Index by author
February 01, 2011; Volume 39,Issue 2
A
Aarons, Leon
- You have accessCritique of the Two-Fold Measure of Prediction Success for Ratios: Application for the Assessment of Drug-Drug InteractionsEleanor J. Guest, Leon Aarons, J. Brian Houston, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition February 2011, 39 (2) 170-173; DOI: https://doi.org/10.1124/dmd.110.036103
Akiyama, Yuko
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Ando, Yuichi
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
B
Beedanagari, Sudheer Reddy
- You have accessHuman CYP2S1 Metabolizes Cyclooxygenase- and Lipoxygenase-Derived EicosanoidsPeter Bui, Satoshi Imaizumi, Sudheer Reddy Beedanagari, Srinivasa T. Reddy and Oliver HankinsonDrug Metabolism and Disposition February 2011, 39 (2) 180-190; DOI: https://doi.org/10.1124/dmd.110.035121
Bettica, Paolo
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
Bonacorsi, Samuel
- You have accessMetabolism and Disposition of 14C-Labeled Peliglitazar in HumansLifei Wang, Carey Munsick, Sean Chen, Samuel Bonacorsi, Peter T. Cheng, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 228-238; DOI: https://doi.org/10.1124/dmd.110.035089
Bordini, Ellenia
- You have accessTissue Distribution and Characterization of Drug-Related Material in Rats and Dogs after Repeated Oral Administration of CasopitantSabrina Pagliarusco, Silvia Martinucci, Ellenia Bordini, Lidia Miraglia, Domenico Cufari, Luca Ferrari and Mario PellegattiDrug Metabolism and Disposition February 2011, 39 (2) 283-293; DOI: https://doi.org/10.1124/dmd.110.035063
Borell, Hubert
- You have accessCYP4F Enzymes Are Responsible for the Elimination of Fingolimod (FTY720), a Novel Treatment of Relapsing Multiple SclerosisYi Jin, Markus Zollinger, Hubert Borell, Alfred Zimmerlin and Christopher J. PattenDrug Metabolism and Disposition February 2011, 39 (2) 191-198; DOI: https://doi.org/10.1124/dmd.110.035378
Boriss, Hinnerk
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
Bottner, Pernilla
- You have accessEffects of Ketoconazole on the In Vivo Biotransformation and Hepatobiliary Transport of the Thrombin Inhibitor AZD0837 in PigsElin M. Matsson, Johan E. Palm, Ulf G. Eriksson, Pernilla Bottner, Anna Lundahl, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition February 2011, 39 (2) 239-246; DOI: https://doi.org/10.1124/dmd.110.035022
Boyle, Gary
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
Braggio, Simone
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
Bui, Peter
- You have accessHuman CYP2S1 Metabolizes Cyclooxygenase- and Lipoxygenase-Derived EicosanoidsPeter Bui, Satoshi Imaizumi, Sudheer Reddy Beedanagari, Srinivasa T. Reddy and Oliver HankinsonDrug Metabolism and Disposition February 2011, 39 (2) 180-190; DOI: https://doi.org/10.1124/dmd.110.035121
Burdette, Doug
- You have accessElucidation of a Novel Bioactivation Pathway of a 3,4-Unsubstituted Isoxazole in Human Liver Microsomes: Formation of a Glutathione Adduct of a Cyanoacrolein Derivative after Isoxazole Ring OpeningJian Yu, James J. Folmer, Valerie Hoesch, James Doherty, James B. Campbell and Doug BurdetteDrug Metabolism and Disposition February 2011, 39 (2) 302-311; DOI: https://doi.org/10.1124/dmd.110.036285
Butters, Caroline
- You have accessThe Utility of In Vitro Data in Making Accurate Predictions of Human P-Glycoprotein-Mediated Drug-Drug Interactions: A Case Study for AZD5672Robert Elsby, Michael Gillen, Caroline Butters, Gemma Imisson, Pradeep Sharma, Veronica Smith and Dominic D. SurryDrug Metabolism and Disposition February 2011, 39 (2) 275-282; DOI: https://doi.org/10.1124/dmd.110.035881
C
Campbell, James B.
- You have accessElucidation of a Novel Bioactivation Pathway of a 3,4-Unsubstituted Isoxazole in Human Liver Microsomes: Formation of a Glutathione Adduct of a Cyanoacrolein Derivative after Isoxazole Ring OpeningJian Yu, James J. Folmer, Valerie Hoesch, James Doherty, James B. Campbell and Doug BurdetteDrug Metabolism and Disposition February 2011, 39 (2) 302-311; DOI: https://doi.org/10.1124/dmd.110.036285
Casabó, V. G.
- You have accessA Pharmacokinetic Model for Evaluating the Impact of Hepatic and Intestinal First-Pass Loss of Saquinavir in the RatR. Lledó-García, A. Nácher, V. G. Casabó and M. Merino-SanjuánDrug Metabolism and Disposition February 2011, 39 (2) 294-301; DOI: https://doi.org/10.1124/dmd.110.034488
Cederbaum, Arthur I.
- You have accessEthanol Induction of CYP2A5: Permissive Role for CYP2E1Yongke Lu, Jian Zhuge, Defeng Wu and Arthur I. CederbaumDrug Metabolism and Disposition February 2011, 39 (2) 330-336; DOI: https://doi.org/10.1124/dmd.110.035691
Chen, Sean
- You have accessMetabolism and Disposition of 14C-Labeled Peliglitazar in HumansLifei Wang, Carey Munsick, Sean Chen, Samuel Bonacorsi, Peter T. Cheng, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 228-238; DOI: https://doi.org/10.1124/dmd.110.035089
Chen, Xiaohui
- You have accessAttenuation of Intestinal Absorption by Major Efflux Transporters: Quantitative Tools and Strategies Using a Caco-2 ModelXuena Lin, Suzanne Skolnik, Xiaohui Chen and Jianling WangDrug Metabolism and Disposition February 2011, 39 (2) 265-274; DOI: https://doi.org/10.1124/dmd.110.034629
Cheng, Peter T.
