Index by author
August 01, 2008; Volume 36,Issue 8
A
Abbara, Chadi
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Abel, E. Dale
- You have accessDeletion of the NADPH-Cytochrome P450 Reductase Gene in Cardiomyocytes Does Not Protect Mice against Doxorubicin-Mediated Acute Cardiac ToxicityCheng Fang, Jun Gu, Fang Xie, Melissa Behr, Weizhu Yang, E. Dale Abel and Xinxin DingDrug Metabolism and Disposition August 2008, 36 (8) 1722-1728; DOI: https://doi.org/10.1124/dmd.108.021881
Aidasani, Divesh
- You have accessIn Vitro Drug-Drug Interaction Screens for Canine Veterinary Medicines: Evaluation of Cytochrome P450 Reversible InhibitionDivesh Aidasani, Matthew J. Zaya, Phyllis B. Malpas and Charles W. LocusonDrug Metabolism and Disposition August 2008, 36 (8) 1512-1518; DOI: https://doi.org/10.1124/dmd.108.021196
Aitio, Olli
- You have accessRegio- and Stereospecific N-Glucuronidation of Medetomidine: The Differences between UDP Glucuronosyltransferase (UGT) 1A4 and UGT2B10 Account for the Complex Kinetics of Human Liver MicrosomesSanna Kaivosaari, Päivi Toivonen, Olli Aitio, Julius Sipilä, Mikko Koskinen, Jarmo S. Salonen and Moshe FinelDrug Metabolism and Disposition August 2008, 36 (8) 1529-1537; DOI: https://doi.org/10.1124/dmd.108.021709
Aloysius, Herve A.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Aoki, Toshiko
- You have accessRole of Organic Anion Transporters in the Pharmacokinetics of Zonampanel, an α-Amino-3-hydroxy-5-methylisoxazole-4-propionate Receptor Antagonist, in RatsTsuyoshi Minematsu, Tadashi Hashimoto, Toshiko Aoki, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2008, 36 (8) 1496-1504; DOI: https://doi.org/10.1124/dmd.107.019828
Arison, Byron H.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Augustine, Lisa M.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
B
Baba, Takahiko
- You have accessIdentification of the Transporters Involved in the Hepatobiliary Transport and Intestinal Efflux of Methyl 1-(3,4-Dimethoxyphenyl)-3-(3-ethylvaleryl)-4-hydroxy-6,7,8-trimethoxy-2-naphthoate (S-8921) Glucuronide, a Pharmacologically Active Metabolite of S-8921Shingo Sakamoto, Hiroyuki Kusuhara, Kazutoshi Horie, Kohji Takahashi, Takahiko Baba, Jun Ishizaki and Yuichi SugiyamaDrug Metabolism and Disposition August 2008, 36 (8) 1553-1561; DOI: https://doi.org/10.1124/dmd.108.020511
Bachmann, Kenneth
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Bae, Soo Kyung
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Behr, Melissa
- You have accessDeletion of the NADPH-Cytochrome P450 Reductase Gene in Cardiomyocytes Does Not Protect Mice against Doxorubicin-Mediated Acute Cardiac ToxicityCheng Fang, Jun Gu, Fang Xie, Melissa Behr, Weizhu Yang, E. Dale Abel and Xinxin DingDrug Metabolism and Disposition August 2008, 36 (8) 1722-1728; DOI: https://doi.org/10.1124/dmd.108.021881
Beijnen, Jos H.
- You have accessExtensive Metabolism and Hepatic Accumulation of Gemcitabine After Multiple Oral and Intravenous Administration in MiceStephan A. Veltkamp, Dick Pluim, Olaf van Tellingen, Jos H. Beijnen and Jan H. M. SchellensDrug Metabolism and Disposition August 2008, 36 (8) 1606-1615; DOI: https://doi.org/10.1124/dmd.108.021048
Besnard, Madeleine
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Blizzard, Timothy A.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Boldt, Sherri
- You have accessA Combined Model for Predicting CYP3A4 Clinical Net Drug-Drug Interaction Based on CYP3A4 Inhibition, Inactivation, and Induction Determined in VitroOdette A. Fahmi, Tristan S. Maurer, Mary Kish, Edwin Cardenas, Sherri Boldt and David NettletonDrug Metabolism and Disposition August 2008, 36 (8) 1698-1708; DOI: https://doi.org/10.1124/dmd.107.018663
Bonhomme-Faivre, Laurence
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Bourasset, Fanchon
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Bourdet, David L.
- You have accessMechanisms Underlying Saturable Intestinal Absorption of MetforminWilliam R. Proctor, David L. Bourdet and Dhiren R. ThakkerDrug Metabolism and Disposition August 2008, 36 (8) 1650-1658; DOI: https://doi.org/10.1124/dmd.107.020180
C
Callery, Patrick S.
- You have accessMetabolism of the Cysteine S-Conjugate of Busulfan Involves a β-Lyase ReactionArthur J. L. Cooper, Islam R. Younis, Zoya V. Niatsetskaya, Boris F. Krasnikov, John T. Pinto, William P. Petros and Patrick S. CalleryDrug Metabolism and Disposition August 2008, 36 (8) 1546-1552; DOI: https://doi.org/10.1124/dmd.108.020768
Cao, Shan
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Cardenas, Edwin
- You have accessA Combined Model for Predicting CYP3A4 Clinical Net Drug-Drug Interaction Based on CYP3A4 Inhibition, Inactivation, and Induction Determined in VitroOdette A. Fahmi, Tristan S. Maurer, Mary Kish, Edwin Cardenas, Sherri Boldt and David NettletonDrug Metabolism and Disposition August 2008, 36 (8) 1698-1708; DOI: https://doi.org/10.1124/dmd.107.018663
Cashman, John R.
- You have accessCurcuminoids Inhibit Multiple Human Cytochromes P450, UDP-Glucuronosyltransferase, and Sulfotransferase Enzymes, whereas Piperine Is a Relatively Selective CYP3A4 InhibitorLaurie P. Volak, Senait Ghirmai, John R. Cashman and Michael H. CourtDrug Metabolism and Disposition August 2008, 36 (8) 1594-1605; DOI: https://doi.org/10.1124/dmd.108.020552
Chacun, Helène
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Chen, Hao
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Chen, Ping
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Chen, Yao
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Cherrington, Nathan J.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Chupka, Jonathan
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Cintrat, Jean-Christophe
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Clogston, Jeffrey D.
- You have accessRapid Distribution of Liposomal Short-Chain Ceramide in Vitro and in VivoBanu S. Zolnik, Stephan T. Stern, James M. Kaiser, Yasser Heakal, Jeffrey D. Clogston, Mark Kester and Scott E. McNeilDrug Metabolism and Disposition August 2008, 36 (8) 1709-1715; DOI: https://doi.org/10.1124/dmd.107.019679
Cooper, Arthur J. L.
- You have accessMetabolism of the Cysteine S-Conjugate of Busulfan Involves a β-Lyase ReactionArthur J. L. Cooper, Islam R. Younis, Zoya V. Niatsetskaya, Boris F. Krasnikov, John T. Pinto, William P. Petros and Patrick S. CalleryDrug Metabolism and Disposition August 2008, 36 (8) 1546-1552; DOI: https://doi.org/10.1124/dmd.108.020768
Correia, Maria Almira
- You have accessPathways of Carbamazepine Bioactivation in Vitro. III. The Role of Human Cytochrome P450 Enzymes in the Formation of 2,3-DihydroxycarbamazepineRobin E. Pearce, Wei Lu, YongQiang Wang, Jack P. Uetrecht, Maria Almira Correia and J. Steven LeederDrug Metabolism and Disposition August 2008, 36 (8) 1637-1649; DOI: https://doi.org/10.1124/dmd.107.019562
Court, Michael H.
