Index by author
January 01, 2011; Volume 39,Issue 1
A
Ačimovič, Jure
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Ahn, Taeho
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Alton, Kevin B.
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
Amano, Nobuyuki
- You have accessQuantitative Investigation of the Impact of P-Glycoprotein Inhibition on Drug Transport across Blood-Brain Barrier in RatsHiroshi Sugimoto, Hideki Hirabayashi, Yoshiaki Kimura, Atsutoshi Furuta, Nobuyuki Amano and Toshiya MoriwakiDrug Metabolism and Disposition January 2011, 39 (1) 8-14; DOI: https://doi.org/10.1124/dmd.110.035774
Auld, Douglas S.
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Austin, Christopher P.
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Azuma, Junichi
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
B
Babalola, Kathlene
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Belič, Ales
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Bi, Yi-an
- You have accessCharacterization of Digoxin Uptake in Sandwich-Cultured Human HepatocytesEmi Kimoto, Jonathan Chupka, Yongling Xiao, Yi-an Bi and David B. DuignanDrug Metabolism and Disposition January 2011, 39 (1) 47-53; DOI: https://doi.org/10.1124/dmd.110.034298
Bjorkhem, Ingemar
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Boado, Ruben J.
- You have accessBrain-Penetrating Tumor Necrosis Factor Decoy Receptor in the MouseQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition January 2011, 39 (1) 71-76; DOI: https://doi.org/10.1124/dmd.110.036012
Boulos, Nidal
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Butcher, Neville J.
- You have accessHistone Deacetylase Inhibitors Increase Human Arylamine N-Acetyltransferase-1 Expression in Human Tumor CellsScott Paterson, Kok L. Sin, Jacky M. Tiang, Rodney F. Minchin and Neville J. ButcherDrug Metabolism and Disposition January 2011, 39 (1) 77-82; DOI: https://doi.org/10.1124/dmd.110.036202
C
Chaudhary, Inder
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Chen, Stephanie
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Chen, Zecheng
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Cheng, Peter T.
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Cho, Joo-Youn
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Chowdhury, Swapan K.
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
Chung, Jae Yong
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Chupka, Jonathan
- You have accessCharacterization of Digoxin Uptake in Sandwich-Cultured Human HepatocytesEmi Kimoto, Jonathan Chupka, Yongling Xiao, Yi-an Bi and David B. DuignanDrug Metabolism and Disposition January 2011, 39 (1) 47-53; DOI: https://doi.org/10.1124/dmd.110.034298
D
Dehnhardt, Christoph
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Deng, Yangmei
- You have accessActivation of the Acute Inflammatory Response Alters Cytochrome P450 Expression and Eicosanoid MetabolismKatherine N. Theken, Yangmei Deng, M. Alison Kannon, Tricia M. Miller, Samuel M. Poloyac and Craig R. LeeDrug Metabolism and Disposition January 2011, 39 (1) 22-29; DOI: https://doi.org/10.1124/dmd.110.035287
Desta, Zeruesenay
- You have accessIn Vitro Cytochrome P450-Mediated Metabolism of ExemestaneLandry K. Kamdem, David A. Flockhart and Zeruesenay DestaDrug Metabolism and Disposition January 2011, 39 (1) 98-105; DOI: https://doi.org/10.1124/dmd.110.032276
Dickmann, Leslie
- You have accessPregnancy Decreases Rat CYP1A2 Activity and ExpressionAlysa A. Walker, Leslie Dickmann and Nina IsoherranenDrug Metabolism and Disposition January 2011, 39 (1) 4-7; DOI: https://doi.org/10.1124/dmd.110.035766
Duignan, David B.
- You have accessCharacterization of Digoxin Uptake in Sandwich-Cultured Human HepatocytesEmi Kimoto, Jonathan Chupka, Yongling Xiao, Yi-an Bi and David B. DuignanDrug Metabolism and Disposition January 2011, 39 (1) 47-53; DOI: https://doi.org/10.1124/dmd.110.034298
Dyer, Michael A.
