Index by author
September 01, 2010; Volume 38,Issue 9
A
Ahmad, Syed
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Aida, Yoshie
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Al Khansa, Ihab
- You have accessLiverbeads: A Practical and Relevant In Vitro Model for Gene Induction InvestigationsIhab Al Khansa, Olivier Blanck, André Guillouzo and Rémi BarsDrug Metabolism and Disposition September 2010, 38 (9) 1598-1604; DOI: https://doi.org/10.1124/dmd.110.033753
Amundsen, Rune
- You have accessCyclosporine A, but Not Tacrolimus, Shows Relevant Inhibition of Organic Anion-Transporting Protein 1B1-Mediated Transport of AtorvastatinRune Amundsen, Hege Christensen, Behnaz Zabihyan and Anders ÅsbergDrug Metabolism and Disposition September 2010, 38 (9) 1499-1504; DOI: https://doi.org/10.1124/dmd.110.032268
Annaert, Pieter
- You have accessIn Situ Intestinal Perfusion in Knockout Mice Demonstrates Inhibition of Intestinal P-Glycoprotein by Ritonavir Causing Increased Darunavir AbsorptionNico Holmstock, Raf Mols, Pieter Annaert and Patrick AugustijnsDrug Metabolism and Disposition September 2010, 38 (9) 1407-1410; DOI: https://doi.org/10.1124/dmd.110.032771
Arakawa, Shingo
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Åsberg, Anders
- You have accessCyclosporine A, but Not Tacrolimus, Shows Relevant Inhibition of Organic Anion-Transporting Protein 1B1-Mediated Transport of AtorvastatinRune Amundsen, Hege Christensen, Behnaz Zabihyan and Anders ÅsbergDrug Metabolism and Disposition September 2010, 38 (9) 1499-1504; DOI: https://doi.org/10.1124/dmd.110.032268
Augustijns, Patrick
- You have accessIn Situ Intestinal Perfusion in Knockout Mice Demonstrates Inhibition of Intestinal P-Glycoprotein by Ritonavir Causing Increased Darunavir AbsorptionNico Holmstock, Raf Mols, Pieter Annaert and Patrick AugustijnsDrug Metabolism and Disposition September 2010, 38 (9) 1407-1410; DOI: https://doi.org/10.1124/dmd.110.032771
B
Baierl, Juergen
- You have accessThe Dipeptidyl Peptidase-4 Inhibitor Linagliptin Exhibits Time- and Dose-Dependent Localization in Kidney, Liver, and Intestine after Intravenous Dosing: Results from High Resolution Autoradiography in RatsAndreas Greischel, Rudolf Binder and Juergen BaierlDrug Metabolism and Disposition September 2010, 38 (9) 1443-1448; DOI: https://doi.org/10.1124/dmd.110.034199
Balani, Suresh K.
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Balbo, Silvia
- You have accessPreferential Glutathione Conjugation of a Reverse Diol Epoxide Compared with a Bay Region Diol Epoxide of Benzo[a]pyrene in Human HepatocytesPramod Upadhyaya, J. Bradley Hochalter, Silvia Balbo, Edward J. McIntee and Stephen S. HechtDrug Metabolism and Disposition September 2010, 38 (9) 1397-1402; DOI: https://doi.org/10.1124/dmd.110.034181
Baldwin, William S.
- You have accessConstitutive Androgen Receptor-Null Mice Are Sensitive to the Toxic Effects of Parathion: Association with Reduced Cytochrome P450-Mediated Parathion MetabolismLinda C. Mota, Juan P. Hernandez and William S. BaldwinDrug Metabolism and Disposition September 2010, 38 (9) 1582-1588; DOI: https://doi.org/10.1124/dmd.110.032961
Bars, Rémi
- You have accessLiverbeads: A Practical and Relevant In Vitro Model for Gene Induction InvestigationsIhab Al Khansa, Olivier Blanck, André Guillouzo and Rémi BarsDrug Metabolism and Disposition September 2010, 38 (9) 1598-1604; DOI: https://doi.org/10.1124/dmd.110.033753
Belvin, Marcia
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Binder, Rudolf
- You have accessThe Dipeptidyl Peptidase-4 Inhibitor Linagliptin Exhibits Time- and Dose-Dependent Localization in Kidney, Liver, and Intestine after Intravenous Dosing: Results from High Resolution Autoradiography in RatsAndreas Greischel, Rudolf Binder and Juergen BaierlDrug Metabolism and Disposition September 2010, 38 (9) 1443-1448; DOI: https://doi.org/10.1124/dmd.110.034199
Blanck, Olivier
- You have accessLiverbeads: A Practical and Relevant In Vitro Model for Gene Induction InvestigationsIhab Al Khansa, Olivier Blanck, André Guillouzo and Rémi BarsDrug Metabolism and Disposition September 2010, 38 (9) 1598-1604; DOI: https://doi.org/10.1124/dmd.110.033753
Boldt, Sherri
- You have accessCytochrome P450 3A4 mRNA Is a More Reliable Marker than CYP3A4 Activity for Detecting Pregnane X Receptor-Activated Induction of Drug-Metabolizing EnzymesOdette A. Fahmi, Mary Kish, Sherri Boldt and R. Scott ObachDrug Metabolism and Disposition September 2010, 38 (9) 1605-1611; DOI: https://doi.org/10.1124/dmd.110.033126
Bradford, Delia
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Bungay, Peter
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Butler, Kathleen
- You have accessAbsorption, Distribution, Metabolism, and Excretion of Ticagrelor in Healthy SubjectsRenli Teng, Stuart Oliver, Martin A. Hayes and Kathleen ButlerDrug Metabolism and Disposition September 2010, 38 (9) 1514-1521; DOI: https://doi.org/10.1124/dmd.110.032250
C
Castell, José V.
- You have accessMetabolite Formation Kinetics and Intrinsic Clearance of Phenacetin, Tolbutamide, Alprazolam, and Midazolam in Adenoviral Cytochrome P450-Transfected HepG2 Cells and Comparison with Hepatocytes and In VivoM. Teresa Donato, David Hallifax, Laura Picazo, José V. Castell, J. Brian Houston, M. José Gomez-Lechón and Agustin LahozDrug Metabolism and Disposition September 2010, 38 (9) 1449-1455; DOI: https://doi.org/10.1124/dmd.110.033605
Chandrasekaran, Appavu
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Chen, Chao
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
Chen, Michael
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Chen, Taosheng
- You have accessProtein Phosphatase 2Cβl Regulates Human Pregnane X Receptor-Mediated CYP3A4 Gene Expression in HepG2 Liver Carcinoma CellsSatyanarayana R. Pondugula, Alexander A. Tong, Jing Wu, Jimmy Cui and Taosheng ChenDrug Metabolism and Disposition September 2010, 38 (9) 1411-1416; DOI: https://doi.org/10.1124/dmd.110.032128
Chiba, Koji
- You have accessEffect of the CYP2D6*10 Genotype on Tolterodine PharmacokineticsMasayo Oishi, Koji Chiba, Bimal Malhotra and Toshio SuwaDrug Metabolism and Disposition September 2010, 38 (9) 1456-1463; DOI: https://doi.org/10.1124/dmd.110.033407
Cho, Sool Yeon
- You have accessDiscontinuous Drug Binding to Proteins: Binding of an Antineoplastic Benzyl Styryl Sulfone to Albumin and Enzymes In Vitro and in Phase I Clinical TrialsSool Yeon Cho, Takao Ohnuma, Lewis R. Silverman, James F. Holland and John RobozDrug Metabolism and Disposition September 2010, 38 (9) 1480-1485; DOI: https://doi.org/10.1124/dmd.110.033001
Christensen, Hege
- You have accessCyclosporine A, but Not Tacrolimus, Shows Relevant Inhibition of Organic Anion-Transporting Protein 1B1-Mediated Transport of AtorvastatinRune Amundsen, Hege Christensen, Behnaz Zabihyan and Anders ÅsbergDrug Metabolism and Disposition September 2010, 38 (9) 1499-1504; DOI: https://doi.org/10.1124/dmd.110.032268
Chuang, Bei-Ching
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Claessens, Adam J.
