Index by author
June 01, 2011; Volume 39,Issue 6
A
Arthur, Evan J.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
B
Balani, Suresh K.
- You have accessA Refined Cytochrome P450 IC50 Shift Assay for Reliably Identifying CYP3A Time-Dependent InhibitorsPing Li, Chuang Lu, Suresh K. Balani and Liang-Shang GanDrug Metabolism and Disposition June 2011, 39 (6) 1054-1057; DOI: https://doi.org/10.1124/dmd.111.038208
Banerjee, Subhashis
- You have accessSuppression of Cytochrome P450 Reductase (POR) Expression in Hepatoma Cells Replicates the Hepatic Lipidosis Observed in Hepatic POR-Null MiceTodd D. Porter, Subhashis Banerjee, Elzbieta I. Stolarczyk and Ling ZouDrug Metabolism and Disposition June 2011, 39 (6) 966-973; DOI: https://doi.org/10.1124/dmd.111.038562
Behr, Melissa
- You have accessThe Tissue-Specific Toxicity of Methimazole in the Mouse Olfactory Mucosa Is Partly Mediated through Target-Tissue Metabolic Activation by CYP2A5Fang Xie, Xin Zhou, Mary Beth Genter, Melissa Behr, Jun Gu and Xinxin DingDrug Metabolism and Disposition June 2011, 39 (6) 947-951; DOI: https://doi.org/10.1124/dmd.110.037895
Black, W. Cameron
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Brot, Nathan
- You have accessStudies on the Metabolism and Biological Activity of the Epimers of SulindacDavid Brunell, Daphna Sagher, Shailaja Kesaraju, Nathan Brot and Herbert WeissbachDrug Metabolism and Disposition June 2011, 39 (6) 1014-1021; DOI: https://doi.org/10.1124/dmd.110.037663
Brunell, David
- You have accessStudies on the Metabolism and Biological Activity of the Epimers of SulindacDavid Brunell, Daphna Sagher, Shailaja Kesaraju, Nathan Brot and Herbert WeissbachDrug Metabolism and Disposition June 2011, 39 (6) 1014-1021; DOI: https://doi.org/10.1124/dmd.110.037663
Buhimschi, Catalin S.
- You have accessATP-Binding Cassette Transporter Expression in Human Placenta as a Function of Pregnancy ConditionCifford W. Mason, Irina A. Buhimschi, Catalin S. Buhimschi, Yafeng Dong, Carl P. Weiner and Peter W. SwaanDrug Metabolism and Disposition June 2011, 39 (6) 1000-1007; DOI: https://doi.org/10.1124/dmd.111.038166
Buhimschi, Irina A.
- You have accessATP-Binding Cassette Transporter Expression in Human Placenta as a Function of Pregnancy ConditionCifford W. Mason, Irina A. Buhimschi, Catalin S. Buhimschi, Yafeng Dong, Carl P. Weiner and Peter W. SwaanDrug Metabolism and Disposition June 2011, 39 (6) 1000-1007; DOI: https://doi.org/10.1124/dmd.111.038166
Butler, Brendan F.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
C
Chan, Eric Chun Yong
- You have accessMetabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by LapatinibHideo Takakusa, Michelle D. Wahlin, Chunsheng Zhao, Kelsey L. Hanson, Lee Sun New, Eric Chun Yong Chan and Sidney D. NelsonDrug Metabolism and Disposition June 2011, 39 (6) 1022-1030; DOI: https://doi.org/10.1124/dmd.110.037531
Chauret, Nathalie
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Chen, Xiaoyan
- You have accessIdentification of Amiodarone Metabolites in Human Bile by Ultraperformance Liquid Chromatography/Quadrupole Time-of-Flight Mass SpectrometryPan Deng, Tiangeng You, Xiaoyan Chen, Tao Yuan, Haihua Huang and Dafang ZhongDrug Metabolism and Disposition June 2011, 39 (6) 1058-1069; DOI: https://doi.org/10.1124/dmd.110.037671
Chen, Yung-Hsiang
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Collier, Ann C.
- You have accessComplex Drug Interactions of HIV Protease Inhibitors 1: Inactivation, Induction, and Inhibition of Cytochrome P450 3A by Ritonavir or NelfinavirBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition June 2011, 39 (6) 1070-1078; DOI: https://doi.org/10.1124/dmd.110.037523
Czendlik, C.