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
E
Espina, Robert
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
F
Farah, Nadia
- You have accessA Baeyer-Villiger Oxidation Specifically Catalyzed by Human Flavin-Containing Monooxygenase 5W. George Lai, Nadia Farah, George A. Moniz and Y. Nancy WongDrug Metabolism and Disposition January 2011, 39 (1) 61-70; DOI: https://doi.org/10.1124/dmd.110.035360
Flockhart, David A.
- You have accessIn Vitro Cytochrome P450-Mediated Metabolism of ExemestaneLandry K. Kamdem, David A. Flockhart and Zeruesenay DestaDrug Metabolism and Disposition January 2011, 39 (1) 98-105; DOI: https://doi.org/10.1124/dmd.110.032276
Fujio, Yasushi
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
Fujiwara, Ryoichi
- You have accessToxicological Evaluation of Acyl Glucuronides of Nonsteroidal Anti-Inflammatory Drugs Using Human Embryonic Kidney 293 Cells Stably Expressing Human UDP-Glucuronosyltransferase and Human HepatocytesToshihisa Koga, Ryoichi Fujiwara, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition January 2011, 39 (1) 54-60; DOI: https://doi.org/10.1124/dmd.110.035600
Furuta, Atsutoshi
- You have accessQuantitative Investigation of the Impact of P-Glycoprotein Inhibition on Drug Transport across Blood-Brain Barrier in RatsHiroshi Sugimoto, Hideki Hirabayashi, Yoshiaki Kimura, Atsutoshi Furuta, Nobuyuki Amano and Toshiya MoriwakiDrug Metabolism and Disposition January 2011, 39 (1) 8-14; DOI: https://doi.org/10.1124/dmd.110.035774
G
Gao, Lan
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
Ghosal, Anima
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
Grey, Anne K. Mullen
- You have accessThe Aryl Hydrocarbon Receptor Pathway and the Response to 3-Methylcholanthrene Are Altered in the Liver of Adrenalectomized RatsAnne K. Mullen Grey and David S. RiddickDrug Metabolism and Disposition January 2011, 39 (1) 83-91; DOI: https://doi.org/10.1124/dmd.110.035584
Grube, Markus
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Guitton, Jérôme
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Guy, R. Kiplin
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
H
Haruta, Tsunemitsu
- You have accessOrganic Cation Transporter-Mediated Renal Secretion of Ipratropium and Tiotropium in Rats and HumansTakeo Nakanishi, Tsunemitsu Haruta, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition January 2011, 39 (1) 117-122; DOI: https://doi.org/10.1124/dmd.110.035402
Hirabayashi, Hideki
- You have accessQuantitative Investigation of the Impact of P-Glycoprotein Inhibition on Drug Transport across Blood-Brain Barrier in RatsHiroshi Sugimoto, Hideki Hirabayashi, Yoshiaki Kimura, Atsutoshi Furuta, Nobuyuki Amano and Toshiya MoriwakiDrug Metabolism and Disposition January 2011, 39 (1) 8-14; DOI: https://doi.org/10.1124/dmd.110.035774
Huang, Ruili
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Hübner, Tobias
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Hui, Eric Ka-Wai
- You have accessBrain-Penetrating Tumor Necrosis Factor Decoy Receptor in the MouseQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition January 2011, 39 (1) 71-76; DOI: https://doi.org/10.1124/dmd.110.036012
Humphreys, W. Griffith
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
I
Isoherranen, Nina
- You have accessPregnancy Decreases Rat CYP1A2 Activity and ExpressionAlysa A. Walker, Leslie Dickmann and Nina IsoherranenDrug Metabolism and Disposition January 2011, 39 (1) 4-7; DOI: https://doi.org/10.1124/dmd.110.035766
J
Jang, In-Jin
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Jedlitschky, Gabriele
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Jung, Heung-Chae
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
K
Kamdem, Landry K.
