaki Tanoue, Kazumi Sugihara, Tae Inoue, Toru Horie and Shigeru OhtaDrug Metabolism and Disposition July 2008, 36 (7) 1202-1205; DOI: https://doi.org/10.1124/dmd.107.019075
Tracy, Timothy S.
- You have accessDifferential Genotype Dependent Inhibition of CYP2C9 in HumansVikas Kumar, Richard C. Brundage, William S. Oetting, Ilo E. Leppik and Timothy S. TracyDrug Metabolism and Disposition July 2008, 36 (7) 1242-1248; DOI: https://doi.org/10.1124/dmd.108.020396
Tsuchiya, Naoko
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
Tsuda-Tsukimoto, Minoru
- You have accessEffect of Plasma Protein Binding on in Vitro-in Vivo Correlation of Biliary Excretion of Drugs Evaluated by Sandwich-Cultured Rat HepatocytesHajime Fukuda, Rikiya Ohashi, Minoru Tsuda-Tsukimoto and Ikumi TamaiDrug Metabolism and Disposition July 2008, 36 (7) 1275-1282; DOI: https://doi.org/10.1124/dmd.107.019026
W
Wang, Guangji
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Wang, Lifei
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
Watanabe, Akito
- You have accessDown-Regulation of a Hepatic Transporter Multidrug Resistance-Associated Protein 2 Is Involved in Alteration of Pharmacokinetics of Glycyrrhizin and Its Metabolites in a Rat Model of Chronic Liver InjuryToshiaki Makino, Nobuhiro Ohtake, Akito Watanabe, Naoko Tsuchiya, Sachiko Imamura, Seiichi Iizuka, Makoto Inoue and Hajime MizukamiDrug Metabolism and Disposition July 2008, 36 (7) 1438-1443; DOI: https://doi.org/10.1124/dmd.108.021089
Waters, Nigel J.
- You have accessTrend Analysis of a Database of Intravenous Pharmacokinetic Parameters in Humans for 670 Drug CompoundsR. Scott Obach, Franco Lombardo and Nigel J. WatersDrug Metabolism and Disposition July 2008, 36 (7) 1385-1405; DOI: https://doi.org/10.1124/dmd.108.020479
Webborn, Peter J. H.
- You have accessPrediction of the Pharmacokinetics of Atorvastatin, Cerivastatin, and Indomethacin Using Kinetic Models Applied to Isolated Rat HepatocytesStuart W. Paine, Alison J. Parker, Philip Gardiner, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition July 2008, 36 (7) 1365-1374; DOI: https://doi.org/10.1124/dmd.107.019455
Williams, Eric T.
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Wolf, C. Roland
- You have accessFunctional Expression and Comparative Characterization of Nine Murine Cytochromes P450 by Fluorescent Inhibition ScreeningLesley A. McLaughlin, Leslie J. Dickmann, C. Roland Wolf and Colin J. HendersonDrug Metabolism and Disposition July 2008, 36 (7) 1322-1331; DOI: https://doi.org/10.1124/dmd.108.021261
Wrighton, Steven A.
- You have accessThe Biotransformation of Prasugrel, a New Thienopyridine Prodrug, by the Human Carboxylesterases 1 and 2Eric T. Williams, Karen O. Jones, G. Douglas Ponsler, Shane M. Lowery, Everett J. Perkins, Steven A. Wrighton, Kenneth J. Ruterbories, Miho Kazui and Nagy A. FaridDrug Metabolism and Disposition July 2008, 36 (7) 1227-1232; DOI: https://doi.org/10.1124/dmd.107.020248
Wu, Chiyuan
- You have accessMetabolism and Disposition of Dasatinib after Oral Administration to HumansLisa J. Christopher, Donghui Cui, Chiyuan Wu, Roger Luo, James A. Manning, Samuel J. Bonacorsi, Michael Lago, Alban Allentoff, Francis Y. F. Lee, Betty McCann, Susan Galbraith, Donald P. Reitberg, Kan He, Anthony Barros, Anne Blackwood-Chirchir, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1357-1364; DOI: https://doi.org/10.1124/dmd.107.018267
Wu, Ellen Y.
- You have accessDrug Transporter and Cytochrome P450 mRNA Expression in Human Ocular Barriers: Implications for Ocular Drug DispositionTao Zhang, Cathie D. Xiang, David Gale, Samantha Carreiro, Ellen Y. Wu and Eric Y. ZhangDrug Metabolism and Disposition July 2008, 36 (7) 1300-1307; DOI: https://doi.org/10.1124/dmd.108.021121
Wurm, Robert M.
- You have accessAn in Vitro Mechanistic Study to Elucidate the Desipramine/Bupropion Clinical Drug-Drug InteractionMelinda J. Reese, Robert M. Wurm, Keith T. Muir, Grant T. Generaux, Lisa St. John-Williams and Donavon J. McconnDrug Metabolism and Disposition July 2008, 36 (7) 1198-1201; DOI: https://doi.org/10.1124/dmd.107.020198
X
Xiang, Cathie D.