- You have accessPharmacokinetics of the Monohydroxy Derivative of Oxcarbazepine and Its Enantiomers after a Single Intravenous Dose Given as Racemate Compared with a Single Oral Dose of OxcarbazepineG. Flesch, C. Czendlik, D. Renard and P. LloydDrug Metabolism and Disposition June 2011, 39 (6) 1103-1110; DOI: https://doi.org/10.1124/dmd.109.030593
D
D'Agostino, Jaime
- You have accessRole of Intestinal Cytochrome P450 (P450) in Modulating the Bioavailability of Oral Lovastatin: Insights from Studies on the Intestinal Epithelium-Specific P450 Reductase Knockout MouseYi Zhu, Jaime D'Agostino and Qing-Yu ZhangDrug Metabolism and Disposition June 2011, 39 (6) 939-943; DOI: https://doi.org/10.1124/dmd.110.037861
Day, Stephen
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Debori, Yasuyuki
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Deese, Alan
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Deng, Pan
- You have accessIdentification of Amiodarone Metabolites in Human Bile by Ultraperformance Liquid Chromatography/Quadrupole Time-of-Flight Mass SpectrometryPan Deng, Tiangeng You, Xiaoyan Chen, Tao Yuan, Haihua Huang and Dafang ZhongDrug Metabolism and Disposition June 2011, 39 (6) 1058-1069; DOI: https://doi.org/10.1124/dmd.110.037671
Denton, Rebecca
- You have accessPrediction of Human Renal Clearance from Preclinical Species for a Diverse Set of Drugs That Exhibit Both Active Secretion and Net ReabsorptionStuart W. Paine, Karelle Ménochet, Rebecca Denton, Dermot F. McGinnity and Robert J. RileyDrug Metabolism and Disposition June 2011, 39 (6) 1008-1013; DOI: https://doi.org/10.1124/dmd.110.037267
Diffenderfer, Laura E.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
Ding, Xinxin
- You have accessThe Tissue-Specific Toxicity of Methimazole in the Mouse Olfactory Mucosa Is Partly Mediated through Target-Tissue Metabolic Activation by CYP2A5Fang Xie, Xin Zhou, Mary Beth Genter, Melissa Behr, Jun Gu and Xinxin DingDrug Metabolism and Disposition June 2011, 39 (6) 947-951; DOI: https://doi.org/10.1124/dmd.110.037895
Dong, Yafeng
- You have accessATP-Binding Cassette Transporter Expression in Human Placenta as a Function of Pregnancy ConditionCifford W. Mason, Irina A. Buhimschi, Catalin S. Buhimschi, Yafeng Dong, Carl P. Weiner and Peter W. SwaanDrug Metabolism and Disposition June 2011, 39 (6) 1000-1007; DOI: https://doi.org/10.1124/dmd.111.038166
F
Faller, Bernard
- You have accessCYP3A Time-Dependent Inhibition Risk Assessment Validated with 400 Reference DrugsAlfred Zimmerlin, Markus Trunzer and Bernard FallerDrug Metabolism and Disposition June 2011, 39 (6) 1039-1046; DOI: https://doi.org/10.1124/dmd.110.037911
Flesch, G.
- You have accessPharmacokinetics of the Monohydroxy Derivative of Oxcarbazepine and Its Enantiomers after a Single Intravenous Dose Given as Racemate Compared with a Single Oral Dose of OxcarbazepineG. Flesch, C. Czendlik, D. Renard and P. LloydDrug Metabolism and Disposition June 2011, 39 (6) 1103-1110; DOI: https://doi.org/10.1124/dmd.109.030593
Fletke, Kyle J.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
Fromm, Martin F.
- You have accessInfluence of Non-Steroidal Anti-Inflammatory Drugs on Organic Anion Transporting Polypeptide (OATP) 1B1- and OATP1B3-Mediated Drug TransportJuergen Kindla, Fabian Müller, Maren Mieth, Martin F. Fromm and Jörg KönigDrug Metabolism and Disposition June 2011, 39 (6) 1047-1053; DOI: https://doi.org/10.1124/dmd.110.037622
- You have accessRole of Organic Anion-Transporting Polypeptides for Cellular Mesalazine (5-Aminosalicylic Acid) UptakeJörg König, Hartmut Glaeser, Markus Keiser, Kathrin Mandery, Ulrich Klotz and Martin F. FrommDrug Metabolism and Disposition June 2011, 39 (6) 1097-1102; DOI: https://doi.org/10.1124/dmd.110.034991
Fukuda, Hajime
- You have accessQuantitative Time-Lapse Imaging-Based Analysis of Drug-Drug Interaction Mediated by Hepatobiliary Transporter, Multidrug Resistance-Associated Protein 2, in Sandwich-Cultured Rat HepatocytesTakeo Nakanishi, Yuta Shibue, Yoko Fukuyama, Kenji Yoshida, Hajime Fukuda, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition June 2011, 39 (6) 984-991; DOI: https://doi.org/10.1124/dmd.111.038059