- You have accessIn Vitro Cytochrome P450-Mediated Metabolism of ExemestaneLandry K. Kamdem, David A. Flockhart and Zeruesenay DestaDrug Metabolism and Disposition January 2011, 39 (1) 98-105; DOI: https://doi.org/10.1124/dmd.110.032276
Kang, Ji-Yeon
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Kannon, M. Alison
- You have accessActivation of the Acute Inflammatory Response Alters Cytochrome P450 Expression and Eicosanoid MetabolismKatherine N. Theken, Yangmei Deng, M. Alison Kannon, Tricia M. Miller, Samuel M. Poloyac and Craig R. LeeDrug Metabolism and Disposition January 2011, 39 (1) 22-29; DOI: https://doi.org/10.1124/dmd.110.035287
Kim, Dong-Hyun
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Kim, Dooil
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Kim, Jung-Ryul
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Kim, Keon-Hee
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Kimoto, Emi
- You have accessCharacterization of Digoxin Uptake in Sandwich-Cultured Human HepatocytesEmi Kimoto, Jonathan Chupka, Yongling Xiao, Yi-an Bi and David B. DuignanDrug Metabolism and Disposition January 2011, 39 (1) 47-53; DOI: https://doi.org/10.1124/dmd.110.034298
Kimura, Yoshiaki
- You have accessQuantitative Investigation of the Impact of P-Glycoprotein Inhibition on Drug Transport across Blood-Brain Barrier in RatsHiroshi Sugimoto, Hideki Hirabayashi, Yoshiaki Kimura, Atsutoshi Furuta, Nobuyuki Amano and Toshiya MoriwakiDrug Metabolism and Disposition January 2011, 39 (1) 8-14; DOI: https://doi.org/10.1124/dmd.110.035774
Kishnani, Narendra S.
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
Kocjan, Darko
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Köck, Kathleen
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Koga, Toshihisa
- You have accessToxicological Evaluation of Acyl Glucuronides of Nonsteroidal Anti-Inflammatory Drugs Using Human Embryonic Kidney 293 Cells Stably Expressing Human UDP-Glucuronosyltransferase and Human HepatocytesToshihisa Koga, Ryoichi Fujiwara, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition January 2011, 39 (1) 54-60; DOI: https://doi.org/10.1124/dmd.110.035600
Korošec, Tina
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Kowalczyk, Dariusz W.
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Kroemer, Heyo K.
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
L
Lai, W. George
- You have accessA Baeyer-Villiger Oxidation Specifically Catalyzed by Human Flavin-Containing Monooxygenase 5W. George Lai, Nadia Farah, George A. Moniz and Y. Nancy WongDrug Metabolism and Disposition January 2011, 39 (1) 61-70; DOI: https://doi.org/10.1124/dmd.110.035360
Lee, Craig R.
- You have accessActivation of the Acute Inflammatory Response Alters Cytochrome P450 Expression and Eicosanoid MetabolismKatherine N. Theken, Yangmei Deng, M. Alison Kannon, Tricia M. Miller, Samuel M. Poloyac and Craig R. LeeDrug Metabolism and Disposition January 2011, 39 (1) 22-29; DOI: https://doi.org/10.1124/dmd.110.035287
Lee, Young Ju
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Lerch, Markus M.
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Li, Wenying
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Lim, Hyeong-Seok
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Lim, Kyoung Soo
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Lu, Jeff Zhiqiang
- You have accessBrain-Penetrating Tumor Necrosis Factor Decoy Receptor in the MouseQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition January 2011, 39 (1) 71-76; DOI: https://doi.org/10.1124/dmd.110.036012
Lu, Min
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Lu, Xiaowen
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
M
Maeda, Makiko
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
Mallari, Jeremy
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Mansour, Tarek
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Mayerle, Julia
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Mews, Steffen
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Miller, Laura
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Miller, Tricia M.