- You have accessCurcuminoids Inhibit Multiple Human Cytochromes P450, UDP-Glucuronosyltransferase, and Sulfotransferase Enzymes, whereas Piperine Is a Relatively Selective CYP3A4 InhibitorLaurie P. Volak, Senait Ghirmai, John R. Cashman and Michael H. CourtDrug Metabolism and Disposition August 2008, 36 (8) 1594-1605; DOI: https://doi.org/10.1124/dmd.108.020552
Couvreur, Patrick
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
D
Dannecker, Robert
- You have accessThe Macrolide Everolimus Forms an Unusual Metabolite in Animals and Humans: Identification of a Phosphocholine EsterMarkus Zollinger, Claudia Sayer, Robert Dannecker, Walter Schuler and Richard SedraniDrug Metabolism and Disposition August 2008, 36 (8) 1457-1460; DOI: https://doi.org/10.1124/dmd.108.020651
Dauvin, Angélique
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Declèves, Xavier
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Deroussent, Alain
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Desmaële, Didier
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Ding, Xinxin
- You have accessDeletion of the NADPH-Cytochrome P450 Reductase Gene in Cardiomyocytes Does Not Protect Mice against Doxorubicin-Mediated Acute Cardiac ToxicityCheng Fang, Jun Gu, Fang Xie, Melissa Behr, Weizhu Yang, E. Dale Abel and Xinxin DingDrug Metabolism and Disposition August 2008, 36 (8) 1722-1728; DOI: https://doi.org/10.1124/dmd.108.021881
Divakaran, Karthika
- You have accessDevelopmental Changes in Human Liver CYP2D6 ExpressionJeffrey C. Stevens, Sandra A. Marsh, Matthew J. Zaya, Karen J. Regina, Karthika Divakaran, Min Le and Ronald N. HinesDrug Metabolism and Disposition August 2008, 36 (8) 1587-1593; DOI: https://doi.org/10.1124/dmd.108.021873
Du, Feifei
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Duan, Jian-Dong
- You have accessAssessment of the Medicines Lidocaine, Prilocaine, and Their Metabolites, 2,6-Dimethylaniline and 2-Methylaniline, for DNA Adduct Formation in Rat TissuesJian-Dong Duan, Alan M. Jeffrey and Gary M. WilliamsDrug Metabolism and Disposition August 2008, 36 (8) 1470-1475; DOI: https://doi.org/10.1124/dmd.107.019950
Dubernet, Catherine
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
E
Ekins, Sean
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Elipe, Maria V. Silva
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Elmquist, William F.
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
Eriksson, Ulf G.
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
F
Faetkenheuer, Gerd
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
Fahmi, Odette A.
- You have accessA Combined Model for Predicting CYP3A4 Clinical Net Drug-Drug Interaction Based on CYP3A4 Inhibition, Inactivation, and Induction Determined in VitroOdette A. Fahmi, Tristan S. Maurer, Mary Kish, Edwin Cardenas, Sherri Boldt and David NettletonDrug Metabolism and Disposition August 2008, 36 (8) 1698-1708; DOI: https://doi.org/10.1124/dmd.107.018663
Faidley, Terry D.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Fang, Cheng
- You have accessDeletion of the NADPH-Cytochrome P450 Reductase Gene in Cardiomyocytes Does Not Protect Mice against Doxorubicin-Mediated Acute Cardiac ToxicityCheng Fang, Jun Gu, Fang Xie, Melissa Behr, Weizhu Yang, E. Dale Abel and Xinxin DingDrug Metabolism and Disposition August 2008, 36 (8) 1722-1728; DOI: https://doi.org/10.1124/dmd.108.021881
Farinotti, Robert
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Ferreira, Humberto
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Finel, Moshe
- You have accessRegio- and Stereospecific N-Glucuronidation of Medetomidine: The Differences between UDP Glucuronosyltransferase (UGT) 1A4 and UGT2B10 Account for the Complex Kinetics of Human Liver MicrosomesSanna Kaivosaari, Päivi Toivonen, Olli Aitio, Julius Sipilä, Mikko Koskinen, Jarmo S. Salonen and Moshe FinelDrug Metabolism and Disposition August 2008, 36 (8) 1529-1537; DOI: https://doi.org/10.1124/dmd.108.021709
Fisher, Craig D.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Forsell, Patrik
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
Freudenthaler, Stefan
- You have accessEffects of Ketoconazole and Quinidine on Pharmacokinetics of Pactimibe and Its Plasma Metabolite, R-125528, in HumansMasakatsu Kotsuma, Taro Tokui, Stefan Freudenthaler and Kenji NishimuraDrug Metabolism and Disposition August 2008, 36 (8) 1505-1511; DOI: https://doi.org/10.1124/dmd.108.021394
Fritsch, Holger
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
Fujiwara, Ryoichi
- You have accessExpression of UGT1A and UGT2B mRNA in Human Normal Tissues and Various Cell LinesAkiko Nakamura, Miki Nakajima, Hiroyuki Yamanaka, Ryoichi Fujiwara and Tsuyoshi YokoiDrug Metabolism and Disposition August 2008, 36 (8) 1461-1464; DOI: https://doi.org/10.1124/dmd.108.021428
Furuta, Takashi
- You have accessPlasma Profiling of Intact Isoflavone Metabolites by High-Performance Liquid Chromatography and Mass Spectrometric Identification of Flavone Glycosides Daidzin and Genistin in Human Plasma after Administration of KinakoKaori Hosoda, Takashi Furuta, Akitomo Yokokawa, Kenichiro Ogura, Akira Hiratsuka and Kazuo IshiiDrug Metabolism and Disposition August 2008, 36 (8) 1485-1495; DOI: https://doi.org/10.1124/dmd.108.021006
G
Gao, Xiumei
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Ghirmai, Senait
- You have accessCurcuminoids Inhibit Multiple Human Cytochromes P450, UDP-Glucuronosyltransferase, and Sulfotransferase Enzymes, whereas Piperine Is a Relatively Selective CYP3A4 InhibitorLaurie P. Volak, Senait Ghirmai, John R. Cashman and Michael H. CourtDrug Metabolism and Disposition August 2008, 36 (8) 1594-1605; DOI: https://doi.org/10.1124/dmd.108.020552
Giri, Nagdeep
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
Gonin, Patrick
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Grime, Ken
- You have accessFunctional Consequences of Active Hepatic Uptake on Cytochrome P450 Inhibition in Rat and Human HepatocytesKen Grime, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition August 2008, 36 (8) 1670-1678; DOI: https://doi.org/10.1124/dmd.108.021055
Gu, Jun
- You have accessDeletion of the NADPH-Cytochrome P450 Reductase Gene in Cardiomyocytes Does Not Protect Mice against Doxorubicin-Mediated Acute Cardiac ToxicityCheng Fang, Jun Gu, Fang Xie, Melissa Behr, Weizhu Yang, E. Dale Abel and Xinxin DingDrug Metabolism and Disposition August 2008, 36 (8) 1722-1728; DOI: https://doi.org/10.1124/dmd.108.021881
Guo, Dong
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
H
Hartmann, Pia
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
Hashimoto, Tadashi
- You have accessRole of Organic Anion Transporters in the Pharmacokinetics of Zonampanel, an α-Amino-3-hydroxy-5-methylisoxazole-4-propionate Receptor Antagonist, in RatsTsuyoshi Minematsu, Tadashi Hashimoto, Toshiko Aoki, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2008, 36 (8) 1496-1504; DOI: https://doi.org/10.1124/dmd.107.019828
Hawke, Roy L.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
He, Yi-Jing
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Heakal, Yasser
- You have accessRapid Distribution of Liposomal Short-Chain Ceramide in Vitro and in VivoBanu S. Zolnik, Stephan T. Stern, James M. Kaiser, Yasser Heakal, Jeffrey D. Clogston, Mark Kester and Scott E. McNeilDrug Metabolism and Disposition August 2008, 36 (8) 1709-1715; DOI: https://doi.org/10.1124/dmd.107.019679
Hines, Ronald N.
