Index by author
October 01, 2011; Volume 39,Issue 10
A
Ahn, Sunjoo
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Anger, Gregory J.
- You have accessMechanisms of Reduced Maternal and Fetal Lopinavir Exposure in a Rat Model of Gestational DiabetesGregory J. Anger and Micheline Piquette-MillerDrug Metabolism and Disposition October 2011, 39 (10) 1850-1859; DOI: https://doi.org/10.1124/dmd.111.040626
Antoun, Joseph
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
Aoki, Katsuyuki
- You have accessPharmacokinetics of Daikenchuto, a Traditional Japanese Medicine (Kampo) after Single Oral Administration to Healthy Japanese VolunteersMasaya Munekage, Hiroyuki Kitagawa, Kengo Ichikawa, Junko Watanabe, Katsuyuki Aoki, Toru Kono and Kazuhiro HanazakiDrug Metabolism and Disposition October 2011, 39 (10) 1784-1788; DOI: https://doi.org/10.1124/dmd.111.040097
Asanuma, Kimie
- You have accessPharmacokinetic and Pharmacodynamic Modeling of the Effect of an Sodium-Glucose Cotransporter Inhibitor, Phlorizin, on Renal Glucose Transport in RatsKoji Yamaguchi, Motohiro Kato, Masayuki Suzuki, Kimie Asanuma, Yoshinori Aso, Sachiya Ikeda and Masaki IshigaiDrug Metabolism and Disposition October 2011, 39 (10) 1801-1807; DOI: https://doi.org/10.1124/dmd.111.040048
Aso, Yoshinori
- You have accessPharmacokinetic and Pharmacodynamic Modeling of the Effect of an Sodium-Glucose Cotransporter Inhibitor, Phlorizin, on Renal Glucose Transport in RatsKoji Yamaguchi, Motohiro Kato, Masayuki Suzuki, Kimie Asanuma, Yoshinori Aso, Sachiya Ikeda and Masaki IshigaiDrug Metabolism and Disposition October 2011, 39 (10) 1801-1807; DOI: https://doi.org/10.1124/dmd.111.040048
Awwad, Michel
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
B
Backman, Janne T.
- You have accessDose-Dependent Interaction between Gemfibrozil and Repaglinide in Humans: Strong Inhibition of CYP2C8 with Subtherapeutic Gemfibrozil DosesJohanna Honkalammi, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition October 2011, 39 (10) 1977-1986; DOI: https://doi.org/10.1124/dmd.111.040931
Baumgardner, Matthew
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Bennett, Mark K.
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Bergström, Moa Andresen
- You have accessBioactivation Pathways of the Cannabinoid Receptor 1 Antagonist RimonabantMoa Andresen Bergström, Emre M. Isin, Neal Castagnoli and Claire E. MilneDrug Metabolism and Disposition October 2011, 39 (10) 1823-1832; DOI: https://doi.org/10.1124/dmd.111.039412
Billheimer, D. Dean
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
Boggs, Jason
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Bratton, Stacie M.
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Bui, Khanh H.
- You have accessIn Vitro and In Vivo Metabolism of a Selective δ-Opioid ReceptorJian Guo, Chungang Gu, Diansong Zhou, Charles S. Elmore, Khanh H. Bui and Scott W. GrimmDrug Metabolism and Disposition October 2011, 39 (10) 1883-1894; DOI: https://doi.org/10.1124/dmd.111.040980
Burks, Scott R.
- You have accessClearance and Biodistribution of Liposomally Encapsulated Nitroxides: A Model for Targeted Delivery of Electron Paramagnetic Resonance Imaging Probes to TumorsScott R. Burks, Eric A. Legenzov, Gerald M. Rosen and Joseph P. Y. KaoDrug Metabolism and Disposition October 2011, 39 (10) 1961-1966; DOI: https://doi.org/10.1124/dmd.111.039636
C
Castagnoli, Neal
- You have accessBioactivation Pathways of the Cannabinoid Receptor 1 Antagonist RimonabantMoa Andresen Bergström, Emre M. Isin, Neal Castagnoli and Claire E. MilneDrug Metabolism and Disposition October 2011, 39 (10) 1823-1832; DOI: https://doi.org/10.1124/dmd.111.039412
Cerec, Virginie
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
Chen, Jianjun
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Chen, Leon
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
Cherrington, Nathan J.
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
Chimalakonda, Krishna C.
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Coelho, Catarina
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Coraggio, Melis
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Corlu, Anne
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
Cronenberger, Carol
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Currie, Kevin S.
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
D
Dalton, James T.