- You have accessMetabolism and Disposition of 14C-Labeled Peliglitazar in HumansLifei Wang, Carey Munsick, Sean Chen, Samuel Bonacorsi, Peter T. Cheng, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 228-238; DOI: https://doi.org/10.1124/dmd.110.035089
Corbioli, Silvia
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
Cufari, Domenico
- You have accessTissue Distribution and Characterization of Drug-Related Material in Rats and Dogs after Repeated Oral Administration of CasopitantSabrina Pagliarusco, Silvia Martinucci, Ellenia Bordini, Lidia Miraglia, Domenico Cufari, Luca Ferrari and Mario PellegattiDrug Metabolism and Disposition February 2011, 39 (2) 283-293; DOI: https://doi.org/10.1124/dmd.110.035063
D
Doherty, James
- You have accessElucidation of a Novel Bioactivation Pathway of a 3,4-Unsubstituted Isoxazole in Human Liver Microsomes: Formation of a Glutathione Adduct of a Cyanoacrolein Derivative after Isoxazole Ring OpeningJian Yu, James J. Folmer, Valerie Hoesch, James Doherty, James B. Campbell and Doug BurdetteDrug Metabolism and Disposition February 2011, 39 (2) 302-311; DOI: https://doi.org/10.1124/dmd.110.036285
E
Ekins, Sean
- You have accessIdentification and Validation of Novel Human Pregnane X Receptor Activators among Prescribed Drugs via Ligand-Based Virtual ScreeningYongmei Pan, Linhao Li, Gregory Kim, Sean Ekins, Hongbing Wang and Peter W. SwaanDrug Metabolism and Disposition February 2011, 39 (2) 337-344; DOI: https://doi.org/10.1124/dmd.110.035808
Elsby, Robert
- You have accessThe Utility of In Vitro Data in Making Accurate Predictions of Human P-Glycoprotein-Mediated Drug-Drug Interactions: A Case Study for AZD5672Robert Elsby, Michael Gillen, Caroline Butters, Gemma Imisson, Pradeep Sharma, Veronica Smith and Dominic D. SurryDrug Metabolism and Disposition February 2011, 39 (2) 275-282; DOI: https://doi.org/10.1124/dmd.110.035881
Eriksson, Ulf G.
- You have accessEffects of Ketoconazole on the In Vivo Biotransformation and Hepatobiliary Transport of the Thrombin Inhibitor AZD0837 in PigsElin M. Matsson, Johan E. Palm, Ulf G. Eriksson, Pernilla Bottner, Anna Lundahl, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition February 2011, 39 (2) 239-246; DOI: https://doi.org/10.1124/dmd.110.035022
F
Ferrari, Luca
- You have accessTissue Distribution and Characterization of Drug-Related Material in Rats and Dogs after Repeated Oral Administration of CasopitantSabrina Pagliarusco, Silvia Martinucci, Ellenia Bordini, Lidia Miraglia, Domenico Cufari, Luca Ferrari and Mario PellegattiDrug Metabolism and Disposition February 2011, 39 (2) 283-293; DOI: https://doi.org/10.1124/dmd.110.035063
Folmer, James J.
- You have accessElucidation of a Novel Bioactivation Pathway of a 3,4-Unsubstituted Isoxazole in Human Liver Microsomes: Formation of a Glutathione Adduct of a Cyanoacrolein Derivative after Isoxazole Ring OpeningJian Yu, James J. Folmer, Valerie Hoesch, James Doherty, James B. Campbell and Doug BurdetteDrug Metabolism and Disposition February 2011, 39 (2) 302-311; DOI: https://doi.org/10.1124/dmd.110.036285
Fontana, Stefano
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
Forsgard, Niklas
- You have accessMorphine Brain Pharmacokinetics at Very Low Concentrations Studied with Accelerator Mass Spectrometry and Liquid Chromatography-Tandem Mass SpectrometryMuhammad Waqas Sadiq, Mehran Salehpour, Niklas Forsgard, Göran Possnert and Margareta Hammarlund-UdenaesDrug Metabolism and Disposition February 2011, 39 (2) 174-179; DOI: https://doi.org/10.1124/dmd.110.036434
Fransson, Martin N.
- You have accessInfluence of Cremophor EL and Genetic Polymorphisms on the Pharmacokinetics of Paclitaxel and Its Metabolites Using a Mechanism-Based ModelMartin N. Fransson, Henrik Gréen, Jan-Eric Litton and Lena E. FribergDrug Metabolism and Disposition February 2011, 39 (2) 247-255; DOI: https://doi.org/10.1124/dmd.110.035394
Friberg, Lena E.
- You have accessInfluence of Cremophor EL and Genetic Polymorphisms on the Pharmacokinetics of Paclitaxel and Its Metabolites Using a Mechanism-Based ModelMartin N. Fransson, Henrik Gréen, Jan-Eric Litton and Lena E. FribergDrug Metabolism and Disposition February 2011, 39 (2) 247-255; DOI: https://doi.org/10.1124/dmd.110.035394
Fujita, Ken-ichi
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
G
Galetin, Aleksandra
- You have accessCritique of the Two-Fold Measure of Prediction Success for Ratios: Application for the Assessment of Drug-Drug InteractionsEleanor J. Guest, Leon Aarons, J. Brian Houston, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition February 2011, 39 (2) 170-173; DOI: https://doi.org/10.1124/dmd.110.036103
Gillen, Michael
- You have accessThe Utility of In Vitro Data in Making Accurate Predictions of Human P-Glycoprotein-Mediated Drug-Drug Interactions: A Case Study for AZD5672Robert Elsby, Michael Gillen, Caroline Butters, Gemma Imisson, Pradeep Sharma, Veronica Smith and Dominic D. SurryDrug Metabolism and Disposition February 2011, 39 (2) 275-282; DOI: https://doi.org/10.1124/dmd.110.035881
Gréen, Henrik
- You have accessInfluence of Cremophor EL and Genetic Polymorphisms on the Pharmacokinetics of Paclitaxel and Its Metabolites Using a Mechanism-Based ModelMartin N. Fransson, Henrik Gréen, Jan-Eric Litton and Lena E. FribergDrug Metabolism and Disposition February 2011, 39 (2) 247-255; DOI: https://doi.org/10.1124/dmd.110.035394
Grossman, Scott J.