Fukuyama, Yoko
- You have accessQuantitative Time-Lapse Imaging-Based Analysis of Drug-Drug Interaction Mediated by Hepatobiliary Transporter, Multidrug Resistance-Associated Protein 2, in Sandwich-Cultured Rat HepatocytesTakeo Nakanishi, Yuta Shibue, Yoko Fukuyama, Kenji Yoshida, Hajime Fukuda, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition June 2011, 39 (6) 984-991; DOI: https://doi.org/10.1124/dmd.111.038059
Furge, Laura Lowe
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
G
Gan, Liang-Shang
- You have accessA Refined Cytochrome P450 IC50 Shift Assay for Reliably Identifying CYP3A Time-Dependent InhibitorsPing Li, Chuang Lu, Suresh K. Balani and Liang-Shang GanDrug Metabolism and Disposition June 2011, 39 (6) 1054-1057; DOI: https://doi.org/10.1124/dmd.111.038208
Genter, Mary Beth
- You have accessThe Tissue-Specific Toxicity of Methimazole in the Mouse Olfactory Mucosa Is Partly Mediated through Target-Tissue Metabolic Activation by CYP2A5Fang Xie, Xin Zhou, Mary Beth Genter, Melissa Behr, Jun Gu and Xinxin DingDrug Metabolism and Disposition June 2011, 39 (6) 947-951; DOI: https://doi.org/10.1124/dmd.110.037895
Glaeser, Hartmut
- You have accessRole of Organic Anion-Transporting Polypeptides for Cellular Mesalazine (5-Aminosalicylic Acid) UptakeJörg König, Hartmut Glaeser, Markus Keiser, Kathrin Mandery, Ulrich Klotz and Martin F. FrommDrug Metabolism and Disposition June 2011, 39 (6) 1097-1102; DOI: https://doi.org/10.1124/dmd.110.034991
Gu, Jun
- You have accessThe Tissue-Specific Toxicity of Methimazole in the Mouse Olfactory Mucosa Is Partly Mediated through Target-Tissue Metabolic Activation by CYP2A5Fang Xie, Xin Zhou, Mary Beth Genter, Melissa Behr, Jun Gu and Xinxin DingDrug Metabolism and Disposition June 2011, 39 (6) 947-951; DOI: https://doi.org/10.1124/dmd.110.037895
Guengerich, F. Peter
- You have accessCytochrome P450 2S1 is Reduced by NADPH-Cytochrome P450 ReductaseYi Xiao, Raku Shinkyo and F. Peter GuengerichDrug Metabolism and Disposition June 2011, 39 (6) 944-946; DOI: https://doi.org/10.1124/dmd.111.039321
H
Hanson, Kelsey L.
- You have accessMetabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by LapatinibHideo Takakusa, Michelle D. Wahlin, Chunsheng Zhao, Kelsey L. Hanson, Lee Sun New, Eric Chun Yong Chan and Sidney D. NelsonDrug Metabolism and Disposition June 2011, 39 (6) 1022-1030; DOI: https://doi.org/10.1124/dmd.110.037531
Hop, Cornelis E. C. A.
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Horikawa, Masato
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
Horita, Shigeru
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Hsi, David J.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
Hu, Zhuohan
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Huang, Haihua
- You have accessIdentification of Amiodarone Metabolites in Human Bile by Ultraperformance Liquid Chromatography/Quadrupole Time-of-Flight Mass SpectrometryPan Deng, Tiangeng You, Xiaoyan Chen, Tao Yuan, Haihua Huang and Dafang ZhongDrug Metabolism and Disposition June 2011, 39 (6) 1058-1069; DOI: https://doi.org/10.1124/dmd.110.037671
I
Ishiwata, Norihisa
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
K
Kassahun, Kelem
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Kato, Yukio
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
Keiser, Markus
- You have accessRole of Organic Anion-Transporting Polypeptides for Cellular Mesalazine (5-Aminosalicylic Acid) UptakeJörg König, Hartmut Glaeser, Markus Keiser, Kathrin Mandery, Ulrich Klotz and Martin F. FrommDrug Metabolism and Disposition June 2011, 39 (6) 1097-1102; DOI: https://doi.org/10.1124/dmd.110.034991
Kesaraju, Shailaja
- You have accessStudies on the Metabolism and Biological Activity of the Epimers of SulindacDavid Brunell, Daphna Sagher, Shailaja Kesaraju, Nathan Brot and Herbert WeissbachDrug Metabolism and Disposition June 2011, 39 (6) 1014-1021; DOI: https://doi.org/10.1124/dmd.110.037663
Kharasch, Evan D.
