Index by author
August 01, 2009; Volume 37,Issue 8
A
Ajetunmobi, Jumoke
- You have accessCharacterizing the Effects of Common UDP Glucuronosyltransferase (UGT) 1A6 and UGT1A1 Polymorphisms on cis- and trans-Resveratrol GlucuronidationOtito Frances Iwuchukwu, Jumoke Ajetunmobi, Din Ung and Swati NagarDrug Metabolism and Disposition August 2009, 37 (8) 1726-1732; DOI: https://doi.org/10.1124/dmd.109.027391
Aoki, Yasuhiro
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
B
Barron, Denis
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
Benninghoff, Abby D.
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Bordini, Ellenia
- You have accessDisposition and Metabolism of Radiolabeled Casopitant in HumansMario Pellegatti, Ellenia Bordini, Patrizia Fizzotti, Andy Roberts and Brendan M. JohnsonDrug Metabolism and Disposition August 2009, 37 (8) 1635-1645; DOI: https://doi.org/10.1124/dmd.109.026781
Boudinot, F. Douglas
- You have accessBinding of Lopinavir to Human α1-Acid Glycoprotein and Serum AlbuminAbhishek Gulati, F. Douglas Boudinot and Phillip M. GerkDrug Metabolism and Disposition August 2009, 37 (8) 1572-1575; DOI: https://doi.org/10.1124/dmd.109.026708
Braeuning, Albert
- You have accessThe Glycogen Synthase Kinase Inhibitor 3-(2,4-Dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione (SB216763) Is a Partial Agonist of the Aryl Hydrocarbon ReceptorAlbert Braeuning and Albrecht BuchmannDrug Metabolism and Disposition August 2009, 37 (8) 1576-1580; DOI: https://doi.org/10.1124/dmd.109.027821
Braithwaite, Robin A.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Buchmann, Albrecht
- You have accessThe Glycogen Synthase Kinase Inhibitor 3-(2,4-Dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione (SB216763) Is a Partial Agonist of the Aryl Hydrocarbon ReceptorAlbert Braeuning and Albrecht BuchmannDrug Metabolism and Disposition August 2009, 37 (8) 1576-1580; DOI: https://doi.org/10.1124/dmd.109.027821
C
Capparelli, Edmund
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
Cavin, Christophe
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
Chang, Shu-Ying
- You have accessFurther Assessment of 17α-Ethinyl Estradiol as an Inhibitor of Different Human Cytochrome P450 Forms in VitroShu-Ying Chang, Cliff Chen, Zheng Yang and A. David RodriguesDrug Metabolism and Disposition August 2009, 37 (8) 1667-1675; DOI: https://doi.org/10.1124/dmd.109.026997
Chen, Cliff
- You have accessFurther Assessment of 17α-Ethinyl Estradiol as an Inhibitor of Different Human Cytochrome P450 Forms in VitroShu-Ying Chang, Cliff Chen, Zheng Yang and A. David RodriguesDrug Metabolism and Disposition August 2009, 37 (8) 1667-1675; DOI: https://doi.org/10.1124/dmd.109.026997
Cheng, Jie
- You have accessRifampicin-Activated Human Pregnane X Receptor and CYP3A4 Induction Enhance Acetaminophen-Induced ToxicityJie Cheng, Xiaochao Ma, Kristopher W. Krausz, Jeffrey R. Idle and Frank J. GonzalezDrug Metabolism and Disposition August 2009, 37 (8) 1611-1621; DOI: https://doi.org/10.1124/dmd.109.027565
Chikada, Tsubasa
- You have accessInvolvement of Vitamin D Receptor in the Intestinal Induction of Human ABCB1Shuko Tachibana, Kouichi Yoshinari, Tsubasa Chikada, Takayoshi Toriyabe, Kiyoshi Nagata and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1604-1610; DOI: https://doi.org/10.1124/dmd.109.027219
Cook, Jack
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
Cowan, David A.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Crozier, Alan
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
D
Darekar, Amanda
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
Davern, Timothy J.
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
de Waart, Dirk R.
- You have accessComplex Pharmacokinetic Behavior of Ezetimibe Depends on Abcc2, Abcc3, and Abcg2Dirk R. de Waart, Maria L. H. Vlaming, Cindy Kunne, Alfred H. Schinkel and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition August 2009, 37 (8) 1698-1702; DOI: https://doi.org/10.1124/dmd.108.026146
Dickins, Maurice
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
E
Elferink, Ronald P. J. Oude
- You have accessComplex Pharmacokinetic Behavior of Ezetimibe Depends on Abcc2, Abcc3, and Abcg2Dirk R. de Waart, Maria L. H. Vlaming, Cindy Kunne, Alfred H. Schinkel and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition August 2009, 37 (8) 1698-1702; DOI: https://doi.org/10.1124/dmd.108.026146
Elliot, Simon P.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Enomoto, Shigeki
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
F
Fahmi, Odette A.
