Index by author
March 01, 2011; Volume 39,Issue 3
A
Abe, Koji
- You have accessDecreased Hepatic Breast Cancer Resistance Protein Expression and Function in Multidrug Resistance-Associated Protein 2-Deficient (TR−) RatsWei Yue, Jin Kyung Lee, Koji Abe, Yuichi Sugiyama and Kim L. R. BrouwerDrug Metabolism and Disposition March 2011, 39 (3) 441-447; DOI: https://doi.org/10.1124/dmd.110.035188
Ahlin, Gustav
- You have accessMeasurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate MethodsMarkus Fridén, Fredrik Bergström, Hong Wan, Mikael Rehngren, Gustav Ahlin, Margareta Hammarlund-Udenaes and Ulf BredbergDrug Metabolism and Disposition March 2011, 39 (3) 353-362; DOI: https://doi.org/10.1124/dmd.110.035998
Akhlaghi, Fatemeh
- You have accessDiabetes Mellitus Reduces Activity of Human UDP-Glucuronosyltransferase 2B7 in Liver and Kidney Leading to Decreased Formation of Mycophenolic Acid Acyl-Glucuronide MetaboliteMiroslav Dostalek, Michael H. Court, Suwagmani Hazarika and Fatemeh AkhlaghiDrug Metabolism and Disposition March 2011, 39 (3) 448-455; DOI: https://doi.org/10.1124/dmd.110.036608
Alton, Kevin B.
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
An, Guohua
- You have accessThe Bioflavonoid Kaempferol Is an Abcg2 Substrate and Inhibits Abcg2-Mediated Quercetin EffluxGuohua An, Jorge Gallegos and Marilyn E. MorrisDrug Metabolism and Disposition March 2011, 39 (3) 426-432; DOI: https://doi.org/10.1124/dmd.110.035212
Anderson, Peter L.
- You have accessAtazanavir Metabolism According to CYP3A5 Status: An In Vitro-In Vivo AssessmentMichael F. Wempe and Peter L. AndersonDrug Metabolism and Disposition March 2011, 39 (3) 522-527; DOI: https://doi.org/10.1124/dmd.110.036178
Auriola, Seppo
- You have accessSimple, Direct, and Informative Method for the Assessment of CYP2C19 Enzyme Inactivation KineticsKaisa A. Salminen, Jukka Leppänen, Jarkko I. Venäläinen, Markku Pasanen, Seppo Auriola, Risto O. Juvonen and Hannu RaunioDrug Metabolism and Disposition March 2011, 39 (3) 412-418; DOI: https://doi.org/10.1124/dmd.110.036376
Aw, Chiu Cheong
- You have accessPharmacokinetic and Pharmacodynamic Properties of Cholinesterase Inhibitors Donepezil, Tacrine, and Galantamine in Aged and Young Lister Hooded RatsCatherine W. Goh, Chiu Cheong Aw, Jasinda H. Lee, Christopher P. Chen and Edward R. BrowneDrug Metabolism and Disposition March 2011, 39 (3) 402-411; DOI: https://doi.org/10.1124/dmd.110.035964
B
Bergström, Fredrik
- You have accessMeasurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate MethodsMarkus Fridén, Fredrik Bergström, Hong Wan, Mikael Rehngren, Gustav Ahlin, Margareta Hammarlund-Udenaes and Ulf BredbergDrug Metabolism and Disposition March 2011, 39 (3) 353-362; DOI: https://doi.org/10.1124/dmd.110.035998
Bhadhprasit, Wattanaporn
- You have accessHepatocyte Nuclear Factor 4α Regulates Expression of the Mouse Female-Specific Cyp3a41 Gene in the LiverWattanaporn Bhadhprasit, Tsutomu Sakuma, Yuki Kawasaki and Nobuo NemotoDrug Metabolism and Disposition March 2011, 39 (3) 490-497; DOI: https://doi.org/10.1124/dmd.110.035980
Bonomo, Fiorenza
- You have accessCasopitant: In Vitro Data and SimCyp Simulation to Predict In Vivo Metabolic Interactions Involving Cytochrome P450 3A4Paola Motta, Nicoletta Pons, Sabrina Pagliarusco, Mario Pellegatti and Fiorenza BonomoDrug Metabolism and Disposition March 2011, 39 (3) 363-372; DOI: https://doi.org/10.1124/dmd.110.035071
Branham, William
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Bredberg, Ulf
- You have accessMeasurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate MethodsMarkus Fridén, Fredrik Bergström, Hong Wan, Mikael Rehngren, Gustav Ahlin, Margareta Hammarlund-Udenaes and Ulf BredbergDrug Metabolism and Disposition March 2011, 39 (3) 353-362; DOI: https://doi.org/10.1124/dmd.110.035998
Brouwer, Kim L. R.
- You have accessDecreased Hepatic Breast Cancer Resistance Protein Expression and Function in Multidrug Resistance-Associated Protein 2-Deficient (TR−) RatsWei Yue, Jin Kyung Lee, Koji Abe, Yuichi Sugiyama and Kim L. R. BrouwerDrug Metabolism and Disposition March 2011, 39 (3) 441-447; DOI: https://doi.org/10.1124/dmd.110.035188
Browne, Edward R.