- You have accessDrug Transporter and Cytochrome P450 mRNA Expression in Human Ocular Barriers: Implications for Ocular Drug DispositionTao Zhang, Cathie D. Xiang, David Gale, Samantha Carreiro, Ellen Y. Wu and Eric Y. ZhangDrug Metabolism and Disposition July 2008, 36 (7) 1300-1307; DOI: https://doi.org/10.1124/dmd.108.021121
Y
Yamamoto, Yukio
- You have accessThe Antiapoptotic Factor Growth Arrest and DNA-Damage-Inducible 45 β Regulates the Nuclear Receptor Constitutive Active/Androstane Receptor-Mediated TranscriptionYukio Yamamoto and Masahiko NegishiDrug Metabolism and Disposition July 2008, 36 (7) 1189-1193; DOI: https://doi.org/10.1124/dmd.108.020628
Yamamura, Yoshikazu
- You have accessInhibitory Effects of Terpenoids on Multidrug Resistance-Associated Protein 2- and Breast Cancer Resistance Protein-Mediated TransportNaoko Yoshida, Tappei Takada, Yoshikazu Yamamura, Isao Adachi, Hiroshi Suzuki and Junichi KawakamiDrug Metabolism and Disposition July 2008, 36 (7) 1206-1211; DOI: https://doi.org/10.1124/dmd.107.019513
Yamazaki, Shinji
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
Ye, Zhi-wei
- You have accessCellular Accumulation of Cholyl-Glycylamido-Fluorescein in Sandwich-Cultured Rat Hepatocytes: Kinetic Characterization, Transport Mechanisms, and Effect of Human Immunodeficiency Virus Protease InhibitorsZhi-wei Ye, Patrick Augustijns and Pieter AnnaertDrug Metabolism and Disposition July 2008, 36 (7) 1315-1321; DOI: https://doi.org/10.1124/dmd.107.019398
Yoshida, Naoko
- You have accessInhibitory Effects of Terpenoids on Multidrug Resistance-Associated Protein 2- and Breast Cancer Resistance Protein-Mediated TransportNaoko Yoshida, Tappei Takada, Yoshikazu Yamamura, Isao Adachi, Hiroshi Suzuki and Junichi KawakamiDrug Metabolism and Disposition July 2008, 36 (7) 1206-1211; DOI: https://doi.org/10.1124/dmd.107.019513
Z
Zhang, Donglu
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
Zhang, Eric Y.
- You have accessDrug Transporter and Cytochrome P450 mRNA Expression in Human Ocular Barriers: Implications for Ocular Drug DispositionTao Zhang, Cathie D. Xiang, David Gale, Samantha Carreiro, Ellen Y. Wu and Eric Y. ZhangDrug Metabolism and Disposition July 2008, 36 (7) 1300-1307; DOI: https://doi.org/10.1124/dmd.108.021121
Zhang, Haiying
- You have accessBiotransformation of [14C]Dasatinib: In Vitro Studies in Rat, Monkey, and Human and Disposition after Administration to Rats and MonkeysLisa J. Christopher, Donghui Cui, Wenying Li, Anthony Barros, Vinod K. Arora, Haiying Zhang, Lifei Wang, Donglu Zhang, James A. Manning, Kan He, Anthony M. Fletcher, Marc Ogan, Michael Lago, Samuel J. Bonacorsi, W. Griffith Humphreys and Ramaswamy A. IyerDrug Metabolism and Disposition July 2008, 36 (7) 1341-1356; DOI: https://doi.org/10.1124/dmd.107.018234
Zhang, Rong
- You have accessInhibitory Effects of Seven Components of Danshen Extract on Catalytic Activity of Cytochrome P450 Enzyme in Human Liver MicrosomesFurong Qiu, Rong Zhang, Jianguo Sun, Jiye A, Haiping Hao, Ying Peng, Hua Ai and Guangji WangDrug Metabolism and Disposition July 2008, 36 (7) 1308-1314; DOI: https://doi.org/10.1124/dmd.108.021030
Zhang, Tao
- You have accessDrug Transporter and Cytochrome P450 mRNA Expression in Human Ocular Barriers: Implications for Ocular Drug DispositionTao Zhang, Cathie D. Xiang, David Gale, Samantha Carreiro, Ellen Y. Wu and Eric Y. ZhangDrug Metabolism and Disposition July 2008, 36 (7) 1300-1307; DOI: https://doi.org/10.1124/dmd.108.021121
Zhang, Wenxia
- You have accessEffects of Spice Constituents on P-Glycoprotein-Mediated Transport and CYP3A4-Mediated Metabolism in VitroWenxia Zhang and Lee-Yong LimDrug Metabolism and Disposition July 2008, 36 (7) 1283-1290; DOI: https://doi.org/10.1124/dmd.107.019737
Zhou, Sue
- You have accessBioactivation of Flutamide Metabolites by Human Liver MicrosomesPing Kang, Deepak Dalvie, Evan Smith, Sue Zhou, Alan Deese and James A. NiemanDrug Metabolism and Disposition July 2008, 36 (7) 1425-1437; DOI: https://doi.org/10.1124/dmd.108.020370
Zou, Helen Y.
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Biomarker Response and Tumor Growth Inhibition to an Orally Available cMet Kinase Inhibitor in Human Tumor Xenograft Mouse ModelsShinji Yamazaki, Judith Skaptason, David Romero, Joseph H. Lee, Helen Y. Zou, James G. Christensen, Jeffrey R. Koup, Bill J. Smith and Tatiana KoudriakovaDrug Metabolism and Disposition July 2008, 36 (7) 1267-1274; DOI: https://doi.org/10.1124/dmd.107.019711
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