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
Fizzotti, Patrizia
- You have accessDisposition and Metabolism of Radiolabeled Casopitant in HumansMario Pellegatti, Ellenia Bordini, Patrizia Fizzotti, Andy Roberts and Brendan M. JohnsonDrug Metabolism and Disposition August 2009, 37 (8) 1635-1645; DOI: https://doi.org/10.1124/dmd.109.026781
Frost, Charles
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Fujita, Shoichi
- You have accessThe Importance of Heterogeneous Nuclear Ribonucleoprotein K on Cytochrome P450 2D2 Gene Regulation: Its Binding Is Reduced in Dark Agouti RatsNoriaki Sakai, Kentaro Q. Sakamoto, Shoichi Fujita and Mayumi IshizukaDrug Metabolism and Disposition August 2009, 37 (8) 1703-1710; DOI: https://doi.org/10.1124/dmd.109.027284
Fujiwara, Ryoichi
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Fukami, Tatsuki
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Fukano, Y.
- You have accessDisposition and Metabolism of a Novel Prostanoid Antiglaucoma Medication, Tafluprost, Following Ocular Administration to RatsY. Fukano and K. KawazuDrug Metabolism and Disposition August 2009, 37 (8) 1622-1634; DOI: https://doi.org/10.1124/dmd.108.024885
Furnes, Bjarte
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
G
Gerk, Phillip M.
- You have accessBinding of Lopinavir to Human α1-Acid Glycoprotein and Serum AlbuminAbhishek Gulati, F. Douglas Boudinot and Phillip M. GerkDrug Metabolism and Disposition August 2009, 37 (8) 1572-1575; DOI: https://doi.org/10.1124/dmd.109.026708
Gonzalez, Frank J.
- You have accessRifampicin-Activated Human Pregnane X Receptor and CYP3A4 Induction Enhance Acetaminophen-Induced ToxicityJie Cheng, Xiaochao Ma, Kristopher W. Krausz, Jeffrey R. Idle and Frank J. GonzalezDrug Metabolism and Disposition August 2009, 37 (8) 1611-1621; DOI: https://doi.org/10.1124/dmd.109.027565
Gorski, J. Christopher
- You have accessSemiphysiologically Based Pharmacokinetic Models for the Inhibition of Midazolam Clearance by Diltiazem and Its Major MetaboliteXin Zhang, Sara K. Quinney, J. Christopher Gorski, David R. Jones and Stephen D. HallDrug Metabolism and Disposition August 2009, 37 (8) 1587-1597; DOI: https://doi.org/10.1124/dmd.109.026658
Grafström, Roland C.
- You have accessThe Ontogeny, Distribution, and Regulation of Alcohol Dehydrogenase 3: Implications for Pulmonary PhysiologyChad M. Thompson, Babasaheb Sonawane and Roland C. GrafströmDrug Metabolism and Disposition August 2009, 37 (8) 1565-1571; DOI: https://doi.org/10.1124/dmd.109.027904
Grossman, Scott J.
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Gu, Zheming
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Gulati, Abhishek
- You have accessBinding of Lopinavir to Human α1-Acid Glycoprotein and Serum AlbuminAbhishek Gulati, F. Douglas Boudinot and Phillip M. GerkDrug Metabolism and Disposition August 2009, 37 (8) 1572-1575; DOI: https://doi.org/10.1124/dmd.109.026708
Guo, Feng
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
H
Halket, John M.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Hall, Stephen D.
- You have accessSemiphysiologically Based Pharmacokinetic Models for the Inhibition of Midazolam Clearance by Diltiazem and Its Major MetaboliteXin Zhang, Sara K. Quinney, J. Christopher Gorski, David R. Jones and Stephen D. HallDrug Metabolism and Disposition August 2009, 37 (8) 1587-1597; DOI: https://doi.org/10.1124/dmd.109.026658
Hao, Feng
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
He, Kan
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Henderson, Marilyn C.
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Hinson, Jack A.