- You have accessPharmacokinetic and Pharmacodynamic Properties of Cholinesterase Inhibitors Donepezil, Tacrine, and Galantamine in Aged and Young Lister Hooded RatsCatherine W. Goh, Chiu Cheong Aw, Jasinda H. Lee, Christopher P. Chen and Edward R. BrowneDrug Metabolism and Disposition March 2011, 39 (3) 402-411; DOI: https://doi.org/10.1124/dmd.110.035964
C
Chen, Christopher P.
- You have accessPharmacokinetic and Pharmacodynamic Properties of Cholinesterase Inhibitors Donepezil, Tacrine, and Galantamine in Aged and Young Lister Hooded RatsCatherine W. Goh, Chiu Cheong Aw, Jasinda H. Lee, Christopher P. Chen and Edward R. BrowneDrug Metabolism and Disposition March 2011, 39 (3) 402-411; DOI: https://doi.org/10.1124/dmd.110.035964
Chen, Guanming
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Chen, Ling-Jen
- You have accessDisposition and Metabolism of Cumene in F344 Rats and B6C3F1 MiceLing-Jen Chen, Christopher J. Wegerski, Daniel J. Kramer, Leslie A. Thomas, Jacob D. McDonald, Kelly J. Dix and J. Michael SandersDrug Metabolism and Disposition March 2011, 39 (3) 498-509; DOI: https://doi.org/10.1124/dmd.110.034769
Chen, Xiaoyan
- You have accessIdentification of 20(S)-Protopanaxadiol Metabolites in Human Liver Microsomes and Human HepatocytesLiang Li, Xiaoyan Chen, Dan Li and Dafang ZhongDrug Metabolism and Disposition March 2011, 39 (3) 472-483; DOI: https://doi.org/10.1124/dmd.110.036723
Chen, Yuan
- You have accessUtility of Intersystem Extrapolation Factors in Early Reaction Phenotyping and the Quantitative Extrapolation of Human Liver Microsomal Intrinsic Clearance Using Recombinant Cytochromes P450Yuan Chen, Liling Liu, Khanh Nguyen and Adrian J. FretlandDrug Metabolism and Disposition March 2011, 39 (3) 373-382; DOI: https://doi.org/10.1124/dmd.110.035147
Chowdhury, Swapan K.
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
Claxton, Christopher R. J.
- You have accessControl and Measurement of Plasma pH in Equilibrium Dialysis: Influence on Drug Plasma Protein BindingRuth E. Curran, Christopher R. J. Claxton, Laura Hutchison, Paul J. Harradine, Iain J. Martin and Peter LittlewoodDrug Metabolism and Disposition March 2011, 39 (3) 551-557; DOI: https://doi.org/10.1124/dmd.110.036988
Court, Michael H.
- You have accessDiabetes Mellitus Reduces Activity of Human UDP-Glucuronosyltransferase 2B7 in Liver and Kidney Leading to Decreased Formation of Mycophenolic Acid Acyl-Glucuronide MetaboliteMiroslav Dostalek, Michael H. Court, Suwagmani Hazarika and Fatemeh AkhlaghiDrug Metabolism and Disposition March 2011, 39 (3) 448-455; DOI: https://doi.org/10.1124/dmd.110.036608
Curran, Ruth E.
- You have accessControl and Measurement of Plasma pH in Equilibrium Dialysis: Influence on Drug Plasma Protein BindingRuth E. Curran, Christopher R. J. Claxton, Laura Hutchison, Paul J. Harradine, Iain J. Martin and Peter LittlewoodDrug Metabolism and Disposition March 2011, 39 (3) 551-557; DOI: https://doi.org/10.1124/dmd.110.036988
D
Dalvie, Deepak
- You have accessComparison of In Vitro Metabolism of Ticlopidine by Human Cytochrome P450 2B6 and Rabbit Cytochrome P450 2B4Jyothi C. Talakad, Manish B. Shah, Gregory S. Walker, Cathie Xiang, James R. Halpert and Deepak DalvieDrug Metabolism and Disposition March 2011, 39 (3) 539-550; DOI: https://doi.org/10.1124/dmd.110.037101
Deng, Helen
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Dial, Stacey
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Dix, Kelly J.
- You have accessDisposition and Metabolism of Cumene in F344 Rats and B6C3F1 MiceLing-Jen Chen, Christopher J. Wegerski, Daniel J. Kramer, Leslie A. Thomas, Jacob D. McDonald, Kelly J. Dix and J. Michael SandersDrug Metabolism and Disposition March 2011, 39 (3) 498-509; DOI: https://doi.org/10.1124/dmd.110.034769
Dostalek, Miroslav
- You have accessDiabetes Mellitus Reduces Activity of Human UDP-Glucuronosyltransferase 2B7 in Liver and Kidney Leading to Decreased Formation of Mycophenolic Acid Acyl-Glucuronide MetaboliteMiroslav Dostalek, Michael H. Court, Suwagmani Hazarika and Fatemeh AkhlaghiDrug Metabolism and Disposition March 2011, 39 (3) 448-455; DOI: https://doi.org/10.1124/dmd.110.036608
F
Fang, Jia-Long
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Finel, Moshe
- You have accessEffects of Cell Differentiation and Assay Conditions on the UDP-Glucuronosyltransferase Activity in Caco-2 CellsHongbo Zhang, Ari Tolonen, Timo Rousu, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition March 2011, 39 (3) 456-464; DOI: https://doi.org/10.1124/dmd.110.036582
Fretland, Adrian J.
