Index by author
July 01, 2011; Volume 39,Issue 7
A
Andersson, Tommy B.
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Aso, Yoshinori
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
B
Berg, Anna-Lena
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Boado, Ruben J.
- You have accessChronic Dosing of Mice with a Transferrin Receptor Monoclonal Antibody-Glial-Derived Neurotrophic Factor Fusion ProteinQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition July 2011, 39 (7) 1149-1154; DOI: https://doi.org/10.1124/dmd.111.038349
Bode, Chris
- You have accessUse of Transporter Knockdown Caco-2 Cells to Investigate the In Vitro Efflux of Statin DrugsJibin Li, Donna A. Volpe, Ying Wang, Wei Zhang, Chris Bode, Albert Owen and Ismael J. HidalgoDrug Metabolism and Disposition July 2011, 39 (7) 1196-1202; DOI: https://doi.org/10.1124/dmd.111.038075
Bowersox, S. Scott
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
C
Caron, Patrick
- You have accessIn Vitro Investigation of Human UDP-Glucuronosyltransferase Isoforms Responsible for Tacrolimus Glucuronidation: Predominant Contribution of UGT1A4Isabelle Laverdière, Patrick Caron, Mario Harvey, Éric Lévesque and Chantal GuillemetteDrug Metabolism and Disposition July 2011, 39 (7) 1127-1130; DOI: https://doi.org/10.1124/dmd.111.039040
Celma, Carles
- You have accessIn Vitro Metabolism of Irosustat, a Novel Steroid Sulfatase Inhibitor: Interspecies Comparison, Metabolite Identification, and Metabolic Enzyme IdentificationVerònica Ventura, Josep Solà, Carles Celma, Concepción Peraire and Rosendo ObachDrug Metabolism and Disposition July 2011, 39 (7) 1235-1246; DOI: https://doi.org/10.1124/dmd.111.038315
Chang, George
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
Cheatham, Steve F.
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Coleman, Renee
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
D
Danhof, Meindert
- You have accessA Semiphysiological Population Model for Prediction of the Pharmacokinetics of Drugs under Liver and Renal Disease ConditionsAshley Strougo, Ashraf Yassen, Walter Krauwinkel, Meindert Danhof and Jan FreijerDrug Metabolism and Disposition July 2011, 39 (7) 1278-1287; DOI: https://doi.org/10.1124/dmd.110.037838
Darnell, Malin
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Davies, Adrian M.
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
Davis, John
- You have accessApplication of Physiologically Based Pharmacokinetic Modeling to Understanding the Clinical Pharmacokinetics of UK-369,003Kenny J. Watson, John Davis and Hannah M. JonesDrug Metabolism and Disposition July 2011, 39 (7) 1203-1213; DOI: https://doi.org/10.1124/dmd.111.038224
Delzer, Juergen
- You have accessDisposition and Drug-Drug Interaction Potential of Veliparib (ABT-888), a Novel and Potent Inhibitor of Poly(ADP-ribose) PolymeraseXiaofeng Li, Juergen Delzer, Richard Voorman, Sonia M. de Morais and Yanbin LaoDrug Metabolism and Disposition July 2011, 39 (7) 1161-1169; DOI: https://doi.org/10.1124/dmd.110.037820
de Morais, Sonia M.
- You have accessDisposition and Drug-Drug Interaction Potential of Veliparib (ABT-888), a Novel and Potent Inhibitor of Poly(ADP-ribose) PolymeraseXiaofeng Li, Juergen Delzer, Richard Voorman, Sonia M. de Morais and Yanbin LaoDrug Metabolism and Disposition July 2011, 39 (7) 1161-1169; DOI: https://doi.org/10.1124/dmd.110.037820
Di, Li
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
Dillnér, Birgitta
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Dinter-Heidorn, Heike
- You have accessCannabinoid Type 1 Receptor Antagonists Modulate Transport Activity of Multidrug Resistance-Associated Proteins MRP1, MRP2, MRP3, and MRP4Hanneke G. M. Wittgen, Jeroen J. M. W. van den Heuvel, Petra H. H. van den Broek, Heike Dinter-Heidorn, Jan B. Koenderink and Frans G. M. RusselDrug Metabolism and Disposition July 2011, 39 (7) 1294-1302; DOI: https://doi.org/10.1124/dmd.110.037812
Druzgala, Pascal
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
Duran, Marinus
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
E
Ellis, Dave
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
F
Fischer, Thomas
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
Foti, Robert S.