- You have accessCYP2D6 Mediates 4-Hydroxylation of Clonidine In Vitro: Implication for Pregnancy-Induced Changes in Clonidine ClearanceAdam J. Claessens, Linda J. Risler, Sara Eyal, Danny D. Shen, Thomas R. Easterling and Mary F. HebertDrug Metabolism and Disposition September 2010, 38 (9) 1393-1396; DOI: https://doi.org/10.1124/dmd.110.033878
Covas, Maria-Isabel
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
Cui, Jimmy
- You have accessProtein Phosphatase 2Cβl Regulates Human Pregnane X Receptor-Mediated CYP3A4 Gene Expression in HepG2 Liver Carcinoma CellsSatyanarayana R. Pondugula, Alexander A. Tong, Jing Wu, Jimmy Cui and Taosheng ChenDrug Metabolism and Disposition September 2010, 38 (9) 1411-1416; DOI: https://doi.org/10.1124/dmd.110.032128
D
de la Torre, Rafael
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
DeMaio, William
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Donato, M. Teresa
- You have accessMetabolite Formation Kinetics and Intrinsic Clearance of Phenacetin, Tolbutamide, Alprazolam, and Midazolam in Adenoviral Cytochrome P450-Transfected HepG2 Cells and Comparison with Hepatocytes and In VivoM. Teresa Donato, David Hallifax, Laura Picazo, José V. Castell, J. Brian Houston, M. José Gomez-Lechón and Agustin LahozDrug Metabolism and Disposition September 2010, 38 (9) 1449-1455; DOI: https://doi.org/10.1124/dmd.110.033605
Dreifinger, Tali
- You have accessRole of P-Glycoprotein in Region-Specific Gastrointestinal Absorption of Talinolol in RatsLeonid Kagan, Tali Dreifinger, Donald E. Mager and Amnon HoffmanDrug Metabolism and Disposition September 2010, 38 (9) 1560-1566; DOI: https://doi.org/10.1124/dmd.110.033019
E
Easterling, Thomas R.
- You have accessCYP2D6 Mediates 4-Hydroxylation of Clonidine In Vitro: Implication for Pregnancy-Induced Changes in Clonidine ClearanceAdam J. Claessens, Linda J. Risler, Sara Eyal, Danny D. Shen, Thomas R. Easterling and Mary F. HebertDrug Metabolism and Disposition September 2010, 38 (9) 1393-1396; DOI: https://doi.org/10.1124/dmd.110.033878
Ebner, Thomas
- You have accessDabigatran Acylglucuronide, the Major Human Metabolite of Dabigatran: In Vitro Formation, Stability, and Pharmacological ActivityThomas Ebner, Klaus Wagner and Wolfgang WienenDrug Metabolism and Disposition September 2010, 38 (9) 1567-1575; DOI: https://doi.org/10.1124/dmd.110.033696
Edgar, Kyle A.
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Eyal, Sara
- You have accessCYP2D6 Mediates 4-Hydroxylation of Clonidine In Vitro: Implication for Pregnancy-Induced Changes in Clonidine ClearanceAdam J. Claessens, Linda J. Risler, Sara Eyal, Danny D. Shen, Thomas R. Easterling and Mary F. HebertDrug Metabolism and Disposition September 2010, 38 (9) 1393-1396; DOI: https://doi.org/10.1124/dmd.110.033878
F
Fahmi, Odette A.
- You have accessCytochrome P450 3A4 mRNA Is a More Reliable Marker than CYP3A4 Activity for Detecting Pregnane X Receptor-Activated Induction of Drug-Metabolizing EnzymesOdette A. Fahmi, Mary Kish, Sherri Boldt and R. Scott ObachDrug Metabolism and Disposition September 2010, 38 (9) 1605-1611; DOI: https://doi.org/10.1124/dmd.110.033126
Farré, Magí
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
Feidt, Diana M.
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Fitó, Montserat
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
Fujimoto, Kazunori
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Fukami, Tatsuki
- You have accessArylacetamide Deacetylase Is a Determinant Enzyme for the Difference in Hydrolase Activities of Phenacetin and AcetaminophenAkinobu Watanabe, Tatsuki Fukami, Shiori Takahashi, Yuki Kobayashi, Nao Nakagawa, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition September 2010, 38 (9) 1532-1537; DOI: https://doi.org/10.1124/dmd.110.033720
Fukuda, Hajime
- You have accessEstimation of Transporters Involved in the Hepatobiliary Transport of TA-0201CA Using Sandwich-Cultured Rat Hepatocytes from Normal and Multidrug Resistance-Associated Protein 2-Deficient RatsHajime Fukuda, Rikiya Ohashi, Noriko Ohashi, Hikaru Yabuuchi and Ikumi TamaiDrug Metabolism and Disposition September 2010, 38 (9) 1505-1513; DOI: https://doi.org/10.1124/dmd.110.033258
G
Gomez-Lechón, M. José
- You have accessMetabolite Formation Kinetics and Intrinsic Clearance of Phenacetin, Tolbutamide, Alprazolam, and Midazolam in Adenoviral Cytochrome P450-Transfected HepG2 Cells and Comparison with Hepatocytes and In VivoM. Teresa Donato, David Hallifax, Laura Picazo, José V. Castell, J. Brian Houston, M. José Gomez-Lechón and Agustin LahozDrug Metabolism and Disposition September 2010, 38 (9) 1449-1455; DOI: https://doi.org/10.1124/dmd.110.033605
Greischel, Andreas
- You have accessThe Dipeptidyl Peptidase-4 Inhibitor Linagliptin Exhibits Time- and Dose-Dependent Localization in Kidney, Liver, and Intestine after Intravenous Dosing: Results from High Resolution Autoradiography in RatsAndreas Greischel, Rudolf Binder and Juergen BaierlDrug Metabolism and Disposition September 2010, 38 (9) 1443-1448; DOI: https://doi.org/10.1124/dmd.110.034199
Guillouzo, André
- You have accessLiverbeads: A Practical and Relevant In Vitro Model for Gene Induction InvestigationsIhab Al Khansa, Olivier Blanck, André Guillouzo and Rémi BarsDrug Metabolism and Disposition September 2010, 38 (9) 1598-1604; DOI: https://doi.org/10.1124/dmd.110.033753
H
Hallifax, David
- You have accessMetabolite Formation Kinetics and Intrinsic Clearance of Phenacetin, Tolbutamide, Alprazolam, and Midazolam in Adenoviral Cytochrome P450-Transfected HepG2 Cells and Comparison with Hepatocytes and In VivoM. Teresa Donato, David Hallifax, Laura Picazo, José V. Castell, J. Brian Houston, M. José Gomez-Lechón and Agustin LahozDrug Metabolism and Disposition September 2010, 38 (9) 1449-1455; DOI: https://doi.org/10.1124/dmd.110.033605
Hayes, Martin A.