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Davis, John
- You have accessMeasurement of Binding of Basic Drugs to Acidic Phospholipids Using Surface Plasmon Resonance and Incorporation of the Data into Mechanistic Tissue Composition Equations to Predict Steady-State Volume of DistributionHelen Small, Iain Gardner, Hannah M. Jones, John Davis and Malcolm RowlandDrug Metabolism and Disposition October 2011, 39 (10) 1789-1793; DOI: https://doi.org/10.1124/dmd.111.040253
Davis, John C.
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Day, Jeffrey S.
- You have accessEfflux Transport Is an Important Determinant of Ethinylestradiol Glucuronide and Ethinylestradiol Sulfate PharmacokineticsMaciej J. Zamek-Gliszczynski, Jeffrey S. Day, Kathleen M. Hillgren and Diane L. PhillipsDrug Metabolism and Disposition October 2011, 39 (10) 1794-1800; DOI: https://doi.org/10.1124/dmd.111.040162
Deese, Alan
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Dineva, Anna
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Dowty, Martin
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
E
Elmore, Charles S.
- You have accessIn Vitro and In Vivo Metabolism of a Selective δ-Opioid ReceptorJian Guo, Chungang Gu, Diansong Zhou, Charles S. Elmore, Khanh H. Bui and Scott W. GrimmDrug Metabolism and Disposition October 2011, 39 (10) 1883-1894; DOI: https://doi.org/10.1124/dmd.111.040980
F
Fahmi, Odette A.
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Fang, Ying
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Fields, Owen
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Fisher, Craig D.
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
Fountain, Scott
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
G
Galetin, Aleksandra
- You have accessPredictive Utility of In Vitro Rifampin Induction Data Generated in Fresh and Cryopreserved Human Hepatocytes, Fa2N-4, and HepaRG CellsIan E. Templeton, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition October 2011, 39 (10) 1921-1929; DOI: https://doi.org/10.1124/dmd.111.040824
- You have accessKinetic Characterization of Rat Hepatic Uptake of 16 Actively Transported DrugsYoshiyuki Yabe, Aleksandra Galetin and J. Brian HoustonDrug Metabolism and Disposition October 2011, 39 (10) 1808-1814; DOI: https://doi.org/10.1124/dmd.111.040477
Gao, Song
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
Garattini, Enrico
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Gardiner, Philip
- You have accessThe Impact of Hepatic Uptake on the Pharmacokinetics of Organic AnionsPhilip Gardiner and Stuart W. PaineDrug Metabolism and Disposition October 2011, 39 (10) 1930-1938; DOI: https://doi.org/10.1124/dmd.111.039842
Gardner, Iain
- You have accessMeasurement of Binding of Basic Drugs to Acidic Phospholipids Using Surface Plasmon Resonance and Incorporation of the Data into Mechanistic Tissue Composition Equations to Predict Steady-State Volume of DistributionHelen Small, Iain Gardner, Hannah M. Jones, John Davis and Malcolm RowlandDrug Metabolism and Disposition October 2011, 39 (10) 1789-1793; DOI: https://doi.org/10.1124/dmd.111.040253
Glaise, Denise
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
Gong, Ping
- You have accessThioacetamide Intoxication Triggers Transcriptional Up-Regulation but Enzyme Inactivation of UDP-GlucuronosyltransferasesHaiping Hao, Lifang Zhang, Shan Jiang, Shiqing Sun, Ping Gong, Yuan Xie, Xueyan Zhou and Guangji WangDrug Metabolism and Disposition October 2011, 39 (10) 1815-1822; DOI: https://doi.org/10.1124/dmd.111.039172
Gopaul, Sashi
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Grimm, Scott W.
- You have accessIn Vitro and In Vivo Metabolism of a Selective δ-Opioid ReceptorJian Guo, Chungang Gu, Diansong Zhou, Charles S. Elmore, Khanh H. Bui and Scott W. GrimmDrug Metabolism and Disposition October 2011, 39 (10) 1883-1894; DOI: https://doi.org/10.1124/dmd.111.040980
Gu, Chungang
- You have accessIn Vitro and In Vivo Metabolism of a Selective δ-Opioid ReceptorJian Guo, Chungang Gu, Diansong Zhou, Charles S. Elmore, Khanh H. Bui and Scott W. GrimmDrug Metabolism and Disposition October 2011, 39 (10) 1883-1894; DOI: https://doi.org/10.1124/dmd.111.040980
Guguen-Guillouzo, Christiane
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
Guo, Jian
- You have accessIn Vitro and In Vivo Metabolism of a Selective δ-Opioid ReceptorJian Guo, Chungang Gu, Diansong Zhou, Charles S. Elmore, Khanh H. Bui and Scott W. GrimmDrug Metabolism and Disposition October 2011, 39 (10) 1883-1894; DOI: https://doi.org/10.1124/dmd.111.040980
H
Halladay, Jason S.