- You have accessDevelopmental Changes in Human Liver CYP2D6 ExpressionJeffrey C. Stevens, Sandra A. Marsh, Matthew J. Zaya, Karen J. Regina, Karthika Divakaran, Min Le and Ronald N. HinesDrug Metabolism and Disposition August 2008, 36 (8) 1587-1593; DOI: https://doi.org/10.1124/dmd.108.021873
Hiratsuka, Akira
- You have accessPlasma Profiling of Intact Isoflavone Metabolites by High-Performance Liquid Chromatography and Mass Spectrometric Identification of Flavone Glycosides Daidzin and Genistin in Human Plasma after Administration of KinakoKaori Hosoda, Takashi Furuta, Akitomo Yokokawa, Kenichiro Ogura, Akira Hiratsuka and Kazuo IshiiDrug Metabolism and Disposition August 2008, 36 (8) 1485-1495; DOI: https://doi.org/10.1124/dmd.108.021006
Horie, Kazutoshi
- You have accessIdentification of the Transporters Involved in the Hepatobiliary Transport and Intestinal Efflux of Methyl 1-(3,4-Dimethoxyphenyl)-3-(3-ethylvaleryl)-4-hydroxy-6,7,8-trimethoxy-2-naphthoate (S-8921) Glucuronide, a Pharmacologically Active Metabolite of S-8921Shingo Sakamoto, Hiroyuki Kusuhara, Kazutoshi Horie, Kohji Takahashi, Takahiko Baba, Jun Ishizaki and Yuichi SugiyamaDrug Metabolism and Disposition August 2008, 36 (8) 1553-1561; DOI: https://doi.org/10.1124/dmd.108.020511
Hosoda, Kaori
- You have accessPlasma Profiling of Intact Isoflavone Metabolites by High-Performance Liquid Chromatography and Mass Spectrometric Identification of Flavone Glycosides Daidzin and Genistin in Human Plasma after Administration of KinakoKaori Hosoda, Takashi Furuta, Akitomo Yokokawa, Kenichiro Ogura, Akira Hiratsuka and Kazuo IshiiDrug Metabolism and Disposition August 2008, 36 (8) 1485-1495; DOI: https://doi.org/10.1124/dmd.108.021006
Hosten, Benoît
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Hu, Dong-Li
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Huang, Wendong
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Huang, Yuhong
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
I
Ishii, Kazuo
- You have accessPlasma Profiling of Intact Isoflavone Metabolites by High-Performance Liquid Chromatography and Mass Spectrometric Identification of Flavone Glycosides Daidzin and Genistin in Human Plasma after Administration of KinakoKaori Hosoda, Takashi Furuta, Akitomo Yokokawa, Kenichiro Ogura, Akira Hiratsuka and Kazuo IshiiDrug Metabolism and Disposition August 2008, 36 (8) 1485-1495; DOI: https://doi.org/10.1124/dmd.108.021006
Ishizaki, Jun
- You have accessIdentification of the Transporters Involved in the Hepatobiliary Transport and Intestinal Efflux of Methyl 1-(3,4-Dimethoxyphenyl)-3-(3-ethylvaleryl)-4-hydroxy-6,7,8-trimethoxy-2-naphthoate (S-8921) Glucuronide, a Pharmacologically Active Metabolite of S-8921Shingo Sakamoto, Hiroyuki Kusuhara, Kazutoshi Horie, Kohji Takahashi, Takahiko Baba, Jun Ishizaki and Yuichi SugiyamaDrug Metabolism and Disposition August 2008, 36 (8) 1553-1561; DOI: https://doi.org/10.1124/dmd.108.020511
J
Jackson, Jonathan P.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Jeffrey, Alan M.
- You have accessAssessment of the Medicines Lidocaine, Prilocaine, and Their Metabolites, 2,6-Dimethylaniline and 2-Methylaniline, for DNA Adduct Formation in Rat TissuesJian-Dong Duan, Alan M. Jeffrey and Gary M. WilliamsDrug Metabolism and Disposition August 2008, 36 (8) 1470-1475; DOI: https://doi.org/10.1124/dmd.107.019950
Jung, Norma
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
K
Kaiser, James M.
- You have accessRapid Distribution of Liposomal Short-Chain Ceramide in Vitro and in VivoBanu S. Zolnik, Stephan T. Stern, James M. Kaiser, Yasser Heakal, Jeffrey D. Clogston, Mark Kester and Scott E. McNeilDrug Metabolism and Disposition August 2008, 36 (8) 1709-1715; DOI: https://doi.org/10.1124/dmd.107.019679
Kaivosaari, Sanna
- You have accessRegio- and Stereospecific N-Glucuronidation of Medetomidine: The Differences between UDP Glucuronosyltransferase (UGT) 1A4 and UGT2B10 Account for the Complex Kinetics of Human Liver MicrosomesSanna Kaivosaari, Päivi Toivonen, Olli Aitio, Julius Sipilä, Mikko Koskinen, Jarmo S. Salonen and Moshe FinelDrug Metabolism and Disposition August 2008, 36 (8) 1529-1537; DOI: https://doi.org/10.1124/dmd.108.021709
Kamimura, Hidetaka
- You have accessRole of Organic Anion Transporters in the Pharmacokinetics of Zonampanel, an α-Amino-3-hydroxy-5-methylisoxazole-4-propionate Receptor Antagonist, in RatsTsuyoshi Minematsu, Tadashi Hashimoto, Toshiko Aoki, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2008, 36 (8) 1496-1504; DOI: https://doi.org/10.1124/dmd.107.019828
Kashuba, Angela D. M.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Kester, Mark
- You have accessRapid Distribution of Liposomal Short-Chain Ceramide in Vitro and in VivoBanu S. Zolnik, Stephan T. Stern, James M. Kaiser, Yasser Heakal, Jeffrey D. Clogston, Mark Kester and Scott E. McNeilDrug Metabolism and Disposition August 2008, 36 (8) 1709-1715; DOI: https://doi.org/10.1124/dmd.107.019679
Khoury, Hania
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Kim, Hyunmi
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Kim, Min-Jung
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Kirchheiner, Julia
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Kish, Mary
- You have accessA Combined Model for Predicting CYP3A4 Clinical Net Drug-Drug Interaction Based on CYP3A4 Inhibition, Inactivation, and Induction Determined in VitroOdette A. Fahmi, Tristan S. Maurer, Mary Kish, Edwin Cardenas, Sherri Boldt and David NettletonDrug Metabolism and Disposition August 2008, 36 (8) 1698-1708; DOI: https://doi.org/10.1124/dmd.107.018663
Kitagaki, Shinji
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
Klaassen, Curtis D.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Knispel, Meike
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
Knutson, Lars
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
Koskinen, Mikko
- You have accessRegio- and Stereospecific N-Glucuronidation of Medetomidine: The Differences between UDP Glucuronosyltransferase (UGT) 1A4 and UGT2B10 Account for the Complex Kinetics of Human Liver MicrosomesSanna Kaivosaari, Päivi Toivonen, Olli Aitio, Julius Sipilä, Mikko Koskinen, Jarmo S. Salonen and Moshe FinelDrug Metabolism and Disposition August 2008, 36 (8) 1529-1537; DOI: https://doi.org/10.1124/dmd.108.021709
Kotsuma, Masakatsu
- You have accessEffects of Ketoconazole and Quinidine on Pharmacokinetics of Pactimibe and Its Plasma Metabolite, R-125528, in HumansMasakatsu Kotsuma, Taro Tokui, Stefan Freudenthaler and Kenji NishimuraDrug Metabolism and Disposition August 2008, 36 (8) 1505-1511; DOI: https://doi.org/10.1124/dmd.108.021394
Krasnikov, Boris F.