- You have accessAbsorption, Distribution, Metabolism, and Excretion of Ticagrelor in Healthy SubjectsRenli Teng, Stuart Oliver, Martin A. Hayes and Kathleen ButlerDrug Metabolism and Disposition September 2010, 38 (9) 1514-1521; DOI: https://doi.org/10.1124/dmd.110.032250
Hebert, Mary F.
- You have accessCYP2D6 Mediates 4-Hydroxylation of Clonidine In Vitro: Implication for Pregnancy-Induced Changes in Clonidine ClearanceAdam J. Claessens, Linda J. Risler, Sara Eyal, Danny D. Shen, Thomas R. Easterling and Mary F. HebertDrug Metabolism and Disposition September 2010, 38 (9) 1393-1396; DOI: https://doi.org/10.1124/dmd.110.033878
- You have accessIncreased Glyburide Clearance in the Pregnant Mouse ModelLin Zhou, Yi Zhang, Mary F. Hebert, Jashvant D. Unadkat and Qingcheng MaoDrug Metabolism and Disposition September 2010, 38 (9) 1403-1406; DOI: https://doi.org/10.1124/dmd.110.033837
Hecht, Stephen S.
- You have accessPreferential Glutathione Conjugation of a Reverse Diol Epoxide Compared with a Bay Region Diol Epoxide of Benzo[a]pyrene in Human HepatocytesPramod Upadhyaya, J. Bradley Hochalter, Silvia Balbo, Edward J. McIntee and Stephen S. HechtDrug Metabolism and Disposition September 2010, 38 (9) 1397-1402; DOI: https://doi.org/10.1124/dmd.110.034181
Hernandez, Juan P.
- You have accessConstitutive Androgen Receptor-Null Mice Are Sensitive to the Toxic Effects of Parathion: Association with Reduced Cytochrome P450-Mediated Parathion MetabolismLinda C. Mota, Juan P. Hernandez and William S. BaldwinDrug Metabolism and Disposition September 2010, 38 (9) 1582-1588; DOI: https://doi.org/10.1124/dmd.110.032961
Heyde, Bruce R.
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Hochalter, J. Bradley
- You have accessPreferential Glutathione Conjugation of a Reverse Diol Epoxide Compared with a Bay Region Diol Epoxide of Benzo[a]pyrene in Human HepatocytesPramod Upadhyaya, J. Bradley Hochalter, Silvia Balbo, Edward J. McIntee and Stephen S. HechtDrug Metabolism and Disposition September 2010, 38 (9) 1397-1402; DOI: https://doi.org/10.1124/dmd.110.034181
Hoffman, Amnon
- You have accessRole of P-Glycoprotein in Region-Specific Gastrointestinal Absorption of Talinolol in RatsLeonid Kagan, Tali Dreifinger, Donald E. Mager and Amnon HoffmanDrug Metabolism and Disposition September 2010, 38 (9) 1560-1566; DOI: https://doi.org/10.1124/dmd.110.033019
Hofmann, Ute
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Holland, James F.
- You have accessDiscontinuous Drug Binding to Proteins: Binding of an Antineoplastic Benzyl Styryl Sulfone to Albumin and Enzymes In Vitro and in Phase I Clinical TrialsSool Yeon Cho, Takao Ohnuma, Lewis R. Silverman, James F. Holland and John RobozDrug Metabolism and Disposition September 2010, 38 (9) 1480-1485; DOI: https://doi.org/10.1124/dmd.110.033001
Holmstock, Nico
- You have accessIn Situ Intestinal Perfusion in Knockout Mice Demonstrates Inhibition of Intestinal P-Glycoprotein by Ritonavir Causing Increased Darunavir AbsorptionNico Holmstock, Raf Mols, Pieter Annaert and Patrick AugustijnsDrug Metabolism and Disposition September 2010, 38 (9) 1407-1410; DOI: https://doi.org/10.1124/dmd.110.032771
Horiguchi, Norio
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
Houston, J. Brian
- You have accessMetabolite Formation Kinetics and Intrinsic Clearance of Phenacetin, Tolbutamide, Alprazolam, and Midazolam in Adenoviral Cytochrome P450-Transfected HepG2 Cells and Comparison with Hepatocytes and In VivoM. Teresa Donato, David Hallifax, Laura Picazo, José V. Castell, J. Brian Houston, M. José Gomez-Lechón and Agustin LahozDrug Metabolism and Disposition September 2010, 38 (9) 1449-1455; DOI: https://doi.org/10.1124/dmd.110.033605
Hu, Yiding
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Hultin, Theresa
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
I
Ichikawa, Takeshi
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
J
Janjetovic, Zorica
- You have accessPurified Mouse CYP27B1 Can Hydroxylate 20,23-Dihydroxyvitamin D3, Producing 1α,20,23-Trihydroxyvitamin D3, Which Has Altered Biological ActivityEdith K. Y. Tang, Wei Li, Zorica Janjetovic, Minh N. Nguyen, Zhao Wang, Andrzej Slominski and Robert C. TuckeyDrug Metabolism and Disposition September 2010, 38 (9) 1553-1559; DOI: https://doi.org/10.1124/dmd.110.034389
Joglar, Jesús
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
K
Kagan, Leonid
- You have accessRole of P-Glycoprotein in Region-Specific Gastrointestinal Absorption of Talinolol in RatsLeonid Kagan, Tali Dreifinger, Donald E. Mager and Amnon HoffmanDrug Metabolism and Disposition September 2010, 38 (9) 1560-1566; DOI: https://doi.org/10.1124/dmd.110.033019
Kakizaki, Satoru
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
Kawai, Ryota
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Khymenets, Olha
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
Kish, Mary
- You have accessCytochrome P450 3A4 mRNA Is a More Reliable Marker than CYP3A4 Activity for Detecting Pregnane X Receptor-Activated Induction of Drug-Metabolizing EnzymesOdette A. Fahmi, Mary Kish, Sherri Boldt and R. Scott ObachDrug Metabolism and Disposition September 2010, 38 (9) 1605-1611; DOI: https://doi.org/10.1124/dmd.110.033126
Kitagaki, Shinji
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Kiyosawa, Naoki
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Klein, Kathrin
