Index by author
March 01, 2012; Volume 40,Issue 3
A
Aleksunes, Lauren M.
- You have accessExpression of Organic Anion Transporter 2 in the Human Kidney and Its Potential Role in the Tubular Secretion of Guanine-Containing Antiviral DrugsYaofeng Cheng, Arpine Vapurcuyan, Mohammad Shahidullah, Lauren M. Aleksunes and Ryan M. PelisDrug Metabolism and Disposition March 2012, 40 (3) 617-624; DOI: https://doi.org/10.1124/dmd.111.042036
Almeida, Reinaldo
- You have accessInvestigation of Figopitant and Its Metabolites in Rat Tissue by Combining Whole-Body Autoradiography with Liquid Extraction Surface Analysis Mass SpectrometrySimone Schadt, Susanne Kallbach, Reinaldo Almeida and Jan SandelDrug Metabolism and Disposition March 2012, 40 (3) 419-425; DOI: https://doi.org/10.1124/dmd.111.043562
Amano, Nobuyuki
- You have accessIn Vivo Biliary Clearance Should Be Predicted by Intrinsic Biliary Clearance in Sandwich-Cultured HepatocytesMasanori Nakakariya, Midori Ono, Nobuyuki Amano, Toshiya Moriwaki, Kazuya Maeda and Yuichi SugiyamaDrug Metabolism and Disposition March 2012, 40 (3) 602-609; DOI: https://doi.org/10.1124/dmd.111.042101
Ando, Yoshinori
- You have accessChanges in Expression of Drug-Metabolizing Enzymes by Single-Walled Carbon Nanotubes in Human Respiratory Tract CellsKotaro Hitoshi, Miki Katoh, Tomoko Suzuki, Yoshinori Ando and Masayuki NadaiDrug Metabolism and Disposition March 2012, 40 (3) 579-587; DOI: https://doi.org/10.1124/dmd.111.043455
Anwar-Mohamed, Anwar
- You have accessInhibition of Heme Oxygenase-1 Partially Reverses the Arsenite-Mediated Decrease of CYP1A1, CYP1A2, CYP3A23, and CYP3A2 Catalytic Activity in Isolated Rat HepatocytesAnwar Anwar-Mohamed, Lars-Oliver Klotz and Ayman O. S. El-KadiDrug Metabolism and Disposition March 2012, 40 (3) 504-514; DOI: https://doi.org/10.1124/dmd.111.042564
Arakawa, Shingo
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
B
Baldisseri, Donna M.
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
Bello, Carlo
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
Bernhardt, Rita
- You have accessThe Effects of Rosuvastatin and the CYP51A1 Inhibitor LEK-935 on the Proteome of Primary Human HepatocytesMartin Wörner, Katja Melchior, Katalin Monostory, Jean-Marc Pascussi, Christian G. Huber and Rita BernhardtDrug Metabolism and Disposition March 2012, 40 (3) 414-418; DOI: https://doi.org/10.1124/dmd.111.040402
Block, Wiebke
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
Bu, Hai-Zhi
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
Buckley, Brian
- You have accessInhibition of Genistein Glucuronidation by Bisphenol A in Human and Rat Liver MicrosomesJanis L. Coughlin, Paul E. Thomas and Brian BuckleyDrug Metabolism and Disposition March 2012, 40 (3) 481-485; DOI: https://doi.org/10.1124/dmd.111.042366
Bundgaard, Christoffer
- You have accessSpecies Comparison of In Vivo P-Glycoprotein-Mediated Brain Efflux Using mdr1a-Deficient Rats and MiceChristoffer Bundgaard, Christian Jes Nyberg Jensen and Mats GarmerDrug Metabolism and Disposition March 2012, 40 (3) 461-466; DOI: https://doi.org/10.1124/dmd.111.043083
C
Canet, Mark J.
- You have accessMolecular Mechanism of Altered Ezetimibe Disposition in Nonalcoholic SteatohepatitisRhiannon N. Hardwick, Craig D. Fisher, Stephanie M. Street, Mark J. Canet and Nathan J. CherringtonDrug Metabolism and Disposition March 2012, 40 (3) 450-460; DOI: https://doi.org/10.1124/dmd.111.041095
Chen, Jianjun
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
Chen, Xiaoyan
- You have accessMetabolism and Pharmacokinetics of Morinidazole in Humans: Identification of Diastereoisomeric Morpholine N+-Glucuronides Catalyzed by UDP Glucuronosyltransferase 1A9Ruina Gao, Liang Li, Cen Xie, Xingxing Diao, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition March 2012, 40 (3) 556-567; DOI: https://doi.org/10.1124/dmd.111.042689
Cheng, Yaofeng
- You have accessExpression of Organic Anion Transporter 2 in the Human Kidney and Its Potential Role in the Tubular Secretion of Guanine-Containing Antiviral DrugsYaofeng Cheng, Arpine Vapurcuyan, Mohammad Shahidullah, Lauren M. Aleksunes and Ryan M. PelisDrug Metabolism and Disposition March 2012, 40 (3) 617-624; DOI: https://doi.org/10.1124/dmd.111.042036
Cherrington, Nathan J.
- You have accessMolecular Mechanism of Altered Ezetimibe Disposition in Nonalcoholic SteatohepatitisRhiannon N. Hardwick, Craig D. Fisher, Stephanie M. Street, Mark J. Canet and Nathan J. CherringtonDrug Metabolism and Disposition March 2012, 40 (3) 450-460; DOI: https://doi.org/10.1124/dmd.111.041095
Clark, Alan J.
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Collier, Ann C.