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
Hippalgaonkar, Ketan
- You have accessVitreal Kinetics of Quinidine in Rabbits in the Presence of Topically Coadministered P-Glycoprotein Substrates/ModulatorsSoumyajit Majumdar, Ketan Hippalgaonkar and Ramesh SrirangamDrug Metabolism and Disposition August 2009, 37 (8) 1718-1725; DOI: https://doi.org/10.1124/dmd.108.026450
Hsu, Fong-Fu
- You have accessIdentification of New 2-Amino-3-methylimidazo[4,5-f]quinoline Urinary Metabolites from β-Naphthoflavone-Treated MiceVijaya M. Lakshmi, Fong-Fu Hsu and Terry V. ZenserDrug Metabolism and Disposition August 2009, 37 (8) 1690-1697; DOI: https://doi.org/10.1124/dmd.109.027342
Humphreys, W. Griffith
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Hurst, Susan
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
Hyland, Ruth
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
I
Idle, Jeffrey R.
- You have accessRifampicin-Activated Human Pregnane X Receptor and CYP3A4 Induction Enhance Acetaminophen-Induced ToxicityJie Cheng, Xiaochao Ma, Kristopher W. Krausz, Jeffrey R. Idle and Frank J. GonzalezDrug Metabolism and Disposition August 2009, 37 (8) 1611-1621; DOI: https://doi.org/10.1124/dmd.109.027565
Ikushiro, Shin-ichi
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Ishizuka, Mayumi
- You have accessThe Importance of Heterogeneous Nuclear Ribonucleoprotein K on Cytochrome P450 2D2 Gene Regulation: Its Binding Is Reduced in Dark Agouti RatsNoriaki Sakai, Kentaro Q. Sakamoto, Shoichi Fujita and Mayumi IshizukaDrug Metabolism and Disposition August 2009, 37 (8) 1703-1710; DOI: https://doi.org/10.1124/dmd.109.027284
Iwatsubo, Takafumi
- You have accessIdentification of Human Metabolites of (–)-N-{2-[(R)-3-(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidino]ethyl}-4-fluorobenzamide (YM758), a Novel If Channel Inhibitor, and Investigation of the Transporter-Mediated Renal and Hepatic Excretion of These MetabolitesKen-ichi Umehara, Nobuaki Shirai, Takafumi Iwatsubo, Kiyoshi Noguchi, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2009, 37 (8) 1646-1657; DOI: https://doi.org/10.1124/dmd.108.026294
Iwuchukwu, Otito Frances
- You have accessCharacterizing the Effects of Common UDP Glucuronosyltransferase (UGT) 1A6 and UGT1A1 Polymorphisms on cis- and trans-Resveratrol GlucuronidationOtito Frances Iwuchukwu, Jumoke Ajetunmobi, Din Ung and Swati NagarDrug Metabolism and Disposition August 2009, 37 (8) 1726-1732; DOI: https://doi.org/10.1124/dmd.109.027391
Izukawa, Takeshi
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
J
James, Laura P.
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
Johnson, Brendan M.
- You have accessDisposition and Metabolism of Radiolabeled Casopitant in HumansMario Pellegatti, Ellenia Bordini, Patrizia Fizzotti, Andy Roberts and Brendan M. JohnsonDrug Metabolism and Disposition August 2009, 37 (8) 1635-1645; DOI: https://doi.org/10.1124/dmd.109.026781
Jones, David R.
- You have accessSemiphysiologically Based Pharmacokinetic Models for the Inhibition of Midazolam Clearance by Diltiazem and Its Major MetaboliteXin Zhang, Sara K. Quinney, J. Christopher Gorski, David R. Jones and Stephen D. HallDrug Metabolism and Disposition August 2009, 37 (8) 1587-1597; DOI: https://doi.org/10.1124/dmd.109.026658
K
Kamimura, Hidetaka
- You have accessIdentification of Human Metabolites of (–)-N-{2-[(R)-3-(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidino]ethyl}-4-fluorobenzamide (YM758), a Novel If Channel Inhibitor, and Investigation of the Transporter-Mediated Renal and Hepatic Excretion of These MetabolitesKen-ichi Umehara, Nobuaki Shirai, Takafumi Iwatsubo, Kiyoshi Noguchi, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2009, 37 (8) 1646-1657; DOI: https://doi.org/10.1124/dmd.108.026294
Kano, Takashi
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Karplus, P. Andrew
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Kawazu, K.
- You have accessDisposition and Metabolism of a Novel Prostanoid Antiglaucoma Medication, Tafluprost, Following Ocular Administration to RatsY. Fukano and K. KawazuDrug Metabolism and Disposition August 2009, 37 (8) 1622-1634; DOI: https://doi.org/10.1124/dmd.108.024885
Kicman, Andrew T.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Knabb, Robert M.
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Kobayashi, Shoko
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Krausz, Kristopher W.
