Index by author
January 01, 2013; Volume 41,Issue 1
A
Aasa, Jenny
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
Abad-Santos, Francisco
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
Agarwal, Sagar
- You have accessFunction of the Blood-Brain Barrier and Restriction of Drug Delivery to Invasive Glioma Cells: Findings in an Orthotopic Rat Xenograft Model of GliomaSagar Agarwal, Pooja Manchanda, Michael A. Vogelbaum, John R. Ohlfest and William F. ElmquistDrug Metabolism and Disposition January 2013, 41 (1) 33-39; DOI: https://doi.org/10.1124/dmd.112.048322
Akamine, Yumiko
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
Alhonen, Leena
- You have accessMetabolism of Triethylenetetramine and 1,12-Diamino-3,6,9-Triazadodecane by the Spermidine/Spermine-N1-Acetyltransferase and Thialysine AcetyltransferaseMervi T. Hyvönen, Janne Weisell, Alex R. Khomutov, Leena Alhonen, Jouko Vepsäläinen and Tuomo A. KeinänenDrug Metabolism and Disposition January 2013, 41 (1) 30-32; DOI: https://doi.org/10.1124/dmd.112.047274
Alsina, Melissa
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Anderson, Erica R.
- You have accessDifferential Influences of Ethanol on Early Exposure to Racemic Methylphenidate Compared with Dexmethylphenidate in HumansKennerly S. Patrick, Arthur B. Straughn, Owen T. Reeves, Hilary Bernstein, Guinevere H. Bell, Erica R. Anderson and Robert J. MalcolmDrug Metabolism and Disposition January 2013, 41 (1) 197-205; DOI: https://doi.org/10.1124/dmd.112.048595
B
Backman, Janne T.
- You have accessAutoinhibition of CYP3A4 Leads to Important Role of CYP2C8 in Imatinib Metabolism: Variability in CYP2C8 Activity May Alter Plasma Concentrations and ResponseAnne M. Filppula, Mikko Neuvonen, Jouko Laitila, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2013, 41 (1) 50-59; DOI: https://doi.org/10.1124/dmd.112.048017
Badros, Ashraf
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Bal, Jo
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Baranczewski, Pawel
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
Barr, John T.
- You have accessEvidence for Substrate-Dependent Inhibition Profiles for Human Liver Aldehyde OxidaseJohn T. Barr and Jeffrey P. JonesDrug Metabolism and Disposition January 2013, 41 (1) 24-29; DOI: https://doi.org/10.1124/dmd.112.048546
Beaumont, Claire
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Bell, Guinevere H.
- You have accessDifferential Influences of Ethanol on Early Exposure to Racemic Methylphenidate Compared with Dexmethylphenidate in HumansKennerly S. Patrick, Arthur B. Straughn, Owen T. Reeves, Hilary Bernstein, Guinevere H. Bell, Erica R. Anderson and Robert J. MalcolmDrug Metabolism and Disposition January 2013, 41 (1) 197-205; DOI: https://doi.org/10.1124/dmd.112.048595
Bernstein, Hilary
- You have accessDifferential Influences of Ethanol on Early Exposure to Racemic Methylphenidate Compared with Dexmethylphenidate in HumansKennerly S. Patrick, Arthur B. Straughn, Owen T. Reeves, Hilary Bernstein, Guinevere H. Bell, Erica R. Anderson and Robert J. MalcolmDrug Metabolism and Disposition January 2013, 41 (1) 197-205; DOI: https://doi.org/10.1124/dmd.112.048595
Berry, Loren M.
- You have accessImpact of Hydrolysis-Mediated Clearance on the Pharmacokinetics of Novel Anaplastic Lymphoma Kinase InhibitorsYohannes Teffera, Loren M. Berry, Rachael L. Brake, Richard T. Lewis, Douglas C. Saffran, Earl Moore, Jingzhou Liu and Zhiyang ZhaoDrug Metabolism and Disposition January 2013, 41 (1) 238-247; DOI: https://doi.org/10.1124/dmd.112.047993
Bjelland, Thor Wilhelm
- You have accessEffects of Hypothermia on the Disposition of Morphine, Midazolam, Fentanyl, and Propofol in Intensive Care Unit PatientsThor Wilhelm Bjelland, Pål Klepstad, Bjørn Olav Haugen, Turid Nilsen and Ola DaleDrug Metabolism and Disposition January 2013, 41 (1) 214-223; DOI: https://doi.org/10.1124/dmd.112.045567
Bomba, Darrin
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Bottlaender, Michel
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Brake, Rachael L.
- You have accessImpact of Hydrolysis-Mediated Clearance on the Pharmacokinetics of Novel Anaplastic Lymphoma Kinase InhibitorsYohannes Teffera, Loren M. Berry, Rachael L. Brake, Richard T. Lewis, Douglas C. Saffran, Earl Moore, Jingzhou Liu and Zhiyang ZhaoDrug Metabolism and Disposition January 2013, 41 (1) 238-247; DOI: https://doi.org/10.1124/dmd.112.047993
Brouwer, Kim L. R.
- You have accessCombination Lopinavir and Ritonavir Alter Exogenous and Endogenous Bile Acid Disposition in Sandwich-Cultured Rat HepatocytesLaToya M. Griffin, Paul B. Watkins, Cassandra H. Perry, Robert L. St. Claire and Kim L. R. BrouwerDrug Metabolism and Disposition January 2013, 41 (1) 188-196; DOI: https://doi.org/10.1124/dmd.112.047225
Bueters, Tjerk
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
Bushey, Ryan T.