- You have accessComplex Drug Interactions of the HIV Protease Inhibitors 3: Effect of Simultaneous or Staggered Dosing of Digoxin and Ritonavir, Nelfinavir, Rifampin, or BupropionBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition March 2012, 40 (3) 610-616; DOI: https://doi.org/10.1124/dmd.111.042705
Coughlin, Janis L.
- You have accessInhibition of Genistein Glucuronidation by Bisphenol A in Human and Rat Liver MicrosomesJanis L. Coughlin, Paul E. Thomas and Brian BuckleyDrug Metabolism and Disposition March 2012, 40 (3) 481-485; DOI: https://doi.org/10.1124/dmd.111.042366
D
Dalvie, Deepak
- You have accessUse of a Multistaged Time-Dependent Inhibition Assay to Assess the Impact of Intestinal Metabolism on Drug-Drug Interaction PotentialMichael Zientek and Deepak DalvieDrug Metabolism and Disposition March 2012, 40 (3) 467-473; DOI: https://doi.org/10.1124/dmd.111.043257
de Waart, Dirk R.
- You have accessOral Availability of Cefadroxil Depends on ABCC3 and ABCC4Dirk R. de Waart, Koen van de Wetering, Cindy Kunne, Suzanne Duijst, Coen C. Paulusma and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition March 2012, 40 (3) 515-521; DOI: https://doi.org/10.1124/dmd.111.041731
Diao, Xingxing
- You have accessMetabolism and Pharmacokinetics of Morinidazole in Humans: Identification of Diastereoisomeric Morpholine N+-Glucuronides Catalyzed by UDP Glucuronosyltransferase 1A9Ruina Gao, Liang Li, Cen Xie, Xingxing Diao, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition March 2012, 40 (3) 556-567; DOI: https://doi.org/10.1124/dmd.111.042689
Dong, Peipei
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Duijst, Suzanne
- You have accessOral Availability of Cefadroxil Depends on ABCC3 and ABCC4Dirk R. de Waart, Koen van de Wetering, Cindy Kunne, Suzanne Duijst, Coen C. Paulusma and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition March 2012, 40 (3) 515-521; DOI: https://doi.org/10.1124/dmd.111.041731
E
Eggers, Karen
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
El-Kadi, Ayman O. S.
- You have accessInhibition of Heme Oxygenase-1 Partially Reverses the Arsenite-Mediated Decrease of CYP1A1, CYP1A2, CYP3A23, and CYP3A2 Catalytic Activity in Isolated Rat HepatocytesAnwar Anwar-Mohamed, Lars-Oliver Klotz and Ayman O. S. El-KadiDrug Metabolism and Disposition March 2012, 40 (3) 504-514; DOI: https://doi.org/10.1124/dmd.111.042564
Endo, Seiko
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
F
Fang, Zhongze
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Finel, Moshe
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Fischer, Thomas
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
Fisher, Craig D.
- You have accessMolecular Mechanism of Altered Ezetimibe Disposition in Nonalcoholic SteatohepatitisRhiannon N. Hardwick, Craig D. Fisher, Stephanie M. Street, Mark J. Canet and Nathan J. CherringtonDrug Metabolism and Disposition March 2012, 40 (3) 450-460; DOI: https://doi.org/10.1124/dmd.111.041095
Fujimoto, Kazunori
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
Fukahori, Aiko
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
G
Gallo, M. A.
- You have accessPolychlorinated Biphenyl Congeners that Increase the Glucuronidation and Biliary Excretion of Thyroxine Are Distinct from the Congeners that Enhance the Serum Disappearance of ThyroxineL. A. Martin, D. T. Wilson, K. R. Reuhl, M. A. Gallo and C. D. KlaassenDrug Metabolism and Disposition March 2012, 40 (3) 588-595; DOI: https://doi.org/10.1124/dmd.111.042796
Gao, Hongying
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Gao, Ruina
- You have accessMetabolism and Pharmacokinetics of Morinidazole in Humans: Identification of Diastereoisomeric Morpholine N+-Glucuronides Catalyzed by UDP Glucuronosyltransferase 1A9Ruina Gao, Liang Li, Cen Xie, Xingxing Diao, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition March 2012, 40 (3) 556-567; DOI: https://doi.org/10.1124/dmd.111.042689
Garmer, Mats
- You have accessSpecies Comparison of In Vivo P-Glycoprotein-Mediated Brain Efflux Using mdr1a-Deficient Rats and MiceChristoffer Bundgaard, Christian Jes Nyberg Jensen and Mats GarmerDrug Metabolism and Disposition March 2012, 40 (3) 461-466; DOI: https://doi.org/10.1124/dmd.111.043083
Gates, Leah A.
- You have accessTrapping of cis-2-Butene-1,4-dial to Measure Furan Metabolism in Human Liver Microsomes by Cytochrome P450 EnzymesLeah A. Gates, Ding Lu and Lisa A. PetersonDrug Metabolism and Disposition March 2012, 40 (3) 596-601; DOI: https://doi.org/10.1124/dmd.111.043679
Ge, Guangbo
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
H
Hardwick, Rhiannon N.