- You have accessRifampicin-Activated Human Pregnane X Receptor and CYP3A4 Induction Enhance Acetaminophen-Induced ToxicityJie Cheng, Xiaochao Ma, Kristopher W. Krausz, Jeffrey R. Idle and Frank J. GonzalezDrug Metabolism and Disposition August 2009, 37 (8) 1611-1621; DOI: https://doi.org/10.1124/dmd.109.027565
Krueger, Sharon K.
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Kunne, Cindy
- You have accessComplex Pharmacokinetic Behavior of Ezetimibe Depends on Abcc2, Abcc3, and Abcg2Dirk R. de Waart, Maria L. H. Vlaming, Cindy Kunne, Alfred H. Schinkel and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition August 2009, 37 (8) 1698-1702; DOI: https://doi.org/10.1124/dmd.108.026146
L
Lakshmi, Vijaya M.
- You have accessIdentification of New 2-Amino-3-methylimidazo[4,5-f]quinoline Urinary Metabolites from β-Naphthoflavone-Treated MiceVijaya M. Lakshmi, Fong-Fu Hsu and Terry V. ZenserDrug Metabolism and Disposition August 2009, 37 (8) 1690-1697; DOI: https://doi.org/10.1124/dmd.109.027342
Lee, William M.
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
Letzig, Lynda
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
Li, Albert P.
- You have accessEvaluation of Luciferin-Isopropyl Acetal as a CYP3A4 Substrate for Human Hepatocytes: Effects of Organic Solvents, Cytochrome P450 (P450) Inhibitors, and P450 InducersAlbert P. LiDrug Metabolism and Disposition August 2009, 37 (8) 1598-1603; DOI: https://doi.org/10.1124/dmd.109.027268
Locuson, Charles W.
- You have accessCYP2D6-CYP2C9 Protein-Protein Interactions and Isoform-Selective Effects on Substrate Binding and CatalysisMurali Subramanian, Michael Low, Charles W. Locuson and Timothy S. TracyDrug Metabolism and Disposition August 2009, 37 (8) 1682-1689; DOI: https://doi.org/10.1124/dmd.109.026500
Low, Michael
- You have accessCYP2D6-CYP2C9 Protein-Protein Interactions and Isoform-Selective Effects on Substrate Binding and CatalysisMurali Subramanian, Michael Low, Charles W. Locuson and Timothy S. TracyDrug Metabolism and Disposition August 2009, 37 (8) 1682-1689; DOI: https://doi.org/10.1124/dmd.109.026500
M
Ma, Xiaochao
- You have accessRifampicin-Activated Human Pregnane X Receptor and CYP3A4 Induction Enhance Acetaminophen-Induced ToxicityJie Cheng, Xiaochao Ma, Kristopher W. Krausz, Jeffrey R. Idle and Frank J. GonzalezDrug Metabolism and Disposition August 2009, 37 (8) 1611-1621; DOI: https://doi.org/10.1124/dmd.109.027565
Majumdar, Soumyajit
- You have accessVitreal Kinetics of Quinidine in Rabbits in the Presence of Topically Coadministered P-Glycoprotein Substrates/ModulatorsSoumyajit Majumdar, Ketan Hippalgaonkar and Ramesh SrirangamDrug Metabolism and Disposition August 2009, 37 (8) 1718-1725; DOI: https://doi.org/10.1124/dmd.108.026450
Maxwell, Brad D.
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Mitroka, James
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Morimoto, Kaori
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Mullen, William
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
N
Nagar, Swati
- You have accessCharacterizing the Effects of Common UDP Glucuronosyltransferase (UGT) 1A6 and UGT1A1 Polymorphisms on cis- and trans-Resveratrol GlucuronidationOtito Frances Iwuchukwu, Jumoke Ajetunmobi, Din Ung and Swati NagarDrug Metabolism and Disposition August 2009, 37 (8) 1726-1732; DOI: https://doi.org/10.1124/dmd.109.027391
Nagata, Kiyoshi
- You have accessInvolvement of Vitamin D Receptor in the Intestinal Induction of Human ABCB1Shuko Tachibana, Kouichi Yoshinari, Tsubasa Chikada, Takayoshi Toriyabe, Kiyoshi Nagata and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1604-1610; DOI: https://doi.org/10.1124/dmd.109.027219
Nakajima, Miki
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Noguchi, Kiyoshi
- You have accessIdentification of Human Metabolites of (–)-N-{2-[(R)-3-(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidino]ethyl}-4-fluorobenzamide (YM758), a Novel If Channel Inhibitor, and Investigation of the Transporter-Mediated Renal and Hepatic Excretion of These MetabolitesKen-ichi Umehara, Nobuaki Shirai, Takafumi Iwatsubo, Kiyoshi Noguchi, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2009, 37 (8) 1646-1657; DOI: https://doi.org/10.1124/dmd.108.026294
O
Obach, R. Scott
- You have accessGlycerolysis of Acyl Glucuronides as an Artifact of in Vitro Drug Metabolism IncubationsR. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1581-1586; DOI: https://doi.org/10.1124/dmd.109.027953
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
Ogihara, Takuo
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
P
Parkin, Mark C.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Pellegatti, Mario
- You have accessDisposition and Metabolism of Radiolabeled Casopitant in HumansMario Pellegatti, Ellenia Bordini, Patrizia Fizzotti, Andy Roberts and Brendan M. JohnsonDrug Metabolism and Disposition August 2009, 37 (8) 1635-1645; DOI: https://doi.org/10.1124/dmd.109.026781
Phipps, Alex
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
Plowchalk, David
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
Q
Quinney, Sara K.