- You have accessActivation of the Acute Inflammatory Response Alters Cytochrome P450 Expression and Eicosanoid MetabolismKatherine N. Theken, Yangmei Deng, M. Alison Kannon, Tricia M. Miller, Samuel M. Poloyac and Craig R. LeeDrug Metabolism and Disposition January 2011, 39 (1) 22-29; DOI: https://doi.org/10.1124/dmd.110.035287
Minchin, Rodney F.
- You have accessHistone Deacetylase Inhibitors Increase Human Arylamine N-Acetyltransferase-1 Expression in Human Tumor CellsScott Paterson, Kok L. Sin, Jacky M. Tiang, Rodney F. Minchin and Neville J. ButcherDrug Metabolism and Disposition January 2011, 39 (1) 77-82; DOI: https://doi.org/10.1124/dmd.110.036202
Moeller, Timothy A.
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Moniz, George A.
- You have accessA Baeyer-Villiger Oxidation Specifically Catalyzed by Human Flavin-Containing Monooxygenase 5W. George Lai, Nadia Farah, George A. Moniz and Y. Nancy WongDrug Metabolism and Disposition January 2011, 39 (1) 61-70; DOI: https://doi.org/10.1124/dmd.110.035360
Monostory, Katalin
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Moriwaki, Toshiya
- You have accessQuantitative Investigation of the Impact of P-Glycoprotein Inhibition on Drug Transport across Blood-Brain Barrier in RatsHiroshi Sugimoto, Hideki Hirabayashi, Yoshiaki Kimura, Atsutoshi Furuta, Nobuyuki Amano and Toshiya MoriwakiDrug Metabolism and Disposition January 2011, 39 (1) 8-14; DOI: https://doi.org/10.1124/dmd.110.035774
Mutlib, Abdul
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
N
Nakajima, Miki
- You have accessToxicological Evaluation of Acyl Glucuronides of Nonsteroidal Anti-Inflammatory Drugs Using Human Embryonic Kidney 293 Cells Stably Expressing Human UDP-Glucuronosyltransferase and Human HepatocytesToshihisa Koga, Ryoichi Fujiwara, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition January 2011, 39 (1) 54-60; DOI: https://doi.org/10.1124/dmd.110.035600
Nakanishi, Takeo
- You have accessOrganic Cation Transporter-Mediated Renal Secretion of Ipratropium and Tiotropium in Rats and HumansTakeo Nakanishi, Tsunemitsu Haruta, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition January 2011, 39 (1) 117-122; DOI: https://doi.org/10.1124/dmd.110.035402
Nambaru, Praveen K.
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Nemeth, Katie
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Nonen, Shinpei
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
O
Obermeier, Mary
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
P
Pan, Jae-Gu
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Panetta, John C.
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Pardridge, William M.
- You have accessBrain-Penetrating Tumor Necrosis Factor Decoy Receptor in the MouseQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition January 2011, 39 (1) 71-76; DOI: https://doi.org/10.1124/dmd.110.036012
Park, Ki Deok
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Park, Seon Ha
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Park, Sun-Ha
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Pascussi, Jean-Marc
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Paterson, Scott
- You have accessHistone Deacetylase Inhibitors Increase Human Arylamine N-Acetyltransferase-1 Expression in Human Tumor CellsScott Paterson, Kok L. Sin, Jacky M. Tiang, Rodney F. Minchin and Neville J. ButcherDrug Metabolism and Disposition January 2011, 39 (1) 77-82; DOI: https://doi.org/10.1124/dmd.110.036202
Payen, Léa
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Penner, Natalia
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
Poloyac, Samuel M.