- You have accessImportance of UDP-Glucuronosyltransferases 2A2 and 2A3 in Tobacco Carcinogen MetabolismRyan T. Bushey, Douglas F. Dluzen and Philip LazarusDrug Metabolism and Disposition January 2013, 41 (1) 170-179; DOI: https://doi.org/10.1124/dmd.112.049171
C
Cabaleiro, Teresa
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
Chen, Chi
- You have accessCharacterization of Differential Cocaine Metabolism in Mouse and Rat through Metabolomics-Guided Metabolite ProfilingDan Yao, Xiaolei Shi, Lei Wang, Blake A. Gosnell and Chi ChenDrug Metabolism and Disposition January 2013, 41 (1) 79-88; DOI: https://doi.org/10.1124/dmd.112.048678
Chen, Li
- You have accessDiscovery and Characterization of Novel, Potent, and Selective Cytochrome P450 2J2 InhibitorsShuang Ren, Juan Zeng, Ye Mei, John Z. H. Zhang, S. Frank Yan, Jian Fei and Li ChenDrug Metabolism and Disposition January 2013, 41 (1) 60-71; DOI: https://doi.org/10.1124/dmd.112.048264
Chiang, John Y. L.
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
D
Dale, Ola
- You have accessEffects of Hypothermia on the Disposition of Morphine, Midazolam, Fentanyl, and Propofol in Intensive Care Unit PatientsThor Wilhelm Bjelland, Pål Klepstad, Bjørn Olav Haugen, Turid Nilsen and Ola DaleDrug Metabolism and Disposition January 2013, 41 (1) 214-223; DOI: https://doi.org/10.1124/dmd.112.045567
Dalton, James T.
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Damont, Annelaure
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Ding, Xinxin
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
- You have accessGeneration and Characterization of a Novel Cyp2a(4/5)bgs-Null Mouse ModelYuan Wei, Lei Li, Xin Zhou, Qing-Yu Zhang, Anwar Dunbar, Fang Liu, Kerri Kluetzman, Weizhu Yang and Xinxin DingDrug Metabolism and Disposition January 2013, 41 (1) 132-140; DOI: https://doi.org/10.1124/dmd.112.048736
Distrutti, Eleonora
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Dluzen, Douglas F.
- You have accessImportance of UDP-Glucuronosyltransferases 2A2 and 2A3 in Tobacco Carcinogen MetabolismRyan T. Bushey, Douglas F. Dluzen and Philip LazarusDrug Metabolism and Disposition January 2013, 41 (1) 170-179; DOI: https://doi.org/10.1124/dmd.112.049171
Dollé, Frédéric
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Dunbar, Anwar
- You have accessGeneration and Characterization of a Novel Cyp2a(4/5)bgs-Null Mouse ModelYuan Wei, Lei Li, Xin Zhou, Qing-Yu Zhang, Anwar Dunbar, Fang Liu, Kerri Kluetzman, Weizhu Yang and Xinxin DingDrug Metabolism and Disposition January 2013, 41 (1) 132-140; DOI: https://doi.org/10.1124/dmd.112.048736
E
Ebner, Thomas
- You have accessEvaluation and Prediction of Potential Drug-Drug Interactions of Linagliptin Using In Vitro Cell Culture MethodsNaoki Ishiguro, Hidetada Shimizu, Wataru Kishimoto, Thomas Ebner and Olaf SchaeferDrug Metabolism and Disposition January 2013, 41 (1) 149-158; DOI: https://doi.org/10.1124/dmd.112.048470
Eklund, Göran
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
Elmquist, William F.
- You have accessFunction of the Blood-Brain Barrier and Restriction of Drug Delivery to Invasive Glioma Cells: Findings in an Orthotopic Rat Xenograft Model of GliomaSagar Agarwal, Pooja Manchanda, Michael A. Vogelbaum, John R. Ohlfest and William F. ElmquistDrug Metabolism and Disposition January 2013, 41 (1) 33-39; DOI: https://doi.org/10.1124/dmd.112.048322
Emmons, Amanda J.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
F
Fang, Ying
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Fei, Jian
- You have accessDiscovery and Characterization of Novel, Potent, and Selective Cytochrome P450 2J2 InhibitorsShuang Ren, Juan Zeng, Ye Mei, John Z. H. Zhang, S. Frank Yan, Jian Fei and Li ChenDrug Metabolism and Disposition January 2013, 41 (1) 60-71; DOI: https://doi.org/10.1124/dmd.112.048264
Felgate, Clive C.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Filppula, Anne M.
- You have accessAutoinhibition of CYP3A4 Leads to Important Role of CYP2C8 in Imatinib Metabolism: Variability in CYP2C8 Activity May Alter Plasma Concentrations and ResponseAnne M. Filppula, Mikko Neuvonen, Jouko Laitila, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2013, 41 (1) 50-59; DOI: https://doi.org/10.1124/dmd.112.048017
Finn, Robert D.
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Fiorucci, Stefano
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Flück, Christa E.
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Fukizawa, Shinya
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
G
Gosnell, Blake A.