- You have accessTissue Distribution and Elimination of [14C]Apixaban in RatsLifei Wang, Kan He, Brad Maxwell, Scott J. Grossman, Larry M. Tremaine, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 256-264; DOI: https://doi.org/10.1124/dmd.110.036442
Gschwind, Hans-Peter
- You have accessAbsorption and Disposition of the Sphingosine 1-Phosphate Receptor Modulator Fingolimod (FTY720) in Healthy Volunteers: A Case of Xenobiotic Biotransformation Following Endogenous Metabolic PathwaysMarkus Zollinger, Hans-Peter Gschwind, Yi Jin, Claudia Sayer, Frédéric Zécri and Stefan HartmannDrug Metabolism and Disposition February 2011, 39 (2) 199-207; DOI: https://doi.org/10.1124/dmd.110.035907
Guest, Eleanor J.
- You have accessCritique of the Two-Fold Measure of Prediction Success for Ratios: Application for the Assessment of Drug-Drug InteractionsEleanor J. Guest, Leon Aarons, J. Brian Houston, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition February 2011, 39 (2) 170-173; DOI: https://doi.org/10.1124/dmd.110.036103
H
Hagihara, Katsunobu
- You have accessGlutaredoxin and Thioredoxin Can Be Involved in Producing the Pharmacologically Active Metabolite of a Thienopyridine Antiplatelet Agent, PrasugrelKatsunobu Hagihara, Miho Kazui, Atsushi Kurihara, Kazuishi Kubota and Toshihiko IkedaDrug Metabolism and Disposition February 2011, 39 (2) 208-214; DOI: https://doi.org/10.1124/dmd.110.035196
Hammarlund-Udenaes, Margareta
- You have accessMorphine Brain Pharmacokinetics at Very Low Concentrations Studied with Accelerator Mass Spectrometry and Liquid Chromatography-Tandem Mass SpectrometryMuhammad Waqas Sadiq, Mehran Salehpour, Niklas Forsgard, Göran Possnert and Margareta Hammarlund-UdenaesDrug Metabolism and Disposition February 2011, 39 (2) 174-179; DOI: https://doi.org/10.1124/dmd.110.036434
Hankinson, Oliver
- You have accessHuman CYP2S1 Metabolizes Cyclooxygenase- and Lipoxygenase-Derived EicosanoidsPeter Bui, Satoshi Imaizumi, Sudheer Reddy Beedanagari, Srinivasa T. Reddy and Oliver HankinsonDrug Metabolism and Disposition February 2011, 39 (2) 180-190; DOI: https://doi.org/10.1124/dmd.110.035121
Hartmann, Stefan
- You have accessAbsorption and Disposition of the Sphingosine 1-Phosphate Receptor Modulator Fingolimod (FTY720) in Healthy Volunteers: A Case of Xenobiotic Biotransformation Following Endogenous Metabolic PathwaysMarkus Zollinger, Hans-Peter Gschwind, Yi Jin, Claudia Sayer, Frédéric Zécri and Stefan HartmannDrug Metabolism and Disposition February 2011, 39 (2) 199-207; DOI: https://doi.org/10.1124/dmd.110.035907
He, Kan
- You have accessTissue Distribution and Elimination of [14C]Apixaban in RatsLifei Wang, Kan He, Brad Maxwell, Scott J. Grossman, Larry M. Tremaine, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 256-264; DOI: https://doi.org/10.1124/dmd.110.036442
Helmdach, Lydia
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
Hirose, Takashi
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Hoesch, Valerie
- You have accessElucidation of a Novel Bioactivation Pathway of a 3,4-Unsubstituted Isoxazole in Human Liver Microsomes: Formation of a Glutathione Adduct of a Cyanoacrolein Derivative after Isoxazole Ring OpeningJian Yu, James J. Folmer, Valerie Hoesch, James Doherty, James B. Campbell and Doug BurdetteDrug Metabolism and Disposition February 2011, 39 (2) 302-311; DOI: https://doi.org/10.1124/dmd.110.036285
Hollenberg, Paul F.