- You have accessSemiphysiologically Based Pharmacokinetic Models for the Inhibition of Midazolam Clearance by Diltiazem and Its Major MetaboliteXin Zhang, Sara K. Quinney, J. Christopher Gorski, David R. Jones and Stephen D. HallDrug Metabolism and Disposition August 2009, 37 (8) 1587-1597; DOI: https://doi.org/10.1124/dmd.109.026658
R
Raghavan, Nirmala
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Roberts, Andy
- You have accessDisposition and Metabolism of Radiolabeled Casopitant in HumansMario Pellegatti, Ellenia Bordini, Patrizia Fizzotti, Andy Roberts and Brendan M. JohnsonDrug Metabolism and Disposition August 2009, 37 (8) 1635-1645; DOI: https://doi.org/10.1124/dmd.109.026781
Roberts, Dean W.
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
Rodrigues, A. David
- You have accessFurther Assessment of 17α-Ethinyl Estradiol as an Inhibitor of Different Human Cytochrome P450 Forms in VitroShu-Ying Chang, Cliff Chen, Zheng Yang and A. David RodriguesDrug Metabolism and Disposition August 2009, 37 (8) 1667-1675; DOI: https://doi.org/10.1124/dmd.109.026997
S
Sakai, Noriaki
- You have accessThe Importance of Heterogeneous Nuclear Ribonucleoprotein K on Cytochrome P450 2D2 Gene Regulation: Its Binding Is Reduced in Dark Agouti RatsNoriaki Sakai, Kentaro Q. Sakamoto, Shoichi Fujita and Mayumi IshizukaDrug Metabolism and Disposition August 2009, 37 (8) 1703-1710; DOI: https://doi.org/10.1124/dmd.109.027284
Sakaki, Toshiyuki
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Sakamoto, Kentaro Q.
- You have accessThe Importance of Heterogeneous Nuclear Ribonucleoprotein K on Cytochrome P450 2D2 Gene Regulation: Its Binding Is Reduced in Dark Agouti RatsNoriaki Sakai, Kentaro Q. Sakamoto, Shoichi Fujita and Mayumi IshizukaDrug Metabolism and Disposition August 2009, 37 (8) 1703-1710; DOI: https://doi.org/10.1124/dmd.109.027284
Schinkel, Alfred H.
- You have accessComplex Pharmacokinetic Behavior of Ezetimibe Depends on Abcc2, Abcc3, and Abcg2Dirk R. de Waart, Maria L. H. Vlaming, Cindy Kunne, Alfred H. Schinkel and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition August 2009, 37 (8) 1698-1702; DOI: https://doi.org/10.1124/dmd.108.026146
Schlenk, Daniel
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Schuster, Alan
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Senggunprai, Laddawan
- You have accessSelective Role of Sulfotransferase 2A1 (SULT2A1) in the N-Sulfoconjugation of Quinolone Drugs in HumansLaddawan Senggunprai, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1711-1717; DOI: https://doi.org/10.1124/dmd.109.027441
Shirai, Nobuaki
- You have accessIdentification of Human Metabolites of (–)-N-{2-[(R)-3-(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidino]ethyl}-4-fluorobenzamide (YM758), a Novel If Channel Inhibitor, and Investigation of the Transporter-Mediated Renal and Hepatic Excretion of These MetabolitesKen-ichi Umehara, Nobuaki Shirai, Takafumi Iwatsubo, Kiyoshi Noguchi, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2009, 37 (8) 1646-1657; DOI: https://doi.org/10.1124/dmd.108.026294
Shirasaka, Yoshiyuki
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Siddens, Lisbeth K.
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Simpson, Pippa M.