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Knobeloch, Daniel
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Kobayashi, Nobuhiro
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
Kobayashi, Yasuna
- You have accessActivation of Cyclosporin A Transport by a Novel λ Light Chain of Human Ig Surface Antigen-Related Gene in Xenopus laevis OocytesYasuna Kobayashi, Takahiro Umemoto, Masayuki Ohbayashi, Noriko Kohyama, Yutaka Sanada and Toshinori YamamotoDrug Metabolism and Disposition September 2010, 38 (9) 1427-1435; DOI: https://doi.org/10.1124/dmd.109.030916
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Kobayashi, Yuki
- You have accessArylacetamide Deacetylase Is a Determinant Enzyme for the Difference in Hydrolase Activities of Phenacetin and AcetaminophenAkinobu Watanabe, Tatsuki Fukami, Shiori Takahashi, Yuki Kobayashi, Nao Nakagawa, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition September 2010, 38 (9) 1532-1537; DOI: https://doi.org/10.1124/dmd.110.033720
Kohara, Sakae
- You have accessCynomolgus Monkey CYP2D44 Newly Identified in Liver, Metabolizes Bufuralol, and DextromethorphanYasuhiro Uno, Shotaro Uehara, Sakae Kohara, Norie Murayama and Hiroshi YamazakiDrug Metabolism and Disposition September 2010, 38 (9) 1486-1492; DOI: https://doi.org/10.1124/dmd.110.033274
Kohyama, Noriko
- You have accessActivation of Cyclosporin A Transport by a Novel λ Light Chain of Human Ig Surface Antigen-Related Gene in Xenopus laevis OocytesYasuna Kobayashi, Takahiro Umemoto, Masayuki Ohbayashi, Noriko Kohyama, Yutaka Sanada and Toshinori YamamotoDrug Metabolism and Disposition September 2010, 38 (9) 1427-1435; DOI: https://doi.org/10.1124/dmd.109.030916
Kose, Noriko
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Kubota, Kazuishi
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
L
Lahoz, Agustin
- You have accessMetabolite Formation Kinetics and Intrinsic Clearance of Phenacetin, Tolbutamide, Alprazolam, and Midazolam in Adenoviral Cytochrome P450-Transfected HepG2 Cells and Comparison with Hepatocytes and In VivoM. Teresa Donato, David Hallifax, Laura Picazo, José V. Castell, J. Brian Houston, M. José Gomez-Lechón and Agustin LahozDrug Metabolism and Disposition September 2010, 38 (9) 1449-1455; DOI: https://doi.org/10.1124/dmd.110.033605
Lai, Yurong
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Lee, David
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Lee, Frank W.
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Lee, Leslie B.
- You have accessRole of P-Glycoprotein and Breast Cancer Resistance Protein-1 in the Brain Penetration and Brain Pharmacodynamic Activity of the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Leslie B. Lee, Jodie Pang, Emile G. Plise and Xiaolin ZhangDrug Metabolism and Disposition September 2010, 38 (9) 1422-1426; DOI: https://doi.org/10.1124/dmd.110.034256
Li, Wei
- You have accessPurified Mouse CYP27B1 Can Hydroxylate 20,23-Dihydroxyvitamin D3, Producing 1α,20,23-Trihydroxyvitamin D3, Which Has Altered Biological ActivityEdith K. Y. Tang, Wei Li, Zorica Janjetovic, Minh N. Nguyen, Zhao Wang, Andrzej Slominski and Robert C. TuckeyDrug Metabolism and Disposition September 2010, 38 (9) 1553-1559; DOI: https://doi.org/10.1124/dmd.110.034389
Liao, Mingxiang
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Liu, Duan
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
M
Maejima, Takanori
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Mager, Donald E.
- You have accessRole of P-Glycoprotein in Region-Specific Gastrointestinal Absorption of Talinolol in RatsLeonid Kagan, Tali Dreifinger, Donald E. Mager and Amnon HoffmanDrug Metabolism and Disposition September 2010, 38 (9) 1560-1566; DOI: https://doi.org/10.1124/dmd.110.033019
Malhotra, Bimal
- You have accessEffect of the CYP2D6*10 Genotype on Tolterodine PharmacokineticsMasayo Oishi, Koji Chiba, Bimal Malhotra and Toshio SuwaDrug Metabolism and Disposition September 2010, 38 (9) 1456-1463; DOI: https://doi.org/10.1124/dmd.110.033407
Manabe, Sunao
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Mandrell, Kathy M.
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Mao, Qingcheng
- You have accessIncreased Glyburide Clearance in the Pregnant Mouse ModelLin Zhou, Yi Zhang, Mary F. Hebert, Jashvant D. Unadkat and Qingcheng MaoDrug Metabolism and Disposition September 2010, 38 (9) 1403-1406; DOI: https://doi.org/10.1124/dmd.110.033837
McIntee, Edward J.
- You have accessPreferential Glutathione Conjugation of a Reverse Diol Epoxide Compared with a Bay Region Diol Epoxide of Benzo[a]pyrene in Human HepatocytesPramod Upadhyaya, J. Bradley Hochalter, Silvia Balbo, Edward J. McIntee and Stephen S. HechtDrug Metabolism and Disposition September 2010, 38 (9) 1397-1402; DOI: https://doi.org/10.1124/dmd.110.034181
Miura, Shin-ichi
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
Miyakoshi, Naoki
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Mols, Raf
- You have accessIn Situ Intestinal Perfusion in Knockout Mice Demonstrates Inhibition of Intestinal P-Glycoprotein by Ritonavir Causing Increased Darunavir AbsorptionNico Holmstock, Raf Mols, Pieter Annaert and Patrick AugustijnsDrug Metabolism and Disposition September 2010, 38 (9) 1407-1410; DOI: https://doi.org/10.1124/dmd.110.032771
Mori, Masatomo
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
Morrison, Jodi
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Mota, Linda C.