- You have accessInactivation of Cytochrome P450 (P450) 3A4 but not P450 3A5 by OSI-930, a Thiophene-Containing Anticancer DrugHsia-lien Lin, Haoming Zhang, Christine Medower, Paul F. Hollenberg and William W. JohnsonDrug Metabolism and Disposition February 2011, 39 (2) 345-350; DOI: https://doi.org/10.1124/dmd.110.034074
Houston, J. Brian
- You have accessCritique of the Two-Fold Measure of Prediction Success for Ratios: Application for the Assessment of Drug-Drug InteractionsEleanor J. Guest, Leon Aarons, J. Brian Houston, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition February 2011, 39 (2) 170-173; DOI: https://doi.org/10.1124/dmd.110.036103
Humphreys, W. Griffith
- You have accessMetabolism and Disposition of 14C-Labeled Peliglitazar in HumansLifei Wang, Carey Munsick, Sean Chen, Samuel Bonacorsi, Peter T. Cheng, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 228-238; DOI: https://doi.org/10.1124/dmd.110.035089
- You have accessTissue Distribution and Elimination of [14C]Apixaban in RatsLifei Wang, Kan He, Brad Maxwell, Scott J. Grossman, Larry M. Tremaine, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 256-264; DOI: https://doi.org/10.1124/dmd.110.036442
I
Ichikawa, Wataru
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Ikeda, Toshihiko
- You have accessGlutaredoxin and Thioredoxin Can Be Involved in Producing the Pharmacologically Active Metabolite of a Thienopyridine Antiplatelet Agent, PrasugrelKatsunobu Hagihara, Miho Kazui, Atsushi Kurihara, Kazuishi Kubota and Toshihiko IkedaDrug Metabolism and Disposition February 2011, 39 (2) 208-214; DOI: https://doi.org/10.1124/dmd.110.035196
Imaizumi, Satoshi
- You have accessHuman CYP2S1 Metabolizes Cyclooxygenase- and Lipoxygenase-Derived EicosanoidsPeter Bui, Satoshi Imaizumi, Sudheer Reddy Beedanagari, Srinivasa T. Reddy and Oliver HankinsonDrug Metabolism and Disposition February 2011, 39 (2) 180-190; DOI: https://doi.org/10.1124/dmd.110.035121
Imisson, Gemma
- You have accessThe Utility of In Vitro Data in Making Accurate Predictions of Human P-Glycoprotein-Mediated Drug-Drug Interactions: A Case Study for AZD5672Robert Elsby, Michael Gillen, Caroline Butters, Gemma Imisson, Pradeep Sharma, Veronica Smith and Dominic D. SurryDrug Metabolism and Disposition February 2011, 39 (2) 275-282; DOI: https://doi.org/10.1124/dmd.110.035881
Ishida, Hiroo
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
J
Jeong, Hyunyoung
- You have accessAltered Cytochrome P450 Expression in Mice during PregnancyKwi Hye Koh, Hui Xie, Ai-Ming Yu and Hyunyoung JeongDrug Metabolism and Disposition February 2011, 39 (2) 165-169; DOI: https://doi.org/10.1124/dmd.110.035790
Jin, Yi
- You have accessCYP4F Enzymes Are Responsible for the Elimination of Fingolimod (FTY720), a Novel Treatment of Relapsing Multiple SclerosisYi Jin, Markus Zollinger, Hubert Borell, Alfred Zimmerlin and Christopher J. PattenDrug Metabolism and Disposition February 2011, 39 (2) 191-198; DOI: https://doi.org/10.1124/dmd.110.035378
- You have accessAbsorption and Disposition of the Sphingosine 1-Phosphate Receptor Modulator Fingolimod (FTY720) in Healthy Volunteers: A Case of Xenobiotic Biotransformation Following Endogenous Metabolic PathwaysMarkus Zollinger, Hans-Peter Gschwind, Yi Jin, Claudia Sayer, Frédéric Zécri and Stefan HartmannDrug Metabolism and Disposition February 2011, 39 (2) 199-207; DOI: https://doi.org/10.1124/dmd.110.035907
Johnson, William W.
- You have accessInactivation of Cytochrome P450 (P450) 3A4 but not P450 3A5 by OSI-930, a Thiophene-Containing Anticancer DrugHsia-lien Lin, Haoming Zhang, Christine Medower, Paul F. Hollenberg and William W. JohnsonDrug Metabolism and Disposition February 2011, 39 (2) 345-350; DOI: https://doi.org/10.1124/dmd.110.034074
K
Kawara, Kaori
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Kazui, Miho
- You have accessGlutaredoxin and Thioredoxin Can Be Involved in Producing the Pharmacologically Active Metabolite of a Thienopyridine Antiplatelet Agent, PrasugrelKatsunobu Hagihara, Miho Kazui, Atsushi Kurihara, Kazuishi Kubota and Toshihiko IkedaDrug Metabolism and Disposition February 2011, 39 (2) 208-214; DOI: https://doi.org/10.1124/dmd.110.035196
Kim, Gregory
- You have accessIdentification and Validation of Novel Human Pregnane X Receptor Activators among Prescribed Drugs via Ligand-Based Virtual ScreeningYongmei Pan, Linhao Li, Gregory Kim, Sean Ekins, Hongbing Wang and Peter W. SwaanDrug Metabolism and Disposition February 2011, 39 (2) 337-344; DOI: https://doi.org/10.1124/dmd.110.035808
Knutson, Lars
- You have accessEffects of Ketoconazole on the In Vivo Biotransformation and Hepatobiliary Transport of the Thrombin Inhibitor AZD0837 in PigsElin M. Matsson, Johan E. Palm, Ulf G. Eriksson, Pernilla Bottner, Anna Lundahl, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition February 2011, 39 (2) 239-246; DOI: https://doi.org/10.1124/dmd.110.035022
Koh, Kwi Hye
- You have accessAltered Cytochrome P450 Expression in Mice during PregnancyKwi Hye Koh, Hui Xie, Ai-Ming Yu and Hyunyoung JeongDrug Metabolism and Disposition February 2011, 39 (2) 165-169; DOI: https://doi.org/10.1124/dmd.110.035790
Kubota, Kazuishi
- You have accessGlutaredoxin and Thioredoxin Can Be Involved in Producing the Pharmacologically Active Metabolite of a Thienopyridine Antiplatelet Agent, PrasugrelKatsunobu Hagihara, Miho Kazui, Atsushi Kurihara, Kazuishi Kubota and Toshihiko IkedaDrug Metabolism and Disposition February 2011, 39 (2) 208-214; DOI: https://doi.org/10.1124/dmd.110.035196
Kurihara, Atsushi