- You have accessMechanism-Based Inactivation of Cytochrome P450 3A4 by Mibefradil through Heme DestructionRobert S. Foti, Dan A. Rock, Josh T. Pearson, Jan L. Wahlstrom and Larry C. WienkersDrug Metabolism and Disposition July 2011, 39 (7) 1188-1195; DOI: https://doi.org/10.1124/dmd.111.038505
Freijer, Jan
- You have accessA Semiphysiological Population Model for Prediction of the Pharmacokinetics of Drugs under Liver and Renal Disease ConditionsAshley Strougo, Ashraf Yassen, Walter Krauwinkel, Meindert Danhof and Jan FreijerDrug Metabolism and Disposition July 2011, 39 (7) 1278-1287; DOI: https://doi.org/10.1124/dmd.110.037838
G
Gannon, Shawn A.
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Gerlach, Jörg C.
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Guillemette, Chantal
- You have accessIn Vitro Investigation of Human UDP-Glucuronosyltransferase Isoforms Responsible for Tacrolimus Glucuronidation: Predominant Contribution of UGT1A4Isabelle Laverdière, Patrick Caron, Mario Harvey, Éric Lévesque and Chantal GuillemetteDrug Metabolism and Disposition July 2011, 39 (7) 1127-1130; DOI: https://doi.org/10.1124/dmd.111.039040
H
Halpert, James R.
- You have accessStructure and Function of Cytochromes P450 2B: From Mechanism-Based Inactivators to X-Ray Crystal Structures and BackJames R. HalpertDrug Metabolism and Disposition July 2011, 39 (7) 1113-1121; DOI: https://doi.org/10.1124/dmd.111.039719
Han, Xing
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Harvey, Mario
- You have accessIn Vitro Investigation of Human UDP-Glucuronosyltransferase Isoforms Responsible for Tacrolimus Glucuronidation: Predominant Contribution of UGT1A4Isabelle Laverdière, Patrick Caron, Mario Harvey, Éric Lévesque and Chantal GuillemetteDrug Metabolism and Disposition July 2011, 39 (7) 1127-1130; DOI: https://doi.org/10.1124/dmd.111.039040
Hashizume, Takanori
- You have accessIn Vitro Investigation of the Glutathione Transferase M1 and T1 Null Genotypes as Risk Factors for Troglitazone-Induced Liver InjuryToru Usui, Takanori Hashizume, Takashi Katsumata, Tsuyoshi Yokoi and Setsuko KomuroDrug Metabolism and Disposition July 2011, 39 (7) 1303-1310; DOI: https://doi.org/10.1124/dmd.111.038661
Hayashi, Mike
- You have accessSimulation of Clinical Drug-Drug Interactions from Hepatocyte CYP3A4 Induction Data and Its Potential Utility in Trial DesignsYang Xu, Yihong Zhou, Mike Hayashi, Magang Shou and Gary L. SkilesDrug Metabolism and Disposition July 2011, 39 (7) 1139-1148; DOI: https://doi.org/10.1124/dmd.111.038067
Hidalgo, Ismael J.
- You have accessUse of Transporter Knockdown Caco-2 Cells to Investigate the In Vitro Efflux of Statin DrugsJibin Li, Donna A. Volpe, Ying Wang, Wei Zhang, Chris Bode, Albert Owen and Ismael J. HidalgoDrug Metabolism and Disposition July 2011, 39 (7) 1196-1202; DOI: https://doi.org/10.1124/dmd.111.038075
Himmelstein, Matthew W.
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Honda, Kokichi
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Hough, Lindsay B.
- You have accessEffects of Acetylenic Epoxygenase Inhibitors on Recombinant Cytochrome P450sMelissa A. VanAlstine and Lindsay B. HoughDrug Metabolism and Disposition July 2011, 39 (7) 1221-1226; DOI: https://doi.org/10.1124/dmd.110.037424
Huang, Youping
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
Hui, Eric Ka-Wai
- You have accessChronic Dosing of Mice with a Transferrin Receptor Monoclonal Antibody-Glial-Derived Neurotrophic Factor Fusion ProteinQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition July 2011, 39 (7) 1149-1154; DOI: https://doi.org/10.1124/dmd.111.038349
I
IJlst, Lodewijk
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
Imai, Teruko
- You have accessPrediction of Human Intestinal Absorption of the Prodrug Temocapril by In Situ Single-Pass Perfusion Using Rat Intestine with Modified Hydrolase ActivityTakaaki Nozawa and Teruko ImaiDrug Metabolism and Disposition July 2011, 39 (7) 1263-1269; DOI: https://doi.org/10.1124/dmd.110.037937
Ishigai, Masaki
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
Iwabuchi, Haruo
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
Izumi, Takashi
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
J
Jepson, Gary W.
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Jiang, Xi-Ling
- You have accessNonlinear Pharmacokinetics of 5-Methoxy-N,N-dimethyltryptamine in MiceHong-Wu Shen, Xi-Ling Jiang and Ai-Ming YuDrug Metabolism and Disposition July 2011, 39 (7) 1227-1234; DOI: https://doi.org/10.1124/dmd.111.039107
Jones, Hannah M.