- You have accessPharmacokinetics of Acetaminophen-Protein Adducts in Adults with Acetaminophen Overdose and Acute Liver FailureLaura P. James, Lynda Letzig, Pippa M. Simpson, Edmund Capparelli, Dean W. Roberts, Jack A. Hinson, Timothy J. Davern and William M. LeeDrug Metabolism and Disposition August 2009, 37 (8) 1779-1784; DOI: https://doi.org/10.1124/dmd.108.026195
Smith, Norman W.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Sonawane, Babasaheb
- You have accessThe Ontogeny, Distribution, and Regulation of Alcohol Dehydrogenase 3: Implications for Pulmonary PhysiologyChad M. Thompson, Babasaheb Sonawane and Roland C. GrafströmDrug Metabolism and Disposition August 2009, 37 (8) 1565-1571; DOI: https://doi.org/10.1124/dmd.109.027904
Srirangam, Ramesh
- You have accessVitreal Kinetics of Quinidine in Rabbits in the Presence of Topically Coadministered P-Glycoprotein Substrates/ModulatorsSoumyajit Majumdar, Ketan Hippalgaonkar and Ramesh SrirangamDrug Metabolism and Disposition August 2009, 37 (8) 1718-1725; DOI: https://doi.org/10.1124/dmd.108.026450
Stalmach, Angélique
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
Steiling, Heike
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
Steventon, Glyn B.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
Subramanian, Murali
- You have accessCYP2D6-CYP2C9 Protein-Protein Interactions and Isoform-Selective Effects on Substrate Binding and CatalysisMurali Subramanian, Michael Low, Charles W. Locuson and Timothy S. TracyDrug Metabolism and Disposition August 2009, 37 (8) 1682-1689; DOI: https://doi.org/10.1124/dmd.109.026500
T
Tachibana, Shuko
- You have accessInvolvement of Vitamin D Receptor in the Intestinal Induction of Human ABCB1Shuko Tachibana, Kouichi Yoshinari, Tsubasa Chikada, Takayoshi Toriyabe, Kiyoshi Nagata and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1604-1610; DOI: https://doi.org/10.1124/dmd.109.027219
Takamiya, Masataka
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Takeda, Shuso
- You have accessCannabidiol-2′,6′-Dimethyl Ether, a Cannabidiol Derivative, Is a Highly Potent and Selective 15-Lipoxygenase InhibitorShuso Takeda, Noriyuki Usami, Ikuo Yamamoto and Kazuhito WatanabeDrug Metabolism and Disposition August 2009, 37 (8) 1733-1737; DOI: https://doi.org/10.1124/dmd.109.026930
Tamai, Ikumi
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Thompson, Chad M.
- You have accessThe Ontogeny, Distribution, and Regulation of Alcohol Dehydrogenase 3: Implications for Pulmonary PhysiologyChad M. Thompson, Babasaheb Sonawane and Roland C. GrafströmDrug Metabolism and Disposition August 2009, 37 (8) 1565-1571; DOI: https://doi.org/10.1124/dmd.109.027904
Toriyabe, Takayoshi
- You have accessInvolvement of Vitamin D Receptor in the Intestinal Induction of Human ABCB1Shuko Tachibana, Kouichi Yoshinari, Tsubasa Chikada, Takayoshi Toriyabe, Kiyoshi Nagata and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1604-1610; DOI: https://doi.org/10.1124/dmd.109.027219
Tracy, Timothy S.
- You have accessCYP2D6-CYP2C9 Protein-Protein Interactions and Isoform-Selective Effects on Substrate Binding and CatalysisMurali Subramanian, Michael Low, Charles W. Locuson and Timothy S. TracyDrug Metabolism and Disposition August 2009, 37 (8) 1682-1689; DOI: https://doi.org/10.1124/dmd.109.026500
Turfus, Sophie C.