- You have accessGlutaredoxin and Thioredoxin Can Be Involved in Producing the Pharmacologically Active Metabolite of a Thienopyridine Antiplatelet Agent, PrasugrelKatsunobu Hagihara, Miho Kazui, Atsushi Kurihara, Kazuishi Kubota and Toshihiko IkedaDrug Metabolism and Disposition February 2011, 39 (2) 208-214; DOI: https://doi.org/10.1124/dmd.110.035196
L
Lennernäs, Hans
- You have accessEffects of Ketoconazole on the In Vivo Biotransformation and Hepatobiliary Transport of the Thrombin Inhibitor AZD0837 in PigsElin M. Matsson, Johan E. Palm, Ulf G. Eriksson, Pernilla Bottner, Anna Lundahl, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition February 2011, 39 (2) 239-246; DOI: https://doi.org/10.1124/dmd.110.035022
Li, Linhao
- You have accessIdentification and Validation of Novel Human Pregnane X Receptor Activators among Prescribed Drugs via Ligand-Based Virtual ScreeningYongmei Pan, Linhao Li, Gregory Kim, Sean Ekins, Hongbing Wang and Peter W. SwaanDrug Metabolism and Disposition February 2011, 39 (2) 337-344; DOI: https://doi.org/10.1124/dmd.110.035808
Lin, Hsia-lien
- You have accessInactivation of Cytochrome P450 (P450) 3A4 but not P450 3A5 by OSI-930, a Thiophene-Containing Anticancer DrugHsia-lien Lin, Haoming Zhang, Christine Medower, Paul F. Hollenberg and William W. JohnsonDrug Metabolism and Disposition February 2011, 39 (2) 345-350; DOI: https://doi.org/10.1124/dmd.110.034074
Lin, Xuena
- You have accessAttenuation of Intestinal Absorption by Major Efflux Transporters: Quantitative Tools and Strategies Using a Caco-2 ModelXuena Lin, Suzanne Skolnik, Xiaohui Chen and Jianling WangDrug Metabolism and Disposition February 2011, 39 (2) 265-274; DOI: https://doi.org/10.1124/dmd.110.034629
Litton, Jan-Eric
- You have accessInfluence of Cremophor EL and Genetic Polymorphisms on the Pharmacokinetics of Paclitaxel and Its Metabolites Using a Mechanism-Based ModelMartin N. Fransson, Henrik Gréen, Jan-Eric Litton and Lena E. FribergDrug Metabolism and Disposition February 2011, 39 (2) 247-255; DOI: https://doi.org/10.1124/dmd.110.035394
Lledó-García, R.
- You have accessA Pharmacokinetic Model for Evaluating the Impact of Hepatic and Intestinal First-Pass Loss of Saquinavir in the RatR. Lledó-García, A. Nácher, V. G. Casabó and M. Merino-SanjuánDrug Metabolism and Disposition February 2011, 39 (2) 294-301; DOI: https://doi.org/10.1124/dmd.110.034488
Longhi, Raffaele
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
Lu, Yongke
- You have accessEthanol Induction of CYP2A5: Permissive Role for CYP2E1Yongke Lu, Jian Zhuge, Defeng Wu and Arthur I. CederbaumDrug Metabolism and Disposition February 2011, 39 (2) 330-336; DOI: https://doi.org/10.1124/dmd.110.035691
Lundahl, Anna
- You have accessEffects of Ketoconazole on the In Vivo Biotransformation and Hepatobiliary Transport of the Thrombin Inhibitor AZD0837 in PigsElin M. Matsson, Johan E. Palm, Ulf G. Eriksson, Pernilla Bottner, Anna Lundahl, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition February 2011, 39 (2) 239-246; DOI: https://doi.org/10.1124/dmd.110.035022
M
Martinucci, Silvia
- You have accessTissue Distribution and Characterization of Drug-Related Material in Rats and Dogs after Repeated Oral Administration of CasopitantSabrina Pagliarusco, Silvia Martinucci, Ellenia Bordini, Lidia Miraglia, Domenico Cufari, Luca Ferrari and Mario PellegattiDrug Metabolism and Disposition February 2011, 39 (2) 283-293; DOI: https://doi.org/10.1124/dmd.110.035063
Matsson, Elin M.
- You have accessEffects of Ketoconazole on the In Vivo Biotransformation and Hepatobiliary Transport of the Thrombin Inhibitor AZD0837 in PigsElin M. Matsson, Johan E. Palm, Ulf G. Eriksson, Pernilla Bottner, Anna Lundahl, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition February 2011, 39 (2) 239-246; DOI: https://doi.org/10.1124/dmd.110.035022
Maxwell, Brad
- You have accessTissue Distribution and Elimination of [14C]Apixaban in RatsLifei Wang, Kan He, Brad Maxwell, Scott J. Grossman, Larry M. Tremaine, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 256-264; DOI: https://doi.org/10.1124/dmd.110.036442
Medower, Christine
- You have accessInactivation of Cytochrome P450 (P450) 3A4 but not P450 3A5 by OSI-930, a Thiophene-Containing Anticancer DrugHsia-lien Lin, Haoming Zhang, Christine Medower, Paul F. Hollenberg and William W. JohnsonDrug Metabolism and Disposition February 2011, 39 (2) 345-350; DOI: https://doi.org/10.1124/dmd.110.034074
Merino-Sanjuán, M.
- You have accessA Pharmacokinetic Model for Evaluating the Impact of Hepatic and Intestinal First-Pass Loss of Saquinavir in the RatR. Lledó-García, A. Nácher, V. G. Casabó and M. Merino-SanjuánDrug Metabolism and Disposition February 2011, 39 (2) 294-301; DOI: https://doi.org/10.1124/dmd.110.034488
Miraglia, Lidia
- You have accessTissue Distribution and Characterization of Drug-Related Material in Rats and Dogs after Repeated Oral Administration of CasopitantSabrina Pagliarusco, Silvia Martinucci, Ellenia Bordini, Lidia Miraglia, Domenico Cufari, Luca Ferrari and Mario PellegattiDrug Metabolism and Disposition February 2011, 39 (2) 283-293; DOI: https://doi.org/10.1124/dmd.110.035063
Miwa, Keisuke
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Miya, Toshimichi
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Mizuno, Keiko
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Munsick, Carey
- You have accessMetabolism and Disposition of 14C-Labeled Peliglitazar in HumansLifei Wang, Carey Munsick, Sean Chen, Samuel Bonacorsi, Peter T. Cheng, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 228-238; DOI: https://doi.org/10.1124/dmd.110.035089
N
Nácher, A.