- You have accessApplication of Physiologically Based Pharmacokinetic Modeling to Understanding the Clinical Pharmacokinetics of UK-369,003Kenny J. Watson, John Davis and Hannah M. JonesDrug Metabolism and Disposition July 2011, 39 (7) 1203-1213; DOI: https://doi.org/10.1124/dmd.111.038224
K
Kato, Motohiro
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
Katsumata, Takashi
- You have accessIn Vitro Investigation of the Glutathione Transferase M1 and T1 Null Genotypes as Risk Factors for Troglitazone-Induced Liver InjuryToru Usui, Takanori Hashizume, Takashi Katsumata, Tsuyoshi Yokoi and Setsuko KomuroDrug Metabolism and Disposition July 2011, 39 (7) 1303-1310; DOI: https://doi.org/10.1124/dmd.111.038661
Koda, Hiroko
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
Koenderink, Jan B.
- You have accessCannabinoid Type 1 Receptor Antagonists Modulate Transport Activity of Multidrug Resistance-Associated Proteins MRP1, MRP2, MRP3, and MRP4Hanneke G. M. Wittgen, Jeroen J. M. W. van den Heuvel, Petra H. H. van den Broek, Heike Dinter-Heidorn, Jan B. Koenderink and Frans G. M. RusselDrug Metabolism and Disposition July 2011, 39 (7) 1294-1302; DOI: https://doi.org/10.1124/dmd.110.037812
Komuro, Setsuko
- You have accessIn Vitro Investigation of the Glutathione Transferase M1 and T1 Null Genotypes as Risk Factors for Troglitazone-Induced Liver InjuryToru Usui, Takanori Hashizume, Takashi Katsumata, Tsuyoshi Yokoi and Setsuko KomuroDrug Metabolism and Disposition July 2011, 39 (7) 1303-1310; DOI: https://doi.org/10.1124/dmd.111.038661
Krauwinkel, Walter
- You have accessA Semiphysiological Population Model for Prediction of the Pharmacokinetics of Drugs under Liver and Renal Disease ConditionsAshley Strougo, Ashraf Yassen, Walter Krauwinkel, Meindert Danhof and Jan FreijerDrug Metabolism and Disposition July 2011, 39 (7) 1278-1287; DOI: https://doi.org/10.1124/dmd.110.037838
Kumaraswamy, Padmapriya
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
L
Lao, Yanbin
- You have accessDisposition and Drug-Drug Interaction Potential of Veliparib (ABT-888), a Novel and Potent Inhibitor of Poly(ADP-ribose) PolymeraseXiaofeng Li, Juergen Delzer, Richard Voorman, Sonia M. de Morais and Yanbin LaoDrug Metabolism and Disposition July 2011, 39 (7) 1161-1169; DOI: https://doi.org/10.1124/dmd.110.037820
Laverdière, Isabelle
- You have accessIn Vitro Investigation of Human UDP-Glucuronosyltransferase Isoforms Responsible for Tacrolimus Glucuronidation: Predominant Contribution of UGT1A4Isabelle Laverdière, Patrick Caron, Mario Harvey, Éric Lévesque and Chantal GuillemetteDrug Metabolism and Disposition July 2011, 39 (7) 1127-1130; DOI: https://doi.org/10.1124/dmd.111.039040
Leslie, Elaine M.
- You have accessGlutathione Transferase P1 Interacts Strongly with the Inner Leaflet of the Plasma MembraneSohail S. Qazi, Anaida Osoria Pérez, Medica Sam and Elaine M. LeslieDrug Metabolism and Disposition July 2011, 39 (7) 1122-1126; DOI: https://doi.org/10.1124/dmd.111.039362
Lévesque, Éric
- You have accessIn Vitro Investigation of Human UDP-Glucuronosyltransferase Isoforms Responsible for Tacrolimus Glucuronidation: Predominant Contribution of UGT1A4Isabelle Laverdière, Patrick Caron, Mario Harvey, Éric Lévesque and Chantal GuillemetteDrug Metabolism and Disposition July 2011, 39 (7) 1127-1130; DOI: https://doi.org/10.1124/dmd.111.039040
Li, Jibin
- You have accessUse of Transporter Knockdown Caco-2 Cells to Investigate the In Vitro Efflux of Statin DrugsJibin Li, Donna A. Volpe, Ying Wang, Wei Zhang, Chris Bode, Albert Owen and Ismael J. HidalgoDrug Metabolism and Disposition July 2011, 39 (7) 1196-1202; DOI: https://doi.org/10.1124/dmd.111.038075
Li, Xiaofeng
- You have accessDisposition and Drug-Drug Interaction Potential of Veliparib (ABT-888), a Novel and Potent Inhibitor of Poly(ADP-ribose) PolymeraseXiaofeng Li, Juergen Delzer, Richard Voorman, Sonia M. de Morais and Yanbin LaoDrug Metabolism and Disposition July 2011, 39 (7) 1161-1169; DOI: https://doi.org/10.1124/dmd.110.037820
Lightning, Luke K.