- You have accessUtility of Intersystem Extrapolation Factors in Early Reaction Phenotyping and the Quantitative Extrapolation of Human Liver Microsomal Intrinsic Clearance Using Recombinant Cytochromes P450Yuan Chen, Liling Liu, Khanh Nguyen and Adrian J. FretlandDrug Metabolism and Disposition March 2011, 39 (3) 373-382; DOI: https://doi.org/10.1124/dmd.110.035147
Freund, Amy
- You have accessValidation of Isolated Metabolites from Drug Metabolism Studies as Analytical Standards by Quantitative NMRGregory S. Walker, Tim F. Ryder, Raman Sharma, Evan B. Smith and Amy FreundDrug Metabolism and Disposition March 2011, 39 (3) 433-440; DOI: https://doi.org/10.1124/dmd.110.036343
Fridén, Markus
- You have accessMeasurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate MethodsMarkus Fridén, Fredrik Bergström, Hong Wan, Mikael Rehngren, Gustav Ahlin, Margareta Hammarlund-Udenaes and Ulf BredbergDrug Metabolism and Disposition March 2011, 39 (3) 353-362; DOI: https://doi.org/10.1124/dmd.110.035998
G
Gahir, Sarabjit S.
- You have accessGestational and Pregnane X Receptor-Mediated Regulation of Placental ATP-Binding Cassette Drug Transporters in MiceSarabjit S. Gahir and Micheline Piquette-MillerDrug Metabolism and Disposition March 2011, 39 (3) 465-471; DOI: https://doi.org/10.1124/dmd.110.034983
Gallegos, Jorge
- You have accessThe Bioflavonoid Kaempferol Is an Abcg2 Substrate and Inhibits Abcg2-Mediated Quercetin EffluxGuohua An, Jorge Gallegos and Marilyn E. MorrisDrug Metabolism and Disposition March 2011, 39 (3) 426-432; DOI: https://doi.org/10.1124/dmd.110.035212
Ghosal, Anima
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
Goh, Catherine W.
- You have accessPharmacokinetic and Pharmacodynamic Properties of Cholinesterase Inhibitors Donepezil, Tacrine, and Galantamine in Aged and Young Lister Hooded RatsCatherine W. Goh, Chiu Cheong Aw, Jasinda H. Lee, Christopher P. Chen and Edward R. BrowneDrug Metabolism and Disposition March 2011, 39 (3) 402-411; DOI: https://doi.org/10.1124/dmd.110.035964
Green, Bridgett
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Gu, Chunyan
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
Guo, Lei
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
H
Halpert, James R.
- You have accessComparison of In Vitro Metabolism of Ticlopidine by Human Cytochrome P450 2B6 and Rabbit Cytochrome P450 2B4Jyothi C. Talakad, Manish B. Shah, Gregory S. Walker, Cathie Xiang, James R. Halpert and Deepak DalvieDrug Metabolism and Disposition March 2011, 39 (3) 539-550; DOI: https://doi.org/10.1124/dmd.110.037101
Hammarlund-Udenaes, Margareta
- You have accessMeasurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate MethodsMarkus Fridén, Fredrik Bergström, Hong Wan, Mikael Rehngren, Gustav Ahlin, Margareta Hammarlund-Udenaes and Ulf BredbergDrug Metabolism and Disposition March 2011, 39 (3) 353-362; DOI: https://doi.org/10.1124/dmd.110.035998
Harradine, Paul J.
- You have accessControl and Measurement of Plasma pH in Equilibrium Dialysis: Influence on Drug Plasma Protein BindingRuth E. Curran, Christopher R. J. Claxton, Laura Hutchison, Paul J. Harradine, Iain J. Martin and Peter LittlewoodDrug Metabolism and Disposition March 2011, 39 (3) 551-557; DOI: https://doi.org/10.1124/dmd.110.036988
Hazarika, Suwagmani
- You have accessDiabetes Mellitus Reduces Activity of Human UDP-Glucuronosyltransferase 2B7 in Liver and Kidney Leading to Decreased Formation of Mycophenolic Acid Acyl-Glucuronide MetaboliteMiroslav Dostalek, Michael H. Court, Suwagmani Hazarika and Fatemeh AkhlaghiDrug Metabolism and Disposition March 2011, 39 (3) 448-455; DOI: https://doi.org/10.1124/dmd.110.036608
Hirvonen, Jouni
- You have accessEffects of Cell Differentiation and Assay Conditions on the UDP-Glucuronosyltransferase Activity in Caco-2 CellsHongbo Zhang, Ari Tolonen, Timo Rousu, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition March 2011, 39 (3) 456-464; DOI: https://doi.org/10.1124/dmd.110.036582
Horinouchi, Hirohisa
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
Hu, Nan
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Hutchison, Laura
- You have accessControl and Measurement of Plasma pH in Equilibrium Dialysis: Influence on Drug Plasma Protein BindingRuth E. Curran, Christopher R. J. Claxton, Laura Hutchison, Paul J. Harradine, Iain J. Martin and Peter LittlewoodDrug Metabolism and Disposition March 2011, 39 (3) 551-557; DOI: https://doi.org/10.1124/dmd.110.036988
I
Iwao, Yasunori
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
J
Jones, Hannah M.