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Hanazaki, Kazuhiro
- You have accessPharmacokinetics of Daikenchuto, a Traditional Japanese Medicine (Kampo) after Single Oral Administration to Healthy Japanese VolunteersMasaya Munekage, Hiroyuki Kitagawa, Kengo Ichikawa, Junko Watanabe, Katsuyuki Aoki, Toru Kono and Kazuhiro HanazakiDrug Metabolism and Disposition October 2011, 39 (10) 1784-1788; DOI: https://doi.org/10.1124/dmd.111.040097
Hao, Haiping
- You have accessThioacetamide Intoxication Triggers Transcriptional Up-Regulation but Enzyme Inactivation of UDP-GlucuronosyltransferasesHaiping Hao, Lifang Zhang, Shan Jiang, Shiqing Sun, Ping Gong, Yuan Xie, Xueyan Zhou and Guangji WangDrug Metabolism and Disposition October 2011, 39 (10) 1815-1822; DOI: https://doi.org/10.1124/dmd.111.039172
Hardwick, Rhiannon N.
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
Hildebrandt, Peter
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Hillgren, Kathleen M.
- You have accessEfflux Transport Is an Important Determinant of Ethinylestradiol Glucuronide and Ethinylestradiol Sulfate PharmacokineticsMaciej J. Zamek-Gliszczynski, Jeffrey S. Day, Kathleen M. Hillgren and Diane L. PhillipsDrug Metabolism and Disposition October 2011, 39 (10) 1794-1800; DOI: https://doi.org/10.1124/dmd.111.040162
Hirasawa, Noriyasu
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Hiratsuka, Masahiro
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Honda, Masashi
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Hong, Lan
- You have accessBrain Regional Pharmacokinetics of p-Aminosalicylic Acid and Its N-Acetylated Metabolite: Effectiveness in Chelating Brain ManganeseLan Hong, Wendy Jiang, Hao Pan, Yueming Jiang, Su Zeng and Wei ZhengDrug Metabolism and Disposition October 2011, 39 (10) 1904-1909; DOI: https://doi.org/10.1124/dmd.111.040915
Honkalammi, Johanna
- You have accessDose-Dependent Interaction between Gemfibrozil and Repaglinide in Humans: Strong Inhibition of CYP2C8 with Subtherapeutic Gemfibrozil DosesJohanna Honkalammi, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition October 2011, 39 (10) 1977-1986; DOI: https://doi.org/10.1124/dmd.111.040931
Hop, Cornelis E. C. A.
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Houston, J. Brian
- You have accessPredictive Utility of In Vitro Rifampin Induction Data Generated in Fresh and Cryopreserved Human Hepatocytes, Fa2N-4, and HepaRG CellsIan E. Templeton, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition October 2011, 39 (10) 1921-1929; DOI: https://doi.org/10.1124/dmd.111.040824
- You have accessKinetic Characterization of Rat Hepatic Uptake of 16 Actively Transported DrugsYoshiyuki Yabe, Aleksandra Galetin and J. Brian HoustonDrug Metabolism and Disposition October 2011, 39 (10) 1808-1814; DOI: https://doi.org/10.1124/dmd.111.040477
Hu, Ming
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
Hunt, C. Anthony
- You have accessEnabling Clearance Predictions to Emerge from In Silico Actions of Quasi-Autonomous Hepatocyte ComponentsShahab Sheikh-Bahaei and C. Anthony HuntDrug Metabolism and Disposition October 2011, 39 (10) 1910-1920; DOI: https://doi.org/10.1124/dmd.111.038703
Hurst, Susan
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
I
Ichikawa, Kengo
- You have accessPharmacokinetics of Daikenchuto, a Traditional Japanese Medicine (Kampo) after Single Oral Administration to Healthy Japanese VolunteersMasaya Munekage, Hiroyuki Kitagawa, Kengo Ichikawa, Junko Watanabe, Katsuyuki Aoki, Toru Kono and Kazuhiro HanazakiDrug Metabolism and Disposition October 2011, 39 (10) 1784-1788; DOI: https://doi.org/10.1124/dmd.111.040097
Ikeda, Sachiya
- You have accessPharmacokinetic and Pharmacodynamic Modeling of the Effect of an Sodium-Glucose Cotransporter Inhibitor, Phlorizin, on Renal Glucose Transport in RatsKoji Yamaguchi, Motohiro Kato, Masayuki Suzuki, Kimie Asanuma, Yoshinori Aso, Sachiya Ikeda and Masaki IshigaiDrug Metabolism and Disposition October 2011, 39 (10) 1801-1807; DOI: https://doi.org/10.1124/dmd.111.040048
Ishigai, Masaki
- You have accessPharmacokinetic and Pharmacodynamic Modeling of the Effect of an Sodium-Glucose Cotransporter Inhibitor, Phlorizin, on Renal Glucose Transport in RatsKoji Yamaguchi, Motohiro Kato, Masayuki Suzuki, Kimie Asanuma, Yoshinori Aso, Sachiya Ikeda and Masaki IshigaiDrug Metabolism and Disposition October 2011, 39 (10) 1801-1807; DOI: https://doi.org/10.1124/dmd.111.040048
Ishizuka, Tomoko
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
Isin, Emre M.