- You have accessConstitutive Androgen Receptor-Null Mice Are Sensitive to the Toxic Effects of Parathion: Association with Reduced Cytochrome P450-Mediated Parathion MetabolismLinda C. Mota, Juan P. Hernandez and William S. BaldwinDrug Metabolism and Disposition September 2010, 38 (9) 1582-1588; DOI: https://doi.org/10.1124/dmd.110.032961
Mukai, Chisato
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Muñoz-Aguayo, Daniel
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
Murayama, Norie
- You have accessCynomolgus Monkey CYP2D44 Newly Identified in Liver, Metabolizes Bufuralol, and DextromethorphanYasuhiro Uno, Shotaro Uehara, Sakae Kohara, Norie Murayama and Hiroshi YamazakiDrug Metabolism and Disposition September 2010, 38 (9) 1486-1492; DOI: https://doi.org/10.1124/dmd.110.033274
N
Nakagawa, Nao
- You have accessArylacetamide Deacetylase Is a Determinant Enzyme for the Difference in Hydrolase Activities of Phenacetin and AcetaminophenAkinobu Watanabe, Tatsuki Fukami, Shiori Takahashi, Yuki Kobayashi, Nao Nakagawa, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition September 2010, 38 (9) 1532-1537; DOI: https://doi.org/10.1124/dmd.110.033720
Nakai, Daisuke
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
Nakajima, Miki
- You have accessArylacetamide Deacetylase Is a Determinant Enzyme for the Difference in Hydrolase Activities of Phenacetin and AcetaminophenAkinobu Watanabe, Tatsuki Fukami, Shiori Takahashi, Yuki Kobayashi, Nao Nakagawa, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition September 2010, 38 (9) 1532-1537; DOI: https://doi.org/10.1124/dmd.110.033720
Nakashima, Emi
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Nan, Yefei
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
Nguyen, Minh N.
- You have accessPurified Mouse CYP27B1 Can Hydroxylate 20,23-Dihydroxyvitamin D3, Producing 1α,20,23-Trihydroxyvitamin D3, Which Has Altered Biological ActivityEdith K. Y. Tang, Wei Li, Zorica Janjetovic, Minh N. Nguyen, Zhao Wang, Andrzej Slominski and Robert C. TuckeyDrug Metabolism and Disposition September 2010, 38 (9) 1553-1559; DOI: https://doi.org/10.1124/dmd.110.034389
Nishimura, Tomohiro
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
O
Obach, R. Scott
- You have accessCytochrome P450 3A4 mRNA Is a More Reliable Marker than CYP3A4 Activity for Detecting Pregnane X Receptor-Activated Induction of Drug-Metabolizing EnzymesOdette A. Fahmi, Mary Kish, Sherri Boldt and R. Scott ObachDrug Metabolism and Disposition September 2010, 38 (9) 1605-1611; DOI: https://doi.org/10.1124/dmd.110.033126
Ochi, Kaori
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Oganesian, Aram
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Ogura, Yuji
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
Ohashi, Noriko
- You have accessEstimation of Transporters Involved in the Hepatobiliary Transport of TA-0201CA Using Sandwich-Cultured Rat Hepatocytes from Normal and Multidrug Resistance-Associated Protein 2-Deficient RatsHajime Fukuda, Rikiya Ohashi, Noriko Ohashi, Hikaru Yabuuchi and Ikumi TamaiDrug Metabolism and Disposition September 2010, 38 (9) 1505-1513; DOI: https://doi.org/10.1124/dmd.110.033258
Ohashi, Rikiya
- You have accessEstimation of Transporters Involved in the Hepatobiliary Transport of TA-0201CA Using Sandwich-Cultured Rat Hepatocytes from Normal and Multidrug Resistance-Associated Protein 2-Deficient RatsHajime Fukuda, Rikiya Ohashi, Noriko Ohashi, Hikaru Yabuuchi and Ikumi TamaiDrug Metabolism and Disposition September 2010, 38 (9) 1505-1513; DOI: https://doi.org/10.1124/dmd.110.033258
Ohbayashi, Masayuki
- You have accessActivation of Cyclosporin A Transport by a Novel λ Light Chain of Human Ig Surface Antigen-Related Gene in Xenopus laevis OocytesYasuna Kobayashi, Takahiro Umemoto, Masayuki Ohbayashi, Noriko Kohyama, Yutaka Sanada and Toshinori YamamotoDrug Metabolism and Disposition September 2010, 38 (9) 1427-1435; DOI: https://doi.org/10.1124/dmd.109.030916
Ohnuma, Takao
- You have accessDiscontinuous Drug Binding to Proteins: Binding of an Antineoplastic Benzyl Styryl Sulfone to Albumin and Enzymes In Vitro and in Phase I Clinical TrialsSool Yeon Cho, Takao Ohnuma, Lewis R. Silverman, James F. Holland and John RobozDrug Metabolism and Disposition September 2010, 38 (9) 1480-1485; DOI: https://doi.org/10.1124/dmd.110.033001
Oishi, Masayo
- You have accessEffect of the CYP2D6*10 Genotype on Tolterodine PharmacokineticsMasayo Oishi, Koji Chiba, Bimal Malhotra and Toshio SuwaDrug Metabolism and Disposition September 2010, 38 (9) 1456-1463; DOI: https://doi.org/10.1124/dmd.110.033407
Okazaki, Osamu
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
Oliver, Stuart
- You have accessAbsorption, Distribution, Metabolism, and Excretion of Ticagrelor in Healthy SubjectsRenli Teng, Stuart Oliver, Martin A. Hayes and Kathleen ButlerDrug Metabolism and Disposition September 2010, 38 (9) 1514-1521; DOI: https://doi.org/10.1124/dmd.110.032250
P
Pang, Jodie
- You have accessRole of P-Glycoprotein and Breast Cancer Resistance Protein-1 in the Brain Penetration and Brain Pharmacodynamic Activity of the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Leslie B. Lee, Jodie Pang, Emile G. Plise and Xiaolin ZhangDrug Metabolism and Disposition September 2010, 38 (9) 1422-1426; DOI: https://doi.org/10.1124/dmd.110.034256
Park, SeongHee
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Picazo, Laura
- You have accessMetabolite Formation Kinetics and Intrinsic Clearance of Phenacetin, Tolbutamide, Alprazolam, and Midazolam in Adenoviral Cytochrome P450-Transfected HepG2 Cells and Comparison with Hepatocytes and In VivoM. Teresa Donato, David Hallifax, Laura Picazo, José V. Castell, J. Brian Houston, M. José Gomez-Lechón and Agustin LahozDrug Metabolism and Disposition September 2010, 38 (9) 1449-1455; DOI: https://doi.org/10.1124/dmd.110.033605
Plise, Emile G.
- You have accessRole of P-Glycoprotein and Breast Cancer Resistance Protein-1 in the Brain Penetration and Brain Pharmacodynamic Activity of the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Leslie B. Lee, Jodie Pang, Emile G. Plise and Xiaolin ZhangDrug Metabolism and Disposition September 2010, 38 (9) 1422-1426; DOI: https://doi.org/10.1124/dmd.110.034256
Pondugula, Satyanarayana R.
- You have accessProtein Phosphatase 2Cβl Regulates Human Pregnane X Receptor-Mediated CYP3A4 Gene Expression in HepG2 Liver Carcinoma CellsSatyanarayana R. Pondugula, Alexander A. Tong, Jing Wu, Jimmy Cui and Taosheng ChenDrug Metabolism and Disposition September 2010, 38 (9) 1411-1416; DOI: https://doi.org/10.1124/dmd.110.032128
Prior, Wei Wei
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Pujadas, Mitona
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
R
Raczynski, Arek R.
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Reding, Matthew T.
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Riedmaier, Stephan
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Risler, Linda J.