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
Juvonen, Risto O.
- You have accessSimple, Direct, and Informative Method for the Assessment of CYP2C19 Enzyme Inactivation KineticsKaisa A. Salminen, Jukka Leppänen, Jarkko I. Venäläinen, Markku Pasanen, Seppo Auriola, Risto O. Juvonen and Hannu RaunioDrug Metabolism and Disposition March 2011, 39 (3) 412-418; DOI: https://doi.org/10.1124/dmd.110.036376
K
Kadowaki, Daisuke
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
Kaput, Jim
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Kawasaki, Yuki
- You have accessHepatocyte Nuclear Factor 4α Regulates Expression of the Mouse Female-Specific Cyp3a41 Gene in the LiverWattanaporn Bhadhprasit, Tsutomu Sakuma, Yuki Kawasaki and Nobuo NemotoDrug Metabolism and Disposition March 2011, 39 (3) 490-497; DOI: https://doi.org/10.1124/dmd.110.035980
Kim, Richard B.
- You have accessEndoxifen, the Active Metabolite of Tamoxifen, Is a Substrate of the Efflux Transporter P-Glycoprotein (Multidrug Resistance 1)Wendy A. Teft, Sara E. Mansell and Richard B. KimDrug Metabolism and Disposition March 2011, 39 (3) 558-562; DOI: https://doi.org/10.1124/dmd.110.036160
Kishnani, Narendra S.
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
Kobayashi, Koichi
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
Koudriakova, Tatiana
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
Kramer, Daniel J.
- You have accessDisposition and Metabolism of Cumene in F344 Rats and B6C3F1 MiceLing-Jen Chen, Christopher J. Wegerski, Daniel J. Kramer, Leslie A. Thomas, Jacob D. McDonald, Kelly J. Dix and J. Michael SandersDrug Metabolism and Disposition March 2011, 39 (3) 498-509; DOI: https://doi.org/10.1124/dmd.110.034769
L
Lee, Jasinda H.
- You have accessPharmacokinetic and Pharmacodynamic Properties of Cholinesterase Inhibitors Donepezil, Tacrine, and Galantamine in Aged and Young Lister Hooded RatsCatherine W. Goh, Chiu Cheong Aw, Jasinda H. Lee, Christopher P. Chen and Edward R. BrowneDrug Metabolism and Disposition March 2011, 39 (3) 402-411; DOI: https://doi.org/10.1124/dmd.110.035964
Lee, Jin Kyung
- You have accessDecreased Hepatic Breast Cancer Resistance Protein Expression and Function in Multidrug Resistance-Associated Protein 2-Deficient (TR−) RatsWei Yue, Jin Kyung Lee, Koji Abe, Yuichi Sugiyama and Kim L. R. BrouwerDrug Metabolism and Disposition March 2011, 39 (3) 441-447; DOI: https://doi.org/10.1124/dmd.110.035188
Leppänen, Jukka
- You have accessSimple, Direct, and Informative Method for the Assessment of CYP2C19 Enzyme Inactivation KineticsKaisa A. Salminen, Jukka Leppänen, Jarkko I. Venäläinen, Markku Pasanen, Seppo Auriola, Risto O. Juvonen and Hannu RaunioDrug Metabolism and Disposition March 2011, 39 (3) 412-418; DOI: https://doi.org/10.1124/dmd.110.036376
Li, Dan
- You have accessIdentification of 20(S)-Protopanaxadiol Metabolites in Human Liver Microsomes and Human HepatocytesLiang Li, Xiaoyan Chen, Dan Li and Dafang ZhongDrug Metabolism and Disposition March 2011, 39 (3) 472-483; DOI: https://doi.org/10.1124/dmd.110.036723
Li, Feng
- You have accessCYP3A-Mediated Generation of Aldehyde and Hydrazine in Atazanavir MetabolismFeng Li, Jie Lu, Laiyou Wang and Xiaochao MaDrug Metabolism and Disposition March 2011, 39 (3) 394-401; DOI: https://doi.org/10.1124/dmd.110.036327
Li, Liang
- You have accessIdentification of 20(S)-Protopanaxadiol Metabolites in Human Liver Microsomes and Human HepatocytesLiang Li, Xiaoyan Chen, Dan Li and Dafang ZhongDrug Metabolism and Disposition March 2011, 39 (3) 472-483; DOI: https://doi.org/10.1124/dmd.110.036723
Littlewood, Peter
- You have accessControl and Measurement of Plasma pH in Equilibrium Dialysis: Influence on Drug Plasma Protein BindingRuth E. Curran, Christopher R. J. Claxton, Laura Hutchison, Paul J. Harradine, Iain J. Martin and Peter LittlewoodDrug Metabolism and Disposition March 2011, 39 (3) 551-557; DOI: https://doi.org/10.1124/dmd.110.036988
Liu, Haiyan
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Liu, Jie
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Liu, Li
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Liu, Liling
- You have accessUtility of Intersystem Extrapolation Factors in Early Reaction Phenotyping and the Quantitative Extrapolation of Human Liver Microsomal Intrinsic Clearance Using Recombinant Cytochromes P450Yuan Chen, Liling Liu, Khanh Nguyen and Adrian J. FretlandDrug Metabolism and Disposition March 2011, 39 (3) 373-382; DOI: https://doi.org/10.1124/dmd.110.035147
Liu, Xiang
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Liu, Xiaodong
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Lu, Jie
- You have accessCYP3A-Mediated Generation of Aldehyde and Hydrazine in Atazanavir MetabolismFeng Li, Jie Lu, Laiyou Wang and Xiaochao MaDrug Metabolism and Disposition March 2011, 39 (3) 394-401; DOI: https://doi.org/10.1124/dmd.110.036327
M
Ma, Xiaochao
- You have accessCYP3A-Mediated Generation of Aldehyde and Hydrazine in Atazanavir MetabolismFeng Li, Jie Lu, Laiyou Wang and Xiaochao MaDrug Metabolism and Disposition March 2011, 39 (3) 394-401; DOI: https://doi.org/10.1124/dmd.110.036327
Mansell, Sara E.