- You have accessBioactivation Pathways of the Cannabinoid Receptor 1 Antagonist RimonabantMoa Andresen Bergström, Emre M. Isin, Neal Castagnoli and Claire E. MilneDrug Metabolism and Disposition October 2011, 39 (10) 1823-1832; DOI: https://doi.org/10.1124/dmd.111.039412
J
Jackson, Jonathan P.
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
James, Laura P.
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Jiang, Jing
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Jiang, Shan
- You have accessThioacetamide Intoxication Triggers Transcriptional Up-Regulation but Enzyme Inactivation of UDP-GlucuronosyltransferasesHaiping Hao, Lifang Zhang, Shan Jiang, Shiqing Sun, Ping Gong, Yuan Xie, Xueyan Zhou and Guangji WangDrug Metabolism and Disposition October 2011, 39 (10) 1815-1822; DOI: https://doi.org/10.1124/dmd.111.039172
Jiang, Wendy
- You have accessBrain Regional Pharmacokinetics of p-Aminosalicylic Acid and Its N-Acetylated Metabolite: Effectiveness in Chelating Brain ManganeseLan Hong, Wendy Jiang, Hao Pan, Yueming Jiang, Su Zeng and Wei ZhengDrug Metabolism and Disposition October 2011, 39 (10) 1904-1909; DOI: https://doi.org/10.1124/dmd.111.040915
Jiang, Yueming
- You have accessBrain Regional Pharmacokinetics of p-Aminosalicylic Acid and Its N-Acetylated Metabolite: Effectiveness in Chelating Brain ManganeseLan Hong, Wendy Jiang, Hao Pan, Yueming Jiang, Su Zeng and Wei ZhengDrug Metabolism and Disposition October 2011, 39 (10) 1904-1909; DOI: https://doi.org/10.1124/dmd.111.040915
Jiang, Zhihong
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
Jones, Hannah M.
- You have accessMeasurement of Binding of Basic Drugs to Acidic Phospholipids Using Surface Plasmon Resonance and Incorporation of the Data into Mechanistic Tissue Composition Equations to Predict Steady-State Volume of DistributionHelen Small, Iain Gardner, Hannah M. Jones, John Davis and Malcolm RowlandDrug Metabolism and Disposition October 2011, 39 (10) 1789-1793; DOI: https://doi.org/10.1124/dmd.111.040253
K
Kao, Joseph P. Y.
- You have accessClearance and Biodistribution of Liposomally Encapsulated Nitroxides: A Model for Targeted Delivery of Electron Paramagnetic Resonance Imaging Probes to TumorsScott R. Burks, Eric A. Legenzov, Gerald M. Rosen and Joseph P. Y. KaoDrug Metabolism and Disposition October 2011, 39 (10) 1961-1966; DOI: https://doi.org/10.1124/dmd.111.039636
Kato, Motohiro
- You have accessPharmacokinetic and Pharmacodynamic Modeling of the Effect of an Sodium-Glucose Cotransporter Inhibitor, Phlorizin, on Renal Glucose Transport in RatsKoji Yamaguchi, Motohiro Kato, Masayuki Suzuki, Kimie Asanuma, Yoshinori Aso, Sachiya Ikeda and Masaki IshigaiDrug Metabolism and Disposition October 2011, 39 (10) 1801-1807; DOI: https://doi.org/10.1124/dmd.111.040048
Kawai, Kenji
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
Khojasteh, S. Cyrus
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Kirk, Christopher J.
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Kitagawa, Hiroyuki
- You have accessPharmacokinetics of Daikenchuto, a Traditional Japanese Medicine (Kampo) after Single Oral Administration to Healthy Japanese VolunteersMasaya Munekage, Hiroyuki Kitagawa, Kengo Ichikawa, Junko Watanabe, Katsuyuki Aoki, Toru Kono and Kazuhiro HanazakiDrug Metabolism and Disposition October 2011, 39 (10) 1784-1788; DOI: https://doi.org/10.1124/dmd.111.040097
Klimecki, Walter T.