- You have accessActivation of the Acute Inflammatory Response Alters Cytochrome P450 Expression and Eicosanoid MetabolismKatherine N. Theken, Yangmei Deng, M. Alison Kannon, Tricia M. Miller, Samuel M. Poloyac and Craig R. LeeDrug Metabolism and Disposition January 2011, 39 (1) 22-29; DOI: https://doi.org/10.1124/dmd.110.035287
R
Raghavan, Nirmala
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Ramanathan, Ragu
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
- You have accessIdentification of Human Liver Cytochrome P450 Enzymes Involved in the Metabolism of SCH 530348 (Vorapaxar), a Potent Oral Thrombin Protease-Activated Receptor 1 AntagonistAnima Ghosal, Xiaowen Lu, Natalia Penner, Lan Gao, Ragu Ramanathan, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition January 2011, 39 (1) 30-38; DOI: https://doi.org/10.1124/dmd.110.035493
Riddick, David S.
- You have accessThe Aryl Hydrocarbon Receptor Pathway and the Response to 3-Methylcholanthrene Are Altered in the Liver of Adrenalectomized RatsAnne K. Mullen Grey and David S. RiddickDrug Metabolism and Disposition January 2011, 39 (1) 83-91; DOI: https://doi.org/10.1124/dmd.110.035584
Rimmbach, Christian
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Ritter, Christoph A.
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Rosskopf, Dieter
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Roussel, Martine F.
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Rozman, Damjana
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
S
Sakamuru, Srilatha
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Scatina, JoAnn
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Seliškar, Matej
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
Sendler, Matthias
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Shiga, Ryota
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
Shin, Sang-Goo
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Shinn, Paul
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Shirasaka, Yoshiyuki
- You have accessOrganic Cation Transporter-Mediated Renal Secretion of Ipratropium and Tiotropium in Rats and HumansTakeo Nakanishi, Tsunemitsu Haruta, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition January 2011, 39 (1) 117-122; DOI: https://doi.org/10.1124/dmd.110.035402
Shukla, Sunita J.
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Sin, Kok L.
- You have accessHistone Deacetylase Inhibitors Increase Human Arylamine N-Acetyltransferase-1 Expression in Human Tumor CellsScott Paterson, Kok L. Sin, Jacky M. Tiang, Rodney F. Minchin and Neville J. ButcherDrug Metabolism and Disposition January 2011, 39 (1) 77-82; DOI: https://doi.org/10.1124/dmd.110.036202
Stewart, Clinton F.
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Sugimoto, Hiroshi
- You have accessQuantitative Investigation of the Impact of P-Glycoprotein Inhibition on Drug Transport across Blood-Brain Barrier in RatsHiroshi Sugimoto, Hideki Hirabayashi, Yoshiaki Kimura, Atsutoshi Furuta, Nobuyuki Amano and Toshiya MoriwakiDrug Metabolism and Disposition January 2011, 39 (1) 8-14; DOI: https://doi.org/10.1124/dmd.110.035774
Sugiura, Chika
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
Szabo, Pal
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
T
Tagen, Michael
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Talaat, Rasmy
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Tamai, Ikumi
- You have accessOrganic Cation Transporter-Mediated Renal Secretion of Ipratropium and Tiotropium in Rats and HumansTakeo Nakanishi, Tsunemitsu Haruta, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition January 2011, 39 (1) 117-122; DOI: https://doi.org/10.1124/dmd.110.035402
Tao, Shiwei
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Theken, Katherine N.
- You have accessActivation of the Acute Inflammatory Response Alters Cytochrome P450 Expression and Eicosanoid MetabolismKatherine N. Theken, Yangmei Deng, M. Alison Kannon, Tricia M. Miller, Samuel M. Poloyac and Craig R. LeeDrug Metabolism and Disposition January 2011, 39 (1) 22-29; DOI: https://doi.org/10.1124/dmd.110.035287
Throm, Stacy
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Tiang, Jacky M.