- You have accessCharacterization of Differential Cocaine Metabolism in Mouse and Rat through Metabolomics-Guided Metabolite ProfilingDan Yao, Xiaolei Shi, Lei Wang, Blake A. Gosnell and Chi ChenDrug Metabolism and Disposition January 2013, 41 (1) 79-88; DOI: https://doi.org/10.1124/dmd.112.048678
Goutal, Sébastien
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Griffin, LaToya M.
- You have accessCombination Lopinavir and Ritonavir Alter Exogenous and Endogenous Bile Acid Disposition in Sandwich-Cultured Rat HepatocytesLaToya M. Griffin, Paul B. Watkins, Cassandra H. Perry, Robert L. St. Claire and Kim L. R. BrouwerDrug Metabolism and Disposition January 2013, 41 (1) 188-196; DOI: https://doi.org/10.1124/dmd.112.047225
Grillo, Mark P.
- You have accessInteraction of γ-Glutamyltranspeptidase with Ibuprofen-S-Acyl-Glutathione In Vitro and In Vivo in HumanMark P. Grillo, Michelle Tadano Lohr and Smriti KheraDrug Metabolism and Disposition January 2013, 41 (1) 111-121; DOI: https://doi.org/10.1124/dmd.112.048645
Gu, Jun
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Guo, Grace L.
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
H
Harrell, Andrew W.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Haugen, Bjørn Olav
- You have accessEffects of Hypothermia on the Disposition of Morphine, Midazolam, Fentanyl, and Propofol in Intensive Care Unit PatientsThor Wilhelm Bjelland, Pål Klepstad, Bjørn Olav Haugen, Turid Nilsen and Ola DaleDrug Metabolism and Disposition January 2013, 41 (1) 214-223; DOI: https://doi.org/10.1124/dmd.112.045567
Henderson, Colin J.
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Hollenberg, Paul F.
- You have accessInteractions between CYP2E1 and CYP2B4: Effects on Affinity for NADPH-Cytochrome P450 Reductase and Substrate MetabolismCesar Kenaan, Erin V. Shea, Hsia-lien Lin, Haoming Zhang, Matthew J. Pratt-Hyatt and Paul F. HollenbergDrug Metabolism and Disposition January 2013, 41 (1) 101-110; DOI: https://doi.org/10.1124/dmd.112.046094
Hu, Yin
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
Hyvönen, Mervi T.
- You have accessMetabolism of Triethylenetetramine and 1,12-Diamino-3,6,9-Triazadodecane by the Spermidine/Spermine-N1-Acetyltransferase and Thialysine AcetyltransferaseMervi T. Hyvönen, Janne Weisell, Alex R. Khomutov, Leena Alhonen, Jouko Vepsäläinen and Tuomo A. KeinänenDrug Metabolism and Disposition January 2013, 41 (1) 30-32; DOI: https://doi.org/10.1124/dmd.112.047274
I
Ikejiri, Kazuaki
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
Imai, Satoki
- You have accessDNA Methylation and Histone Modification Profiles of Mouse Organic Anion Transporting PolypeptidesSatoki Imai, Ryota Kikuchi, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 72-78; DOI: https://doi.org/10.1124/dmd.112.047969
Imai, Teruko
- You have accessPharmacokinetic Mechanism Involved in the Prolonged High Retention of Laninamivir in Mouse Respiratory Tissues after Intranasal Administration of its Prodrug Laninamivir OctanoateKumiko Koyama, Daisuke Nakai, Makoto Takahashi, Naoko Nakai, Nobuhiro Kobayashi, Teruko Imai and Takashi IzumiDrug Metabolism and Disposition January 2013, 41 (1) 180-187; DOI: https://doi.org/10.1124/dmd.112.048280
Infante, Jeffrey R.
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Ishiguro, Naoki
- You have accessEvaluation and Prediction of Potential Drug-Drug Interactions of Linagliptin Using In Vitro Cell Culture MethodsNaoki Ishiguro, Hidetada Shimizu, Wataru Kishimoto, Thomas Ebner and Olaf SchaeferDrug Metabolism and Disposition January 2013, 41 (1) 149-158; DOI: https://doi.org/10.1124/dmd.112.048470
Izumi, Takashi
- You have accessPharmacokinetic Mechanism Involved in the Prolonged High Retention of Laninamivir in Mouse Respiratory Tissues after Intranasal Administration of its Prodrug Laninamivir OctanoateKumiko Koyama, Daisuke Nakai, Makoto Takahashi, Naoko Nakai, Nobuhiro Kobayashi, Teruko Imai and Takashi IzumiDrug Metabolism and Disposition January 2013, 41 (1) 180-187; DOI: https://doi.org/10.1124/dmd.112.048280
J
Jones, Jeffrey P.
- You have accessEvidence for Substrate-Dependent Inhibition Profiles for Human Liver Aldehyde OxidaseJohn T. Barr and Jeffrey P. JonesDrug Metabolism and Disposition January 2013, 41 (1) 24-29; DOI: https://doi.org/10.1124/dmd.112.048546
Jones, Ryan D.