- You have accessMetabolism of the Cysteine S-Conjugate of Busulfan Involves a β-Lyase ReactionArthur J. L. Cooper, Islam R. Younis, Zoya V. Niatsetskaya, Boris F. Krasnikov, John T. Pinto, William P. Petros and Patrick S. CalleryDrug Metabolism and Disposition August 2008, 36 (8) 1546-1552; DOI: https://doi.org/10.1124/dmd.108.020768
Kusuhara, Hiroyuki
- You have accessIdentification of the Transporters Involved in the Hepatobiliary Transport and Intestinal Efflux of Methyl 1-(3,4-Dimethoxyphenyl)-3-(3-ethylvaleryl)-4-hydroxy-6,7,8-trimethoxy-2-naphthoate (S-8921) Glucuronide, a Pharmacologically Active Metabolite of S-8921Shingo Sakamoto, Hiroyuki Kusuhara, Kazutoshi Horie, Kohji Takahashi, Takahiko Baba, Jun Ishizaki and Yuichi SugiyamaDrug Metabolism and Disposition August 2008, 36 (8) 1553-1561; DOI: https://doi.org/10.1124/dmd.108.020511
L
Lamba, Jatinder K.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Laugier, Christelle
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Le, Min
- You have accessDevelopmental Changes in Human Liver CYP2D6 ExpressionJeffrey C. Stevens, Sandra A. Marsh, Matthew J. Zaya, Karen J. Regina, Karthika Divakaran, Min Le and Ronald N. HinesDrug Metabolism and Disposition August 2008, 36 (8) 1587-1593; DOI: https://doi.org/10.1124/dmd.108.021873
Leeder, J. Steven
- You have accessPathways of Carbamazepine Bioactivation in Vitro. III. The Role of Human Cytochrome P450 Enzymes in the Formation of 2,3-DihydroxycarbamazepineRobin E. Pearce, Wei Lu, YongQiang Wang, Jack P. Uetrecht, Maria Almira Correia and J. Steven LeederDrug Metabolism and Disposition August 2008, 36 (8) 1637-1649; DOI: https://doi.org/10.1124/dmd.107.019562
Lehmann, Clara
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
Lennernäs, Hans
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
Lepêtre-Mouelhi, Sinda
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Li, Chuan
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Li, Qing
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Li, Wei
- You have accessUDP-Glucuronosyltransferase 1A6 Is the Major Isozyme Responsible for Protocatechuic Aldehyde Glucuronidation in Human Liver MicrosomesHui-Xin Liu, Yong Liu, Jiang-Wei Zhang, Wei Li, Hong-Tao Liu and Ling YangDrug Metabolism and Disposition August 2008, 36 (8) 1562-1569; DOI: https://doi.org/10.1124/dmd.108.020560
Li, Zhong-Yu
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Lichti-Kaiser, Kristin
- You have accessThe Traditional Chinese Herbal Remedy Tian Xian Activates Pregnane X Receptor and Induces CYP3A Gene Expression in HepatocytesKristin Lichti-Kaiser and Jeff L. StaudingerDrug Metabolism and Disposition August 2008, 36 (8) 1538-1545; DOI: https://doi.org/10.1124/dmd.108.021774
Liu, Changxiao
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Liu, Hong-Tao
- You have accessUDP-Glucuronosyltransferase 1A6 Is the Major Isozyme Responsible for Protocatechuic Aldehyde Glucuronidation in Human Liver MicrosomesHui-Xin Liu, Yong Liu, Jiang-Wei Zhang, Wei Li, Hong-Tao Liu and Ling YangDrug Metabolism and Disposition August 2008, 36 (8) 1562-1569; DOI: https://doi.org/10.1124/dmd.108.020560
Liu, Hui-Xin
- You have accessUDP-Glucuronosyltransferase 1A6 Is the Major Isozyme Responsible for Protocatechuic Aldehyde Glucuronidation in Human Liver MicrosomesHui-Xin Liu, Yong Liu, Jiang-Wei Zhang, Wei Li, Hong-Tao Liu and Ling YangDrug Metabolism and Disposition August 2008, 36 (8) 1562-1569; DOI: https://doi.org/10.1124/dmd.108.020560
Liu, Kwang-Hyeon
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Liu, Yong
- You have accessUDP-Glucuronosyltransferase 1A6 Is the Major Isozyme Responsible for Protocatechuic Aldehyde Glucuronidation in Human Liver MicrosomesHui-Xin Liu, Yong Liu, Jiang-Wei Zhang, Wei Li, Hong-Tao Liu and Ling YangDrug Metabolism and Disposition August 2008, 36 (8) 1562-1569; DOI: https://doi.org/10.1124/dmd.108.020560
Locuson, Charles W.
- You have accessIn Vitro Drug-Drug Interaction Screens for Canine Veterinary Medicines: Evaluation of Cytochrome P450 Reversible InhibitionDivesh Aidasani, Matthew J. Zaya, Phyllis B. Malpas and Charles W. LocusonDrug Metabolism and Disposition August 2008, 36 (8) 1512-1518; DOI: https://doi.org/10.1124/dmd.108.021196
Logren, Ulrika
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
Lu, Tong
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Lu, Wei
- You have accessPeroxidase-Mediated Bioactivation of Hydroxylated Metabolites of Carbamazepine and PhenytoinWei Lu and Jack P. UetrechtDrug Metabolism and Disposition August 2008, 36 (8) 1624-1636; DOI: https://doi.org/10.1124/dmd.107.019554
- You have accessPathways of Carbamazepine Bioactivation in Vitro. III. The Role of Human Cytochrome P450 Enzymes in the Formation of 2,3-DihydroxycarbamazepineRobin E. Pearce, Wei Lu, YongQiang Wang, Jack P. Uetrecht, Maria Almira Correia and J. Steven LeederDrug Metabolism and Disposition August 2008, 36 (8) 1637-1649; DOI: https://doi.org/10.1124/dmd.107.019562
M
Maher, Jonathan M.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Malpas, Phyllis B.
- You have accessIn Vitro Drug-Drug Interaction Screens for Canine Veterinary Medicines: Evaluation of Cytochrome P450 Reversible InhibitionDivesh Aidasani, Matthew J. Zaya, Phyllis B. Malpas and Charles W. LocusonDrug Metabolism and Disposition August 2008, 36 (8) 1512-1518; DOI: https://doi.org/10.1124/dmd.108.021196
Marsh, Sandra A.
- You have accessDevelopmental Changes in Human Liver CYP2D6 ExpressionJeffrey C. Stevens, Sandra A. Marsh, Matthew J. Zaya, Karen J. Regina, Karthika Divakaran, Min Le and Ronald N. HinesDrug Metabolism and Disposition August 2008, 36 (8) 1587-1593; DOI: https://doi.org/10.1124/dmd.108.021873
Maurer, Tristan S.
- You have accessA Combined Model for Predicting CYP3A4 Clinical Net Drug-Drug Interaction Based on CYP3A4 Inhibition, Inactivation, and Induction Determined in VitroOdette A. Fahmi, Tristan S. Maurer, Mary Kish, Edwin Cardenas, Sherri Boldt and David NettletonDrug Metabolism and Disposition August 2008, 36 (8) 1698-1708; DOI: https://doi.org/10.1124/dmd.107.018663
McNeil, Scott E.