- You have accessComplex Drug Interactions of HIV Protease Inhibitors 1: Inactivation, Induction, and Inhibition of Cytochrome P450 3A by Ritonavir or NelfinavirBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition June 2011, 39 (6) 1070-1078; DOI: https://doi.org/10.1124/dmd.110.037523
Khojasteh, S. Cyrus
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Kindla, Juergen
- You have accessInfluence of Non-Steroidal Anti-Inflammatory Drugs on Organic Anion Transporting Polypeptide (OATP) 1B1- and OATP1B3-Mediated Drug TransportJuergen Kindla, Fabian Müller, Maren Mieth, Martin F. Fromm and Jörg KönigDrug Metabolism and Disposition June 2011, 39 (6) 1047-1053; DOI: https://doi.org/10.1124/dmd.110.037622
Kirby, Brian J.
- You have accessComplex Drug Interactions of HIV Protease Inhibitors 1: Inactivation, Induction, and Inhibition of Cytochrome P450 3A by Ritonavir or NelfinavirBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition June 2011, 39 (6) 1070-1078; DOI: https://doi.org/10.1124/dmd.110.037523
Klotz, Ulrich
- You have accessRole of Organic Anion-Transporting Polypeptides for Cellular Mesalazine (5-Aminosalicylic Acid) UptakeJörg König, Hartmut Glaeser, Markus Keiser, Kathrin Mandery, Ulrich Klotz and Martin F. FrommDrug Metabolism and Disposition June 2011, 39 (6) 1097-1102; DOI: https://doi.org/10.1124/dmd.110.034991
Koeplinger, Kenneth
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Kondo, Tsunenori
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
König, Jörg
- You have accessInfluence of Non-Steroidal Anti-Inflammatory Drugs on Organic Anion Transporting Polypeptide (OATP) 1B1- and OATP1B3-Mediated Drug TransportJuergen Kindla, Fabian Müller, Maren Mieth, Martin F. Fromm and Jörg KönigDrug Metabolism and Disposition June 2011, 39 (6) 1047-1053; DOI: https://doi.org/10.1124/dmd.110.037622
- You have accessRole of Organic Anion-Transporting Polypeptides for Cellular Mesalazine (5-Aminosalicylic Acid) UptakeJörg König, Hartmut Glaeser, Markus Keiser, Kathrin Mandery, Ulrich Klotz and Martin F. FrommDrug Metabolism and Disposition June 2011, 39 (6) 1097-1102; DOI: https://doi.org/10.1124/dmd.110.034991
Kusuhara, Hiroyuki
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
L
Li, Ping
- You have accessA Refined Cytochrome P450 IC50 Shift Assay for Reliably Identifying CYP3A Time-Dependent InhibitorsPing Li, Chuang Lu, Suresh K. Balani and Liang-Shang GanDrug Metabolism and Disposition June 2011, 39 (6) 1054-1057; DOI: https://doi.org/10.1124/dmd.111.038208
Lloyd, P.
- You have accessPharmacokinetics of the Monohydroxy Derivative of Oxcarbazepine and Its Enantiomers after a Single Intravenous Dose Given as Racemate Compared with a Single Oral Dose of OxcarbazepineG. Flesch, C. Czendlik, D. Renard and P. LloydDrug Metabolism and Disposition June 2011, 39 (6) 1103-1110; DOI: https://doi.org/10.1124/dmd.109.030593
Lu, Chuang
- You have accessA Refined Cytochrome P450 IC50 Shift Assay for Reliably Identifying CYP3A Time-Dependent InhibitorsPing Li, Chuang Lu, Suresh K. Balani and Liang-Shang GanDrug Metabolism and Disposition June 2011, 39 (6) 1054-1057; DOI: https://doi.org/10.1124/dmd.111.038208
M
Maeda, Kazuya
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Mandery, Kathrin
- You have accessRole of Organic Anion-Transporting Polypeptides for Cellular Mesalazine (5-Aminosalicylic Acid) UptakeJörg König, Hartmut Glaeser, Markus Keiser, Kathrin Mandery, Ulrich Klotz and Martin F. FrommDrug Metabolism and Disposition June 2011, 39 (6) 1097-1102; DOI: https://doi.org/10.1124/dmd.110.034991
Mason, Cifford W.
- You have accessATP-Binding Cassette Transporter Expression in Human Placenta as a Function of Pregnancy ConditionCifford W. Mason, Irina A. Buhimschi, Catalin S. Buhimschi, Yafeng Dong, Carl P. Weiner and Peter W. SwaanDrug Metabolism and Disposition June 2011, 39 (6) 1000-1007; DOI: https://doi.org/10.1124/dmd.111.038166
Matsubara, Kazuki
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
McGinnity, Dermot F.