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
Lin, Zhen
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
Liston, Theodore E.
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
Lowe, Ezra R.
- You have accessOcular Pharmacokinetics of Mapracorat, a Novel, Selective Glucocorticoid Receptor Agonist, in Rabbits and MonkeysJoel W. Proksch, Ezra R. Lowe and Keith W. WardDrug Metabolism and Disposition July 2011, 39 (7) 1181-1187; DOI: https://doi.org/10.1124/dmd.111.039099
Lu, Jeff Zhiqiang
- You have accessChronic Dosing of Mice with a Transferrin Receptor Monoclonal Antibody-Glial-Derived Neurotrophic Factor Fusion ProteinQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition July 2011, 39 (7) 1149-1154; DOI: https://doi.org/10.1124/dmd.111.038349
Luís, Paula B. M.
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
M
Mingoia, Robert T.
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Mitsui, Tetsuya
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
Miyaji, Yoshihiro
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Mohsen, Al-Walid
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
Mueller, Juergen
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
N
Nabb, Diane L.
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Nakayama, Shintaro
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Nozawa, Takaaki
- You have accessPrediction of Human Intestinal Absorption of the Prodrug Temocapril by In Situ Single-Pass Perfusion Using Rat Intestine with Modified Hydrolase ActivityTakaaki Nozawa and Teruko ImaiDrug Metabolism and Disposition July 2011, 39 (7) 1263-1269; DOI: https://doi.org/10.1124/dmd.110.037937
O
Obach, Rosendo
- You have accessIn Vitro Metabolism of Irosustat, a Novel Steroid Sulfatase Inhibitor: Interspecies Comparison, Metabolite Identification, and Metabolic Enzyme IdentificationVerònica Ventura, Josep Solà, Carles Celma, Concepción Peraire and Rosendo ObachDrug Metabolism and Disposition July 2011, 39 (7) 1235-1246; DOI: https://doi.org/10.1124/dmd.111.038315
Oguchi, Minoru
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
Okazaki, Osamu
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Okudaira, Noriko
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Osoria Pérez, Anaida
- You have accessGlutathione Transferase P1 Interacts Strongly with the Inner Leaflet of the Plasma MembraneSohail S. Qazi, Anaida Osoria Pérez, Medica Sam and Elaine M. LeslieDrug Metabolism and Disposition July 2011, 39 (7) 1122-1126; DOI: https://doi.org/10.1124/dmd.111.039362
Owen, Albert
- You have accessUse of Transporter Knockdown Caco-2 Cells to Investigate the In Vitro Efflux of Statin DrugsJibin Li, Donna A. Volpe, Ying Wang, Wei Zhang, Chris Bode, Albert Owen and Ismael J. HidalgoDrug Metabolism and Disposition July 2011, 39 (7) 1196-1202; DOI: https://doi.org/10.1124/dmd.111.038075
P
Palme, Monica
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
Pardridge, William M.
- You have accessChronic Dosing of Mice with a Transferrin Receptor Monoclonal Antibody-Glial-Derived Neurotrophic Factor Fusion ProteinQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition July 2011, 39 (7) 1149-1154; DOI: https://doi.org/10.1124/dmd.111.038349
Pearson, Josh T.
- You have accessMechanism-Based Inactivation of Cytochrome P450 3A4 by Mibefradil through Heme DestructionRobert S. Foti, Dan A. Rock, Josh T. Pearson, Jan L. Wahlstrom and Larry C. WienkersDrug Metabolism and Disposition July 2011, 39 (7) 1188-1195; DOI: https://doi.org/10.1124/dmd.111.038505
Peraire, Concepción
- You have accessIn Vitro Metabolism of Irosustat, a Novel Steroid Sulfatase Inhibitor: Interspecies Comparison, Metabolite Identification, and Metabolic Enzyme IdentificationVerònica Ventura, Josep Solà, Carles Celma, Concepción Peraire and Rosendo ObachDrug Metabolism and Disposition July 2011, 39 (7) 1235-1246; DOI: https://doi.org/10.1124/dmd.111.038315
Proksch, Joel W.
- You have accessOcular Pharmacokinetics of Mapracorat, a Novel, Selective Glucocorticoid Receptor Agonist, in Rabbits and MonkeysJoel W. Proksch, Ezra R. Lowe and Keith W. WardDrug Metabolism and Disposition July 2011, 39 (7) 1181-1187; DOI: https://doi.org/10.1124/dmd.111.039099
Q
Qazi, Sohail S.