- You have accessRapid Distribution of Liposomal Short-Chain Ceramide in Vitro and in VivoBanu S. Zolnik, Stephan T. Stern, James M. Kaiser, Yasser Heakal, Jeffrey D. Clogston, Mark Kester and Scott E. McNeilDrug Metabolism and Disposition August 2008, 36 (8) 1709-1715; DOI: https://doi.org/10.1124/dmd.107.019679
Merrell, Matthew D.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Michael, Bruce F.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Minematsu, Tsuyoshi
- You have accessRole of Organic Anion Transporters in the Pharmacokinetics of Zonampanel, an α-Amino-3-hydroxy-5-methylisoxazole-4-propionate Receptor Antagonist, in RatsTsuyoshi Minematsu, Tadashi Hashimoto, Toshiko Aoki, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2008, 36 (8) 1496-1504; DOI: https://doi.org/10.1124/dmd.107.019828
Miyakoshi, Naoki
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
Moore, David D.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Moran, Cassandra
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Mukai, Chisato
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
N
Nakajima, Miki
- You have accessExpression of UGT1A and UGT2B mRNA in Human Normal Tissues and Various Cell LinesAkiko Nakamura, Miki Nakajima, Hiroyuki Yamanaka, Ryoichi Fujiwara and Tsuyoshi YokoiDrug Metabolism and Disposition August 2008, 36 (8) 1461-1464; DOI: https://doi.org/10.1124/dmd.108.021428
Nakamura, Akiko
- You have accessExpression of UGT1A and UGT2B mRNA in Human Normal Tissues and Various Cell LinesAkiko Nakamura, Miki Nakajima, Hiroyuki Yamanaka, Ryoichi Fujiwara and Tsuyoshi YokoiDrug Metabolism and Disposition August 2008, 36 (8) 1461-1464; DOI: https://doi.org/10.1124/dmd.108.021428
Nelsen, Andrew C.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Nettleton, David
- You have accessA Combined Model for Predicting CYP3A4 Clinical Net Drug-Drug Interaction Based on CYP3A4 Inhibition, Inactivation, and Induction Determined in VitroOdette A. Fahmi, Tristan S. Maurer, Mary Kish, Edwin Cardenas, Sherri Boldt and David NettletonDrug Metabolism and Disposition August 2008, 36 (8) 1698-1708; DOI: https://doi.org/10.1124/dmd.107.018663
Niatsetskaya, Zoya V.
- You have accessMetabolism of the Cysteine S-Conjugate of Busulfan Involves a β-Lyase ReactionArthur J. L. Cooper, Islam R. Younis, Zoya V. Niatsetskaya, Boris F. Krasnikov, John T. Pinto, William P. Petros and Patrick S. CalleryDrug Metabolism and Disposition August 2008, 36 (8) 1546-1552; DOI: https://doi.org/10.1124/dmd.108.020768
Nishimura, Kenji
- You have accessEffects of Ketoconazole and Quinidine on Pharmacokinetics of Pactimibe and Its Plasma Metabolite, R-125528, in HumansMasakatsu Kotsuma, Taro Tokui, Stefan Freudenthaler and Kenji NishimuraDrug Metabolism and Disposition August 2008, 36 (8) 1505-1511; DOI: https://doi.org/10.1124/dmd.108.021394
Nordgren, Anders
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
O
Ogura, Kenichiro
- You have accessPlasma Profiling of Intact Isoflavone Metabolites by High-Performance Liquid Chromatography and Mass Spectrometric Identification of Flavone Glycosides Daidzin and Genistin in Human Plasma after Administration of KinakoKaori Hosoda, Takashi Furuta, Akitomo Yokokawa, Kenichiro Ogura, Akira Hiratsuka and Kazuo IshiiDrug Metabolism and Disposition August 2008, 36 (8) 1485-1495; DOI: https://doi.org/10.1124/dmd.108.021006
P
Paci, Angelo
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Paine, Mary F.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Pan, Guoyu
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
Pearce, Robin E.
- You have accessPathways of Carbamazepine Bioactivation in Vitro. III. The Role of Human Cytochrome P450 Enzymes in the Formation of 2,3-DihydroxycarbamazepineRobin E. Pearce, Wei Lu, YongQiang Wang, Jack P. Uetrecht, Maria Almira Correia and J. Steven LeederDrug Metabolism and Disposition August 2008, 36 (8) 1637-1649; DOI: https://doi.org/10.1124/dmd.107.019562
Petit, Benoît
- You have accessEffect of Interleukin-2 Pretreatment on Paclitaxel Absorption and Tissue Disposition after Oral and Intravenous Administration in MiceBenoît Hosten, Chadi Abbara, Benoît Petit, Angélique Dauvin, Fanchon Bourasset, Robert Farinotti, Patrick Gonin and Laurence Bonhomme-FaivreDrug Metabolism and Disposition August 2008, 36 (8) 1729-1735; DOI: https://doi.org/10.1124/dmd.107.019091
Petros, William P.
- You have accessMetabolism of the Cysteine S-Conjugate of Busulfan Involves a β-Lyase ReactionArthur J. L. Cooper, Islam R. Younis, Zoya V. Niatsetskaya, Boris F. Krasnikov, John T. Pinto, William P. Petros and Patrick S. CalleryDrug Metabolism and Disposition August 2008, 36 (8) 1546-1552; DOI: https://doi.org/10.1124/dmd.108.020768
Pinto, John T.
- You have accessMetabolism of the Cysteine S-Conjugate of Busulfan Involves a β-Lyase ReactionArthur J. L. Cooper, Islam R. Younis, Zoya V. Niatsetskaya, Boris F. Krasnikov, John T. Pinto, William P. Petros and Patrick S. CalleryDrug Metabolism and Disposition August 2008, 36 (8) 1546-1552; DOI: https://doi.org/10.1124/dmd.108.020768
Pluim, Dick
- You have accessExtensive Metabolism and Hepatic Accumulation of Gemcitabine After Multiple Oral and Intravenous Administration in MiceStephan A. Veltkamp, Dick Pluim, Olaf van Tellingen, Jos H. Beijnen and Jan H. M. SchellensDrug Metabolism and Disposition August 2008, 36 (8) 1606-1615; DOI: https://doi.org/10.1124/dmd.108.021048
Proctor, William R.
- You have accessMechanisms Underlying Saturable Intestinal Absorption of MetforminWilliam R. Proctor, David L. Bourdet and Dhiren R. ThakkerDrug Metabolism and Disposition August 2008, 36 (8) 1650-1658; DOI: https://doi.org/10.1124/dmd.107.020180
R
Ranade, Aarati
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Reddy, L. Harivardhan
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Regina, Karen J.
- You have accessDevelopmental Changes in Human Liver CYP2D6 ExpressionJeffrey C. Stevens, Sandra A. Marsh, Matthew J. Zaya, Karen J. Regina, Karthika Divakaran, Min Le and Ronald N. HinesDrug Metabolism and Disposition August 2008, 36 (8) 1587-1593; DOI: https://doi.org/10.1124/dmd.108.021873
Riley, Robert J.
- You have accessFunctional Consequences of Active Hepatic Uptake on Cytochrome P450 Inhibition in Rat and Human HepatocytesKen Grime, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition August 2008, 36 (8) 1670-1678; DOI: https://doi.org/10.1124/dmd.108.021055
Roberts, Patrick J.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Rollins, Kristan D.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Rousseau, Bernard
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Rubbert, Andrea
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
S
Sakamoto, Shingo
- You have accessIdentification of the Transporters Involved in the Hepatobiliary Transport and Intestinal Efflux of Methyl 1-(3,4-Dimethoxyphenyl)-3-(3-ethylvaleryl)-4-hydroxy-6,7,8-trimethoxy-2-naphthoate (S-8921) Glucuronide, a Pharmacologically Active Metabolite of S-8921Shingo Sakamoto, Hiroyuki Kusuhara, Kazutoshi Horie, Kohji Takahashi, Takahiko Baba, Jun Ishizaki and Yuichi SugiyamaDrug Metabolism and Disposition August 2008, 36 (8) 1553-1561; DOI: https://doi.org/10.1124/dmd.108.020511
Salonen, Jarmo S.