- You have accessEndoxifen, the Active Metabolite of Tamoxifen, Is a Substrate of the Efflux Transporter P-Glycoprotein (Multidrug Resistance 1)Wendy A. Teft, Sara E. Mansell and Richard B. KimDrug Metabolism and Disposition March 2011, 39 (3) 558-562; DOI: https://doi.org/10.1124/dmd.110.036160
Martin, Iain J.
- You have accessControl and Measurement of Plasma pH in Equilibrium Dialysis: Influence on Drug Plasma Protein BindingRuth E. Curran, Christopher R. J. Claxton, Laura Hutchison, Paul J. Harradine, Iain J. Martin and Peter LittlewoodDrug Metabolism and Disposition March 2011, 39 (3) 551-557; DOI: https://doi.org/10.1124/dmd.110.036988
Maruyama, Toru
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
McDonald, Jacob D.
- You have accessDisposition and Metabolism of Cumene in F344 Rats and B6C3F1 MiceLing-Jen Chen, Christopher J. Wegerski, Daniel J. Kramer, Leslie A. Thomas, Jacob D. McDonald, Kelly J. Dix and J. Michael SandersDrug Metabolism and Disposition March 2011, 39 (3) 498-509; DOI: https://doi.org/10.1124/dmd.110.034769
Morris, Marilyn E.
- You have accessThe Bioflavonoid Kaempferol Is an Abcg2 Substrate and Inhibits Abcg2-Mediated Quercetin EffluxGuohua An, Jorge Gallegos and Marilyn E. MorrisDrug Metabolism and Disposition March 2011, 39 (3) 426-432; DOI: https://doi.org/10.1124/dmd.110.035212
Motta, Paola
- You have accessCasopitant: In Vitro Data and SimCyp Simulation to Predict In Vivo Metabolic Interactions Involving Cytochrome P450 3A4Paola Motta, Nicoletta Pons, Sabrina Pagliarusco, Mario Pellegatti and Fiorenza BonomoDrug Metabolism and Disposition March 2011, 39 (3) 363-372; DOI: https://doi.org/10.1124/dmd.110.035071
N
Nemoto, Nobuo
- You have accessHepatocyte Nuclear Factor 4α Regulates Expression of the Mouse Female-Specific Cyp3a41 Gene in the LiverWattanaporn Bhadhprasit, Tsutomu Sakuma, Yuki Kawasaki and Nobuo NemotoDrug Metabolism and Disposition March 2011, 39 (3) 490-497; DOI: https://doi.org/10.1124/dmd.110.035980
Nguyen, Khanh
- You have accessUtility of Intersystem Extrapolation Factors in Early Reaction Phenotyping and the Quantitative Extrapolation of Human Liver Microsomal Intrinsic Clearance Using Recombinant Cytochromes P450Yuan Chen, Liling Liu, Khanh Nguyen and Adrian J. FretlandDrug Metabolism and Disposition March 2011, 39 (3) 373-382; DOI: https://doi.org/10.1124/dmd.110.035147
Ning, Baitang
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
O
Otagiri, Masaki
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
P
Pagliarusco, Sabrina
- You have accessCasopitant: In Vitro Data and SimCyp Simulation to Predict In Vivo Metabolic Interactions Involving Cytochrome P450 3A4Paola Motta, Nicoletta Pons, Sabrina Pagliarusco, Mario Pellegatti and Fiorenza BonomoDrug Metabolism and Disposition March 2011, 39 (3) 363-372; DOI: https://doi.org/10.1124/dmd.110.035071
Pan, Xian
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Pasanen, Markku
- You have accessSimple, Direct, and Informative Method for the Assessment of CYP2C19 Enzyme Inactivation KineticsKaisa A. Salminen, Jukka Leppänen, Jarkko I. Venäläinen, Markku Pasanen, Seppo Auriola, Risto O. Juvonen and Hannu RaunioDrug Metabolism and Disposition March 2011, 39 (3) 412-418; DOI: https://doi.org/10.1124/dmd.110.036376
Pellegatti, Mario