- You have accessA Pharmacokinetic Model for Evaluating the Impact of Hepatic and Intestinal First-Pass Loss of Saquinavir in the RatR. Lledó-García, A. Nácher, V. G. Casabó and M. Merino-SanjuánDrug Metabolism and Disposition February 2011, 39 (2) 294-301; DOI: https://doi.org/10.1124/dmd.110.034488
Nagashima, Fumio
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Narabayashi, Masaru
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Nash, Mike
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
P
Pagliarusco, Sabrina
- You have accessTissue Distribution and Characterization of Drug-Related Material in Rats and Dogs after Repeated Oral Administration of CasopitantSabrina Pagliarusco, Silvia Martinucci, Ellenia Bordini, Lidia Miraglia, Domenico Cufari, Luca Ferrari and Mario PellegattiDrug Metabolism and Disposition February 2011, 39 (2) 283-293; DOI: https://doi.org/10.1124/dmd.110.035063
Palm, Johan E.
- You have accessEffects of Ketoconazole on the In Vivo Biotransformation and Hepatobiliary Transport of the Thrombin Inhibitor AZD0837 in PigsElin M. Matsson, Johan E. Palm, Ulf G. Eriksson, Pernilla Bottner, Anna Lundahl, Lars Knutson and Hans LennernäsDrug Metabolism and Disposition February 2011, 39 (2) 239-246; DOI: https://doi.org/10.1124/dmd.110.035022
Pan, Yongmei
- You have accessIdentification and Validation of Novel Human Pregnane X Receptor Activators among Prescribed Drugs via Ligand-Based Virtual ScreeningYongmei Pan, Linhao Li, Gregory Kim, Sean Ekins, Hongbing Wang and Peter W. SwaanDrug Metabolism and Disposition February 2011, 39 (2) 337-344; DOI: https://doi.org/10.1124/dmd.110.035808
Patten, Christopher J.
- You have accessCYP4F Enzymes Are Responsible for the Elimination of Fingolimod (FTY720), a Novel Treatment of Relapsing Multiple SclerosisYi Jin, Markus Zollinger, Hubert Borell, Alfred Zimmerlin and Christopher J. PattenDrug Metabolism and Disposition February 2011, 39 (2) 191-198; DOI: https://doi.org/10.1124/dmd.110.035378
Pellegatti, Mario
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
- You have accessTissue Distribution and Characterization of Drug-Related Material in Rats and Dogs after Repeated Oral Administration of CasopitantSabrina Pagliarusco, Silvia Martinucci, Ellenia Bordini, Lidia Miraglia, Domenico Cufari, Luca Ferrari and Mario PellegattiDrug Metabolism and Disposition February 2011, 39 (2) 283-293; DOI: https://doi.org/10.1124/dmd.110.035063
Possnert, Göran
- You have accessMorphine Brain Pharmacokinetics at Very Low Concentrations Studied with Accelerator Mass Spectrometry and Liquid Chromatography-Tandem Mass SpectrometryMuhammad Waqas Sadiq, Mehran Salehpour, Niklas Forsgard, Göran Possnert and Margareta Hammarlund-UdenaesDrug Metabolism and Disposition February 2011, 39 (2) 174-179; DOI: https://doi.org/10.1124/dmd.110.036434
R
Reddy, Srinivasa T.
- You have accessHuman CYP2S1 Metabolizes Cyclooxygenase- and Lipoxygenase-Derived EicosanoidsPeter Bui, Satoshi Imaizumi, Sudheer Reddy Beedanagari, Srinivasa T. Reddy and Oliver HankinsonDrug Metabolism and Disposition February 2011, 39 (2) 180-190; DOI: https://doi.org/10.1124/dmd.110.035121
Remmel, Rory P.
- You have accessCorrelation between Bilirubin Glucuronidation and Estradiol-3-Gluronidation in the Presence of Model UDP-Glucuronosyltransferase 1A1 Substrates/InhibitorsJin Zhou, Timothy S. Tracy and Rory P. RemmelDrug Metabolism and Disposition February 2011, 39 (2) 322-329; DOI: https://doi.org/10.1124/dmd.110.035030
Renzulli, Cecilia
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
Rostami-Hodjegan, Amin
- You have accessCritique of the Two-Fold Measure of Prediction Success for Ratios: Application for the Assessment of Drug-Drug InteractionsEleanor J. Guest, Leon Aarons, J. Brian Houston, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition February 2011, 39 (2) 170-173; DOI: https://doi.org/10.1124/dmd.110.036103
S
Sadiq, Muhammad Waqas
- You have accessMorphine Brain Pharmacokinetics at Very Low Concentrations Studied with Accelerator Mass Spectrometry and Liquid Chromatography-Tandem Mass SpectrometryMuhammad Waqas Sadiq, Mehran Salehpour, Niklas Forsgard, Göran Possnert and Margareta Hammarlund-UdenaesDrug Metabolism and Disposition February 2011, 39 (2) 174-179; DOI: https://doi.org/10.1124/dmd.110.036434
Saji, Shigehira
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Salehpour, Mehran
- You have accessMorphine Brain Pharmacokinetics at Very Low Concentrations Studied with Accelerator Mass Spectrometry and Liquid Chromatography-Tandem Mass SpectrometryMuhammad Waqas Sadiq, Mehran Salehpour, Niklas Forsgard, Göran Possnert and Margareta Hammarlund-UdenaesDrug Metabolism and Disposition February 2011, 39 (2) 174-179; DOI: https://doi.org/10.1124/dmd.110.036434
Sasaki, Yasutsuna
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Sayer, Claudia
- You have accessAbsorption and Disposition of the Sphingosine 1-Phosphate Receptor Modulator Fingolimod (FTY720) in Healthy Volunteers: A Case of Xenobiotic Biotransformation Following Endogenous Metabolic PathwaysMarkus Zollinger, Hans-Peter Gschwind, Yi Jin, Claudia Sayer, Frédéric Zécri and Stefan HartmannDrug Metabolism and Disposition February 2011, 39 (2) 199-207; DOI: https://doi.org/10.1124/dmd.110.035907
Schiller, Jürgen
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
Sharma, Pradeep
- You have accessThe Utility of In Vitro Data in Making Accurate Predictions of Human P-Glycoprotein-Mediated Drug-Drug Interactions: A Case Study for AZD5672Robert Elsby, Michael Gillen, Caroline Butters, Gemma Imisson, Pradeep Sharma, Veronica Smith and Dominic D. SurryDrug Metabolism and Disposition February 2011, 39 (2) 275-282; DOI: https://doi.org/10.1124/dmd.110.035881
Skolnik, Suzanne
- You have accessAttenuation of Intestinal Absorption by Major Efflux Transporters: Quantitative Tools and Strategies Using a Caco-2 ModelXuena Lin, Suzanne Skolnik, Xiaohui Chen and Jianling WangDrug Metabolism and Disposition February 2011, 39 (2) 265-274; DOI: https://doi.org/10.1124/dmd.110.034629
Smith, Veronica
- You have accessThe Utility of In Vitro Data in Making Accurate Predictions of Human P-Glycoprotein-Mediated Drug-Drug Interactions: A Case Study for AZD5672Robert Elsby, Michael Gillen, Caroline Butters, Gemma Imisson, Pradeep Sharma, Veronica Smith and Dominic D. SurryDrug Metabolism and Disposition February 2011, 39 (2) 275-282; DOI: https://doi.org/10.1124/dmd.110.035881
Sugiyama, Minako
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Sunakawa, Yu
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Surry, Dominic D.