- You have accessCarboxylesterases Are Uniquely Expressed among Tissues and Regulated by Nuclear Hormone Receptors in the MouseRyan D. Jones, Anna M. Taylor, Ernest Y. Tong and Joyce J. RepaDrug Metabolism and Disposition January 2013, 41 (1) 40-49; DOI: https://doi.org/10.1124/dmd.112.048397
K
Kagan, Leonid
- You have accessMechanisms of Subcutaneous Absorption of Rituximab in RatsLeonid Kagan and Donald E. MagerDrug Metabolism and Disposition January 2013, 41 (1) 248-255; DOI: https://doi.org/10.1124/dmd.112.048496
Kanamitsu, Kayoko
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
Kassiou, Michael
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Keinänen, Tuomo A.
- You have accessMetabolism of Triethylenetetramine and 1,12-Diamino-3,6,9-Triazadodecane by the Spermidine/Spermine-N1-Acetyltransferase and Thialysine AcetyltransferaseMervi T. Hyvönen, Janne Weisell, Alex R. Khomutov, Leena Alhonen, Jouko Vepsäläinen and Tuomo A. KeinänenDrug Metabolism and Disposition January 2013, 41 (1) 30-32; DOI: https://doi.org/10.1124/dmd.112.047274
Kempsford, Rodger D.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Kenaan, Cesar
- You have accessInteractions between CYP2E1 and CYP2B4: Effects on Affinity for NADPH-Cytochrome P450 Reductase and Substrate MetabolismCesar Kenaan, Erin V. Shea, Hsia-lien Lin, Haoming Zhang, Matthew J. Pratt-Hyatt and Paul F. HollenbergDrug Metabolism and Disposition January 2013, 41 (1) 101-110; DOI: https://doi.org/10.1124/dmd.112.046094
Khera, Smriti
- You have accessInteraction of γ-Glutamyltranspeptidase with Ibuprofen-S-Acyl-Glutathione In Vitro and In Vivo in HumanMark P. Grillo, Michelle Tadano Lohr and Smriti KheraDrug Metabolism and Disposition January 2013, 41 (1) 111-121; DOI: https://doi.org/10.1124/dmd.112.048645
Khomutov, Alex R.
- You have accessMetabolism of Triethylenetetramine and 1,12-Diamino-3,6,9-Triazadodecane by the Spermidine/Spermine-N1-Acetyltransferase and Thialysine AcetyltransferaseMervi T. Hyvönen, Janne Weisell, Alex R. Khomutov, Leena Alhonen, Jouko Vepsäläinen and Tuomo A. KeinänenDrug Metabolism and Disposition January 2013, 41 (1) 30-32; DOI: https://doi.org/10.1124/dmd.112.047274
Kikuchi, Ryota
- You have accessDNA Methylation and Histone Modification Profiles of Mouse Organic Anion Transporting PolypeptidesSatoki Imai, Ryota Kikuchi, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 72-78; DOI: https://doi.org/10.1124/dmd.112.047969
Kirk, Christopher
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Kishimoto, Wataru
- You have accessEvaluation and Prediction of Potential Drug-Drug Interactions of Linagliptin Using In Vitro Cell Culture MethodsNaoki Ishiguro, Hidetada Shimizu, Wataru Kishimoto, Thomas Ebner and Olaf SchaeferDrug Metabolism and Disposition January 2013, 41 (1) 149-158; DOI: https://doi.org/10.1124/dmd.112.048470
Klepstad, Pål
- You have accessEffects of Hypothermia on the Disposition of Morphine, Midazolam, Fentanyl, and Propofol in Intensive Care Unit PatientsThor Wilhelm Bjelland, Pål Klepstad, Bjørn Olav Haugen, Turid Nilsen and Ola DaleDrug Metabolism and Disposition January 2013, 41 (1) 214-223; DOI: https://doi.org/10.1124/dmd.112.045567
Kluetzman, Kerri
- You have accessGeneration and Characterization of a Novel Cyp2a(4/5)bgs-Null Mouse ModelYuan Wei, Lei Li, Xin Zhou, Qing-Yu Zhang, Anwar Dunbar, Fang Liu, Kerri Kluetzman, Weizhu Yang and Xinxin DingDrug Metabolism and Disposition January 2013, 41 (1) 132-140; DOI: https://doi.org/10.1124/dmd.112.048736
Kobayashi, Nobuhiro
- You have accessPharmacokinetic Mechanism Involved in the Prolonged High Retention of Laninamivir in Mouse Respiratory Tissues after Intranasal Administration of its Prodrug Laninamivir OctanoateKumiko Koyama, Daisuke Nakai, Makoto Takahashi, Naoko Nakai, Nobuhiro Kobayashi, Teruko Imai and Takashi IzumiDrug Metabolism and Disposition January 2013, 41 (1) 180-187; DOI: https://doi.org/10.1124/dmd.112.048280
Kong, Bo
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Koyama, Kumiko
- You have accessPharmacokinetic Mechanism Involved in the Prolonged High Retention of Laninamivir in Mouse Respiratory Tissues after Intranasal Administration of its Prodrug Laninamivir OctanoateKumiko Koyama, Daisuke Nakai, Makoto Takahashi, Naoko Nakai, Nobuhiro Kobayashi, Teruko Imai and Takashi IzumiDrug Metabolism and Disposition January 2013, 41 (1) 180-187; DOI: https://doi.org/10.1124/dmd.112.048280
Kusuhara, Hiroyuki
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
- You have accessDNA Methylation and Histone Modification Profiles of Mouse Organic Anion Transporting PolypeptidesSatoki Imai, Ryota Kikuchi, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 72-78; DOI: https://doi.org/10.1124/dmd.112.047969
L
Laitila, Jouko
- You have accessAutoinhibition of CYP3A4 Leads to Important Role of CYP2C8 in Imatinib Metabolism: Variability in CYP2C8 Activity May Alter Plasma Concentrations and ResponseAnne M. Filppula, Mikko Neuvonen, Jouko Laitila, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2013, 41 (1) 50-59; DOI: https://doi.org/10.1124/dmd.112.048017
Lazarus, Philip
- You have accessImportance of UDP-Glucuronosyltransferases 2A2 and 2A3 in Tobacco Carcinogen MetabolismRyan T. Bushey, Douglas F. Dluzen and Philip LazarusDrug Metabolism and Disposition January 2013, 41 (1) 170-179; DOI: https://doi.org/10.1124/dmd.112.049171
Lewis, Richard T.