- You have accessHistone Deacetylase Inhibitors Increase Human Arylamine N-Acetyltransferase-1 Expression in Human Tumor CellsScott Paterson, Kok L. Sin, Jacky M. Tiang, Rodney F. Minchin and Neville J. ButcherDrug Metabolism and Disposition January 2011, 39 (1) 77-82; DOI: https://doi.org/10.1124/dmd.110.036202
U
Urleb, Uroš
- You have accessInhibition of Human Sterol Δ7-Reductase and Other Postlanosterol Enzymes by LK-980, a Novel Inhibitor of Cholesterol SynthesisJure Ačimovič, Tina Korošec, Matej Seliškar, Ingemar Bjorkhem, Katalin Monostory, Pal Szabo, Jean-Marc Pascussi, Ales Belič, Uroš Urleb, Darko Kocjan and Damjana RozmanDrug Metabolism and Disposition January 2011, 39 (1) 39-46; DOI: https://doi.org/10.1124/dmd.110.035840
V
VanLeer, Danielle
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Venkatesan, Aranapakam
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
Vishwanathan, Karthick
- You have accessApplication of Quantitative NMR in Pharmacological Evaluation of Biologically Generated Metabolites: Implications in Drug DiscoveryAbdul Mutlib, Robert Espina, Karthick Vishwanathan, Kathlene Babalola, Zecheng Chen, Christoph Dehnhardt, Aranapakam Venkatesan, Tarek Mansour, Inder Chaudhary, Rasmy Talaat and JoAnn ScatinaDrug Metabolism and Disposition January 2011, 39 (1) 106-116; DOI: https://doi.org/10.1124/dmd.110.032490
W
Walker, Alysa A.
- You have accessPregnancy Decreases Rat CYP1A2 Activity and ExpressionAlysa A. Walker, Leslie Dickmann and Nina IsoherranenDrug Metabolism and Disposition January 2011, 39 (1) 4-7; DOI: https://doi.org/10.1124/dmd.110.035766
Wang, Lifei
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Washio, Ikumi
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
Weiss, Frank U.
- You have accessDrug Efflux Transporter Multidrug Resistance-Associated Protein 5 Affects Sensitivity of Pancreatic Cancer Cell Lines to the Nucleoside Anticancer Drug 5-FluorouracilPraveen K. Nambaru, Tobias Hübner, Kathleen Köck, Steffen Mews, Markus Grube, Léa Payen, Jérôme Guitton, Matthias Sendler, Gabriele Jedlitschky, Christian Rimmbach, Dieter Rosskopf, Dariusz W. Kowalczyk, Heyo K. Kroemer, Frank U. Weiss, Julia Mayerle, Markus M. Lerch and Christoph A. RitterDrug Metabolism and Disposition January 2011, 39 (1) 132-139; DOI: https://doi.org/10.1124/dmd.110.033613
Williams, Richard T.
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Wong, Y. Nancy
- You have accessA Baeyer-Villiger Oxidation Specifically Catalyzed by Human Flavin-Containing Monooxygenase 5W. George Lai, Nadia Farah, George A. Moniz and Y. Nancy WongDrug Metabolism and Disposition January 2011, 39 (1) 61-70; DOI: https://doi.org/10.1124/dmd.110.035360
X
Xia, Menghang
- You have accessIdentification of Clinically Used Drugs That Activate Pregnane X ReceptorsSunita J. Shukla, Srilatha Sakamuru, Ruili Huang, Timothy A. Moeller, Paul Shinn, Danielle VanLeer, Douglas S. Auld, Christopher P. Austin and Menghang XiaDrug Metabolism and Disposition January 2011, 39 (1) 151-159; DOI: https://doi.org/10.1124/dmd.110.035105
Xiao, Yongling
- You have accessCharacterization of Digoxin Uptake in Sandwich-Cultured Human HepatocytesEmi Kimoto, Jonathan Chupka, Yongling Xiao, Yi-an Bi and David B. DuignanDrug Metabolism and Disposition January 2011, 39 (1) 47-53; DOI: https://doi.org/10.1124/dmd.110.034298
