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Research ArticleArticle

Studies to Further Investigate the Inhibition of Human Liver Microsomal CYP2C8 by the Acyl-β-Glucuronide of Gemfibrozil

S. M. Jenkins, T. Zvyaga, S. R. Johnson, J. Hurley, A. Wagner, R. Burrell, W. Turley, J. E. Leet, T. Philip and A. D. Rodrigues
Drug Metabolism and Disposition December 2011, 39 (12) 2421-2430; DOI: https://doi.org/10.1124/dmd.111.041947
S. M. Jenkins
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T. Zvyaga
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S. R. Johnson
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J. Hurley
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A. Wagner
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R. Burrell
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W. Turley
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J. E. Leet
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T. Philip
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Article Information

vol. 39 no. 12 2421-2430
DOI 
https://doi.org/10.1124/dmd.111.041947
PubMed 
21911547

Published By 
American Society for Pharmacology and Experimental Therapeutics
Print ISSN 
0090-9556
Online ISSN 
1521-009X
History 
  • Received July 26, 2011
  • Accepted September 12, 2011
  • Published online November 21, 2011.

Article Versions

  • Earlier version (September 12, 2011 - 10:26).
  • You are viewing the most recent version of this article.
Copyright & Usage 
Copyright © 2011 by The American Society for Pharmacology and Experimental Therapeutics

Author Information

  1. S. M. Jenkins,
  2. T. Zvyaga,
  3. S. R. Johnson,
  4. J. Hurley,
  5. A. Wagner,
  6. R. Burrell,
  7. W. Turley,
  8. J. E. Leet,
  9. T. Philip and
  10. A. D. Rodrigues
  1. Bristol-Myers Squibb Molecular Sciences & Candidate Optimization, Wallingford, Connecticut (S.M.J., T.Z., J.H., A.W., R.B., W.T., J.E.L., T.P.); and Bristol-Myers Squibb Molecular Sciences & Candidate Optimization, Princeton, New Jersey (S.R.J., A.D.R.)
  1. Address correspondence to:
    Dr. Susan M. Jenkins, Bristol-Myers Squibb Company, 5 Research Parkway, Wallingford, CT 06492. E-mail: susan.jenkins{at}bms.com
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Drug Metabolism and Disposition: 39 (12)
Drug Metabolism and Disposition
Vol. 39, Issue 12
1 Dec 2011
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Research ArticleArticle

INHIBITION OF CYP2C8 BY GEMFIBROZIL GLUCURONIDE ANALOGS

S. M. Jenkins, T. Zvyaga, S. R. Johnson, J. Hurley, A. Wagner, R. Burrell, W. Turley, J. E. Leet, T. Philip and A. D. Rodrigues
Drug Metabolism and Disposition December 1, 2011, 39 (12) 2421-2430; DOI: https://doi.org/10.1124/dmd.111.041947

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Research ArticleArticle

INHIBITION OF CYP2C8 BY GEMFIBROZIL GLUCURONIDE ANALOGS

S. M. Jenkins, T. Zvyaga, S. R. Johnson, J. Hurley, A. Wagner, R. Burrell, W. Turley, J. E. Leet, T. Philip and A. D. Rodrigues
Drug Metabolism and Disposition December 1, 2011, 39 (12) 2421-2430; DOI: https://doi.org/10.1124/dmd.111.041947
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