- You have accessImpact of Hydrolysis-Mediated Clearance on the Pharmacokinetics of Novel Anaplastic Lymphoma Kinase InhibitorsYohannes Teffera, Loren M. Berry, Rachael L. Brake, Richard T. Lewis, Douglas C. Saffran, Earl Moore, Jingzhou Liu and Zhiyang ZhaoDrug Metabolism and Disposition January 2013, 41 (1) 238-247; DOI: https://doi.org/10.1124/dmd.112.047993
Li, Jin
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Li, Lei
- You have accessGeneration and Characterization of a Novel Cyp2a(4/5)bgs-Null Mouse ModelYuan Wei, Lei Li, Xin Zhou, Qing-Yu Zhang, Anwar Dunbar, Fang Liu, Kerri Kluetzman, Weizhu Yang and Xinxin DingDrug Metabolism and Disposition January 2013, 41 (1) 132-140; DOI: https://doi.org/10.1124/dmd.112.048736
Lin, Hsia-lien
- You have accessInteractions between CYP2E1 and CYP2B4: Effects on Affinity for NADPH-Cytochrome P450 Reductase and Substrate MetabolismCesar Kenaan, Erin V. Shea, Hsia-lien Lin, Haoming Zhang, Matthew J. Pratt-Hyatt and Paul F. HollenbergDrug Metabolism and Disposition January 2013, 41 (1) 101-110; DOI: https://doi.org/10.1124/dmd.112.046094
Lindgren, Anders
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
Liu, Fang
- You have accessGeneration and Characterization of a Novel Cyp2a(4/5)bgs-Null Mouse ModelYuan Wei, Lei Li, Xin Zhou, Qing-Yu Zhang, Anwar Dunbar, Fang Liu, Kerri Kluetzman, Weizhu Yang and Xinxin DingDrug Metabolism and Disposition January 2013, 41 (1) 132-140; DOI: https://doi.org/10.1124/dmd.112.048736
Liu, Jingzhou
- You have accessImpact of Hydrolysis-Mediated Clearance on the Pharmacokinetics of Novel Anaplastic Lymphoma Kinase InhibitorsYohannes Teffera, Loren M. Berry, Rachael L. Brake, Richard T. Lewis, Douglas C. Saffran, Earl Moore, Jingzhou Liu and Zhiyang ZhaoDrug Metabolism and Disposition January 2013, 41 (1) 238-247; DOI: https://doi.org/10.1124/dmd.112.047993
Lohr, Michelle Tadano
- You have accessInteraction of γ-Glutamyltranspeptidase with Ibuprofen-S-Acyl-Glutathione In Vitro and In Vivo in HumanMark P. Grillo, Michelle Tadano Lohr and Smriti KheraDrug Metabolism and Disposition January 2013, 41 (1) 111-121; DOI: https://doi.org/10.1124/dmd.112.048645
López-Rodríguez, Rosario
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
M
Mager, Donald E.
- You have accessMechanisms of Subcutaneous Absorption of Rituximab in RatsLeonid Kagan and Donald E. MagerDrug Metabolism and Disposition January 2013, 41 (1) 248-255; DOI: https://doi.org/10.1124/dmd.112.048496
Malcolm, Robert J.
- You have accessDifferential Influences of Ethanol on Early Exposure to Racemic Methylphenidate Compared with Dexmethylphenidate in HumansKennerly S. Patrick, Arthur B. Straughn, Owen T. Reeves, Hilary Bernstein, Guinevere H. Bell, Erica R. Anderson and Robert J. MalcolmDrug Metabolism and Disposition January 2013, 41 (1) 197-205; DOI: https://doi.org/10.1124/dmd.112.048595
Malmquist, Jonas
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
Manchanda, Pooja
- You have accessFunction of the Blood-Brain Barrier and Restriction of Drug Delivery to Invasive Glioma Cells: Findings in an Orthotopic Rat Xenograft Model of GliomaSagar Agarwal, Pooja Manchanda, Michael A. Vogelbaum, John R. Ohlfest and William F. ElmquistDrug Metabolism and Disposition January 2013, 41 (1) 33-39; DOI: https://doi.org/10.1124/dmd.112.048322
Maruyama, Toru
- You have accessCarbon Monoxide–Bound Red Blood Cells Protect Red Blood Cell Transfusion-Induced Hepatic Cytochrome P450 Impairment in Hemorrhagic-Shock RatsShigeru Ogaki, Kazuaki Taguchi, Hiroshi Watanabe, Masaki Otagiri and Toru MaruyamaDrug Metabolism and Disposition January 2013, 41 (1) 141-148; DOI: https://doi.org/10.1124/dmd.112.048744
McLaughlin, Lesley A.