- You have accessPrediction of Human Renal Clearance from Preclinical Species for a Diverse Set of Drugs That Exhibit Both Active Secretion and Net ReabsorptionStuart W. Paine, Karelle Ménochet, Rebecca Denton, Dermot F. McGinnity and Robert J. RileyDrug Metabolism and Disposition June 2011, 39 (6) 1008-1013; DOI: https://doi.org/10.1124/dmd.110.037267
McIntosh, Ian
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Ménochet, Karelle
- You have accessPrediction of Human Renal Clearance from Preclinical Species for a Diverse Set of Drugs That Exhibit Both Active Secretion and Net ReabsorptionStuart W. Paine, Karelle Ménochet, Rebecca Denton, Dermot F. McGinnity and Robert J. RileyDrug Metabolism and Disposition June 2011, 39 (6) 1008-1013; DOI: https://doi.org/10.1124/dmd.110.037267
Mieth, Maren
- You have accessInfluence of Non-Steroidal Anti-Inflammatory Drugs on Organic Anion Transporting Polypeptide (OATP) 1B1- and OATP1B3-Mediated Drug TransportJuergen Kindla, Fabian Müller, Maren Mieth, Martin F. Fromm and Jörg KönigDrug Metabolism and Disposition June 2011, 39 (6) 1047-1053; DOI: https://doi.org/10.1124/dmd.110.037622
Mocny, Catherine S.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
More, Vijay R.
- You have accessAlteration of Hepatic but Not Renal Transporter Expression in Diet-Induced Obese MiceVijay R. More and Angela L. SlittDrug Metabolism and Disposition June 2011, 39 (6) 992-999; DOI: https://doi.org/10.1124/dmd.110.037507
Mulder, Teresa
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Müller, Fabian
- You have accessInfluence of Non-Steroidal Anti-Inflammatory Drugs on Organic Anion Transporting Polypeptide (OATP) 1B1- and OATP1B3-Mediated Drug TransportJuergen Kindla, Fabian Müller, Maren Mieth, Martin F. Fromm and Jörg KönigDrug Metabolism and Disposition June 2011, 39 (6) 1047-1053; DOI: https://doi.org/10.1124/dmd.110.037622
N
Nagy, Leslie D.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
Nakamichi, Noritaka
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
Nakanishi, Takeo
- You have accessQuantitative Time-Lapse Imaging-Based Analysis of Drug-Drug Interaction Mediated by Hepatobiliary Transporter, Multidrug Resistance-Associated Protein 2, in Sandwich-Cultured Rat HepatocytesTakeo Nakanishi, Yuta Shibue, Yoko Fukuyama, Kenji Yoshida, Hajime Fukuda, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition June 2011, 39 (6) 984-991; DOI: https://doi.org/10.1124/dmd.111.038059
Nakayama, Hideki
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Nelson, Sidney D.
- You have accessMetabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by LapatinibHideo Takakusa, Michelle D. Wahlin, Chunsheng Zhao, Kelsey L. Hanson, Lee Sun New, Eric Chun Yong Chan and Sidney D. NelsonDrug Metabolism and Disposition June 2011, 39 (6) 1022-1030; DOI: https://doi.org/10.1124/dmd.110.037531
New, Lee Sun
- You have accessMetabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by LapatinibHideo Takakusa, Michelle D. Wahlin, Chunsheng Zhao, Kelsey L. Hanson, Lee Sun New, Eric Chun Yong Chan and Sidney D. NelsonDrug Metabolism and Disposition June 2011, 39 (6) 1022-1030; DOI: https://doi.org/10.1124/dmd.110.037531
Nicoll-Griffith, Deborah
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Nomeir, Amin A.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
O
Ogilvie, Brian W.
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
P
Paine, Stuart W.
- You have accessPrediction of Human Renal Clearance from Preclinical Species for a Diverse Set of Drugs That Exhibit Both Active Secretion and Net ReabsorptionStuart W. Paine, Karelle Ménochet, Rebecca Denton, Dermot F. McGinnity and Robert J. RileyDrug Metabolism and Disposition June 2011, 39 (6) 1008-1013; DOI: https://doi.org/10.1124/dmd.110.037267
Palamanda, Jairam R.
- You have accessSubstituted Imidazole of 5-Fluoro-2-[4-[(2-phenyl-1H-imidazol-5-yl)methyl]-1-piperazinyl]pyrimidine Inactivates Cytochrome P450 2D6 by Protein AdductionLeslie D. Nagy, Catherine S. Mocny, Laura E. Diffenderfer, David J. Hsi, Brendan F. Butler, Evan J. Arthur, Kyle J. Fletke, Jairam R. Palamanda, Amin A. Nomeir and Laura Lowe FurgeDrug Metabolism and Disposition June 2011, 39 (6) 974-983; DOI: https://doi.org/10.1124/dmd.110.037630
Parkinson, Andrew
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Porter, Todd D.