- You have accessMolecular Mechanism of Altered Ezetimibe Disposition in Nonalcoholic SteatohepatitisRhiannon N. Hardwick, Craig D. Fisher, Stephanie M. Street, Mark J. Canet and Nathan J. CherringtonDrug Metabolism and Disposition March 2012, 40 (3) 450-460; DOI: https://doi.org/10.1124/dmd.111.041095
Hasegawa, Maki
- You have accessInvestigation of Drug-Drug Interactions Caused by Human Pregnane X Receptor-Mediated Induction of CYP3A4 and CYP2C Subfamilies in Chimeric Mice with a Humanized LiverMaki Hasegawa, Harunobu Tahara, Ryo Inoue, Masakazu Kakuni, Chise Tateno and Junko UshikiDrug Metabolism and Disposition March 2012, 40 (3) 474-480; DOI: https://doi.org/10.1124/dmd.111.042754
He, Guiyuan
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Helsby, Nuala A.
- You have accessWhich CYP2B6 Variants Have Functional Consequences for Cyclophosphamide Bioactivation?Nuala A. Helsby and Malcolm D. TingleDrug Metabolism and Disposition March 2012, 40 (3) 635-637; DOI: https://doi.org/10.1124/dmd.111.043646
Hitoshi, Kotaro
- You have accessChanges in Expression of Drug-Metabolizing Enzymes by Single-Walled Carbon Nanotubes in Human Respiratory Tract CellsKotaro Hitoshi, Miki Katoh, Tomoko Suzuki, Yoshinori Ando and Masayuki NadaiDrug Metabolism and Disposition March 2012, 40 (3) 579-587; DOI: https://doi.org/10.1124/dmd.111.043455
Honkavaara, Juhana
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
Huber, Christian G.
- You have accessThe Effects of Rosuvastatin and the CYP51A1 Inhibitor LEK-935 on the Proteome of Primary Human HepatocytesMartin Wörner, Katja Melchior, Katalin Monostory, Jean-Marc Pascussi, Christian G. Huber and Rita BernhardtDrug Metabolism and Disposition March 2012, 40 (3) 414-418; DOI: https://doi.org/10.1124/dmd.111.040402
I
Inoue, Ryo
- You have accessInvestigation of Drug-Drug Interactions Caused by Human Pregnane X Receptor-Mediated Induction of CYP3A4 and CYP2C Subfamilies in Chimeric Mice with a Humanized LiverMaki Hasegawa, Harunobu Tahara, Ryo Inoue, Masakazu Kakuni, Chise Tateno and Junko UshikiDrug Metabolism and Disposition March 2012, 40 (3) 474-480; DOI: https://doi.org/10.1124/dmd.111.042754
Isoherranen, Nina
- You have accessStereospecific Metabolism of Itraconazole by CYP3A4: Dioxolane Ring Scission of Azole AntifungalsChi-Chi Peng, Wei Shi, Justin D. Lutz, Kent L. Kunze, Jun O. Liu, Wendel L. Nelson and Nina IsoherranenDrug Metabolism and Disposition March 2012, 40 (3) 426-435; DOI: https://doi.org/10.1124/dmd.111.042739
J
Jensen, Christian Jes Nyberg
- You have accessSpecies Comparison of In Vivo P-Glycoprotein-Mediated Brain Efflux Using mdr1a-Deficient Rats and MiceChristoffer Bundgaard, Christian Jes Nyberg Jensen and Mats GarmerDrug Metabolism and Disposition March 2012, 40 (3) 461-466; DOI: https://doi.org/10.1124/dmd.111.043083
K
Kakuni, Masakazu
- You have accessInvestigation of Drug-Drug Interactions Caused by Human Pregnane X Receptor-Mediated Induction of CYP3A4 and CYP2C Subfamilies in Chimeric Mice with a Humanized LiverMaki Hasegawa, Harunobu Tahara, Ryo Inoue, Masakazu Kakuni, Chise Tateno and Junko UshikiDrug Metabolism and Disposition March 2012, 40 (3) 474-480; DOI: https://doi.org/10.1124/dmd.111.042754
Kallbach, Susanne
- You have accessInvestigation of Figopitant and Its Metabolites in Rat Tissue by Combining Whole-Body Autoradiography with Liquid Extraction Surface Analysis Mass SpectrometrySimone Schadt, Susanne Kallbach, Reinaldo Almeida and Jan SandelDrug Metabolism and Disposition March 2012, 40 (3) 419-425; DOI: https://doi.org/10.1124/dmd.111.043562
Kang, Ping
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
Kato, Ayako
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
Katoh, Miki
- You have accessChanges in Expression of Drug-Metabolizing Enzymes by Single-Walled Carbon Nanotubes in Human Respiratory Tract CellsKotaro Hitoshi, Miki Katoh, Tomoko Suzuki, Yoshinori Ando and Masayuki NadaiDrug Metabolism and Disposition March 2012, 40 (3) 579-587; DOI: https://doi.org/10.1124/dmd.111.043455
Kharasch, Evan D.
- You have accessComplex Drug Interactions of the HIV Protease Inhibitors 3: Effect of Simultaneous or Staggered Dosing of Digoxin and Ritonavir, Nelfinavir, Rifampin, or BupropionBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition March 2012, 40 (3) 610-616; DOI: https://doi.org/10.1124/dmd.111.042705
Kirby, Brian J.
- You have accessComplex Drug Interactions of the HIV Protease Inhibitors 3: Effect of Simultaneous or Staggered Dosing of Digoxin and Ritonavir, Nelfinavir, Rifampin, or BupropionBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition March 2012, 40 (3) 610-616; DOI: https://doi.org/10.1124/dmd.111.042705
Klaassen, C. D.