- You have accessGlutathione Transferase P1 Interacts Strongly with the Inner Leaflet of the Plasma MembraneSohail S. Qazi, Anaida Osoria Pérez, Medica Sam and Elaine M. LeslieDrug Metabolism and Disposition July 2011, 39 (7) 1122-1126; DOI: https://doi.org/10.1124/dmd.111.039362
R
Rao, Satish
- You have accessMetabolism and Pharmacokinetics of Naronapride (ATI-7505), a Serotonin 5-HT4 Receptor Agonist for Gastrointestinal Motility DisordersS. Scott Bowersox, Luke K. Lightning, Satish Rao, Monica Palme, Dave Ellis, Renee Coleman, Adrian M. Davies, Padmapriya Kumaraswamy and Pascal DruzgalaDrug Metabolism and Disposition July 2011, 39 (7) 1170-1180; DOI: https://doi.org/10.1124/dmd.110.037564
Rock, Dan A.
- You have accessMechanism-Based Inactivation of Cytochrome P450 3A4 by Mibefradil through Heme DestructionRobert S. Foti, Dan A. Rock, Josh T. Pearson, Jan L. Wahlstrom and Larry C. WienkersDrug Metabolism and Disposition July 2011, 39 (7) 1188-1195; DOI: https://doi.org/10.1124/dmd.111.038505
Rosebraugh, Matthew
- You have accessReceptor-Based Dosing Optimization of Erythropoietin in Juvenile Sheep after PhlebotomyMatthew Rosebraugh, John A. Widness and Peter Veng-PedersenDrug Metabolism and Disposition July 2011, 39 (7) 1214-1220; DOI: https://doi.org/10.1124/dmd.110.036855
Rossberg, Ingrid
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Ruiter, Jos P. N.
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
Russel, Frans G. M.
- You have accessCannabinoid Type 1 Receptor Antagonists Modulate Transport Activity of Multidrug Resistance-Associated Proteins MRP1, MRP2, MRP3, and MRP4Hanneke G. M. Wittgen, Jeroen J. M. W. van den Heuvel, Petra H. H. van den Broek, Heike Dinter-Heidorn, Jan B. Koenderink and Frans G. M. RusselDrug Metabolism and Disposition July 2011, 39 (7) 1294-1302; DOI: https://doi.org/10.1124/dmd.110.037812
S
Sam, Medica
- You have accessGlutathione Transferase P1 Interacts Strongly with the Inner Leaflet of the Plasma MembraneSohail S. Qazi, Anaida Osoria Pérez, Medica Sam and Elaine M. LeslieDrug Metabolism and Disposition July 2011, 39 (7) 1122-1126; DOI: https://doi.org/10.1124/dmd.111.039362
Schreiter, Thomas
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Scott, Dennis O.
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
Sekiguchi, Nobuo
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
Shen, Hong-Wu
- You have accessNonlinear Pharmacokinetics of 5-Methoxy-N,N-dimethyltryptamine in MiceHong-Wu Shen, Xi-Ling Jiang and Ai-Ming YuDrug Metabolism and Disposition July 2011, 39 (7) 1227-1234; DOI: https://doi.org/10.1124/dmd.111.039107
Shiosakai, Kazuhito
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Shou, Magang
- You have accessSimulation of Clinical Drug-Drug Interactions from Hepatocyte CYP3A4 Induction Data and Its Potential Utility in Trial DesignsYang Xu, Yihong Zhou, Mike Hayashi, Magang Shou and Gary L. SkilesDrug Metabolism and Disposition July 2011, 39 (7) 1139-1148; DOI: https://doi.org/10.1124/dmd.111.038067
Silva, Margarida F. B.
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
Skiles, Gary L.
- You have accessSimulation of Clinical Drug-Drug Interactions from Hepatocyte CYP3A4 Induction Data and Its Potential Utility in Trial DesignsYang Xu, Yihong Zhou, Mike Hayashi, Magang Shou and Gary L. SkilesDrug Metabolism and Disposition July 2011, 39 (7) 1139-1148; DOI: https://doi.org/10.1124/dmd.111.038067
Söderdahl, Therese
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Solà, Josep
- You have accessIn Vitro Metabolism of Irosustat, a Novel Steroid Sulfatase Inhibitor: Interspecies Comparison, Metabolite Identification, and Metabolic Enzyme IdentificationVerònica Ventura, Josep Solà, Carles Celma, Concepción Peraire and Rosendo ObachDrug Metabolism and Disposition July 2011, 39 (7) 1235-1246; DOI: https://doi.org/10.1124/dmd.111.038315
Strougo, Ashley
- You have accessA Semiphysiological Population Model for Prediction of the Pharmacokinetics of Drugs under Liver and Renal Disease ConditionsAshley Strougo, Ashraf Yassen, Walter Krauwinkel, Meindert Danhof and Jan FreijerDrug Metabolism and Disposition July 2011, 39 (7) 1278-1287; DOI: https://doi.org/10.1124/dmd.110.037838
Sugiyama, Daisuke
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Suzuki, Wataru
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Szostek, Bogdan
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
T
Takada, Maiko
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
Takakusa, Hideo
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Takata, Shotaro
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
Tavares de Almeida, Isabel
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
Troutman, Matthew D.
