Inhibition and Stimulation of Intestinal and Hepatic CYP3A Activity: Studies in Humanized CYP3A4 Transgenic Mice Using Triazolam

Division of Molecular Biology, The Netherlands Cancer Institute, Amsterdam, The Netherlands (R.A.B.v.W., R.W.R., A.E.v.H., A.H.S.); Department of Pharmaceutical Sciences, Utrecht University, Utrecht, The Netherlands (R.W.S., J.H.B.); and Department of Pharmacy and Pharmacology, Slotervaart Hospital, Amsterdam, The Netherlands (J.H.B.)

Address correspondence to:
Alfred H. Schinkel,
Division of Molecular Biology, The Netherlands Cancer Institute, Plesmanlaan 121, 1066 CX Amsterdam, The Netherlands.
E-mail: a.schinkel{at}nki.nl

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