- You have accessSuppression of Cytochrome P450 Reductase (POR) Expression in Hepatoma Cells Replicates the Hepatic Lipidosis Observed in Hepatic POR-Null MiceTodd D. Porter, Subhashis Banerjee, Elzbieta I. Stolarczyk and Ling ZouDrug Metabolism and Disposition June 2011, 39 (6) 966-973; DOI: https://doi.org/10.1124/dmd.111.038562
R
Renard, D.
- You have accessPharmacokinetics of the Monohydroxy Derivative of Oxcarbazepine and Its Enantiomers after a Single Intravenous Dose Given as Racemate Compared with a Single Oral Dose of OxcarbazepineG. Flesch, C. Czendlik, D. Renard and P. LloydDrug Metabolism and Disposition June 2011, 39 (6) 1103-1110; DOI: https://doi.org/10.1124/dmd.109.030593
Reynolds, Mark
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Riley, Robert J.
- You have accessPrediction of Human Renal Clearance from Preclinical Species for a Diverse Set of Drugs That Exhibit Both Active Secretion and Net ReabsorptionStuart W. Paine, Karelle Ménochet, Rebecca Denton, Dermot F. McGinnity and Robert J. RileyDrug Metabolism and Disposition June 2011, 39 (6) 1008-1013; DOI: https://doi.org/10.1124/dmd.110.037267
Rosenberg, Elizabeth
- You have accessPharmacokinetics and Metabolism in Rats, Dogs, and Monkeys of the Cathepsin K Inhibitor Odanacatib: Demethylation of a Methylsulfonyl Moiety as a Major Metabolic PathwayKelem Kassahun, W. Cameron Black, Deborah Nicoll-Griffith, Ian McIntosh, Nathalie Chauret, Stephen Day, Elizabeth Rosenberg and Kenneth KoeplingerDrug Metabolism and Disposition June 2011, 39 (6) 1079-1087; DOI: https://doi.org/10.1124/dmd.110.037184
Rudewicz, Patrick J.
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
S
Sagher, Daphna
- You have accessStudies on the Metabolism and Biological Activity of the Epimers of SulindacDavid Brunell, Daphna Sagher, Shailaja Kesaraju, Nathan Brot and Herbert WeissbachDrug Metabolism and Disposition June 2011, 39 (6) 1014-1021; DOI: https://doi.org/10.1124/dmd.110.037663
Shibue, Yuta
- You have accessQuantitative Time-Lapse Imaging-Based Analysis of Drug-Drug Interaction Mediated by Hepatobiliary Transporter, Multidrug Resistance-Associated Protein 2, in Sandwich-Cultured Rat HepatocytesTakeo Nakanishi, Yuta Shibue, Yoko Fukuyama, Kenji Yoshida, Hajime Fukuda, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition June 2011, 39 (6) 984-991; DOI: https://doi.org/10.1124/dmd.111.038059
Shinkyo, Raku
- You have accessCytochrome P450 2S1 is Reduced by NADPH-Cytochrome P450 ReductaseYi Xiao, Raku Shinkyo and F. Peter GuengerichDrug Metabolism and Disposition June 2011, 39 (6) 944-946; DOI: https://doi.org/10.1124/dmd.111.039321
Shirasaka, Yoshiyuki
- You have accessQuantitative Time-Lapse Imaging-Based Analysis of Drug-Drug Interaction Mediated by Hepatobiliary Transporter, Multidrug Resistance-Associated Protein 2, in Sandwich-Cultured Rat HepatocytesTakeo Nakanishi, Yuta Shibue, Yoko Fukuyama, Kenji Yoshida, Hajime Fukuda, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition June 2011, 39 (6) 984-991; DOI: https://doi.org/10.1124/dmd.111.038059
Silver, David L.
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
Slitt, Angela L.
- You have accessAlteration of Hepatic but Not Renal Transporter Expression in Diet-Induced Obese MiceVijay R. More and Angela L. SlittDrug Metabolism and Disposition June 2011, 39 (6) 992-999; DOI: https://doi.org/10.1124/dmd.110.037507
Solon, Eric
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Stolarczyk, Elzbieta I.
- You have accessSuppression of Cytochrome P450 Reductase (POR) Expression in Hepatoma Cells Replicates the Hepatic Lipidosis Observed in Hepatic POR-Null MiceTodd D. Porter, Subhashis Banerjee, Elzbieta I. Stolarczyk and Ling ZouDrug Metabolism and Disposition June 2011, 39 (6) 966-973; DOI: https://doi.org/10.1124/dmd.111.038562
Sugiura, Tomoko
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
Sugiyama, Yuichi
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Swaan, Peter W.