- You have accessCasopitant: In Vitro Data and SimCyp Simulation to Predict In Vivo Metabolic Interactions Involving Cytochrome P450 3A4Paola Motta, Nicoletta Pons, Sabrina Pagliarusco, Mario Pellegatti and Fiorenza BonomoDrug Metabolism and Disposition March 2011, 39 (3) 363-372; DOI: https://doi.org/10.1124/dmd.110.035071
Piquette-Miller, Micheline
- You have accessGestational and Pregnane X Receptor-Mediated Regulation of Placental ATP-Binding Cassette Drug Transporters in MiceSarabjit S. Gahir and Micheline Piquette-MillerDrug Metabolism and Disposition March 2011, 39 (3) 465-471; DOI: https://doi.org/10.1124/dmd.110.034983
Pons, Nicoletta
- You have accessCasopitant: In Vitro Data and SimCyp Simulation to Predict In Vivo Metabolic Interactions Involving Cytochrome P450 3A4Paola Motta, Nicoletta Pons, Sabrina Pagliarusco, Mario Pellegatti and Fiorenza BonomoDrug Metabolism and Disposition March 2011, 39 (3) 363-372; DOI: https://doi.org/10.1124/dmd.110.035071
R
Raunio, Hannu
- You have accessSimple, Direct, and Informative Method for the Assessment of CYP2C19 Enzyme Inactivation KineticsKaisa A. Salminen, Jukka Leppänen, Jarkko I. Venäläinen, Markku Pasanen, Seppo Auriola, Risto O. Juvonen and Hannu RaunioDrug Metabolism and Disposition March 2011, 39 (3) 412-418; DOI: https://doi.org/10.1124/dmd.110.036376
Rehngren, Mikael
- You have accessMeasurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate MethodsMarkus Fridén, Fredrik Bergström, Hong Wan, Mikael Rehngren, Gustav Ahlin, Margareta Hammarlund-Udenaes and Ulf BredbergDrug Metabolism and Disposition March 2011, 39 (3) 353-362; DOI: https://doi.org/10.1124/dmd.110.035998
Romero, David
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
Rousu, Timo
- You have accessEffects of Cell Differentiation and Assay Conditions on the UDP-Glucuronosyltransferase Activity in Caco-2 CellsHongbo Zhang, Ari Tolonen, Timo Rousu, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition March 2011, 39 (3) 456-464; DOI: https://doi.org/10.1124/dmd.110.036582
Ryder, Tim F.
- You have accessValidation of Isolated Metabolites from Drug Metabolism Studies as Analytical Standards by Quantitative NMRGregory S. Walker, Tim F. Ryder, Raman Sharma, Evan B. Smith and Amy FreundDrug Metabolism and Disposition March 2011, 39 (3) 433-440; DOI: https://doi.org/10.1124/dmd.110.036343
S
Sakai, Hiromi
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
Sakuma, Tsutomu
- You have accessHepatocyte Nuclear Factor 4α Regulates Expression of the Mouse Female-Specific Cyp3a41 Gene in the LiverWattanaporn Bhadhprasit, Tsutomu Sakuma, Yuki Kawasaki and Nobuo NemotoDrug Metabolism and Disposition March 2011, 39 (3) 490-497; DOI: https://doi.org/10.1124/dmd.110.035980
Salminen, Kaisa A.
- You have accessSimple, Direct, and Informative Method for the Assessment of CYP2C19 Enzyme Inactivation KineticsKaisa A. Salminen, Jukka Leppänen, Jarkko I. Venäläinen, Markku Pasanen, Seppo Auriola, Risto O. Juvonen and Hannu RaunioDrug Metabolism and Disposition March 2011, 39 (3) 412-418; DOI: https://doi.org/10.1124/dmd.110.036376
Sanders, J. Michael
- You have accessDisposition and Metabolism of Cumene in F344 Rats and B6C3F1 MiceLing-Jen Chen, Christopher J. Wegerski, Daniel J. Kramer, Leslie A. Thomas, Jacob D. McDonald, Kelly J. Dix and J. Michael SandersDrug Metabolism and Disposition March 2011, 39 (3) 498-509; DOI: https://doi.org/10.1124/dmd.110.034769
Shah, Manish B.