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
Koechling, Wolfgang
- You have accessMetabolite Profiles of Degarelix, a New Gonadotropin-Releasing Hormone Receptor Antagonist, in Rat, Dog, and MonkeyAnders Sonesson, Wolfgang Koechling, Jacek Stalewski, László B. Tankó and Birgitte Buur RasmussenDrug Metabolism and Disposition October 2011, 39 (10) 1895-1903; DOI: https://doi.org/10.1124/dmd.111.039883
Kono, Toru
- You have accessPharmacokinetics of Daikenchuto, a Traditional Japanese Medicine (Kampo) after Single Oral Administration to Healthy Japanese VolunteersMasaya Munekage, Hiroyuki Kitagawa, Kengo Ichikawa, Junko Watanabe, Katsuyuki Aoki, Toru Kono and Kazuhiro HanazakiDrug Metabolism and Disposition October 2011, 39 (10) 1784-1788; DOI: https://doi.org/10.1124/dmd.111.040097
Kraynov, Eugenia
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Kuang, Bing
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Kuebler, Peter
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Kurihara, Atsushi
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
L
La, Hank
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Lake, April D.
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
Le, Hoa
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Le, Vi-Huyen
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Legenzov, Eric A.
- You have accessClearance and Biodistribution of Liposomally Encapsulated Nitroxides: A Model for Targeted Delivery of Electron Paramagnetic Resonance Imaging Probes to TumorsScott R. Burks, Eric A. Legenzov, Gerald M. Rosen and Joseph P. Y. KaoDrug Metabolism and Disposition October 2011, 39 (10) 1961-1966; DOI: https://doi.org/10.1124/dmd.111.039636
Leimkühler, Silke
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Lendzian, Friedhelm
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Li, Chien-Ming
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Li, Wei
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Liao, X. Charlene
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Liu, Lichuan
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Loi, Cho-Ming
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Lu, Yan
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Lubach, Joseph W.
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
M
Madec, Stéphanie
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
Mahro, Martin
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Martin, Steven W.
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Matsubara, Yoichi
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Miller, Duane D.
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Milne, Claire E.
- You have accessBioactivation Pathways of the Cannabinoid Receptor 1 Antagonist RimonabantMoa Andresen Bergström, Emre M. Isin, Neal Castagnoli and Claire E. MilneDrug Metabolism and Disposition October 2011, 39 (10) 1823-1832; DOI: https://doi.org/10.1124/dmd.111.039412
Miyaji, Yoshihiro
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
Molineaux, Christopher J.
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Moran, Cindy L.
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Moran, Jeffery H.
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Munekage, Masaya
- You have accessPharmacokinetics of Daikenchuto, a Traditional Japanese Medicine (Kampo) after Single Oral Administration to Healthy Japanese VolunteersMasaya Munekage, Hiroyuki Kitagawa, Kengo Ichikawa, Junko Watanabe, Katsuyuki Aoki, Toru Kono and Kazuhiro HanazakiDrug Metabolism and Disposition October 2011, 39 (10) 1784-1788; DOI: https://doi.org/10.1124/dmd.111.040097
Muroi, Yuka
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
N
Narayanan, Ramesh
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Neuvonen, Pertti J.
- You have accessDose-Dependent Interaction between Gemfibrozil and Repaglinide in Humans: Strong Inhibition of CYP2C8 with Subtherapeutic Gemfibrozil DosesJohanna Honkalammi, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition October 2011, 39 (10) 1977-1986; DOI: https://doi.org/10.1124/dmd.111.040931
Niemi, Mikko
- You have accessDose-Dependent Interaction between Gemfibrozil and Repaglinide in Humans: Strong Inhibition of CYP2C8 with Subtherapeutic Gemfibrozil DosesJohanna Honkalammi, Mikko Niemi, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition October 2011, 39 (10) 1977-1986; DOI: https://doi.org/10.1124/dmd.111.040931
Novak, Petr
- You have accessAnalysis of Global and Absorption, Distribution, Metabolism, and Elimination Gene Expression in the Progressive Stages of Human Nonalcoholic Fatty Liver DiseaseApril D. Lake, Petr Novak, Craig D. Fisher, Jonathan P. Jackson, Rhiannon N. Hardwick, D. Dean Billheimer, Walter T. Klimecki and Nathan J. CherringtonDrug Metabolism and Disposition October 2011, 39 (10) 1954-1960; DOI: https://doi.org/10.1124/dmd.111.040592
O
Oda, Akifumi
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Okazaki, Osamu
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
P
Paine, Stuart W.
- You have accessThe Impact of Hepatic Uptake on the Pharmacokinetics of Organic AnionsPhilip Gardiner and Stuart W. PaineDrug Metabolism and Disposition October 2011, 39 (10) 1930-1938; DOI: https://doi.org/10.1124/dmd.111.039842
Pan, Hao
- You have accessBrain Regional Pharmacokinetics of p-Aminosalicylic Acid and Its N-Acetylated Metabolite: Effectiveness in Chelating Brain ManganeseLan Hong, Wendy Jiang, Hao Pan, Yueming Jiang, Su Zeng and Wei ZhengDrug Metabolism and Disposition October 2011, 39 (10) 1904-1909; DOI: https://doi.org/10.1124/dmd.111.040915
Parke, Deanna N.