- You have accessPolychlorinated Biphenyl Congeners that Increase the Glucuronidation and Biliary Excretion of Thyroxine Are Distinct from the Congeners that Enhance the Serum Disappearance of ThyroxineL. A. Martin, D. T. Wilson, K. R. Reuhl, M. A. Gallo and C. D. KlaassenDrug Metabolism and Disposition March 2012, 40 (3) 588-595; DOI: https://doi.org/10.1124/dmd.111.042796
Klotz, Lars-Oliver
- You have accessInhibition of Heme Oxygenase-1 Partially Reverses the Arsenite-Mediated Decrease of CYP1A1, CYP1A2, CYP3A23, and CYP3A2 Catalytic Activity in Isolated Rat HepatocytesAnwar Anwar-Mohamed, Lars-Oliver Klotz and Ayman O. S. El-KadiDrug Metabolism and Disposition March 2012, 40 (3) 504-514; DOI: https://doi.org/10.1124/dmd.111.042564
Kunne, Cindy
- You have accessOral Availability of Cefadroxil Depends on ABCC3 and ABCC4Dirk R. de Waart, Koen van de Wetering, Cindy Kunne, Suzanne Duijst, Coen C. Paulusma and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition March 2012, 40 (3) 515-521; DOI: https://doi.org/10.1124/dmd.111.041731
Kunze, Kent L.
- You have accessStereospecific Metabolism of Itraconazole by CYP3A4: Dioxolane Ring Scission of Azole AntifungalsChi-Chi Peng, Wei Shi, Justin D. Lutz, Kent L. Kunze, Jun O. Liu, Wendel L. Nelson and Nina IsoherranenDrug Metabolism and Disposition March 2012, 40 (3) 426-435; DOI: https://doi.org/10.1124/dmd.111.042739
Kuusela, Erja
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
L
Lämmer, Marc
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
Li, Liang
- You have accessMetabolism and Pharmacokinetics of Morinidazole in Humans: Identification of Diastereoisomeric Morpholine N+-Glucuronides Catalyzed by UDP Glucuronosyltransferase 1A9Ruina Gao, Liang Li, Cen Xie, Xingxing Diao, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition March 2012, 40 (3) 556-567; DOI: https://doi.org/10.1124/dmd.111.042689
Li, Wei
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
Liang, Sicheng
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Liras, Jennifer
- You have accessExcretion, Metabolism, and Pharmacokinetics of 1-(8-(2-Chlorophenyl)-9-(4-Chlorophenyl)-9H-Purin-6-yl)-4-(Ethylamino)Piperidine-4-Carboxamide, a Selective Cannabinoid Receptor Antagonist, in Healthy Male VolunteersZhuang Miao, Hao Sun, Jennifer Liras and Chandra PrakashDrug Metabolism and Disposition March 2012, 40 (3) 568-578; DOI: https://doi.org/10.1124/dmd.111.043273
Liu, Huixin
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Liu, Jun O.
- You have accessStereospecific Metabolism of Itraconazole by CYP3A4: Dioxolane Ring Scission of Azole AntifungalsChi-Chi Peng, Wei Shi, Justin D. Lutz, Kent L. Kunze, Jun O. Liu, Wendel L. Nelson and Nina IsoherranenDrug Metabolism and Disposition March 2012, 40 (3) 426-435; DOI: https://doi.org/10.1124/dmd.111.042739
Lu, Ding
- You have accessTrapping of cis-2-Butene-1,4-dial to Measure Furan Metabolism in Human Liver Microsomes by Cytochrome P450 EnzymesLeah A. Gates, Ding Lu and Lisa A. PetersonDrug Metabolism and Disposition March 2012, 40 (3) 596-601; DOI: https://doi.org/10.1124/dmd.111.043679
Lütjohann, Dieter
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
Lutz, Justin D.
- You have accessStereospecific Metabolism of Itraconazole by CYP3A4: Dioxolane Ring Scission of Azole AntifungalsChi-Chi Peng, Wei Shi, Justin D. Lutz, Kent L. Kunze, Jun O. Liu, Wendel L. Nelson and Nina IsoherranenDrug Metabolism and Disposition March 2012, 40 (3) 426-435; DOI: https://doi.org/10.1124/dmd.111.042739
M
Maeda, Kazuya
- You have accessIn Vivo Biliary Clearance Should Be Predicted by Intrinsic Biliary Clearance in Sandwich-Cultured HepatocytesMasanori Nakakariya, Midori Ono, Nobuyuki Amano, Toshiya Moriwaki, Kazuya Maeda and Yuichi SugiyamaDrug Metabolism and Disposition March 2012, 40 (3) 602-609; DOI: https://doi.org/10.1124/dmd.111.042101
Martin, L. A.
- You have accessPolychlorinated Biphenyl Congeners that Increase the Glucuronidation and Biliary Excretion of Thyroxine Are Distinct from the Congeners that Enhance the Serum Disappearance of ThyroxineL. A. Martin, D. T. Wilson, K. R. Reuhl, M. A. Gallo and C. D. KlaassenDrug Metabolism and Disposition March 2012, 40 (3) 588-595; DOI: https://doi.org/10.1124/dmd.111.042796
Melchior, Katja
- You have accessThe Effects of Rosuvastatin and the CYP51A1 Inhibitor LEK-935 on the Proteome of Primary Human HepatocytesMartin Wörner, Katja Melchior, Katalin Monostory, Jean-Marc Pascussi, Christian G. Huber and Rita BernhardtDrug Metabolism and Disposition March 2012, 40 (3) 414-418; DOI: https://doi.org/10.1124/dmd.111.040402
Miao, Zhuang
- You have accessExcretion, Metabolism, and Pharmacokinetics of 1-(8-(2-Chlorophenyl)-9-(4-Chlorophenyl)-9H-Purin-6-yl)-4-(Ethylamino)Piperidine-4-Carboxamide, a Selective Cannabinoid Receptor Antagonist, in Healthy Male VolunteersZhuang Miao, Hao Sun, Jennifer Liras and Chandra PrakashDrug Metabolism and Disposition March 2012, 40 (3) 568-578; DOI: https://doi.org/10.1124/dmd.111.043273
Monostory, Katalin
- You have accessThe Effects of Rosuvastatin and the CYP51A1 Inhibitor LEK-935 on the Proteome of Primary Human HepatocytesMartin Wörner, Katja Melchior, Katalin Monostory, Jean-Marc Pascussi, Christian G. Huber and Rita BernhardtDrug Metabolism and Disposition March 2012, 40 (3) 414-418; DOI: https://doi.org/10.1124/dmd.111.040402
Morgan, Edward T.