- You have accessThe Utility of In Vitro Data in Making Accurate Predictions of Human P-Glycoprotein-Mediated Drug-Drug Interactions: A Case Study for AZD5672Robert Elsby, Michael Gillen, Caroline Butters, Gemma Imisson, Pradeep Sharma, Veronica Smith and Dominic D. SurryDrug Metabolism and Disposition February 2011, 39 (2) 275-282; DOI: https://doi.org/10.1124/dmd.110.035881
Swaan, Peter W.
- You have accessIdentification and Validation of Novel Human Pregnane X Receptor Activators among Prescribed Drugs via Ligand-Based Virtual ScreeningYongmei Pan, Linhao Li, Gregory Kim, Sean Ekins, Hongbing Wang and Peter W. SwaanDrug Metabolism and Disposition February 2011, 39 (2) 337-344; DOI: https://doi.org/10.1124/dmd.110.035808
T
Thomas, Steven
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
Tracy, Timothy S.
- You have accessCorrelation between Bilirubin Glucuronidation and Estradiol-3-Gluronidation in the Presence of Model UDP-Glucuronosyltransferase 1A1 Substrates/InhibitorsJin Zhou, Timothy S. Tracy and Rory P. RemmelDrug Metabolism and Disposition February 2011, 39 (2) 322-329; DOI: https://doi.org/10.1124/dmd.110.035030
Tremaine, Larry M.
- You have accessTissue Distribution and Elimination of [14C]Apixaban in RatsLifei Wang, Kan He, Brad Maxwell, Scott J. Grossman, Larry M. Tremaine, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 256-264; DOI: https://doi.org/10.1124/dmd.110.036442
V
Vinco, Federicia
- You have accessBrain Tissue Binding of Drugs: Evaluation and Validation of Solid Supported Porcine Brain Membrane Vesicles (TRANSIL) as a Novel High-Throughput MethodRaffaele Longhi, Silvia Corbioli, Stefano Fontana, Federicia Vinco, Simone Braggio, Lydia Helmdach, Jürgen Schiller and Hinnerk BorissDrug Metabolism and Disposition February 2011, 39 (2) 312-321; DOI: https://doi.org/10.1124/dmd.110.036095
W
Wang, Hongbing
- You have accessIdentification and Validation of Novel Human Pregnane X Receptor Activators among Prescribed Drugs via Ligand-Based Virtual ScreeningYongmei Pan, Linhao Li, Gregory Kim, Sean Ekins, Hongbing Wang and Peter W. SwaanDrug Metabolism and Disposition February 2011, 39 (2) 337-344; DOI: https://doi.org/10.1124/dmd.110.035808
Wang, Jianling
- You have accessAttenuation of Intestinal Absorption by Major Efflux Transporters: Quantitative Tools and Strategies Using a Caco-2 ModelXuena Lin, Suzanne Skolnik, Xiaohui Chen and Jianling WangDrug Metabolism and Disposition February 2011, 39 (2) 265-274; DOI: https://doi.org/10.1124/dmd.110.034629
Wang, Lifei
- You have accessMetabolism and Disposition of 14C-Labeled Peliglitazar in HumansLifei Wang, Carey Munsick, Sean Chen, Samuel Bonacorsi, Peter T. Cheng, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 228-238; DOI: https://doi.org/10.1124/dmd.110.035089
- You have accessTissue Distribution and Elimination of [14C]Apixaban in RatsLifei Wang, Kan He, Brad Maxwell, Scott J. Grossman, Larry M. Tremaine, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 256-264; DOI: https://doi.org/10.1124/dmd.110.036442
Wright, Mark
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
Wu, Defeng
- You have accessEthanol Induction of CYP2A5: Permissive Role for CYP2E1Yongke Lu, Jian Zhuge, Defeng Wu and Arthur I. CederbaumDrug Metabolism and Disposition February 2011, 39 (2) 330-336; DOI: https://doi.org/10.1124/dmd.110.035691
X
Xie, Hui
- You have accessAltered Cytochrome P450 Expression in Mice during PregnancyKwi Hye Koh, Hui Xie, Ai-Ming Yu and Hyunyoung JeongDrug Metabolism and Disposition February 2011, 39 (2) 165-169; DOI: https://doi.org/10.1124/dmd.110.035790
Y
Yamamoto, Wataru
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Yamashita, Keishi
- You have accessDelayed Elimination of SN-38 in Cancer Patients with Severe Renal FailureKen-ichi Fujita, Yu Sunakawa, Keisuke Miwa, Yuko Akiyama, Minako Sugiyama, Kaori Kawara, Hiroo Ishida, Keishi Yamashita, Keiko Mizuno, Shigehira Saji, Wataru Ichikawa, Wataru Yamamoto, Fumio Nagashima, Toshimichi Miya, Masaru Narabayashi, Yuichi Ando, Takashi Hirose and Yasutsuna SasakiDrug Metabolism and Disposition February 2011, 39 (2) 161-164; DOI: https://doi.org/10.1124/dmd.110.035451