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
U
Uchiyama, Minoru
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
Umland, John P.
- You have accessSpecies Independence in Brain Tissue Binding Using Brain HomogenatesLi Di, John P. Umland, George Chang, Youping Huang, Zhen Lin, Dennis O. Scott, Matthew D. Troutman and Theodore E. ListonDrug Metabolism and Disposition July 2011, 39 (7) 1270-1277; DOI: https://doi.org/10.1124/dmd.111.038778
Urbaniak, Thomas
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Usui, Toru
- You have accessIn Vitro Investigation of the Glutathione Transferase M1 and T1 Null Genotypes as Risk Factors for Troglitazone-Induced Liver InjuryToru Usui, Takanori Hashizume, Takashi Katsumata, Tsuyoshi Yokoi and Setsuko KomuroDrug Metabolism and Disposition July 2011, 39 (7) 1303-1310; DOI: https://doi.org/10.1124/dmd.111.038661
V
VanAlstine, Melissa A.
- You have accessEffects of Acetylenic Epoxygenase Inhibitors on Recombinant Cytochrome P450sMelissa A. VanAlstine and Lindsay B. HoughDrug Metabolism and Disposition July 2011, 39 (7) 1221-1226; DOI: https://doi.org/10.1124/dmd.110.037424
van den Broek, Petra H. H.
- You have accessCannabinoid Type 1 Receptor Antagonists Modulate Transport Activity of Multidrug Resistance-Associated Proteins MRP1, MRP2, MRP3, and MRP4Hanneke G. M. Wittgen, Jeroen J. M. W. van den Heuvel, Petra H. H. van den Broek, Heike Dinter-Heidorn, Jan B. Koenderink and Frans G. M. RusselDrug Metabolism and Disposition July 2011, 39 (7) 1294-1302; DOI: https://doi.org/10.1124/dmd.110.037812
van den Heuvel, Jeroen J. M. W.
- You have accessCannabinoid Type 1 Receptor Antagonists Modulate Transport Activity of Multidrug Resistance-Associated Proteins MRP1, MRP2, MRP3, and MRP4Hanneke G. M. Wittgen, Jeroen J. M. W. van den Heuvel, Petra H. H. van den Broek, Heike Dinter-Heidorn, Jan B. Koenderink and Frans G. M. RusselDrug Metabolism and Disposition July 2011, 39 (7) 1294-1302; DOI: https://doi.org/10.1124/dmd.110.037812
Veng-Pedersen, Peter
- You have accessReceptor-Based Dosing Optimization of Erythropoietin in Juvenile Sheep after PhlebotomyMatthew Rosebraugh, John A. Widness and Peter Veng-PedersenDrug Metabolism and Disposition July 2011, 39 (7) 1214-1220; DOI: https://doi.org/10.1124/dmd.110.036855
Ventura, Verònica
- You have accessIn Vitro Metabolism of Irosustat, a Novel Steroid Sulfatase Inhibitor: Interspecies Comparison, Metabolite Identification, and Metabolic Enzyme IdentificationVerònica Ventura, Josep Solà, Carles Celma, Concepción Peraire and Rosendo ObachDrug Metabolism and Disposition July 2011, 39 (7) 1235-1246; DOI: https://doi.org/10.1124/dmd.111.038315
Vockley, Jerry
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
Volpe, Donna A.
- You have accessUse of Transporter Knockdown Caco-2 Cells to Investigate the In Vitro Efflux of Statin DrugsJibin Li, Donna A. Volpe, Ying Wang, Wei Zhang, Chris Bode, Albert Owen and Ismael J. HidalgoDrug Metabolism and Disposition July 2011, 39 (7) 1196-1202; DOI: https://doi.org/10.1124/dmd.111.038075
Voorman, Richard
- You have accessDisposition and Drug-Drug Interaction Potential of Veliparib (ABT-888), a Novel and Potent Inhibitor of Poly(ADP-ribose) PolymeraseXiaofeng Li, Juergen Delzer, Richard Voorman, Sonia M. de Morais and Yanbin LaoDrug Metabolism and Disposition July 2011, 39 (7) 1161-1169; DOI: https://doi.org/10.1124/dmd.110.037820
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Wahlstrom, Jan L.