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Mei, Ye
- You have accessDiscovery and Characterization of Novel, Potent, and Selective Cytochrome P450 2J2 InhibitorsShuang Ren, Juan Zeng, Ye Mei, John Z. H. Zhang, S. Frank Yan, Jian Fei and Li ChenDrug Metabolism and Disposition January 2013, 41 (1) 60-71; DOI: https://doi.org/10.1124/dmd.112.048264
Miura, Masatomo
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
Moore, Earl
- You have accessImpact of Hydrolysis-Mediated Clearance on the Pharmacokinetics of Novel Anaplastic Lymphoma Kinase InhibitorsYohannes Teffera, Loren M. Berry, Rachael L. Brake, Richard T. Lewis, Douglas C. Saffran, Earl Moore, Jingzhou Liu and Zhiyang ZhaoDrug Metabolism and Disposition January 2013, 41 (1) 238-247; DOI: https://doi.org/10.1124/dmd.112.047993
N
Nakai, Daisuke
- You have accessPharmacokinetic Mechanism Involved in the Prolonged High Retention of Laninamivir in Mouse Respiratory Tissues after Intranasal Administration of its Prodrug Laninamivir OctanoateKumiko Koyama, Daisuke Nakai, Makoto Takahashi, Naoko Nakai, Nobuhiro Kobayashi, Teruko Imai and Takashi IzumiDrug Metabolism and Disposition January 2013, 41 (1) 180-187; DOI: https://doi.org/10.1124/dmd.112.048280
Nakai, Naoko
- You have accessPharmacokinetic Mechanism Involved in the Prolonged High Retention of Laninamivir in Mouse Respiratory Tissues after Intranasal Administration of its Prodrug Laninamivir OctanoateKumiko Koyama, Daisuke Nakai, Makoto Takahashi, Naoko Nakai, Nobuhiro Kobayashi, Teruko Imai and Takashi IzumiDrug Metabolism and Disposition January 2013, 41 (1) 180-187; DOI: https://doi.org/10.1124/dmd.112.048280
Narayanan, Ramesh
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Neuvonen, Mikko
- You have accessAutoinhibition of CYP3A4 Leads to Important Role of CYP2C8 in Imatinib Metabolism: Variability in CYP2C8 Activity May Alter Plasma Concentrations and ResponseAnne M. Filppula, Mikko Neuvonen, Jouko Laitila, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2013, 41 (1) 50-59; DOI: https://doi.org/10.1124/dmd.112.048017
Neuvonen, Pertti J.
- You have accessAutoinhibition of CYP3A4 Leads to Important Role of CYP2C8 in Imatinib Metabolism: Variability in CYP2C8 Activity May Alter Plasma Concentrations and ResponseAnne M. Filppula, Mikko Neuvonen, Jouko Laitila, Pertti J. Neuvonen and Janne T. BackmanDrug Metabolism and Disposition January 2013, 41 (1) 50-59; DOI: https://doi.org/10.1124/dmd.112.048017
Nilsen, Turid
- You have accessEffects of Hypothermia on the Disposition of Morphine, Midazolam, Fentanyl, and Propofol in Intensive Care Unit PatientsThor Wilhelm Bjelland, Pål Klepstad, Bjørn Olav Haugen, Turid Nilsen and Ola DaleDrug Metabolism and Disposition January 2013, 41 (1) 214-223; DOI: https://doi.org/10.1124/dmd.112.045567
Novalbos, Jesús
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
O
Ochoa, Dolores
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
Ogaki, Shigeru
- You have accessCarbon Monoxide–Bound Red Blood Cells Protect Red Blood Cell Transfusion-Induced Hepatic Cytochrome P450 Impairment in Hemorrhagic-Shock RatsShigeru Ogaki, Kazuaki Taguchi, Hiroshi Watanabe, Masaki Otagiri and Toru MaruyamaDrug Metabolism and Disposition January 2013, 41 (1) 141-148; DOI: https://doi.org/10.1124/dmd.112.048744
Ohlfest, John R.
- You have accessFunction of the Blood-Brain Barrier and Restriction of Drug Delivery to Invasive Glioma Cells: Findings in an Orthotopic Rat Xenograft Model of GliomaSagar Agarwal, Pooja Manchanda, Michael A. Vogelbaum, John R. Ohlfest and William F. ElmquistDrug Metabolism and Disposition January 2013, 41 (1) 33-39; DOI: https://doi.org/10.1124/dmd.112.048322
Otagiri, Masaki
- You have accessCarbon Monoxide–Bound Red Blood Cells Protect Red Blood Cell Transfusion-Induced Hepatic Cytochrome P450 Impairment in Hemorrhagic-Shock RatsShigeru Ogaki, Kazuaki Taguchi, Hiroshi Watanabe, Masaki Otagiri and Toru MaruyamaDrug Metabolism and Disposition January 2013, 41 (1) 141-148; DOI: https://doi.org/10.1124/dmd.112.048744
P
Pandey, Amit V.
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Papadopoulos, Kyriakos
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Patel, Nainesh H.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Patrick, Kennerly S.