- You have accessCYP2D6 Mediates 4-Hydroxylation of Clonidine In Vitro: Implication for Pregnancy-Induced Changes in Clonidine ClearanceAdam J. Claessens, Linda J. Risler, Sara Eyal, Danny D. Shen, Thomas R. Easterling and Mary F. HebertDrug Metabolism and Disposition September 2010, 38 (9) 1393-1396; DOI: https://doi.org/10.1124/dmd.110.033878
Robins, Russell H.
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Roboz, John
- You have accessDiscontinuous Drug Binding to Proteins: Binding of an Antineoplastic Benzyl Styryl Sulfone to Albumin and Enzymes In Vitro and in Phase I Clinical TrialsSool Yeon Cho, Takao Ohnuma, Lewis R. Silverman, James F. Holland and John RobozDrug Metabolism and Disposition September 2010, 38 (9) 1480-1485; DOI: https://doi.org/10.1124/dmd.110.033001
S
Sai, Yoshimichi
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Salphati, Laurent
- You have accessRole of P-Glycoprotein and Breast Cancer Resistance Protein-1 in the Brain Penetration and Brain Pharmacodynamic Activity of the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Leslie B. Lee, Jodie Pang, Emile G. Plise and Xiaolin ZhangDrug Metabolism and Disposition September 2010, 38 (9) 1422-1426; DOI: https://doi.org/10.1124/dmd.110.034256
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Sampath, Deepak
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Sanada, Yutaka
- You have accessActivation of Cyclosporin A Transport by a Novel λ Light Chain of Human Ig Surface Antigen-Related Gene in Xenopus laevis OocytesYasuna Kobayashi, Takahiro Umemoto, Masayuki Ohbayashi, Noriko Kohyama, Yutaka Sanada and Toshinori YamamotoDrug Metabolism and Disposition September 2010, 38 (9) 1427-1435; DOI: https://doi.org/10.1124/dmd.109.030916
Sato, Ken
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
Scatina, JoAnn
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Schwab, Matthias
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Shen, Danny D.
- You have accessCYP2D6 Mediates 4-Hydroxylation of Clonidine In Vitro: Implication for Pregnancy-Induced Changes in Clonidine ClearanceAdam J. Claessens, Linda J. Risler, Sara Eyal, Danny D. Shen, Thomas R. Easterling and Mary F. HebertDrug Metabolism and Disposition September 2010, 38 (9) 1393-1396; DOI: https://doi.org/10.1124/dmd.110.033878
Shen, Li
- You have accessIn Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in HumansLi Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay and Appavu ChandrasekaranDrug Metabolism and Disposition September 2010, 38 (9) 1471-1479; DOI: https://doi.org/10.1124/dmd.109.030999
Shibaya, Yukari
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Shilliday, F. Barclay
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Shipman, Rob
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Silverman, Lewis R.
- You have accessDiscontinuous Drug Binding to Proteins: Binding of an Antineoplastic Benzyl Styryl Sulfone to Albumin and Enzymes In Vitro and in Phase I Clinical TrialsSool Yeon Cho, Takao Ohnuma, Lewis R. Silverman, James F. Holland and John RobozDrug Metabolism and Disposition September 2010, 38 (9) 1480-1485; DOI: https://doi.org/10.1124/dmd.110.033001
Slominski, Andrzej
- You have accessPurified Mouse CYP27B1 Can Hydroxylate 20,23-Dihydroxyvitamin D3, Producing 1α,20,23-Trihydroxyvitamin D3, Which Has Altered Biological ActivityEdith K. Y. Tang, Wei Li, Zorica Janjetovic, Minh N. Nguyen, Zhao Wang, Andrzej Slominski and Robert C. TuckeyDrug Metabolism and Disposition September 2010, 38 (9) 1553-1559; DOI: https://doi.org/10.1124/dmd.110.034389
Suwa, Toshio
- You have accessEffect of the CYP2D6*10 Genotype on Tolterodine PharmacokineticsMasayo Oishi, Koji Chiba, Bimal Malhotra and Toshio SuwaDrug Metabolism and Disposition September 2010, 38 (9) 1456-1463; DOI: https://doi.org/10.1124/dmd.110.033407
Suzuki, Eiko
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
T
Takagi, Akinori
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Takahashi, Shiori
- You have accessArylacetamide Deacetylase Is a Determinant Enzyme for the Difference in Hydrolase Activities of Phenacetin and AcetaminophenAkinobu Watanabe, Tatsuki Fukami, Shiori Takahashi, Yuki Kobayashi, Nao Nakagawa, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition September 2010, 38 (9) 1532-1537; DOI: https://doi.org/10.1124/dmd.110.033720
Takasaki, Wataru
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Takizawa, Daichi
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
Tamai, Ikumi
- You have accessEstimation of Transporters Involved in the Hepatobiliary Transport of TA-0201CA Using Sandwich-Cultured Rat Hepatocytes from Normal and Multidrug Resistance-Associated Protein 2-Deficient RatsHajime Fukuda, Rikiya Ohashi, Noriko Ohashi, Hikaru Yabuuchi and Ikumi TamaiDrug Metabolism and Disposition September 2010, 38 (9) 1505-1513; DOI: https://doi.org/10.1124/dmd.110.033258
Tanaka, Noriaki
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Tang, Edith K. Y.
- You have accessPurified Mouse CYP27B1 Can Hydroxylate 20,23-Dihydroxyvitamin D3, Producing 1α,20,23-Trihydroxyvitamin D3, Which Has Altered Biological ActivityEdith K. Y. Tang, Wei Li, Zorica Janjetovic, Minh N. Nguyen, Zhao Wang, Andrzej Slominski and Robert C. TuckeyDrug Metabolism and Disposition September 2010, 38 (9) 1553-1559; DOI: https://doi.org/10.1124/dmd.110.034389
Tang, Yitong
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
Teng, Renli
- You have accessAbsorption, Distribution, Metabolism, and Excretion of Ticagrelor in Healthy SubjectsRenli Teng, Stuart Oliver, Martin A. Hayes and Kathleen ButlerDrug Metabolism and Disposition September 2010, 38 (9) 1514-1521; DOI: https://doi.org/10.1124/dmd.110.032250
Thasler, Wolfgang E.
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Thompson, David C.
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Tojima, Hiroki
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
Tomi, Masatoshi
- You have accessProton-Coupled Erythromycin Antiport at Rat Blood-Placenta BarrierYoshimichi Sai, Tomohiro Nishimura, Kaori Ochi, Noriaki Tanaka, Akinori Takagi, Masatoshi Tomi, Noriko Kose, Yasuna Kobayashi, Naoki Miyakoshi, Shinji Kitagaki, Chisato Mukai and Emi NakashimaDrug Metabolism and Disposition September 2010, 38 (9) 1576-1581; DOI: https://doi.org/10.1124/dmd.110.033266
Tong, Alexander A.