- You have accessPharmacokinetic Optimization of 4-Substituted Methoxybenzoyl-aryl-thiazole and 2-Aryl-4-benzoyl-imidazole for Improving Oral BioavailabilityChien-Ming Li, Jianjun Chen, Yan Lu, Ramesh Narayanan, Deanna N. Parke, Wei Li, Sunjoo Ahn, Duane D. Miller and James T. DaltonDrug Metabolism and Disposition October 2011, 39 (10) 1833-1839; DOI: https://doi.org/10.1124/dmd.110.036616
Phillips, Diane L.
- You have accessEfflux Transport Is an Important Determinant of Ethinylestradiol Glucuronide and Ethinylestradiol Sulfate PharmacokineticsMaciej J. Zamek-Gliszczynski, Jeffrey S. Day, Kathleen M. Hillgren and Diane L. PhillipsDrug Metabolism and Disposition October 2011, 39 (10) 1794-1800; DOI: https://doi.org/10.1124/dmd.111.040162
Piquette-Miller, Micheline
- You have accessMechanisms of Reduced Maternal and Fetal Lopinavir Exposure in a Rat Model of Gestational DiabetesGregory J. Anger and Micheline Piquette-MillerDrug Metabolism and Disposition October 2011, 39 (10) 1850-1859; DOI: https://doi.org/10.1124/dmd.111.040626
Plée-Gautier, Emmanuelle
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
R
Radominska-Pandya, Anna
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Rasmussen, Birgitte Buur
- You have accessMetabolite Profiles of Degarelix, a New Gonadotropin-Releasing Hormone Receptor Antagonist, in Rat, Dog, and MonkeyAnders Sonesson, Wolfgang Koechling, Jacek Stalewski, László B. Tankó and Birgitte Buur RasmussenDrug Metabolism and Disposition October 2011, 39 (10) 1895-1903; DOI: https://doi.org/10.1124/dmd.111.039883
Rodrigues, David
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Romão, Maria João
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Rosen, Gerald M.
- You have accessClearance and Biodistribution of Liposomally Encapsulated Nitroxides: A Model for Targeted Delivery of Electron Paramagnetic Resonance Imaging Probes to TumorsScott R. Burks, Eric A. Legenzov, Gerald M. Rosen and Joseph P. Y. KaoDrug Metabolism and Disposition October 2011, 39 (10) 1961-1966; DOI: https://doi.org/10.1124/dmd.111.039636
Rowland, Malcolm
- You have accessMeasurement of Binding of Basic Drugs to Acidic Phospholipids Using Surface Plasmon Resonance and Incorporation of the Data into Mechanistic Tissue Composition Equations to Predict Steady-State Volume of DistributionHelen Small, Iain Gardner, Hannah M. Jones, John Davis and Malcolm RowlandDrug Metabolism and Disposition October 2011, 39 (10) 1789-1793; DOI: https://doi.org/10.1124/dmd.111.040253
S
Saggu, Miguel
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Saigusa, Daisuke
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Saito, Motoko
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
Salaun, Jean-Pierre
- You have accessCYP4F3B Expression Is Associated with Differentiation of HepaRG Human Hepatocytes and Unaffected by Fatty Acid OverloadStéphanie Madec, Virginie Cerec, Emmanuelle Plée-Gautier, Joseph Antoun, Denise Glaise, Jean-Pierre Salaun, Christiane Guguen-Guillouzo and Anne CorluDrug Metabolism and Disposition October 2011, 39 (10) 1987-1996; DOI: https://doi.org/10.1124/dmd.110.036848
Sheikh-Bahaei, Shahab
- You have accessEnabling Clearance Predictions to Emerge from In Silico Actions of Quasi-Autonomous Hepatocyte ComponentsShahab Sheikh-Bahaei and C. Anthony HuntDrug Metabolism and Disposition October 2011, 39 (10) 1910-1920; DOI: https://doi.org/10.1124/dmd.111.038703
Shin, Young
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Small, Helen
- You have accessMeasurement of Binding of Basic Drugs to Acidic Phospholipids Using Surface Plasmon Resonance and Incorporation of the Data into Mechanistic Tissue Composition Equations to Predict Steady-State Volume of DistributionHelen Small, Iain Gardner, Hannah M. Jones, John Davis and Malcolm RowlandDrug Metabolism and Disposition October 2011, 39 (10) 1789-1793; DOI: https://doi.org/10.1124/dmd.111.040253
Sonesson, Anders