- You have accessRegio- and Stereospecific N-Glucuronidation of Medetomidine: The Differences between UDP Glucuronosyltransferase (UGT) 1A4 and UGT2B10 Account for the Complex Kinetics of Human Liver MicrosomesSanna Kaivosaari, Päivi Toivonen, Olli Aitio, Julius Sipilä, Mikko Koskinen, Jarmo S. Salonen and Moshe FinelDrug Metabolism and Disposition August 2008, 36 (8) 1529-1537; DOI: https://doi.org/10.1124/dmd.108.021709
Sayer, Claudia
- You have accessThe Macrolide Everolimus Forms an Unusual Metabolite in Animals and Humans: Identification of a Phosphocholine EsterMarkus Zollinger, Claudia Sayer, Robert Dannecker, Walter Schuler and Richard SedraniDrug Metabolism and Disposition August 2008, 36 (8) 1457-1460; DOI: https://doi.org/10.1124/dmd.108.020651
Schellens, Jan H. M.
- You have accessExtensive Metabolism and Hepatic Accumulation of Gemcitabine After Multiple Oral and Intravenous Administration in MiceStephan A. Veltkamp, Dick Pluim, Olaf van Tellingen, Jos H. Beijnen and Jan H. M. SchellensDrug Metabolism and Disposition August 2008, 36 (8) 1606-1615; DOI: https://doi.org/10.1124/dmd.108.021048
Schuetz, Erin
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Schuetz, Erin G.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Schuler, Walter
- You have accessThe Macrolide Everolimus Forms an Unusual Metabolite in Animals and Humans: Identification of a Phosphocholine EsterMarkus Zollinger, Claudia Sayer, Robert Dannecker, Walter Schuler and Richard SedraniDrug Metabolism and Disposition August 2008, 36 (8) 1457-1460; DOI: https://doi.org/10.1124/dmd.108.020651
Sedrani, Richard
- You have accessThe Macrolide Everolimus Forms an Unusual Metabolite in Animals and Humans: Identification of a Phosphocholine EsterMarkus Zollinger, Claudia Sayer, Robert Dannecker, Walter Schuler and Richard SedraniDrug Metabolism and Disposition August 2008, 36 (8) 1457-1460; DOI: https://doi.org/10.1124/dmd.108.020651
Seo, Kyung-Ah
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Shaik, Naveed
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
Shang, Hongcai
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Shin, Jae-Gook
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Shon, Ji-Hong
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
Shoop, Wesley L.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Sipilä, Julius
- You have accessRegio- and Stereospecific N-Glucuronidation of Medetomidine: The Differences between UDP Glucuronosyltransferase (UGT) 1A4 and UGT2B10 Account for the Complex Kinetics of Human Liver MicrosomesSanna Kaivosaari, Päivi Toivonen, Olli Aitio, Julius Sipilä, Mikko Koskinen, Jarmo S. Salonen and Moshe FinelDrug Metabolism and Disposition August 2008, 36 (8) 1529-1537; DOI: https://doi.org/10.1124/dmd.108.021709
Sjödin, Elin
- You have accessIntestinal and Hepatobiliary Transport of Ximelagatran and Its Metabolites in PigsElin Sjödin, Holger Fritsch, Ulf G. Eriksson, Ulrika Logren, Anders Nordgren, Patrik Forsell, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition August 2008, 36 (8) 1519-1528; DOI: https://doi.org/10.1124/dmd.108.020412
Slitt, Angela L.
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Staudinger, Jeff L.
- You have accessThe Traditional Chinese Herbal Remedy Tian Xian Activates Pregnane X Receptor and Induces CYP3A Gene Expression in HepatocytesKristin Lichti-Kaiser and Jeff L. StaudingerDrug Metabolism and Disposition August 2008, 36 (8) 1538-1545; DOI: https://doi.org/10.1124/dmd.108.021774
Stellbrink, Hans-Juergen
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
Stern, Stephan T.
- You have accessRapid Distribution of Liposomal Short-Chain Ceramide in Vitro and in VivoBanu S. Zolnik, Stephan T. Stern, James M. Kaiser, Yasser Heakal, Jeffrey D. Clogston, Mark Kester and Scott E. McNeilDrug Metabolism and Disposition August 2008, 36 (8) 1709-1715; DOI: https://doi.org/10.1124/dmd.107.019679
Stevens, Jeffrey C.
- You have accessDevelopmental Changes in Human Liver CYP2D6 ExpressionJeffrey C. Stevens, Sandra A. Marsh, Matthew J. Zaya, Karen J. Regina, Karthika Divakaran, Min Le and Ronald N. HinesDrug Metabolism and Disposition August 2008, 36 (8) 1587-1593; DOI: https://doi.org/10.1124/dmd.108.021873
Strom, Stephen
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Sugiyama, Yuichi
- You have accessIdentification of the Transporters Involved in the Hepatobiliary Transport and Intestinal Efflux of Methyl 1-(3,4-Dimethoxyphenyl)-3-(3-ethylvaleryl)-4-hydroxy-6,7,8-trimethoxy-2-naphthoate (S-8921) Glucuronide, a Pharmacologically Active Metabolite of S-8921Shingo Sakamoto, Hiroyuki Kusuhara, Kazutoshi Horie, Kohji Takahashi, Takahiko Baba, Jun Ishizaki and Yuichi SugiyamaDrug Metabolism and Disposition August 2008, 36 (8) 1553-1561; DOI: https://doi.org/10.1124/dmd.108.020511
Sun, Yan
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
T
Takahashi, Kohji
- You have accessIdentification of the Transporters Involved in the Hepatobiliary Transport and Intestinal Efflux of Methyl 1-(3,4-Dimethoxyphenyl)-3-(3-ethylvaleryl)-4-hydroxy-6,7,8-trimethoxy-2-naphthoate (S-8921) Glucuronide, a Pharmacologically Active Metabolite of S-8921Shingo Sakamoto, Hiroyuki Kusuhara, Kazutoshi Horie, Kohji Takahashi, Takahiko Baba, Jun Ishizaki and Yuichi SugiyamaDrug Metabolism and Disposition August 2008, 36 (8) 1553-1561; DOI: https://doi.org/10.1124/dmd.108.020511
Taubert, Dirk
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
Terasaki, Tetsuya
- You have accessInvestigation of the Role of Breast Cancer Resistance Protein (Bcrp/Abcg2) on Pharmacokinetics and Central Nervous System Penetration of Abacavir and Zidovudine in the MouseNagdeep Giri, Naveed Shaik, Guoyu Pan, Tetsuya Terasaki, Chisato Mukai, Shinji Kitagaki, Naoki Miyakoshi and William F. ElmquistDrug Metabolism and Disposition August 2008, 36 (8) 1476-1484; DOI: https://doi.org/10.1124/dmd.108.020974
Thakker, Dhiren R.
- You have accessMechanisms Underlying Saturable Intestinal Absorption of MetforminWilliam R. Proctor, David L. Bourdet and Dhiren R. ThakkerDrug Metabolism and Disposition August 2008, 36 (8) 1650-1658; DOI: https://doi.org/10.1124/dmd.107.020180
Thompson, Donald R.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Toivonen, Päivi
- You have accessRegio- and Stereospecific N-Glucuronidation of Medetomidine: The Differences between UDP Glucuronosyltransferase (UGT) 1A4 and UGT2B10 Account for the Complex Kinetics of Human Liver MicrosomesSanna Kaivosaari, Päivi Toivonen, Olli Aitio, Julius Sipilä, Mikko Koskinen, Jarmo S. Salonen and Moshe FinelDrug Metabolism and Disposition August 2008, 36 (8) 1529-1537; DOI: https://doi.org/10.1124/dmd.108.021709
Tokui, Taro
- You have accessEffects of Ketoconazole and Quinidine on Pharmacokinetics of Pactimibe and Its Plasma Metabolite, R-125528, in HumansMasakatsu Kotsuma, Taro Tokui, Stefan Freudenthaler and Kenji NishimuraDrug Metabolism and Disposition August 2008, 36 (8) 1505-1511; DOI: https://doi.org/10.1124/dmd.108.021394
Tschirret-Guth, Richard A.