- You have accessProtein Phosphatase 2Cβl Regulates Human Pregnane X Receptor-Mediated CYP3A4 Gene Expression in HepG2 Liver Carcinoma CellsSatyanarayana R. Pondugula, Alexander A. Tong, Jing Wu, Jimmy Cui and Taosheng ChenDrug Metabolism and Disposition September 2010, 38 (9) 1411-1416; DOI: https://doi.org/10.1124/dmd.110.032128
Torres, Josep Lluis
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
Touriño, Sonia
- You have accessAntioxidant Activities of Hydroxytyrosol Main Metabolites Do Not Contribute to Beneficial Health Effects after Olive Oil IngestionOlha Khymenets, Montserat Fitó, Sonia Touriño, Daniel Muñoz-Aguayo, Mitona Pujadas, Josep Lluis Torres, Jesús Joglar, Magí Farré, Maria-Isabel Covas and Rafael de la TorreDrug Metabolism and Disposition September 2010, 38 (9) 1417-1421; DOI: https://doi.org/10.1124/dmd.110.032821
Tuckey, Robert C.
- You have accessPurified Mouse CYP27B1 Can Hydroxylate 20,23-Dihydroxyvitamin D3, Producing 1α,20,23-Trihydroxyvitamin D3, Which Has Altered Biological ActivityEdith K. Y. Tang, Wei Li, Zorica Janjetovic, Minh N. Nguyen, Zhao Wang, Andrzej Slominski and Robert C. TuckeyDrug Metabolism and Disposition September 2010, 38 (9) 1553-1559; DOI: https://doi.org/10.1124/dmd.110.034389
U
Uehara, Shotaro
- You have accessCynomolgus Monkey CYP2D44 Newly Identified in Liver, Metabolizes Bufuralol, and DextromethorphanYasuhiro Uno, Shotaro Uehara, Sakae Kohara, Norie Murayama and Hiroshi YamazakiDrug Metabolism and Disposition September 2010, 38 (9) 1486-1492; DOI: https://doi.org/10.1124/dmd.110.033274
Umemoto, Takahiro
- You have accessActivation of Cyclosporin A Transport by a Novel λ Light Chain of Human Ig Surface Antigen-Related Gene in Xenopus laevis OocytesYasuna Kobayashi, Takahiro Umemoto, Masayuki Ohbayashi, Noriko Kohyama, Yutaka Sanada and Toshinori YamamotoDrug Metabolism and Disposition September 2010, 38 (9) 1427-1435; DOI: https://doi.org/10.1124/dmd.109.030916
Unadkat, Jashvant D.
- You have accessIncreased Glyburide Clearance in the Pregnant Mouse ModelLin Zhou, Yi Zhang, Mary F. Hebert, Jashvant D. Unadkat and Qingcheng MaoDrug Metabolism and Disposition September 2010, 38 (9) 1403-1406; DOI: https://doi.org/10.1124/dmd.110.033837
Uno, Yasuhiro
- You have accessCynomolgus Monkey CYP2D44 Newly Identified in Liver, Metabolizes Bufuralol, and DextromethorphanYasuhiro Uno, Shotaro Uehara, Sakae Kohara, Norie Murayama and Hiroshi YamazakiDrug Metabolism and Disposition September 2010, 38 (9) 1486-1492; DOI: https://doi.org/10.1124/dmd.110.033274
Upadhyaya, Pramod
- You have accessPreferential Glutathione Conjugation of a Reverse Diol Epoxide Compared with a Bay Region Diol Epoxide of Benzo[a]pyrene in Human HepatocytesPramod Upadhyaya, J. Bradley Hochalter, Silvia Balbo, Edward J. McIntee and Stephen S. HechtDrug Metabolism and Disposition September 2010, 38 (9) 1397-1402; DOI: https://doi.org/10.1124/dmd.110.034181
W
Wagner, Klaus
- You have accessDabigatran Acylglucuronide, the Major Human Metabolite of Dabigatran: In Vitro Formation, Stability, and Pharmacological ActivityThomas Ebner, Klaus Wagner and Wolfgang WienenDrug Metabolism and Disposition September 2010, 38 (9) 1567-1575; DOI: https://doi.org/10.1124/dmd.110.033696
Wallin, Jeffrey J.
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Wang, Shixiang
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
Wang, Zhao
- You have accessPurified Mouse CYP27B1 Can Hydroxylate 20,23-Dihydroxyvitamin D3, Producing 1α,20,23-Trihydroxyvitamin D3, Which Has Altered Biological ActivityEdith K. Y. Tang, Wei Li, Zorica Janjetovic, Minh N. Nguyen, Zhao Wang, Andrzej Slominski and Robert C. TuckeyDrug Metabolism and Disposition September 2010, 38 (9) 1553-1559; DOI: https://doi.org/10.1124/dmd.110.034389
Watanabe, Akinobu
- You have accessArylacetamide Deacetylase Is a Determinant Enzyme for the Difference in Hydrolase Activities of Phenacetin and AcetaminophenAkinobu Watanabe, Tatsuki Fukami, Shiori Takahashi, Yuki Kobayashi, Nao Nakagawa, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition September 2010, 38 (9) 1532-1537; DOI: https://doi.org/10.1124/dmd.110.033720
Weiss, Thomas S.
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Wienen, Wolfgang
- You have accessDabigatran Acylglucuronide, the Major Human Metabolite of Dabigatran: In Vitro Formation, Stability, and Pharmacological ActivityThomas Ebner, Klaus Wagner and Wolfgang WienenDrug Metabolism and Disposition September 2010, 38 (9) 1567-1575; DOI: https://doi.org/10.1124/dmd.110.033696
Wong, Harvey
- You have accessPharmacokinetic-Pharmacodynamic Modeling of Tumor Growth Inhibition and Biomarker Modulation by the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Harvey Wong, Marcia Belvin, Delia Bradford, Kyle A. Edgar, Wei Wei Prior, Deepak Sampath and Jeffrey J. WallinDrug Metabolism and Disposition September 2010, 38 (9) 1436-1442; DOI: https://doi.org/10.1124/dmd.110.032912
Wu, Jing
- You have accessProtein Phosphatase 2Cβl Regulates Human Pregnane X Receptor-Mediated CYP3A4 Gene Expression in HepG2 Liver Carcinoma CellsSatyanarayana R. Pondugula, Alexander A. Tong, Jing Wu, Jimmy Cui and Taosheng ChenDrug Metabolism and Disposition September 2010, 38 (9) 1411-1416; DOI: https://doi.org/10.1124/dmd.110.032128
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Xia, Cindy Q.