- You have accessMetabolite Profiles of Degarelix, a New Gonadotropin-Releasing Hormone Receptor Antagonist, in Rat, Dog, and MonkeyAnders Sonesson, Wolfgang Koechling, Jacek Stalewski, László B. Tankó and Birgitte Buur RasmussenDrug Metabolism and Disposition October 2011, 39 (10) 1895-1903; DOI: https://doi.org/10.1124/dmd.111.039883
Sowell, C. Gregory
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Stalewski, Jacek
- You have accessMetabolite Profiles of Degarelix, a New Gonadotropin-Releasing Hormone Receptor Antagonist, in Rat, Dog, and MonkeyAnders Sonesson, Wolfgang Koechling, Jacek Stalewski, László B. Tankó and Birgitte Buur RasmussenDrug Metabolism and Disposition October 2011, 39 (10) 1895-1903; DOI: https://doi.org/10.1124/dmd.111.039883
Sun, Shiqing
- You have accessThioacetamide Intoxication Triggers Transcriptional Up-Regulation but Enzyme Inactivation of UDP-GlucuronosyltransferasesHaiping Hao, Lifang Zhang, Shan Jiang, Shiqing Sun, Ping Gong, Yuan Xie, Xueyan Zhou and Guangji WangDrug Metabolism and Disposition October 2011, 39 (10) 1815-1822; DOI: https://doi.org/10.1124/dmd.111.039172
Suzuki, Masayuki
- You have accessPharmacokinetic and Pharmacodynamic Modeling of the Effect of an Sodium-Glucose Cotransporter Inhibitor, Phlorizin, on Renal Glucose Transport in RatsKoji Yamaguchi, Motohiro Kato, Masayuki Suzuki, Kimie Asanuma, Yoshinori Aso, Sachiya Ikeda and Masaki IshigaiDrug Metabolism and Disposition October 2011, 39 (10) 1801-1807; DOI: https://doi.org/10.1124/dmd.111.040048
Suzuki, Naoto
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
T
Tamaki, Yuichiro
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Tankó, László B.
- You have accessMetabolite Profiles of Degarelix, a New Gonadotropin-Releasing Hormone Receptor Antagonist, in Rat, Dog, and MonkeyAnders Sonesson, Wolfgang Koechling, Jacek Stalewski, László B. Tankó and Birgitte Buur RasmussenDrug Metabolism and Disposition October 2011, 39 (10) 1895-1903; DOI: https://doi.org/10.1124/dmd.111.039883
Templeton, Ian E.
- You have accessPredictive Utility of In Vitro Rifampin Induction Data Generated in Fresh and Cryopreserved Human Hepatocytes, Fa2N-4, and HepaRG CellsIan E. Templeton, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition October 2011, 39 (10) 1921-1929; DOI: https://doi.org/10.1124/dmd.111.040824
Teng, Yang
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
Terao, Mineko
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
Tomioka, Yoshihisa
- You have accessFunctional Characterization of CYP2B6 Allelic Variants in Demethylation of Antimalarial ArtemetherMasashi Honda, Yuka Muroi, Yuichiro Tamaki, Daisuke Saigusa, Naoto Suzuki, Yoshihisa Tomioka, Yoichi Matsubara, Akifumi Oda, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition October 2011, 39 (10) 1860-1865; DOI: https://doi.org/10.1124/dmd.111.040352
Trincão, José
- You have accessCharacterization and Crystallization of Mouse Aldehyde Oxidase 3: From Mouse Liver to Escherichia coli Heterologous Protein ExpressionMartin Mahro, Catarina Coelho, José Trincão, David Rodrigues, Mineko Terao, Enrico Garattini, Miguel Saggu, Friedhelm Lendzian, Peter Hildebrandt, Maria João Romão and Silke LeimkühlerDrug Metabolism and Disposition October 2011, 39 (10) 1939-1945; DOI: https://doi.org/10.1124/dmd.111.040873
W
Walter, Sarah
- You have accessDistribution of KAI-9803, a Novel δ-Protein Kinase C Inhibitor, after Intravenous Administration to RatsYoshihiro Miyaji, Sarah Walter, Leon Chen, Atsushi Kurihara, Tomoko Ishizuka, Motoko Saito, Kenji Kawai and Osamu OkazakiDrug Metabolism and Disposition October 2011, 39 (10) 1946-1953; DOI: https://doi.org/10.1124/dmd.111.040725
Wang, Diane
- You have accessHow Current Understanding of Clearance Mechanisms and Pharmacodynamics of Therapeutic Proteins Can Be Applied for Evaluation of Their Drug-Drug Interaction PotentialEugenia Kraynov, Steven W. Martin, Susan Hurst, Odette A. Fahmi, Martin Dowty, Carol Cronenberger, Cho-Ming Loi, Bing Kuang, Owen Fields, Scott Fountain, Michel Awwad and Diane WangDrug Metabolism and Disposition October 2011, 39 (10) 1779-1783; DOI: https://doi.org/10.1124/dmd.111.040808
Wang, Guangji