- You have accessDifferential Influences of Ethanol on Early Exposure to Racemic Methylphenidate Compared with Dexmethylphenidate in HumansKennerly S. Patrick, Arthur B. Straughn, Owen T. Reeves, Hilary Bernstein, Guinevere H. Bell, Erica R. Anderson and Robert J. MalcolmDrug Metabolism and Disposition January 2013, 41 (1) 197-205; DOI: https://doi.org/10.1124/dmd.112.048595
Pearce, Sebastian J.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Pereira, Adrian I.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Perry, Cassandra H.
- You have accessCombination Lopinavir and Ritonavir Alter Exogenous and Endogenous Bile Acid Disposition in Sandwich-Cultured Rat HepatocytesLaToya M. Griffin, Paul B. Watkins, Cassandra H. Perry, Robert L. St. Claire and Kim L. R. BrouwerDrug Metabolism and Disposition January 2013, 41 (1) 188-196; DOI: https://doi.org/10.1124/dmd.112.047225
Peyronneau, Marie-Anne
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Porter, Todd D.
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Pratt-Hyatt, Matthew J.
- You have accessInteractions between CYP2E1 and CYP2B4: Effects on Affinity for NADPH-Cytochrome P450 Reductase and Substrate MetabolismCesar Kenaan, Erin V. Shea, Hsia-lien Lin, Haoming Zhang, Matthew J. Pratt-Hyatt and Paul F. HollenbergDrug Metabolism and Disposition January 2013, 41 (1) 101-110; DOI: https://doi.org/10.1124/dmd.112.046094
Prieto-Pérez, Rocío
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
R
Reeves, Owen T.
- You have accessDifferential Influences of Ethanol on Early Exposure to Racemic Methylphenidate Compared with Dexmethylphenidate in HumansKennerly S. Patrick, Arthur B. Straughn, Owen T. Reeves, Hilary Bernstein, Guinevere H. Bell, Erica R. Anderson and Robert J. MalcolmDrug Metabolism and Disposition January 2013, 41 (1) 197-205; DOI: https://doi.org/10.1124/dmd.112.048595
Ren, Shuang
- You have accessDiscovery and Characterization of Novel, Potent, and Selective Cytochrome P450 2J2 InhibitorsShuang Ren, Juan Zeng, Ye Mei, John Z. H. Zhang, S. Frank Yan, Jian Fei and Li ChenDrug Metabolism and Disposition January 2013, 41 (1) 60-71; DOI: https://doi.org/10.1124/dmd.112.048264
Renga, Barbara
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Repa, Joyce J.
- You have accessCarboxylesterases Are Uniquely Expressed among Tissues and Regulated by Nuclear Hormone Receptors in the MouseRyan D. Jones, Anna M. Taylor, Ernest Y. Tong and Joyce J. RepaDrug Metabolism and Disposition January 2013, 41 (1) 40-49; DOI: https://doi.org/10.1124/dmd.112.048397
Riddick, David S.
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Roberts, Andy D.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Román, Manuel
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
Ronseaux, Sebastien
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
S
Saba, Wadad
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Saffran, Douglas C.
- You have accessImpact of Hydrolysis-Mediated Clearance on the Pharmacokinetics of Novel Anaplastic Lymphoma Kinase InhibitorsYohannes Teffera, Loren M. Berry, Rachael L. Brake, Richard T. Lewis, Douglas C. Saffran, Earl Moore, Jingzhou Liu and Zhiyang ZhaoDrug Metabolism and Disposition January 2013, 41 (1) 238-247; DOI: https://doi.org/10.1124/dmd.112.047993
Schaefer, Olaf
- You have accessEvaluation and Prediction of Potential Drug-Drug Interactions of Linagliptin Using In Vitro Cell Culture MethodsNaoki Ishiguro, Hidetada Shimizu, Wataru Kishimoto, Thomas Ebner and Olaf SchaeferDrug Metabolism and Disposition January 2013, 41 (1) 149-158; DOI: https://doi.org/10.1124/dmd.112.048470
Shea, Erin V.
- You have accessInteractions between CYP2E1 and CYP2B4: Effects on Affinity for NADPH-Cytochrome P450 Reductase and Substrate MetabolismCesar Kenaan, Erin V. Shea, Hsia-lien Lin, Haoming Zhang, Matthew J. Pratt-Hyatt and Paul F. HollenbergDrug Metabolism and Disposition January 2013, 41 (1) 101-110; DOI: https://doi.org/10.1124/dmd.112.046094
Shi, Xiaolei
- You have accessCharacterization of Differential Cocaine Metabolism in Mouse and Rat through Metabolomics-Guided Metabolite ProfilingDan Yao, Xiaolei Shi, Lei Wang, Blake A. Gosnell and Chi ChenDrug Metabolism and Disposition January 2013, 41 (1) 79-88; DOI: https://doi.org/10.1124/dmd.112.048678
Shimizu, Hidetada
- You have accessEvaluation and Prediction of Potential Drug-Drug Interactions of Linagliptin Using In Vitro Cell Culture MethodsNaoki Ishiguro, Hidetada Shimizu, Wataru Kishimoto, Thomas Ebner and Olaf SchaeferDrug Metabolism and Disposition January 2013, 41 (1) 149-158; DOI: https://doi.org/10.1124/dmd.112.048470
Siederer, Sarah K.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
St. Claire, Robert L.