- You have accessATP-Binding Cassette Transporter Expression in Human Placenta as a Function of Pregnancy ConditionCifford W. Mason, Irina A. Buhimschi, Catalin S. Buhimschi, Yafeng Dong, Carl P. Weiner and Peter W. SwaanDrug Metabolism and Disposition June 2011, 39 (6) 1000-1007; DOI: https://doi.org/10.1124/dmd.111.038166
T
Takahashi, Ryan
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
Takakusa, Hideo
- You have accessMetabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by LapatinibHideo Takakusa, Michelle D. Wahlin, Chunsheng Zhao, Kelsey L. Hanson, Lee Sun New, Eric Chun Yong Chan and Sidney D. NelsonDrug Metabolism and Disposition June 2011, 39 (6) 1022-1030; DOI: https://doi.org/10.1124/dmd.110.037531
Takeuchi, Kazuya
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
Tamai, Ikumi
- You have accessQuantitative Time-Lapse Imaging-Based Analysis of Drug-Drug Interaction Mediated by Hepatobiliary Transporter, Multidrug Resistance-Associated Protein 2, in Sandwich-Cultured Rat HepatocytesTakeo Nakanishi, Yuta Shibue, Yoko Fukuyama, Kenji Yoshida, Hajime Fukuda, Yoshiyuki Shirasaka and Ikumi TamaiDrug Metabolism and Disposition June 2011, 39 (6) 984-991; DOI: https://doi.org/10.1124/dmd.111.038059
Thummel, Kenneth E.
- You have accessComplex Drug Interactions of HIV Protease Inhibitors 1: Inactivation, Induction, and Inhibition of Cytochrome P450 3A by Ritonavir or NelfinavirBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition June 2011, 39 (6) 1070-1078; DOI: https://doi.org/10.1124/dmd.110.037523
Trunzer, Markus
- You have accessCYP3A Time-Dependent Inhibition Risk Assessment Validated with 400 Reference DrugsAlfred Zimmerlin, Markus Trunzer and Bernard FallerDrug Metabolism and Disposition June 2011, 39 (6) 1039-1046; DOI: https://doi.org/10.1124/dmd.110.037911
U
Umeda, Saki
- You have accessPharmacokinetics and Hepatic Uptake of Eltrombopag, a Novel Platelet-Increasing AgentKazuya Takeuchi, Tomoko Sugiura, Saki Umeda, Kazuki Matsubara, Masato Horikawa, Noritaka Nakamichi, David L. Silver, Norihisa Ishiwata and Yukio KatoDrug Metabolism and Disposition June 2011, 39 (6) 1088-1096; DOI: https://doi.org/10.1124/dmd.110.037960
Unadkat, Jashvant D.
- You have accessComplex Drug Interactions of HIV Protease Inhibitors 1: Inactivation, Induction, and Inhibition of Cytochrome P450 3A by Ritonavir or NelfinavirBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition June 2011, 39 (6) 1070-1078; DOI: https://doi.org/10.1124/dmd.110.037523
W
Wahlin, Michelle D.
- You have accessMetabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by LapatinibHideo Takakusa, Michelle D. Wahlin, Chunsheng Zhao, Kelsey L. Hanson, Lee Sun New, Eric Chun Yong Chan and Sidney D. NelsonDrug Metabolism and Disposition June 2011, 39 (6) 1022-1030; DOI: https://doi.org/10.1124/dmd.110.037531
Watanabe, Takao
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Watanabe, Tomoko
- You have accessPrediction of the Overall Renal Tubular Secretion and Hepatic Clearance of Anionic Drugs and a Renal Drug-Drug Interaction Involving Organic Anion Transporter 3 in Humans by In Vitro Uptake ExperimentsTakao Watanabe, Hiroyuki Kusuhara, Tomoko Watanabe, Yasuyuki Debori, Kazuya Maeda, Tsunenori Kondo, Hideki Nakayama, Shigeru Horita, Brian W. Ogilvie, Andrew Parkinson, Zhuohan Hu and Yuichi SugiyamaDrug Metabolism and Disposition June 2011, 39 (6) 1031-1038; DOI: https://doi.org/10.1124/dmd.110.036129
Weiner, Carl P.