- You have accessThioacetamide Intoxication Triggers Transcriptional Up-Regulation but Enzyme Inactivation of UDP-GlucuronosyltransferasesHaiping Hao, Lifang Zhang, Shan Jiang, Shiqing Sun, Ping Gong, Yuan Xie, Xueyan Zhou and Guangji WangDrug Metabolism and Disposition October 2011, 39 (10) 1815-1822; DOI: https://doi.org/10.1124/dmd.111.039172
Wang, Jingrong
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
Wang, Zhengping
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Watanabe, Junko
- You have accessPharmacokinetics of Daikenchuto, a Traditional Japanese Medicine (Kampo) after Single Oral Administration to Healthy Japanese VolunteersMasaya Munekage, Hiroyuki Kitagawa, Kengo Ichikawa, Junko Watanabe, Katsuyuki Aoki, Toru Kono and Kazuhiro HanazakiDrug Metabolism and Disposition October 2011, 39 (10) 1784-1788; DOI: https://doi.org/10.1124/dmd.111.040097
Wong, Hansen
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Wong, Harvey
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Wong, Susan
- You have accessSignificant Species Difference in Amide Hydrolysis of GDC-0834, a Novel Potent and Selective Bruton's Tyrosine Kinase InhibitorLichuan Liu, Jason S. Halladay, Young Shin, Susan Wong, Melis Coraggio, Hank La, Matthew Baumgardner, Hoa Le, Sashi Gopaul, Jason Boggs, Peter Kuebler, John C. Davis, X. Charlene Liao, Joseph W. Lubach, Alan Deese, C. Gregory Sowell, Kevin S. Currie, Wendy B. Young, S. Cyrus Khojasteh, Cornelis E. C. A. Hop and Harvey WongDrug Metabolism and Disposition October 2011, 39 (10) 1840-1849; DOI: https://doi.org/10.1124/dmd.111.040840
Wu, Baojian
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
X
Xie, Yuan
- You have accessThioacetamide Intoxication Triggers Transcriptional Up-Regulation but Enzyme Inactivation of UDP-GlucuronosyltransferasesHaiping Hao, Lifang Zhang, Shan Jiang, Shiqing Sun, Ping Gong, Yuan Xie, Xueyan Zhou and Guangji WangDrug Metabolism and Disposition October 2011, 39 (10) 1815-1822; DOI: https://doi.org/10.1124/dmd.111.039172
Y
Yabe, Yoshiyuki
- You have accessKinetic Characterization of Rat Hepatic Uptake of 16 Actively Transported DrugsYoshiyuki Yabe, Aleksandra Galetin and J. Brian HoustonDrug Metabolism and Disposition October 2011, 39 (10) 1808-1814; DOI: https://doi.org/10.1124/dmd.111.040477
Yamaguchi, Koji
- You have accessPharmacokinetic and Pharmacodynamic Modeling of the Effect of an Sodium-Glucose Cotransporter Inhibitor, Phlorizin, on Renal Glucose Transport in RatsKoji Yamaguchi, Motohiro Kato, Masayuki Suzuki, Kimie Asanuma, Yoshinori Aso, Sachiya Ikeda and Masaki IshigaiDrug Metabolism and Disposition October 2011, 39 (10) 1801-1807; DOI: https://doi.org/10.1124/dmd.111.040048
Yang, Jinfu
- You have accessPharmacokinetics, Pharmacodynamics, Metabolism, Distribution, and Excretion of Carfilzomib in RatsJinfu Yang, Zhengping Wang, Ying Fang, Jing Jiang, Frances Zhao, Hansen Wong, Mark K. Bennett, Christopher J. Molineaux and Christopher J. KirkDrug Metabolism and Disposition October 2011, 39 (10) 1873-1882; DOI: https://doi.org/10.1124/dmd.111.039164
Yang, Zhen
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
Yiew, Kan Hui
- You have accessConjugation of Synthetic Cannabinoids JWH-018 and JWH-073, Metabolites by Human UDP-GlucuronosyltransferasesKrishna C. Chimalakonda, Stacie M. Bratton, Vi-Huyen Le, Kan Hui Yiew, Anna Dineva, Cindy L. Moran, Laura P. James, Jeffery H. Moran and Anna Radominska-PandyaDrug Metabolism and Disposition October 2011, 39 (10) 1967-1976; DOI: https://doi.org/10.1124/dmd.111.040709
Yin, Taijun
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
You, Ming
- You have accessEnhancement of Oral Bioavailability of 20(S)-Ginsenoside Rh2 through Improved Understanding of Its Absorption and Efflux MechanismsZhen Yang, Song Gao, Jingrong Wang, Taijun Yin, Yang Teng, Baojian Wu, Ming You, Zhihong Jiang and Ming HuDrug Metabolism and Disposition October 2011, 39 (10) 1866-1872; DOI: https://doi.org/10.1124/dmd.111.040006
Young, Wendy B.
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