- You have accessEditorialEdward T. Morgan,Drug Metabolism and Disposition March 2012, 40 (3) 413; DOI: https://doi.org/10.1124/dmd.111.000009
Moriwaki, Toshiya
- You have accessIn Vivo Biliary Clearance Should Be Predicted by Intrinsic Biliary Clearance in Sandwich-Cultured HepatocytesMasanori Nakakariya, Midori Ono, Nobuyuki Amano, Toshiya Moriwaki, Kazuya Maeda and Yuichi SugiyamaDrug Metabolism and Disposition March 2012, 40 (3) 602-609; DOI: https://doi.org/10.1124/dmd.111.042101
Mueller, Juergen
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
N
Nadai, Masayuki
- You have accessChanges in Expression of Drug-Metabolizing Enzymes by Single-Walled Carbon Nanotubes in Human Respiratory Tract CellsKotaro Hitoshi, Miki Katoh, Tomoko Suzuki, Yoshinori Ando and Masayuki NadaiDrug Metabolism and Disposition March 2012, 40 (3) 579-587; DOI: https://doi.org/10.1124/dmd.111.043455
Nakakariya, Masanori
- You have accessIn Vivo Biliary Clearance Should Be Predicted by Intrinsic Biliary Clearance in Sandwich-Cultured HepatocytesMasanori Nakakariya, Midori Ono, Nobuyuki Amano, Toshiya Moriwaki, Kazuya Maeda and Yuichi SugiyamaDrug Metabolism and Disposition March 2012, 40 (3) 602-609; DOI: https://doi.org/10.1124/dmd.111.042101
Nelson, Wendel L.
- You have accessStereospecific Metabolism of Itraconazole by CYP3A4: Dioxolane Ring Scission of Azole AntifungalsChi-Chi Peng, Wei Shi, Justin D. Lutz, Kent L. Kunze, Jun O. Liu, Wendel L. Nelson and Nina IsoherranenDrug Metabolism and Disposition March 2012, 40 (3) 426-435; DOI: https://doi.org/10.1124/dmd.111.042739
Nguyen, Minh N.
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
O
Obach, R. Scott
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Ono, Midori
- You have accessIn Vivo Biliary Clearance Should Be Predicted by Intrinsic Biliary Clearance in Sandwich-Cultured HepatocytesMasanori Nakakariya, Midori Ono, Nobuyuki Amano, Toshiya Moriwaki, Kazuya Maeda and Yuichi SugiyamaDrug Metabolism and Disposition March 2012, 40 (3) 602-609; DOI: https://doi.org/10.1124/dmd.111.042101
Oswald, Stefan
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
Oude Elferink, Ronald P. J.
- You have accessOral Availability of Cefadroxil Depends on ABCC3 and ABCC4Dirk R. de Waart, Koen van de Wetering, Cindy Kunne, Suzanne Duijst, Coen C. Paulusma and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition March 2012, 40 (3) 515-521; DOI: https://doi.org/10.1124/dmd.111.041731
P
Pascussi, Jean-Marc
- You have accessThe Effects of Rosuvastatin and the CYP51A1 Inhibitor LEK-935 on the Proteome of Primary Human HepatocytesMartin Wörner, Katja Melchior, Katalin Monostory, Jean-Marc Pascussi, Christian G. Huber and Rita BernhardtDrug Metabolism and Disposition March 2012, 40 (3) 414-418; DOI: https://doi.org/10.1124/dmd.111.040402
Patyna, Shem
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
Paulusma, Coen C.
- You have accessOral Availability of Cefadroxil Depends on ABCC3 and ABCC4Dirk R. de Waart, Koen van de Wetering, Cindy Kunne, Suzanne Duijst, Coen C. Paulusma and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition March 2012, 40 (3) 515-521; DOI: https://doi.org/10.1124/dmd.111.041731
Pelis, Ryan M.
- You have accessExpression of Organic Anion Transporter 2 in the Human Kidney and Its Potential Role in the Tubular Secretion of Guanine-Containing Antiviral DrugsYaofeng Cheng, Arpine Vapurcuyan, Mohammad Shahidullah, Lauren M. Aleksunes and Ryan M. PelisDrug Metabolism and Disposition March 2012, 40 (3) 617-624; DOI: https://doi.org/10.1124/dmd.111.042036
Peng, Chi-Chi
- You have accessStereospecific Metabolism of Itraconazole by CYP3A4: Dioxolane Ring Scission of Azole AntifungalsChi-Chi Peng, Wei Shi, Justin D. Lutz, Kent L. Kunze, Jun O. Liu, Wendel L. Nelson and Nina IsoherranenDrug Metabolism and Disposition March 2012, 40 (3) 426-435; DOI: https://doi.org/10.1124/dmd.111.042739
Peng, Geoffrey W.