- You have accessATP-Binding Cassette Transporter Expression in Human Placenta as a Function of Pregnancy ConditionCifford W. Mason, Irina A. Buhimschi, Catalin S. Buhimschi, Yafeng Dong, Carl P. Weiner and Peter W. SwaanDrug Metabolism and Disposition June 2011, 39 (6) 1000-1007; DOI: https://doi.org/10.1124/dmd.111.038166
Weissbach, Herbert
- You have accessStudies on the Metabolism and Biological Activity of the Epimers of SulindacDavid Brunell, Daphna Sagher, Shailaja Kesaraju, Nathan Brot and Herbert WeissbachDrug Metabolism and Disposition June 2011, 39 (6) 1014-1021; DOI: https://doi.org/10.1124/dmd.110.037663
Whittington, Dale
- You have accessComplex Drug Interactions of HIV Protease Inhibitors 1: Inactivation, Induction, and Inhibition of Cytochrome P450 3A by Ritonavir or NelfinavirBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition June 2011, 39 (6) 1070-1078; DOI: https://doi.org/10.1124/dmd.110.037523
Wong, Harvey
- You have accessAbsorption, Distribution, Metabolism, and Excretion of [14C]GDC-0449 (Vismodegib), an Orally Active Hedgehog Pathway Inhibitor, in Rats and Dogs: A Unique Metabolic Pathway via Pyridine Ring OpeningQin Yue, Yung-Hsiang Chen, Teresa Mulder, Alan Deese, Ryan Takahashi, Patrick J. Rudewicz, Mark Reynolds, Eric Solon, Cornelis E. C. A. Hop, Harvey Wong and S. Cyrus KhojastehDrug Metabolism and Disposition June 2011, 39 (6) 952-965; DOI: https://doi.org/10.1124/dmd.110.037374
X
Xiao, Yi
- You have accessCytochrome P450 2S1 is Reduced by NADPH-Cytochrome P450 ReductaseYi Xiao, Raku Shinkyo and F. Peter GuengerichDrug Metabolism and Disposition June 2011, 39 (6) 944-946; DOI: https://doi.org/10.1124/dmd.111.039321
Xie, Fang
- You have accessThe Tissue-Specific Toxicity of Methimazole in the Mouse Olfactory Mucosa Is Partly Mediated through Target-Tissue Metabolic Activation by CYP2A5Fang Xie, Xin Zhou, Mary Beth Genter, Melissa Behr, Jun Gu and Xinxin DingDrug Metabolism and Disposition June 2011, 39 (6) 947-951; DOI: https://doi.org/10.1124/dmd.110.037895
Y
Yoshida, Kenji
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Yuan, Tao
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Zhang, Qing-Yu
- You have accessRole of Intestinal Cytochrome P450 (P450) in Modulating the Bioavailability of Oral Lovastatin: Insights from Studies on the Intestinal Epithelium-Specific P450 Reductase Knockout MouseYi Zhu, Jaime D'Agostino and Qing-Yu ZhangDrug Metabolism and Disposition June 2011, 39 (6) 939-943; DOI: https://doi.org/10.1124/dmd.110.037861
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- You have accessMetabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by LapatinibHideo Takakusa, Michelle D. Wahlin, Chunsheng Zhao, Kelsey L. Hanson, Lee Sun New, Eric Chun Yong Chan and Sidney D. NelsonDrug Metabolism and Disposition June 2011, 39 (6) 1022-1030; DOI: https://doi.org/10.1124/dmd.110.037531
Zhong, Dafang
- You have accessIdentification of Amiodarone Metabolites in Human Bile by Ultraperformance Liquid Chromatography/Quadrupole Time-of-Flight Mass SpectrometryPan Deng, Tiangeng You, Xiaoyan Chen, Tao Yuan, Haihua Huang and Dafang ZhongDrug Metabolism and Disposition June 2011, 39 (6) 1058-1069; DOI: https://doi.org/10.1124/dmd.110.037671
Zhou, Xin
- You have accessThe Tissue-Specific Toxicity of Methimazole in the Mouse Olfactory Mucosa Is Partly Mediated through Target-Tissue Metabolic Activation by CYP2A5Fang Xie, Xin Zhou, Mary Beth Genter, Melissa Behr, Jun Gu and Xinxin DingDrug Metabolism and Disposition June 2011, 39 (6) 947-951; DOI: https://doi.org/10.1124/dmd.110.037895
Zhu, Yi
- You have accessRole of Intestinal Cytochrome P450 (P450) in Modulating the Bioavailability of Oral Lovastatin: Insights from Studies on the Intestinal Epithelium-Specific P450 Reductase Knockout MouseYi Zhu, Jaime D'Agostino and Qing-Yu ZhangDrug Metabolism and Disposition June 2011, 39 (6) 939-943; DOI: https://doi.org/10.1124/dmd.110.037861
Zimmerlin, Alfred
- You have accessCYP3A Time-Dependent Inhibition Risk Assessment Validated with 400 Reference DrugsAlfred Zimmerlin, Markus Trunzer and Bernard FallerDrug Metabolism and Disposition June 2011, 39 (6) 1039-1046; DOI: https://doi.org/10.1124/dmd.110.037911
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- You have accessSuppression of Cytochrome P450 Reductase (POR) Expression in Hepatoma Cells Replicates the Hepatic Lipidosis Observed in Hepatic POR-Null MiceTodd D. Porter, Subhashis Banerjee, Elzbieta I. Stolarczyk and Ling ZouDrug Metabolism and Disposition June 2011, 39 (6) 966-973; DOI: https://doi.org/10.1124/dmd.111.038562
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