- You have accessComparative Disposition and Metabolism of Paraherquamide in Sheep, Gerbils, and DogsHerve A. Aloysius, Maria V. Silva Elipe, Byron H. Arison, Terry D. Faidley, Bruce F. Michael, Timothy A. Blizzard, Donald R. Thompson, Wesley L. Shoop and Richard A. Tschirret-GuthDrug Metabolism and Disposition August 2008, 36 (8) 1659-1669; DOI: https://doi.org/10.1124/dmd.107.019430
Tu, Jiang-Hua
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
U
Uetrecht, Jack P.
- You have accessPeroxidase-Mediated Bioactivation of Hydroxylated Metabolites of Carbamazepine and PhenytoinWei Lu and Jack P. UetrechtDrug Metabolism and Disposition August 2008, 36 (8) 1624-1636; DOI: https://doi.org/10.1124/dmd.107.019554
- You have accessPathways of Carbamazepine Bioactivation in Vitro. III. The Role of Human Cytochrome P450 Enzymes in the Formation of 2,3-DihydroxycarbamazepineRobin E. Pearce, Wei Lu, YongQiang Wang, Jack P. Uetrecht, Maria Almira Correia and J. Steven LeederDrug Metabolism and Disposition August 2008, 36 (8) 1637-1649; DOI: https://doi.org/10.1124/dmd.107.019562
Usui, Takashi
- You have accessRole of Organic Anion Transporters in the Pharmacokinetics of Zonampanel, an α-Amino-3-hydroxy-5-methylisoxazole-4-propionate Receptor Antagonist, in RatsTsuyoshi Minematsu, Tadashi Hashimoto, Toshiko Aoki, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2008, 36 (8) 1496-1504; DOI: https://doi.org/10.1124/dmd.107.019828
V
van Lunzen, Jan
- You have accessRelevance of the Organic Cation Transporters 1 and 2 for Antiretroviral Drug Therapy in Human Immunodeficiency Virus InfectionNorma Jung, Clara Lehmann, Andrea Rubbert, Meike Knispel, Pia Hartmann, Jan van Lunzen, Hans-Juergen Stellbrink, Gerd Faetkenheuer and Dirk TaubertDrug Metabolism and Disposition August 2008, 36 (8) 1616-1623; DOI: https://doi.org/10.1124/dmd.108.020826
van Tellingen, Olaf
- You have accessExtensive Metabolism and Hepatic Accumulation of Gemcitabine After Multiple Oral and Intravenous Administration in MiceStephan A. Veltkamp, Dick Pluim, Olaf van Tellingen, Jos H. Beijnen and Jan H. M. SchellensDrug Metabolism and Disposition August 2008, 36 (8) 1606-1615; DOI: https://doi.org/10.1124/dmd.108.021048
Vassal, Gilles
- You have accessSqualenoylation Favorably Modifies the in Vivo Pharmacokinetics and Biodistribution of Gemcitabine in MiceL. Harivardhan Reddy, Hania Khoury, Angelo Paci, Alain Deroussent, Humberto Ferreira, Catherine Dubernet, Xavier Declèves, Madeleine Besnard, Helène Chacun, Sinda Lepêtre-Mouelhi, Didier Desmaële, Bernard Rousseau, Christelle Laugier, Jean-Christophe Cintrat, Gilles Vassal and Patrick CouvreurDrug Metabolism and Disposition August 2008, 36 (8) 1570-1577; DOI: https://doi.org/10.1124/dmd.108.020735
Veltkamp, Stephan A.
- You have accessExtensive Metabolism and Hepatic Accumulation of Gemcitabine After Multiple Oral and Intravenous Administration in MiceStephan A. Veltkamp, Dick Pluim, Olaf van Tellingen, Jos H. Beijnen and Jan H. M. SchellensDrug Metabolism and Disposition August 2008, 36 (8) 1606-1615; DOI: https://doi.org/10.1124/dmd.108.021048
Venkataramanan, Raman
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Volak, Laurie P.
- You have accessCurcuminoids Inhibit Multiple Human Cytochromes P450, UDP-Glucuronosyltransferase, and Sulfotransferase Enzymes, whereas Piperine Is a Relatively Selective CYP3A4 InhibitorLaurie P. Volak, Senait Ghirmai, John R. Cashman and Michael H. CourtDrug Metabolism and Disposition August 2008, 36 (8) 1594-1605; DOI: https://doi.org/10.1124/dmd.108.020552
W
Wan, Renzhong
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Wang, Dan
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Wang, Fengqing
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Wang, Yi
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Wang, YongQiang
- You have accessPathways of Carbamazepine Bioactivation in Vitro. III. The Role of Human Cytochrome P450 Enzymes in the Formation of 2,3-DihydroxycarbamazepineRobin E. Pearce, Wei Lu, YongQiang Wang, Jack P. Uetrecht, Maria Almira Correia and J. Steven LeederDrug Metabolism and Disposition August 2008, 36 (8) 1637-1649; DOI: https://doi.org/10.1124/dmd.107.019562
Webborn, Peter J. H.
- You have accessFunctional Consequences of Active Hepatic Uptake on Cytochrome P450 Inhibition in Rat and Human HepatocytesKen Grime, Peter J. H. Webborn and Robert J. RileyDrug Metabolism and Disposition August 2008, 36 (8) 1670-1678; DOI: https://doi.org/10.1124/dmd.108.021055
Williams, Eric E.
- You have accessThe Influence of CYP3A5 Genotype on Dexamethasone Induction of CYP3A Activity in African AmericansPatrick J. Roberts, Kristan D. Rollins, Angela D. M. Kashuba, Mary F. Paine, Andrew C. Nelsen, Eric E. Williams, Cassandra Moran, Jatinder K. Lamba, Erin G. Schuetz and Roy L. HawkeDrug Metabolism and Disposition August 2008, 36 (8) 1465-1469; DOI: https://doi.org/10.1124/dmd.107.020065
Williams, Gary M.