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
Peters, Jette
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
Peterson, Lisa A.
- You have accessTrapping of cis-2-Butene-1,4-dial to Measure Furan Metabolism in Human Liver Microsomes by Cytochrome P450 EnzymesLeah A. Gates, Ding Lu and Lisa A. PetersonDrug Metabolism and Disposition March 2012, 40 (3) 596-601; DOI: https://doi.org/10.1124/dmd.111.043679
Pool, William F.
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
Prakash, Chandra
- You have accessExcretion, Metabolism, and Pharmacokinetics of 1-(8-(2-Chlorophenyl)-9-(4-Chlorophenyl)-9H-Purin-6-yl)-4-(Ethylamino)Piperidine-4-Carboxamide, a Selective Cannabinoid Receptor Antagonist, in Healthy Male VolunteersZhuang Miao, Hao Sun, Jennifer Liras and Chandra PrakashDrug Metabolism and Disposition March 2012, 40 (3) 568-578; DOI: https://doi.org/10.1124/dmd.111.043273
R
Raekallio, Marja
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
Ranta-Panula, Ville
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
Restitutti, Flavia
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
Reuhl, K. R.
- You have accessPolychlorinated Biphenyl Congeners that Increase the Glucuronidation and Biliary Excretion of Thyroxine Are Distinct from the Congeners that Enhance the Serum Disappearance of ThyroxineL. A. Martin, D. T. Wilson, K. R. Reuhl, M. A. Gallo and C. D. KlaassenDrug Metabolism and Disposition March 2012, 40 (3) 588-595; DOI: https://doi.org/10.1124/dmd.111.042796
Rinne, Valtteri
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
Ripp, Sharon L.
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
S
Salla, Kati
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
Sandel, Jan
- You have accessInvestigation of Figopitant and Its Metabolites in Rat Tissue by Combining Whole-Body Autoradiography with Liquid Extraction Surface Analysis Mass SpectrometrySimone Schadt, Susanne Kallbach, Reinaldo Almeida and Jan SandelDrug Metabolism and Disposition March 2012, 40 (3) 419-425; DOI: https://doi.org/10.1124/dmd.111.043562
Sato, Kimihiko
- You have accessUnimolecular and Bimolecular Binding System for the Prediction of CYP2D6-Mediated MetabolismKimihiko Sato and Yasushi YamazoeDrug Metabolism and Disposition March 2012, 40 (3) 486-496; DOI: https://doi.org/10.1124/dmd.111.043125
Schadt, Simone
- You have accessInvestigation of Figopitant and Its Metabolites in Rat Tissue by Combining Whole-Body Autoradiography with Liquid Extraction Surface Analysis Mass SpectrometrySimone Schadt, Susanne Kallbach, Reinaldo Almeida and Jan SandelDrug Metabolism and Disposition March 2012, 40 (3) 419-425; DOI: https://doi.org/10.1124/dmd.111.043562
Scheinin, Mika
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
Schildknegt, Klaas
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Shahidullah, Mohammad
- You have accessExpression of Organic Anion Transporter 2 in the Human Kidney and Its Potential Role in the Tubular Secretion of Guanine-Containing Antiviral DrugsYaofeng Cheng, Arpine Vapurcuyan, Mohammad Shahidullah, Lauren M. Aleksunes and Ryan M. PelisDrug Metabolism and Disposition March 2012, 40 (3) 617-624; DOI: https://doi.org/10.1124/dmd.111.042036
Sharma, Raman
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Shi, Wei
- You have accessStereospecific Metabolism of Itraconazole by CYP3A4: Dioxolane Ring Scission of Azole AntifungalsChi-Chi Peng, Wei Shi, Justin D. Lutz, Kent L. Kunze, Jun O. Liu, Wendel L. Nelson and Nina IsoherranenDrug Metabolism and Disposition March 2012, 40 (3) 426-435; DOI: https://doi.org/10.1124/dmd.111.042739
Shinagawa, Akira
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
Siegmund, Werner
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
Slominski, Andrzej T.
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
Speed, Bill
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
Spracklin, Douglas K.
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Street, Stephanie M.
- You have accessMolecular Mechanism of Altered Ezetimibe Disposition in Nonalcoholic SteatohepatitisRhiannon N. Hardwick, Craig D. Fisher, Stephanie M. Street, Mark J. Canet and Nathan J. CherringtonDrug Metabolism and Disposition March 2012, 40 (3) 450-460; DOI: https://doi.org/10.1124/dmd.111.041095
Strelevitz, Timothy J.