- You have accessUse of Human Microsomes and Deuterated Substrates: An Alternative Approach for the Identification of Novel Metabolites of Ketamine by Mass SpectrometrySophie C. Turfus, Mark C. Parkin, David A. Cowan, John M. Halket, Norman W. Smith, Robin A. Braithwaite, Simon P. Elliot, Glyn B. Steventon and Andrew T. KicmanDrug Metabolism and Disposition August 2009, 37 (8) 1769-1778; DOI: https://doi.org/10.1124/dmd.108.026328
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Uchida, Kenichi
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
Umehara, Ken-ichi
- You have accessIdentification of Human Metabolites of (–)-N-{2-[(R)-3-(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidino]ethyl}-4-fluorobenzamide (YM758), a Novel If Channel Inhibitor, and Investigation of the Transporter-Mediated Renal and Hepatic Excretion of These MetabolitesKen-ichi Umehara, Nobuaki Shirai, Takafumi Iwatsubo, Kiyoshi Noguchi, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2009, 37 (8) 1646-1657; DOI: https://doi.org/10.1124/dmd.108.026294
Ung, Din
- You have accessCharacterizing the Effects of Common UDP Glucuronosyltransferase (UGT) 1A6 and UGT1A1 Polymorphisms on cis- and trans-Resveratrol GlucuronidationOtito Frances Iwuchukwu, Jumoke Ajetunmobi, Din Ung and Swati NagarDrug Metabolism and Disposition August 2009, 37 (8) 1726-1732; DOI: https://doi.org/10.1124/dmd.109.027391
Usami, Noriyuki
- You have accessCannabidiol-2′,6′-Dimethyl Ether, a Cannabidiol Derivative, Is a Highly Potent and Selective 15-Lipoxygenase InhibitorShuso Takeda, Noriyuki Usami, Ikuo Yamamoto and Kazuhito WatanabeDrug Metabolism and Disposition August 2009, 37 (8) 1733-1737; DOI: https://doi.org/10.1124/dmd.109.026930
Usui, Takashi
- You have accessIdentification of Human Metabolites of (–)-N-{2-[(R)-3-(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidino]ethyl}-4-fluorobenzamide (YM758), a Novel If Channel Inhibitor, and Investigation of the Transporter-Mediated Renal and Hepatic Excretion of These MetabolitesKen-ichi Umehara, Nobuaki Shirai, Takafumi Iwatsubo, Kiyoshi Noguchi, Takashi Usui and Hidetaka KamimuraDrug Metabolism and Disposition August 2009, 37 (8) 1646-1657; DOI: https://doi.org/10.1124/dmd.108.026294
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VanDyke, Jonathan E.
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Vlaming, Maria L. H.
- You have accessComplex Pharmacokinetic Behavior of Ezetimibe Depends on Abcc2, Abcc3, and Abcg2Dirk R. de Waart, Maria L. H. Vlaming, Cindy Kunne, Alfred H. Schinkel and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition August 2009, 37 (8) 1698-1702; DOI: https://doi.org/10.1124/dmd.108.026146
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Wada, Sho
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Wagatsuma, Tamae
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Wang, Lifei
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Watanabe, Kazuhito
- You have accessCannabidiol-2′,6′-Dimethyl Ether, a Cannabidiol Derivative, Is a Highly Potent and Selective 15-Lipoxygenase InhibitorShuso Takeda, Noriyuki Usami, Ikuo Yamamoto and Kazuhito WatanabeDrug Metabolism and Disposition August 2009, 37 (8) 1733-1737; DOI: https://doi.org/10.1124/dmd.109.026930
Williams, David E.
- You have accessCharacterization of Sulfoxygenation and Structural Implications of Human Flavin-Containing Monooxygenase Isoform 2 (FMO2.1) Variants S195L and N413KSharon K. Krueger, Marilyn C. Henderson, Lisbeth K. Siddens, Jonathan E. VanDyke, Abby D. Benninghoff, P. Andrew Karplus, Bjarte Furnes, Daniel Schlenk and David E. WilliamsDrug Metabolism and Disposition August 2009, 37 (8) 1785-1791; DOI: https://doi.org/10.1124/dmd.109.027201
Williamson, Gary
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
Y
Yabuuchi, Hikaru
- You have accessOseltamivir (Tamiflu) Is a Substrate of Peptide Transporter 1Takuo Ogihara, Takashi Kano, Tamae Wagatsuma, Sho Wada, Hikaru Yabuuchi, Shigeki Enomoto, Kaori Morimoto, Yoshiyuki Shirasaka, Shoko Kobayashi and Ikumi TamaiDrug Metabolism and Disposition August 2009, 37 (8) 1676-1681; DOI: https://doi.org/10.1124/dmd.109.026922
Yamamoto, Ikuo