- You have accessMechanism-Based Inactivation of Cytochrome P450 3A4 by Mibefradil through Heme DestructionRobert S. Foti, Dan A. Rock, Josh T. Pearson, Jan L. Wahlstrom and Larry C. WienkersDrug Metabolism and Disposition July 2011, 39 (7) 1188-1195; DOI: https://doi.org/10.1124/dmd.111.038505
Wanders, Ronald J. A.
- You have accessRole of Isovaleryl-CoA Dehydrogenase and Short Branched-Chain Acyl-CoA Dehydrogenase in the Metabolism of Valproic Acid: Implications for the Branched-Chain Amino Acid Oxidation PathwayPaula B. M. Luís, Jos P. N. Ruiter, Lodewijk IJlst, Isabel Tavares de Almeida, Marinus Duran, Al-Walid Mohsen, Jerry Vockley, Ronald J. A. Wanders and Margarida F. B. SilvaDrug Metabolism and Disposition July 2011, 39 (7) 1155-1160; DOI: https://doi.org/10.1124/dmd.110.037606
Wang, Ying
- You have accessUse of Transporter Knockdown Caco-2 Cells to Investigate the In Vitro Efflux of Statin DrugsJibin Li, Donna A. Volpe, Ying Wang, Wei Zhang, Chris Bode, Albert Owen and Ismael J. HidalgoDrug Metabolism and Disposition July 2011, 39 (7) 1196-1202; DOI: https://doi.org/10.1124/dmd.111.038075
Ward, Keith W.
- You have accessOcular Pharmacokinetics of Mapracorat, a Novel, Selective Glucocorticoid Receptor Agonist, in Rabbits and MonkeysJoel W. Proksch, Ezra R. Lowe and Keith W. WardDrug Metabolism and Disposition July 2011, 39 (7) 1181-1187; DOI: https://doi.org/10.1124/dmd.111.039099
Watanabe, Akiko
- You have accessCombination of GSH Trapping and Time-Dependent Inhibition Assays as a Predictive Method of Drugs Generating Highly Reactive MetabolitesShintaro Nakayama, Hideo Takakusa, Akiko Watanabe, Yoshihiro Miyaji, Wataru Suzuki, Daisuke Sugiyama, Kazuhito Shiosakai, Kokichi Honda, Noriko Okudaira, Takashi Izumi and Osamu OkazakiDrug Metabolism and Disposition July 2011, 39 (7) 1247-1254; DOI: https://doi.org/10.1124/dmd.111.039180
Watanabe, Hiroo
- You have accessQuantitative Prediction of Mechanism-Based Inhibition Caused by Mibefradil in RatsNobuo Sekiguchi, Motohiro Kato, Maiko Takada, Hiroo Watanabe, Shotaro Takata, Tetsuya Mitsui, Yoshinori Aso and Masaki IshigaiDrug Metabolism and Disposition July 2011, 39 (7) 1255-1262; DOI: https://doi.org/10.1124/dmd.110.037903
Watson, Kenny J.
- You have accessApplication of Physiologically Based Pharmacokinetic Modeling to Understanding the Clinical Pharmacokinetics of UK-369,003Kenny J. Watson, John Davis and Hannah M. JonesDrug Metabolism and Disposition July 2011, 39 (7) 1203-1213; DOI: https://doi.org/10.1124/dmd.111.038224
Widness, John A.
- You have accessReceptor-Based Dosing Optimization of Erythropoietin in Juvenile Sheep after PhlebotomyMatthew Rosebraugh, John A. Widness and Peter Veng-PedersenDrug Metabolism and Disposition July 2011, 39 (7) 1214-1220; DOI: https://doi.org/10.1124/dmd.110.036855
Wienkers, Larry C.
- You have accessMechanism-Based Inactivation of Cytochrome P450 3A4 by Mibefradil through Heme DestructionRobert S. Foti, Dan A. Rock, Josh T. Pearson, Jan L. Wahlstrom and Larry C. WienkersDrug Metabolism and Disposition July 2011, 39 (7) 1188-1195; DOI: https://doi.org/10.1124/dmd.111.038505
Wittgen, Hanneke G. M.