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Sugiyama, Yuichi
- You have accessIn Vivo Biliary Clearance Should Be Predicted by Intrinsic Biliary Clearance in Sandwich-Cultured HepatocytesMasanori Nakakariya, Midori Ono, Nobuyuki Amano, Toshiya Moriwaki, Kazuya Maeda and Yuichi SugiyamaDrug Metabolism and Disposition March 2012, 40 (3) 602-609; DOI: https://doi.org/10.1124/dmd.111.042101
Sun, Hao
- You have accessExcretion, Metabolism, and Pharmacokinetics of 1-(8-(2-Chlorophenyl)-9-(4-Chlorophenyl)-9H-Purin-6-yl)-4-(Ethylamino)Piperidine-4-Carboxamide, a Selective Cannabinoid Receptor Antagonist, in Healthy Male VolunteersZhuang Miao, Hao Sun, Jennifer Liras and Chandra PrakashDrug Metabolism and Disposition March 2012, 40 (3) 568-578; DOI: https://doi.org/10.1124/dmd.111.043273
Suzuki, Tomoko
- You have accessChanges in Expression of Drug-Metabolizing Enzymes by Single-Walled Carbon Nanotubes in Human Respiratory Tract CellsKotaro Hitoshi, Miki Katoh, Tomoko Suzuki, Yoshinori Ando and Masayuki NadaiDrug Metabolism and Disposition March 2012, 40 (3) 579-587; DOI: https://doi.org/10.1124/dmd.111.043455
T
Tahara, Harunobu
- You have accessInvestigation of Drug-Drug Interactions Caused by Human Pregnane X Receptor-Mediated Induction of CYP3A4 and CYP2C Subfamilies in Chimeric Mice with a Humanized LiverMaki Hasegawa, Harunobu Tahara, Ryo Inoue, Masakazu Kakuni, Chise Tateno and Junko UshikiDrug Metabolism and Disposition March 2012, 40 (3) 474-480; DOI: https://doi.org/10.1124/dmd.111.042754
Takasaki, Wataru
- You have accessEvaluation of Hepatic Glutathione Transferase Mu 1 and Theta 1 Activities in Humans and Mice Using Genotype InformationShingo Arakawa, Kazunori Fujimoto, Ayako Kato, Seiko Endo, Aiko Fukahori, Akira Shinagawa, Thomas Fischer, Juergen Mueller and Wataru TakasakiDrug Metabolism and Disposition March 2012, 40 (3) 497-503; DOI: https://doi.org/10.1124/dmd.111.042911
Tateno, Chise
- You have accessInvestigation of Drug-Drug Interactions Caused by Human Pregnane X Receptor-Mediated Induction of CYP3A4 and CYP2C Subfamilies in Chimeric Mice with a Humanized LiverMaki Hasegawa, Harunobu Tahara, Ryo Inoue, Masakazu Kakuni, Chise Tateno and Junko UshikiDrug Metabolism and Disposition March 2012, 40 (3) 474-480; DOI: https://doi.org/10.1124/dmd.111.042754
Thomas, Paul E.
- You have accessInhibition of Genistein Glucuronidation by Bisphenol A in Human and Rat Liver MicrosomesJanis L. Coughlin, Paul E. Thomas and Brian BuckleyDrug Metabolism and Disposition March 2012, 40 (3) 481-485; DOI: https://doi.org/10.1124/dmd.111.042366
Thummel, Kenneth E.
- You have accessComplex Drug Interactions of the HIV Protease Inhibitors 3: Effect of Simultaneous or Staggered Dosing of Digoxin and Ritonavir, Nelfinavir, Rifampin, or BupropionBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition March 2012, 40 (3) 610-616; DOI: https://doi.org/10.1124/dmd.111.042705
Tieu, Elaine W.
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
Tingle, Malcolm D.
- You have accessWhich CYP2B6 Variants Have Functional Consequences for Cyclophosphamide Bioactivation?Nuala A. Helsby and Malcolm D. TingleDrug Metabolism and Disposition March 2012, 40 (3) 635-637; DOI: https://doi.org/10.1124/dmd.111.043646
Tremaine, Larry M.
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Tuckey, Robert C.
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
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Unadkat, Jashvant D.
- You have accessComplex Drug Interactions of the HIV Protease Inhibitors 3: Effect of Simultaneous or Staggered Dosing of Digoxin and Ritonavir, Nelfinavir, Rifampin, or BupropionBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition March 2012, 40 (3) 610-616; DOI: https://doi.org/10.1124/dmd.111.042705
Ushiki, Junko
- You have accessInvestigation of Drug-Drug Interactions Caused by Human Pregnane X Receptor-Mediated Induction of CYP3A4 and CYP2C Subfamilies in Chimeric Mice with a Humanized LiverMaki Hasegawa, Harunobu Tahara, Ryo Inoue, Masakazu Kakuni, Chise Tateno and Junko UshikiDrug Metabolism and Disposition March 2012, 40 (3) 474-480; DOI: https://doi.org/10.1124/dmd.111.042754
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Vainio, Outi
- You have accessInfluence of MK-467, a Peripherally Acting α2-Adrenoceptor Antagonist on the Disposition of Intravenous Dexmedetomidine in DogsJuhana Honkavaara, Flavia Restitutti, Marja Raekallio, Kati Salla, Erja Kuusela, Ville Ranta-Panula, Valtteri Rinne, Outi Vainio and Mika ScheininDrug Metabolism and Disposition March 2012, 40 (3) 445-449; DOI: https://doi.org/10.1124/dmd.111.042671
van de Wetering, Koen
- You have accessOral Availability of Cefadroxil Depends on ABCC3 and ABCC4Dirk R. de Waart, Koen van de Wetering, Cindy Kunne, Suzanne Duijst, Coen C. Paulusma and Ronald P. J. Oude ElferinkDrug Metabolism and Disposition March 2012, 40 (3) 515-521; DOI: https://doi.org/10.1124/dmd.111.041731
Vapurcuyan, Arpine
- You have accessExpression of Organic Anion Transporter 2 in the Human Kidney and Its Potential Role in the Tubular Secretion of Guanine-Containing Antiviral DrugsYaofeng Cheng, Arpine Vapurcuyan, Mohammad Shahidullah, Lauren M. Aleksunes and Ryan M. PelisDrug Metabolism and Disposition March 2012, 40 (3) 617-624; DOI: https://doi.org/10.1124/dmd.111.042036
Vaz, Alfin D. N.