Xue, Yongjun
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Y
Yang, Zheng
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Yokoi, Tsuyoshi
- You have accessToxicological Evaluation of Acyl Glucuronides of Nonsteroidal Anti-Inflammatory Drugs Using Human Embryonic Kidney 293 Cells Stably Expressing Human UDP-Glucuronosyltransferase and Human HepatocytesToshihisa Koga, Ryoichi Fujiwara, Miki Nakajima and Tsuyoshi YokoiDrug Metabolism and Disposition January 2011, 39 (1) 54-60; DOI: https://doi.org/10.1124/dmd.110.035600
Yoshida, Mitsuhiro
- You have accessCigarette Smoke Extract Induces CYP2B6 through Constitutive Androstane Receptor in HepatocytesIkumi Washio, Makiko Maeda, Chika Sugiura, Ryota Shiga, Mitsuhiro Yoshida, Shinpei Nonen, Yasushi Fujio and Junichi AzumaDrug Metabolism and Disposition January 2011, 39 (1) 1-3; DOI: https://doi.org/10.1124/dmd.110.034504
Yu, Kyung-Sang
- You have accessEffects of Pregnane X Receptor (NR1I2) and CYP2B6 Genetic Polymorphisms on the Induction of Bupropion Hydroxylation by RifampinJae Yong Chung, Joo-Youn Cho, Hyeong-Seok Lim, Jung-Ryul Kim, Kyung-Sang Yu, Kyoung Soo Lim, Sang-Goo Shin and In-Jin JangDrug Metabolism and Disposition January 2011, 39 (1) 92-97; DOI: https://doi.org/10.1124/dmd.110.035246
Yun, Chul-Ho
- You have accessGeneration of Human Chiral Metabolites of Simvastatin and Lovastatin by Bacterial CYP102A1 MutantsKeon-Hee Kim, Ji-Yeon Kang, Dong-Hyun Kim, Sun-Ha Park, Seon Ha Park, Dooil Kim, Ki Deok Park, Young Ju Lee, Heung-Chae Jung, Jae-Gu Pan, Taeho Ahn and Chul-Ho YunDrug Metabolism and Disposition January 2011, 39 (1) 140-150; DOI: https://doi.org/10.1124/dmd.110.036392
Z
Zhang, Donglu
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Zhang, Fan
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Zhang, Hao
- You have accessPlasma Stability-Dependent Circulation of Acyl Glucuronide Metabolites in Humans: How Circulating Metabolite Profiles of Muraglitazar and Peliglitazar Can Lead to Misleading Risk AssessmentDonglu Zhang, Nirmala Raghavan, Lifei Wang, Yongjun Xue, Mary Obermeier, Stephanie Chen, Shiwei Tao, Hao Zhang, Peter T. Cheng, Wenying Li, Ragu Ramanathan, Zheng Yang and W. Griffith HumphreysDrug Metabolism and Disposition January 2011, 39 (1) 123-131; DOI: https://doi.org/10.1124/dmd.110.035048
Zhang, Jiakun
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
Zhou, Qing-Hui
- You have accessBrain-Penetrating Tumor Necrosis Factor Decoy Receptor in the MouseQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition January 2011, 39 (1) 71-76; DOI: https://doi.org/10.1124/dmd.110.036012
Zhu, Fangyi
- You have accessWhole-Body Physiologically Based Pharmacokinetic Model for Nutlin-3a in Mice after Intravenous and Oral AdministrationFan Zhang, Michael Tagen, Stacy Throm, Jeremy Mallari, Laura Miller, R. Kiplin Guy, Michael A. Dyer, Richard T. Williams, Martine F. Roussel, Katie Nemeth, Fangyi Zhu, Jiakun Zhang, Min Lu, John C. Panetta, Nidal Boulos and Clinton F. StewartDrug Metabolism and Disposition January 2011, 39 (1) 15-21; DOI: https://doi.org/10.1124/dmd.110.035915
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