- You have accessAssessment of the Medicines Lidocaine, Prilocaine, and Their Metabolites, 2,6-Dimethylaniline and 2-Methylaniline, for DNA Adduct Formation in Rat TissuesJian-Dong Duan, Alan M. Jeffrey and Gary M. WilliamsDrug Metabolism and Disposition August 2008, 36 (8) 1470-1475; DOI: https://doi.org/10.1124/dmd.107.019950
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Xie, Fang
- You have accessDeletion of the NADPH-Cytochrome P450 Reductase Gene in Cardiomyocytes Does Not Protect Mice against Doxorubicin-Mediated Acute Cardiac ToxicityCheng Fang, Jun Gu, Fang Xie, Melissa Behr, Weizhu Yang, E. Dale Abel and Xinxin DingDrug Metabolism and Disposition August 2008, 36 (8) 1722-1728; DOI: https://doi.org/10.1124/dmd.108.021881
Xu, Fang
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Y
Yamanaka, Hiroyuki
- You have accessExpression of UGT1A and UGT2B mRNA in Human Normal Tissues and Various Cell LinesAkiko Nakamura, Miki Nakajima, Hiroyuki Yamanaka, Ryoichi Fujiwara and Tsuyoshi YokoiDrug Metabolism and Disposition August 2008, 36 (8) 1461-1464; DOI: https://doi.org/10.1124/dmd.108.021428
Yang, Junling
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Yang, Ling
- You have accessUDP-Glucuronosyltransferase 1A6 Is the Major Isozyme Responsible for Protocatechuic Aldehyde Glucuronidation in Human Liver MicrosomesHui-Xin Liu, Yong Liu, Jiang-Wei Zhang, Wei Li, Hong-Tao Liu and Ling YangDrug Metabolism and Disposition August 2008, 36 (8) 1562-1569; DOI: https://doi.org/10.1124/dmd.108.020560
Yang, Weizhu
- You have accessDeletion of the NADPH-Cytochrome P450 Reductase Gene in Cardiomyocytes Does Not Protect Mice against Doxorubicin-Mediated Acute Cardiac ToxicityCheng Fang, Jun Gu, Fang Xie, Melissa Behr, Weizhu Yang, E. Dale Abel and Xinxin DingDrug Metabolism and Disposition August 2008, 36 (8) 1722-1728; DOI: https://doi.org/10.1124/dmd.108.021881
Yasuda, Kazuto
- You have accessA Comprehensive in Vitro and in Silico Analysis of Antibiotics That Activate Pregnane X Receptor and Induce CYP3A4 in Liver and IntestineKazuto Yasuda, Aarati Ranade, Raman Venkataramanan, Stephen Strom, Jonathan Chupka, Sean Ekins, Erin Schuetz and Kenneth BachmannDrug Metabolism and Disposition August 2008, 36 (8) 1689-1697; DOI: https://doi.org/10.1124/dmd.108.020701
Yokoi, Tsuyoshi
- You have accessExpression of UGT1A and UGT2B mRNA in Human Normal Tissues and Various Cell LinesAkiko Nakamura, Miki Nakajima, Hiroyuki Yamanaka, Ryoichi Fujiwara and Tsuyoshi YokoiDrug Metabolism and Disposition August 2008, 36 (8) 1461-1464; DOI: https://doi.org/10.1124/dmd.108.021428
Yokokawa, Akitomo
- You have accessPlasma Profiling of Intact Isoflavone Metabolites by High-Performance Liquid Chromatography and Mass Spectrometric Identification of Flavone Glycosides Daidzin and Genistin in Human Plasma after Administration of KinakoKaori Hosoda, Takashi Furuta, Akitomo Yokokawa, Kenichiro Ogura, Akira Hiratsuka and Kazuo IshiiDrug Metabolism and Disposition August 2008, 36 (8) 1485-1495; DOI: https://doi.org/10.1124/dmd.108.021006
Younis, Islam R.
- You have accessMetabolism of the Cysteine S-Conjugate of Busulfan Involves a β-Lyase ReactionArthur J. L. Cooper, Islam R. Younis, Zoya V. Niatsetskaya, Boris F. Krasnikov, John T. Pinto, William P. Petros and Patrick S. CalleryDrug Metabolism and Disposition August 2008, 36 (8) 1546-1552; DOI: https://doi.org/10.1124/dmd.108.020768
Z
Zaya, Matthew J.
- You have accessIn Vitro Drug-Drug Interaction Screens for Canine Veterinary Medicines: Evaluation of Cytochrome P450 Reversible InhibitionDivesh Aidasani, Matthew J. Zaya, Phyllis B. Malpas and Charles W. LocusonDrug Metabolism and Disposition August 2008, 36 (8) 1512-1518; DOI: https://doi.org/10.1124/dmd.108.021196
- You have accessDevelopmental Changes in Human Liver CYP2D6 ExpressionJeffrey C. Stevens, Sandra A. Marsh, Matthew J. Zaya, Karen J. Regina, Karthika Divakaran, Min Le and Ronald N. HinesDrug Metabolism and Disposition August 2008, 36 (8) 1587-1593; DOI: https://doi.org/10.1124/dmd.108.021873
Zhang, Boli
- You have accessPlasma and Urinary Tanshinol from Salvia miltiorrhiza (Danshen) Can Be Used as Pharmacokinetic Markers for Cardiotonic Pills, a Cardiovascular Herbal MedicineTong Lu, Junling Yang, Xiumei Gao, Ping Chen, Feifei Du, Yan Sun, Fengqing Wang, Fang Xu, Hongcai Shang, Yuhong Huang, Yi Wang, Renzhong Wan, Changxiao Liu, Boli Zhang and Chuan LiDrug Metabolism and Disposition August 2008, 36 (8) 1578-1586; DOI: https://doi.org/10.1124/dmd.108.021592
Zhang, Jiang-Wei
- You have accessUDP-Glucuronosyltransferase 1A6 Is the Major Isozyme Responsible for Protocatechuic Aldehyde Glucuronidation in Human Liver MicrosomesHui-Xin Liu, Yong Liu, Jiang-Wei Zhang, Wei Li, Hong-Tao Liu and Ling YangDrug Metabolism and Disposition August 2008, 36 (8) 1562-1569; DOI: https://doi.org/10.1124/dmd.108.020560
Zhang, Wei
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Zhang, Youcai
- You have accessThe Nrf2 Activator Oltipraz Also Activates the Constitutive Androstane ReceptorMatthew D. Merrell, Jonathan P. Jackson, Lisa M. Augustine, Craig D. Fisher, Angela L. Slitt, Jonathan M. Maher, Wendong Huang, David D. Moore, Youcai Zhang, Curtis D. Klaassen and Nathan J. CherringtonDrug Metabolism and Disposition August 2008, 36 (8) 1716-1721; DOI: https://doi.org/10.1124/dmd.108.020867
Zhou, Hong-Hao
- You have accessCytochrome P450 2B6 Catalyzes the Formation of Pharmacologically Active Sibutramine (N-{1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutyl}-N,N-dimethylamine) Metabolites in Human Liver MicrosomesSoo Kyung Bae, Shan Cao, Kyung-Ah Seo, Hyunmi Kim, Min-Jung Kim, Ji-Hong Shon, Kwang-Hyeon Liu, Hong-Hao Zhou and Jae-Gook ShinDrug Metabolism and Disposition August 2008, 36 (8) 1679-1688; DOI: https://doi.org/10.1124/dmd.108.020727
- You have accessHepatic Nuclear Factor 1α Inhibitor Ursodeoxycholic Acid Influences Pharmacokinetics of the Organic Anion Transporting Polypeptide 1B1 Substrate Rosuvastatin and BilirubinYi-Jing He, Wei Zhang, Jiang-Hua Tu, Julia Kirchheiner, Yao Chen, Dong Guo, Qing Li, Zhong-Yu Li, Hao Chen, Dong-Li Hu, Dan Wang and Hong-Hao ZhouDrug Metabolism and Disposition August 2008, 36 (8) 1453-1456; DOI: https://doi.org/10.1124/dmd.108.020503
Zollinger, Markus
- You have accessThe Macrolide Everolimus Forms an Unusual Metabolite in Animals and Humans: Identification of a Phosphocholine EsterMarkus Zollinger, Claudia Sayer, Robert Dannecker, Walter Schuler and Richard SedraniDrug Metabolism and Disposition August 2008, 36 (8) 1457-1460; DOI: https://doi.org/10.1124/dmd.108.020651
Zolnik, Banu S.
- You have accessRapid Distribution of Liposomal Short-Chain Ceramide in Vitro and in VivoBanu S. Zolnik, Stephan T. Stern, James M. Kaiser, Yasser Heakal, Jeffrey D. Clogston, Mark Kester and Scott E. McNeilDrug Metabolism and Disposition August 2008, 36 (8) 1709-1715; DOI: https://doi.org/10.1124/dmd.107.019679
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