- You have accessCannabidiol-2′,6′-Dimethyl Ether, a Cannabidiol Derivative, Is a Highly Potent and Selective 15-Lipoxygenase InhibitorShuso Takeda, Noriyuki Usami, Ikuo Yamamoto and Kazuhito WatanabeDrug Metabolism and Disposition August 2009, 37 (8) 1733-1737; DOI: https://doi.org/10.1124/dmd.109.026930
Yamanaka, Hiroyuki
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Yamazoe, Yasushi
- You have accessInvolvement of Vitamin D Receptor in the Intestinal Induction of Human ABCB1Shuko Tachibana, Kouichi Yoshinari, Tsubasa Chikada, Takayoshi Toriyabe, Kiyoshi Nagata and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1604-1610; DOI: https://doi.org/10.1124/dmd.109.027219
- You have accessSelective Role of Sulfotransferase 2A1 (SULT2A1) in the N-Sulfoconjugation of Quinolone Drugs in HumansLaddawan Senggunprai, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1711-1717; DOI: https://doi.org/10.1124/dmd.109.027441
Yang, Zheng
- You have accessFurther Assessment of 17α-Ethinyl Estradiol as an Inhibitor of Different Human Cytochrome P450 Forms in VitroShu-Ying Chang, Cliff Chen, Zheng Yang and A. David RodriguesDrug Metabolism and Disposition August 2009, 37 (8) 1667-1675; DOI: https://doi.org/10.1124/dmd.109.026997
Yokoi, Tsuyoshi
- You have accessQuantitative Analysis of UDP-Glucuronosyltransferase (UGT) 1A and UGT2B Expression Levels in Human LiversTakeshi Izukawa, Miki Nakajima, Ryoichi Fujiwara, Hiroyuki Yamanaka, Tatsuki Fukami, Masataka Takamiya, Yasuhiro Aoki, Shin-ichi Ikushiro, Toshiyuki Sakaki and Tsuyoshi YokoiDrug Metabolism and Disposition August 2009, 37 (8) 1759-1768; DOI: https://doi.org/10.1124/dmd.109.027227
Yokota, Takao
- You have accessMetabolite Profiling of Hydroxycinnamate Derivatives in Plasma and Urine after the Ingestion of Coffee by Humans: Identification of Biomarkers of Coffee ConsumptionAngélique Stalmach, William Mullen, Denis Barron, Kenichi Uchida, Takao Yokota, Christophe Cavin, Heike Steiling, Gary Williamson and Alan CrozierDrug Metabolism and Disposition August 2009, 37 (8) 1749-1758; DOI: https://doi.org/10.1124/dmd.109.028019
Yoshinari, Kouichi
- You have accessInvolvement of Vitamin D Receptor in the Intestinal Induction of Human ABCB1Shuko Tachibana, Kouichi Yoshinari, Tsubasa Chikada, Takayoshi Toriyabe, Kiyoshi Nagata and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1604-1610; DOI: https://doi.org/10.1124/dmd.109.027219
- You have accessSelective Role of Sulfotransferase 2A1 (SULT2A1) in the N-Sulfoconjugation of Quinolone Drugs in HumansLaddawan Senggunprai, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition August 2009, 37 (8) 1711-1717; DOI: https://doi.org/10.1124/dmd.109.027441
Youdim, Kuresh
- You have accessComparison of Different Algorithms for Predicting Clinical Drug-Drug Interactions, Based on the Use of CYP3A4 in Vitro Data: Predictions of Compounds as Precipitants of InteractionOdette A. Fahmi, Susan Hurst, David Plowchalk, Jack Cook, Feng Guo, Kuresh Youdim, Maurice Dickins, Alex Phipps, Amanda Darekar, Ruth Hyland and R. Scott ObachDrug Metabolism and Disposition August 2009, 37 (8) 1658-1666; DOI: https://doi.org/10.1124/dmd.108.026252
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Zenser, Terry V.
- You have accessIdentification of New 2-Amino-3-methylimidazo[4,5-f]quinoline Urinary Metabolites from β-Naphthoflavone-Treated MiceVijaya M. Lakshmi, Fong-Fu Hsu and Terry V. ZenserDrug Metabolism and Disposition August 2009, 37 (8) 1690-1697; DOI: https://doi.org/10.1124/dmd.109.027342
Zhang, Donglu
- You have accessComparative Metabolism of 14C-Labeled Apixaban in Mice, Rats, Rabbits, Dogs, and HumansDonglu Zhang, Kan He, Nirmala Raghavan, Lifei Wang, James Mitroka, Brad D. Maxwell, Robert M. Knabb, Charles Frost, Alan Schuster, Feng Hao, Zheming Gu, W. Griffith Humphreys and Scott J. GrossmanDrug Metabolism and Disposition August 2009, 37 (8) 1738-1748; DOI: https://doi.org/10.1124/dmd.108.025981
Zhang, Xin
- You have accessSemiphysiologically Based Pharmacokinetic Models for the Inhibition of Midazolam Clearance by Diltiazem and Its Major MetaboliteXin Zhang, Sara K. Quinney, J. Christopher Gorski, David R. Jones and Stephen D. HallDrug Metabolism and Disposition August 2009, 37 (8) 1587-1597; DOI: https://doi.org/10.1124/dmd.109.026658
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