- You have accessCannabinoid Type 1 Receptor Antagonists Modulate Transport Activity of Multidrug Resistance-Associated Proteins MRP1, MRP2, MRP3, and MRP4Hanneke G. M. Wittgen, Jeroen J. M. W. van den Heuvel, Petra H. H. van den Broek, Heike Dinter-Heidorn, Jan B. Koenderink and Frans G. M. RusselDrug Metabolism and Disposition July 2011, 39 (7) 1294-1302; DOI: https://doi.org/10.1124/dmd.110.037812
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Xu, Yang
- You have accessSimulation of Clinical Drug-Drug Interactions from Hepatocyte CYP3A4 Induction Data and Its Potential Utility in Trial DesignsYang Xu, Yihong Zhou, Mike Hayashi, Magang Shou and Gary L. SkilesDrug Metabolism and Disposition July 2011, 39 (7) 1139-1148; DOI: https://doi.org/10.1124/dmd.111.038067
Y
Yamamura, Naotoshi
- You have accessIn Vitro Metabolism of Rivoglitazone, a Novel Peroxisome Proliferator-Activated Receptor γ Agonist, in Rat, Monkey, and Human Liver Microsomes and Freshly Isolated HepatocytesMinoru Uchiyama, Hiroko Koda, Thomas Fischer, Juergen Mueller, Naotoshi Yamamura, Minoru Oguchi, Haruo Iwabuchi, Osamu Okazaki and Takashi IzumiDrug Metabolism and Disposition July 2011, 39 (7) 1311-1319; DOI: https://doi.org/10.1124/dmd.111.038729
Yang, Ching-Hui
- You have accessComparative Metabolism of 1,2,3,3,3-Pentafluoropropene in Male and Female Mouse, Rat, Dog, and Human Liver Microsomes and Cytosol and Male Rat Hepatocytes via Oxidative Dehalogenation and Glutathione S-Conjugation PathwaysXing Han, Bogdan Szostek, Ching-Hui Yang, Steve F. Cheatham, Robert T. Mingoia, Diane L. Nabb, Shawn A. Gannon, Matthew W. Himmelstein and Gary W. JepsonDrug Metabolism and Disposition July 2011, 39 (7) 1288-1293; DOI: https://doi.org/10.1124/dmd.111.038299
Yassen, Ashraf
- You have accessA Semiphysiological Population Model for Prediction of the Pharmacokinetics of Drugs under Liver and Renal Disease ConditionsAshley Strougo, Ashraf Yassen, Walter Krauwinkel, Meindert Danhof and Jan FreijerDrug Metabolism and Disposition July 2011, 39 (7) 1278-1287; DOI: https://doi.org/10.1124/dmd.110.037838
Yokoi, Tsuyoshi
- You have accessIn Vitro Investigation of the Glutathione Transferase M1 and T1 Null Genotypes as Risk Factors for Troglitazone-Induced Liver InjuryToru Usui, Takanori Hashizume, Takashi Katsumata, Tsuyoshi Yokoi and Setsuko KomuroDrug Metabolism and Disposition July 2011, 39 (7) 1303-1310; DOI: https://doi.org/10.1124/dmd.111.038661
Yu, Ai-Ming
- You have accessNonlinear Pharmacokinetics of 5-Methoxy-N,N-dimethyltryptamine in MiceHong-Wu Shen, Xi-Ling Jiang and Ai-Ming YuDrug Metabolism and Disposition July 2011, 39 (7) 1227-1234; DOI: https://doi.org/10.1124/dmd.111.039107
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Zeilinger, Katrin
- You have accessCytochrome P450-Dependent Metabolism in HepaRG Cells Cultured in a Dynamic Three-Dimensional BioreactorMalin Darnell, Thomas Schreiter, Katrin Zeilinger, Thomas Urbaniak, Therese Söderdahl, Ingrid Rossberg, Birgitta Dillnér, Anna-Lena Berg, Jörg C. Gerlach and Tommy B. AnderssonDrug Metabolism and Disposition July 2011, 39 (7) 1131-1138; DOI: https://doi.org/10.1124/dmd.110.037721
Zhang, Wei
- You have accessUse of Transporter Knockdown Caco-2 Cells to Investigate the In Vitro Efflux of Statin DrugsJibin Li, Donna A. Volpe, Ying Wang, Wei Zhang, Chris Bode, Albert Owen and Ismael J. HidalgoDrug Metabolism and Disposition July 2011, 39 (7) 1196-1202; DOI: https://doi.org/10.1124/dmd.111.038075
Zhou, Qing-Hui
- You have accessChronic Dosing of Mice with a Transferrin Receptor Monoclonal Antibody-Glial-Derived Neurotrophic Factor Fusion ProteinQing-Hui Zhou, Ruben J. Boado, Eric Ka-Wai Hui, Jeff Zhiqiang Lu and William M. PardridgeDrug Metabolism and Disposition July 2011, 39 (7) 1149-1154; DOI: https://doi.org/10.1124/dmd.111.038349
Zhou, Yihong
- You have accessSimulation of Clinical Drug-Drug Interactions from Hepatocyte CYP3A4 Induction Data and Its Potential Utility in Trial DesignsYang Xu, Yihong Zhou, Mike Hayashi, Magang Shou and Gary L. SkilesDrug Metabolism and Disposition July 2011, 39 (7) 1139-1148; DOI: https://doi.org/10.1124/dmd.111.038067
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