- You have accessComparison of In Vitro Metabolism of Ticlopidine by Human Cytochrome P450 2B6 and Rabbit Cytochrome P450 2B4Jyothi C. Talakad, Manish B. Shah, Gregory S. Walker, Cathie Xiang, James R. Halpert and Deepak DalvieDrug Metabolism and Disposition March 2011, 39 (3) 539-550; DOI: https://doi.org/10.1124/dmd.110.037101
Sharma, Raman
- You have accessValidation of Isolated Metabolites from Drug Metabolism Studies as Analytical Standards by Quantitative NMRGregory S. Walker, Tim F. Ryder, Raman Sharma, Evan B. Smith and Amy FreundDrug Metabolism and Disposition March 2011, 39 (3) 433-440; DOI: https://doi.org/10.1124/dmd.110.036343
Shi, Leming
- You have accessSimilarities and Differences in the Expression of Drug-Metabolizing Enzymes between Human Hepatic Cell Lines and Primary Human HepatocytesLei Guo, Stacey Dial, Leming Shi, William Branham, Jie Liu, Jia-Long Fang, Bridgett Green, Helen Deng, Jim Kaput and Baitang NingDrug Metabolism and Disposition March 2011, 39 (3) 528-538; DOI: https://doi.org/10.1124/dmd.110.035873
Skaptason, Judith
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
Smith, Evan B.
- You have accessValidation of Isolated Metabolites from Drug Metabolism Studies as Analytical Standards by Quantitative NMRGregory S. Walker, Tim F. Ryder, Raman Sharma, Evan B. Smith and Amy FreundDrug Metabolism and Disposition March 2011, 39 (3) 433-440; DOI: https://doi.org/10.1124/dmd.110.036343
Su, Ai-Duen
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
Sugiyama, Yuichi
- You have accessDecreased Hepatic Breast Cancer Resistance Protein Expression and Function in Multidrug Resistance-Associated Protein 2-Deficient (TR−) RatsWei Yue, Jin Kyung Lee, Koji Abe, Yuichi Sugiyama and Kim L. R. BrouwerDrug Metabolism and Disposition March 2011, 39 (3) 441-447; DOI: https://doi.org/10.1124/dmd.110.035188
T
Taguchi, Kazuaki
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
Talakad, Jyothi C.
- You have accessComparison of In Vitro Metabolism of Ticlopidine by Human Cytochrome P450 2B6 and Rabbit Cytochrome P450 2B4Jyothi C. Talakad, Manish B. Shah, Gregory S. Walker, Cathie Xiang, James R. Halpert and Deepak DalvieDrug Metabolism and Disposition March 2011, 39 (3) 539-550; DOI: https://doi.org/10.1124/dmd.110.037101
Tan, Weiwei
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
Teft, Wendy A.
- You have accessEndoxifen, the Active Metabolite of Tamoxifen, Is a Substrate of the Efflux Transporter P-Glycoprotein (Multidrug Resistance 1)Wendy A. Teft, Sara E. Mansell and Richard B. KimDrug Metabolism and Disposition March 2011, 39 (3) 558-562; DOI: https://doi.org/10.1124/dmd.110.036160
Thomas, Leslie A.
- You have accessDisposition and Metabolism of Cumene in F344 Rats and B6C3F1 MiceLing-Jen Chen, Christopher J. Wegerski, Daniel J. Kramer, Leslie A. Thomas, Jacob D. McDonald, Kelly J. Dix and J. Michael SandersDrug Metabolism and Disposition March 2011, 39 (3) 498-509; DOI: https://doi.org/10.1124/dmd.110.034769
Tolonen, Ari
- You have accessEffects of Cell Differentiation and Assay Conditions on the UDP-Glucuronosyltransferase Activity in Caco-2 CellsHongbo Zhang, Ari Tolonen, Timo Rousu, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition March 2011, 39 (3) 456-464; DOI: https://doi.org/10.1124/dmd.110.036582
Tong, Wei
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
V
Vekich, Sylvia
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
Venäläinen, Jarkko I.
- You have accessSimple, Direct, and Informative Method for the Assessment of CYP2C19 Enzyme Inactivation KineticsKaisa A. Salminen, Jukka Leppänen, Jarkko I. Venäläinen, Markku Pasanen, Seppo Auriola, Risto O. Juvonen and Hannu RaunioDrug Metabolism and Disposition March 2011, 39 (3) 412-418; DOI: https://doi.org/10.1124/dmd.110.036376
W
Walker, Gregory S.
- You have accessValidation of Isolated Metabolites from Drug Metabolism Studies as Analytical Standards by Quantitative NMRGregory S. Walker, Tim F. Ryder, Raman Sharma, Evan B. Smith and Amy FreundDrug Metabolism and Disposition March 2011, 39 (3) 433-440; DOI: https://doi.org/10.1124/dmd.110.036343
- You have accessComparison of In Vitro Metabolism of Ticlopidine by Human Cytochrome P450 2B6 and Rabbit Cytochrome P450 2B4Jyothi C. Talakad, Manish B. Shah, Gregory S. Walker, Cathie Xiang, James R. Halpert and Deepak DalvieDrug Metabolism and Disposition March 2011, 39 (3) 539-550; DOI: https://doi.org/10.1124/dmd.110.037101
Wan, Hong
- You have accessMeasurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate MethodsMarkus Fridén, Fredrik Bergström, Hong Wan, Mikael Rehngren, Gustav Ahlin, Margareta Hammarlund-Udenaes and Ulf BredbergDrug Metabolism and Disposition March 2011, 39 (3) 353-362; DOI: https://doi.org/10.1124/dmd.110.035998
Wang, Guangji
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Wang, Laiyou
- You have accessCYP3A-Mediated Generation of Aldehyde and Hydrazine in Atazanavir MetabolismFeng Li, Jie Lu, Laiyou Wang and Xiaochao MaDrug Metabolism and Disposition March 2011, 39 (3) 394-401; DOI: https://doi.org/10.1124/dmd.110.036327
Wang, Xinting
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Watanabe, Hiroshi
- You have accessRepeated Injection of High Doses of Hemoglobin-Encapsulated Liposomes (Hemoglobin Vesicles) Induces Accelerated Blood Clearance in a Hemorrhagic Shock Rat ModelKazuaki Taguchi, Yasunori Iwao, Hiroshi Watanabe, Daisuke Kadowaki, Hiromi Sakai, Koichi Kobayashi, Hirohisa Horinouchi, Toru Maruyama and Masaki OtagiriDrug Metabolism and Disposition March 2011, 39 (3) 484-489; DOI: https://doi.org/10.1124/dmd.110.036913
Wegerski, Christopher J.