Yu, Ai-Ming
- You have accessAltered Cytochrome P450 Expression in Mice during PregnancyKwi Hye Koh, Hui Xie, Ai-Ming Yu and Hyunyoung JeongDrug Metabolism and Disposition February 2011, 39 (2) 165-169; DOI: https://doi.org/10.1124/dmd.110.035790
Yu, Jian
- You have accessElucidation of a Novel Bioactivation Pathway of a 3,4-Unsubstituted Isoxazole in Human Liver Microsomes: Formation of a Glutathione Adduct of a Cyanoacrolein Derivative after Isoxazole Ring OpeningJian Yu, James J. Folmer, Valerie Hoesch, James Doherty, James B. Campbell and Doug BurdetteDrug Metabolism and Disposition February 2011, 39 (2) 302-311; DOI: https://doi.org/10.1124/dmd.110.036285
Z
Zamuner, Stefano
- You have accessDisposition and Metabolism of [14C]SB-649868, an Orexin 1 and 2 Receptor Antagonist, in HumansCecilia Renzulli, Mike Nash, Mark Wright, Steven Thomas, Stefano Zamuner, Mario Pellegatti, Paolo Bettica and Gary BoyleDrug Metabolism and Disposition February 2011, 39 (2) 215-227; DOI: https://doi.org/10.1124/dmd.110.035386
Zécri, Frédéric
- You have accessAbsorption and Disposition of the Sphingosine 1-Phosphate Receptor Modulator Fingolimod (FTY720) in Healthy Volunteers: A Case of Xenobiotic Biotransformation Following Endogenous Metabolic PathwaysMarkus Zollinger, Hans-Peter Gschwind, Yi Jin, Claudia Sayer, Frédéric Zécri and Stefan HartmannDrug Metabolism and Disposition February 2011, 39 (2) 199-207; DOI: https://doi.org/10.1124/dmd.110.035907
Zhang, Donglu
- You have accessMetabolism and Disposition of 14C-Labeled Peliglitazar in HumansLifei Wang, Carey Munsick, Sean Chen, Samuel Bonacorsi, Peter T. Cheng, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 228-238; DOI: https://doi.org/10.1124/dmd.110.035089
- You have accessTissue Distribution and Elimination of [14C]Apixaban in RatsLifei Wang, Kan He, Brad Maxwell, Scott J. Grossman, Larry M. Tremaine, W. Griffith Humphreys and Donglu ZhangDrug Metabolism and Disposition February 2011, 39 (2) 256-264; DOI: https://doi.org/10.1124/dmd.110.036442
Zhang, Haoming
- You have accessInactivation of Cytochrome P450 (P450) 3A4 but not P450 3A5 by OSI-930, a Thiophene-Containing Anticancer DrugHsia-lien Lin, Haoming Zhang, Christine Medower, Paul F. Hollenberg and William W. JohnsonDrug Metabolism and Disposition February 2011, 39 (2) 345-350; DOI: https://doi.org/10.1124/dmd.110.034074
Zhou, Jin
- You have accessCorrelation between Bilirubin Glucuronidation and Estradiol-3-Gluronidation in the Presence of Model UDP-Glucuronosyltransferase 1A1 Substrates/InhibitorsJin Zhou, Timothy S. Tracy and Rory P. RemmelDrug Metabolism and Disposition February 2011, 39 (2) 322-329; DOI: https://doi.org/10.1124/dmd.110.035030
Zhuge, Jian
- You have accessEthanol Induction of CYP2A5: Permissive Role for CYP2E1Yongke Lu, Jian Zhuge, Defeng Wu and Arthur I. CederbaumDrug Metabolism and Disposition February 2011, 39 (2) 330-336; DOI: https://doi.org/10.1124/dmd.110.035691
Zimmerlin, Alfred
- You have accessCYP4F Enzymes Are Responsible for the Elimination of Fingolimod (FTY720), a Novel Treatment of Relapsing Multiple SclerosisYi Jin, Markus Zollinger, Hubert Borell, Alfred Zimmerlin and Christopher J. PattenDrug Metabolism and Disposition February 2011, 39 (2) 191-198; DOI: https://doi.org/10.1124/dmd.110.035378
Zollinger, Markus
- You have accessCYP4F Enzymes Are Responsible for the Elimination of Fingolimod (FTY720), a Novel Treatment of Relapsing Multiple SclerosisYi Jin, Markus Zollinger, Hubert Borell, Alfred Zimmerlin and Christopher J. PattenDrug Metabolism and Disposition February 2011, 39 (2) 191-198; DOI: https://doi.org/10.1124/dmd.110.035378
- You have accessAbsorption and Disposition of the Sphingosine 1-Phosphate Receptor Modulator Fingolimod (FTY720) in Healthy Volunteers: A Case of Xenobiotic Biotransformation Following Endogenous Metabolic PathwaysMarkus Zollinger, Hans-Peter Gschwind, Yi Jin, Claudia Sayer, Frédéric Zécri and Stefan HartmannDrug Metabolism and Disposition February 2011, 39 (2) 199-207; DOI: https://doi.org/10.1124/dmd.110.035907
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