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Xiao, Chaoni
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
Xie, Jin
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Yabuuchi, Hikaru
- You have accessEstimation of Transporters Involved in the Hepatobiliary Transport of TA-0201CA Using Sandwich-Cultured Rat Hepatocytes from Normal and Multidrug Resistance-Associated Protein 2-Deficient RatsHajime Fukuda, Rikiya Ohashi, Noriko Ohashi, Hikaru Yabuuchi and Ikumi TamaiDrug Metabolism and Disposition September 2010, 38 (9) 1505-1513; DOI: https://doi.org/10.1124/dmd.110.033258
Yamaguchi, Takashi
- You have accessMethemoglobinemia Induced by 1,2-Dichloro-4-nitrobenzene in Mice with a Disrupted Glutathione S-Transferase Mu 1 GeneShingo Arakawa, Takanori Maejima, Naoki Kiyosawa, Takashi Yamaguchi, Yukari Shibaya, Yoshie Aida, Ryota Kawai, Kazunori Fujimoto, Sunao Manabe and Wataru TakasakiDrug Metabolism and Disposition September 2010, 38 (9) 1545-1552; DOI: https://doi.org/10.1124/dmd.110.033597
Yamamoto, Toshinori
- You have accessActivation of Cyclosporin A Transport by a Novel λ Light Chain of Human Ig Surface Antigen-Related Gene in Xenopus laevis OocytesYasuna Kobayashi, Takahiro Umemoto, Masayuki Ohbayashi, Noriko Kohyama, Yutaka Sanada and Toshinori YamamotoDrug Metabolism and Disposition September 2010, 38 (9) 1427-1435; DOI: https://doi.org/10.1124/dmd.109.030916
Yamamura, Naotoshi
- You have accessIdentification of Valproic Acid Glucuronide Hydrolase As a Key Enzyme for the Interaction of Valproic Acid with Carbapenem AntibioticsEiko Suzuki, Naotoshi Yamamura, Yuji Ogura, Daisuke Nakai, Kazuishi Kubota, Nobuhiro Kobayashi, Shin-ichi Miura and Osamu OkazakiDrug Metabolism and Disposition September 2010, 38 (9) 1538-1544; DOI: https://doi.org/10.1124/dmd.110.032938
Yamazaki, Hiroshi
- You have accessCynomolgus Monkey CYP2D44 Newly Identified in Liver, Metabolizes Bufuralol, and DextromethorphanYasuhiro Uno, Shotaro Uehara, Sakae Kohara, Norie Murayama and Hiroshi YamazakiDrug Metabolism and Disposition September 2010, 38 (9) 1486-1492; DOI: https://doi.org/10.1124/dmd.110.033274
Yamazaki, Yuichi
- You have accessHistone Deacetylase Inhibitors Induce Cytochrome P450 2B by Activating Nuclear Receptor Constitutive Androstane ReceptorDaichi Takizawa, Satoru Kakizaki, Norio Horiguchi, Hiroki Tojima, Yuichi Yamazaki, Takeshi Ichikawa, Ken Sato and Masatomo MoriDrug Metabolism and Disposition September 2010, 38 (9) 1493-1498; DOI: https://doi.org/10.1124/dmd.110.032854
Yang, Shengtian
- You have accessNovel Metabolic Bioactivation Mechanism for a Series of Anti-Inflammatory Agents (2,5-Diaminothiophene Derivatives) Mediated by Cytochrome P450 EnzymesYiding Hu, Shengtian Yang, F. Barclay Shilliday, Bruce R. Heyde, Kathy M. Mandrell, Russell H. Robins, Jin Xie, Matthew T. Reding, Yurong Lai and David C. ThompsonDrug Metabolism and Disposition September 2010, 38 (9) 1522-1531; DOI: https://doi.org/10.1124/dmd.110.032581
Yokoi, Tsuyoshi
- You have accessArylacetamide Deacetylase Is a Determinant Enzyme for the Difference in Hydrolase Activities of Phenacetin and AcetaminophenAkinobu Watanabe, Tatsuki Fukami, Shiori Takahashi, Yuki Kobayashi, Nao Nakagawa, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition September 2010, 38 (9) 1532-1537; DOI: https://doi.org/10.1124/dmd.110.033720
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Zabihyan, Behnaz
- You have accessCyclosporine A, but Not Tacrolimus, Shows Relevant Inhibition of Organic Anion-Transporting Protein 1B1-Mediated Transport of AtorvastatinRune Amundsen, Hege Christensen, Behnaz Zabihyan and Anders ÅsbergDrug Metabolism and Disposition September 2010, 38 (9) 1499-1504; DOI: https://doi.org/10.1124/dmd.110.032268
Zanger, Ulrich M.
- You have accessProfiling Induction of Cytochrome P450 Enzyme Activity by Statins Using a New Liquid Chromatography-Tandem Mass Spectrometry Cocktail Assay in Human HepatocytesDiana M. Feidt, Kathrin Klein, Ute Hofmann, Stephan Riedmaier, Daniel Knobeloch, Wolfgang E. Thasler, Thomas S. Weiss, Matthias Schwab and Ulrich M. ZangerDrug Metabolism and Disposition September 2010, 38 (9) 1589-1597; DOI: https://doi.org/10.1124/dmd.110.033886
Zhang, Xiaolin
- You have accessRole of P-Glycoprotein and Breast Cancer Resistance Protein-1 in the Brain Penetration and Brain Pharmacodynamic Activity of the Novel Phosphatidylinositol 3-Kinase Inhibitor GDC-0941Laurent Salphati, Leslie B. Lee, Jodie Pang, Emile G. Plise and Xiaolin ZhangDrug Metabolism and Disposition September 2010, 38 (9) 1422-1426; DOI: https://doi.org/10.1124/dmd.110.034256
Zhang, Yi
- You have accessIncreased Glyburide Clearance in the Pregnant Mouse ModelLin Zhou, Yi Zhang, Mary F. Hebert, Jashvant D. Unadkat and Qingcheng MaoDrug Metabolism and Disposition September 2010, 38 (9) 1403-1406; DOI: https://doi.org/10.1124/dmd.110.033837
Zheng, Xiaohui
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
Zhou, Lin
- You have accessIncreased Glyburide Clearance in the Pregnant Mouse ModelLin Zhou, Yi Zhang, Mary F. Hebert, Jashvant D. Unadkat and Qingcheng MaoDrug Metabolism and Disposition September 2010, 38 (9) 1403-1406; DOI: https://doi.org/10.1124/dmd.110.033837
Zhu, Juanli
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
Zhu, Qing
- You have accessInhibition of Hepatic Organic Anion-Transporting Polypeptide by RNA Interference in Sandwich-Cultured Human Hepatocytes: An In Vitro Model to Assess Transporter-Mediated Drug-Drug InteractionsMingxiang Liao, Arek R. Raczynski, Michael Chen, Bei-Ching Chuang, Qing Zhu, Rob Shipman, Jodi Morrison, David Lee, Frank W. Lee, Suresh K. Balani and Cindy Q. XiaDrug Metabolism and Disposition September 2010, 38 (9) 1612-1622; DOI: https://doi.org/10.1124/dmd.110.032995
Zi, Jing
- You have accessMetabolism of Tanshinol Borneol Ester in Rat and Human Liver MicrosomesDuan Liu, Xiaohui Zheng, Yitong Tang, Jing Zi, Yefei Nan, Shixiang Wang, Chaoni Xiao, Juanli Zhu and Chao ChenDrug Metabolism and Disposition September 2010, 38 (9) 1464-1470; DOI: https://doi.org/10.1124/dmd.110.033381
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