- You have accessDeuterium Isotope Effects on Drug Pharmacokinetics. I. System-Dependent Effects of Specific Deuteration with Aldehyde Oxidase Cleared DrugsRaman Sharma, Timothy J. Strelevitz, Hongying Gao, Alan J. Clark, Klaas Schildknegt, R. Scott Obach, Sharon L. Ripp, Douglas K. Spracklin, Larry M. Tremaine and Alfin D. N. VazDrug Metabolism and Disposition March 2012, 40 (3) 625-634; DOI: https://doi.org/10.1124/dmd.111.042770
Venner, Monica
- You have accessClarithromycin Is Absorbed by an Intestinal Uptake Mechanism That Is Sensitive to Major Inhibition by Rifampicin: Results of a Short-Term Drug Interaction Study in FoalsJette Peters, Karen Eggers, Stefan Oswald, Wiebke Block, Dieter Lütjohann, Marc Lämmer, Monica Venner and Werner SiegmundDrug Metabolism and Disposition March 2012, 40 (3) 522-528; DOI: https://doi.org/10.1124/dmd.111.042267
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Whittington, Dale
- You have accessComplex Drug Interactions of the HIV Protease Inhibitors 3: Effect of Simultaneous or Staggered Dosing of Digoxin and Ritonavir, Nelfinavir, Rifampin, or BupropionBrian J. Kirby, Ann C. Collier, Evan D. Kharasch, Dale Whittington, Kenneth E. Thummel and Jashvant D. UnadkatDrug Metabolism and Disposition March 2012, 40 (3) 610-616; DOI: https://doi.org/10.1124/dmd.111.042705
Wilson, D. T.
- You have accessPolychlorinated Biphenyl Congeners that Increase the Glucuronidation and Biliary Excretion of Thyroxine Are Distinct from the Congeners that Enhance the Serum Disappearance of ThyroxineL. A. Martin, D. T. Wilson, K. R. Reuhl, M. A. Gallo and C. D. KlaassenDrug Metabolism and Disposition March 2012, 40 (3) 588-595; DOI: https://doi.org/10.1124/dmd.111.042796
Wörner, Martin
- You have accessThe Effects of Rosuvastatin and the CYP51A1 Inhibitor LEK-935 on the Proteome of Primary Human HepatocytesMartin Wörner, Katja Melchior, Katalin Monostory, Jean-Marc Pascussi, Christian G. Huber and Rita BernhardtDrug Metabolism and Disposition March 2012, 40 (3) 414-418; DOI: https://doi.org/10.1124/dmd.111.040402
Wu, Ellen Y.
- You have accessPharmacokinetics, Distribution, and Metabolism of [14C]Sunitinib in Rats, Monkeys, and HumansBill Speed, Hai-Zhi Bu, William F. Pool, Geoffrey W. Peng, Ellen Y. Wu, Shem Patyna, Carlo Bello and Ping KangDrug Metabolism and Disposition March 2012, 40 (3) 539-555; DOI: https://doi.org/10.1124/dmd.111.042853
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Xie, Cen
- You have accessMetabolism and Pharmacokinetics of Morinidazole in Humans: Identification of Diastereoisomeric Morpholine N+-Glucuronides Catalyzed by UDP Glucuronosyltransferase 1A9Ruina Gao, Liang Li, Cen Xie, Xingxing Diao, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition March 2012, 40 (3) 556-567; DOI: https://doi.org/10.1124/dmd.111.042689
Y
Yamazoe, Yasushi
- You have accessUnimolecular and Bimolecular Binding System for the Prediction of CYP2D6-Mediated MetabolismKimihiko Sato and Yasushi YamazoeDrug Metabolism and Disposition March 2012, 40 (3) 486-496; DOI: https://doi.org/10.1124/dmd.111.043125
Yang, Ling
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Z
Zhang, Hongbo
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Zhang, Yanyan
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Zhong, Dafang
- You have accessMetabolism and Pharmacokinetics of Morinidazole in Humans: Identification of Diastereoisomeric Morpholine N+-Glucuronides Catalyzed by UDP Glucuronosyltransferase 1A9Ruina Gao, Liang Li, Cen Xie, Xingxing Diao, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition March 2012, 40 (3) 556-567; DOI: https://doi.org/10.1124/dmd.111.042689
Zhu, Liangliang
- You have accessCharacterization of Hepatic and Intestinal Glucuronidation of Magnolol: Application of the Relative Activity Factor Approach to Decipher the Contributions of Multiple UDP-Glucuronosyltransferase IsoformsLiangliang Zhu, Guangbo Ge, Hongbo Zhang, Huixin Liu, Guiyuan He, Sicheng Liang, Yanyan Zhang, Zhongze Fang, Peipei Dong, Moshe Finel and Ling YangDrug Metabolism and Disposition March 2012, 40 (3) 529-538; DOI: https://doi.org/10.1124/dmd.111.042192
Zientek, Michael
- You have accessUse of a Multistaged Time-Dependent Inhibition Assay to Assess the Impact of Intestinal Metabolism on Drug-Drug Interaction PotentialMichael Zientek and Deepak DalvieDrug Metabolism and Disposition March 2012, 40 (3) 467-473; DOI: https://doi.org/10.1124/dmd.111.043257
Zjawiony, Jordan K.
- You have accessHuman Cytochrome P450scc (CYP11A1) Catalyzes Epoxide Formation with ErgosterolRobert C. Tuckey, Minh N. Nguyen, Jianjun Chen, Andrzej T. Slominski, Donna M. Baldisseri, Elaine W. Tieu, Jordan K. Zjawiony and Wei LiDrug Metabolism and Disposition March 2012, 40 (3) 436-444; DOI: https://doi.org/10.1124/dmd.111.042515
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