- You have accessDisposition and Metabolism of Cumene in F344 Rats and B6C3F1 MiceLing-Jen Chen, Christopher J. Wegerski, Daniel J. Kramer, Leslie A. Thomas, Jacob D. McDonald, Kelly J. Dix and J. Michael SandersDrug Metabolism and Disposition March 2011, 39 (3) 498-509; DOI: https://doi.org/10.1124/dmd.110.034769
Wempe, Michael F.
- You have accessAtazanavir Metabolism According to CYP3A5 Status: An In Vitro-In Vivo AssessmentMichael F. Wempe and Peter L. AndersonDrug Metabolism and Disposition March 2011, 39 (3) 522-527; DOI: https://doi.org/10.1124/dmd.110.036178
Wilner, Keith D.
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
X
Xiang, Cathie
- You have accessComparison of In Vitro Metabolism of Ticlopidine by Human Cytochrome P450 2B6 and Rabbit Cytochrome P450 2B4Jyothi C. Talakad, Manish B. Shah, Gregory S. Walker, Cathie Xiang, James R. Halpert and Deepak DalvieDrug Metabolism and Disposition March 2011, 39 (3) 539-550; DOI: https://doi.org/10.1124/dmd.110.037101
Xie, Lin
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Xie, Shanshan
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Y
Yamazaki, Shinji
- You have accessPrediction of Oral Pharmacokinetics of cMet Kinase Inhibitors in Humans: Physiologically Based Pharmacokinetic Model Versus Traditional One-Compartment ModelShinji Yamazaki, Judith Skaptason, David Romero, Sylvia Vekich, Hannah M. Jones, Weiwei Tan, Keith D. Wilner and Tatiana KoudriakovaDrug Metabolism and Disposition March 2011, 39 (3) 383-393; DOI: https://doi.org/10.1124/dmd.110.035857
Yuan, Yuan
- You have accessCharacterization of Human Liver Enzymes Involved in the Biotransformation of Boceprevir, a Hepatitis C Virus Protease InhibitorAnima Ghosal, Yuan Yuan, Wei Tong, Ai-Duen Su, Chunyan Gu, Swapan K. Chowdhury, Narendra S. Kishnani and Kevin B. AltonDrug Metabolism and Disposition March 2011, 39 (3) 510-521; DOI: https://doi.org/10.1124/dmd.110.036996
Yue, Wei
- You have accessDecreased Hepatic Breast Cancer Resistance Protein Expression and Function in Multidrug Resistance-Associated Protein 2-Deficient (TR−) RatsWei Yue, Jin Kyung Lee, Koji Abe, Yuichi Sugiyama and Kim L. R. BrouwerDrug Metabolism and Disposition March 2011, 39 (3) 441-447; DOI: https://doi.org/10.1124/dmd.110.035188
Z
Zhang, Hongbo
- You have accessEffects of Cell Differentiation and Assay Conditions on the UDP-Glucuronosyltransferase Activity in Caco-2 CellsHongbo Zhang, Ari Tolonen, Timo Rousu, Jouni Hirvonen and Moshe FinelDrug Metabolism and Disposition March 2011, 39 (3) 456-464; DOI: https://doi.org/10.1124/dmd.110.036582
Zhang, Lulu
- You have accessOpposite Effect of Diabetes Mellitus Induced by Streptozotocin on Oral and Intravenous Pharmacokinetics of Verapamil in RatsNan Hu, Shanshan Xie, Li Liu, Xinting Wang, Xian Pan, Guanming Chen, Lulu Zhang, Haiyan Liu, Xiang Liu, Xiaodong Liu, Lin Xie and Guangji WangDrug Metabolism and Disposition March 2011, 39 (3) 419-425; DOI: https://doi.org/10.1124/dmd.110.035642
Zhong, Dafang
- You have accessIdentification of 20(S)-Protopanaxadiol Metabolites in Human Liver Microsomes and Human HepatocytesLiang Li, Xiaoyan Chen, Dan Li and Dafang ZhongDrug Metabolism and Disposition March 2011, 39 (3) 472-483; DOI: https://doi.org/10.1124/dmd.110.036723
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