- You have accessCombination Lopinavir and Ritonavir Alter Exogenous and Endogenous Bile Acid Disposition in Sandwich-Cultured Rat HepatocytesLaToya M. Griffin, Paul B. Watkins, Cassandra H. Perry, Robert L. St. Claire and Kim L. R. BrouwerDrug Metabolism and Disposition January 2013, 41 (1) 188-196; DOI: https://doi.org/10.1124/dmd.112.047225
Straughn, Arthur B.
- You have accessDifferential Influences of Ethanol on Early Exposure to Racemic Methylphenidate Compared with Dexmethylphenidate in HumansKennerly S. Patrick, Arthur B. Straughn, Owen T. Reeves, Hilary Bernstein, Guinevere H. Bell, Erica R. Anderson and Robert J. MalcolmDrug Metabolism and Disposition January 2013, 41 (1) 197-205; DOI: https://doi.org/10.1124/dmd.112.048595
Sugiyama, Yuichi
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
- You have accessDNA Methylation and Histone Modification Profiles of Mouse Organic Anion Transporting PolypeptidesSatoki Imai, Ryota Kikuchi, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 72-78; DOI: https://doi.org/10.1124/dmd.112.047969
Swanson, Hollie I.
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
T
Taguchi, Kazuaki
- You have accessCarbon Monoxide–Bound Red Blood Cells Protect Red Blood Cell Transfusion-Induced Hepatic Cytochrome P450 Impairment in Hemorrhagic-Shock RatsShigeru Ogaki, Kazuaki Taguchi, Hiroshi Watanabe, Masaki Otagiri and Toru MaruyamaDrug Metabolism and Disposition January 2013, 41 (1) 141-148; DOI: https://doi.org/10.1124/dmd.112.048744
Takahashi, Makoto
- You have accessPharmacokinetic Mechanism Involved in the Prolonged High Retention of Laninamivir in Mouse Respiratory Tissues after Intranasal Administration of its Prodrug Laninamivir OctanoateKumiko Koyama, Daisuke Nakai, Makoto Takahashi, Naoko Nakai, Nobuhiro Kobayashi, Teruko Imai and Takashi IzumiDrug Metabolism and Disposition January 2013, 41 (1) 180-187; DOI: https://doi.org/10.1124/dmd.112.048280
Talegón, María
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
Taylor, Anna M.
- You have accessCarboxylesterases Are Uniquely Expressed among Tissues and Regulated by Nuclear Hormone Receptors in the MouseRyan D. Jones, Anna M. Taylor, Ernest Y. Tong and Joyce J. RepaDrug Metabolism and Disposition January 2013, 41 (1) 40-49; DOI: https://doi.org/10.1124/dmd.112.048397
Teffera, Yohannes
- You have accessImpact of Hydrolysis-Mediated Clearance on the Pharmacokinetics of Novel Anaplastic Lymphoma Kinase InhibitorsYohannes Teffera, Loren M. Berry, Rachael L. Brake, Richard T. Lewis, Douglas C. Saffran, Earl Moore, Jingzhou Liu and Zhiyang ZhaoDrug Metabolism and Disposition January 2013, 41 (1) 238-247; DOI: https://doi.org/10.1124/dmd.112.047993
Thomas, Ann M.
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Tong, Ernest Y.
- You have accessCarboxylesterases Are Uniquely Expressed among Tissues and Regulated by Nuclear Hormone Receptors in the MouseRyan D. Jones, Anna M. Taylor, Ernest Y. Tong and Joyce J. RepaDrug Metabolism and Disposition January 2013, 41 (1) 40-49; DOI: https://doi.org/10.1124/dmd.112.048397
Turek, Dominika
- You have accessEffect of Solvents on the Time-Dependent Inhibition of CYP3A4 and the Biotransformation of AZD3839 in Human Liver Microsomes and HepatocytesJenny Aasa, Yin Hu, Göran Eklund, Anders Lindgren, Pawel Baranczewski, Jonas Malmquist, Dominika Turek and Tjerk BuetersDrug Metabolism and Disposition January 2013, 41 (1) 159-169; DOI: https://doi.org/10.1124/dmd.112.047597
U
Uno, Tsukasa
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
V
Valette, Héric
- You have accessMetabolism and Quantification of [18F]DPA-714, a New TSPO Positron Emission Tomography RadioligandMarie-Anne Peyronneau, Wadad Saba, Sébastien Goutal, Annelaure Damont, Frédéric Dollé, Michael Kassiou, Michel Bottlaender and Héric ValetteDrug Metabolism and Disposition January 2013, 41 (1) 122-131; DOI: https://doi.org/10.1124/dmd.112.046342
Vepsäläinen, Jouko
- You have accessMetabolism of Triethylenetetramine and 1,12-Diamino-3,6,9-Triazadodecane by the Spermidine/Spermine-N1-Acetyltransferase and Thialysine AcetyltransferaseMervi T. Hyvönen, Janne Weisell, Alex R. Khomutov, Leena Alhonen, Jouko Vepsäläinen and Tuomo A. KeinänenDrug Metabolism and Disposition January 2013, 41 (1) 30-32; DOI: https://doi.org/10.1124/dmd.112.047274
Vogelbaum, Michael A.
- You have accessFunction of the Blood-Brain Barrier and Restriction of Drug Delivery to Invasive Glioma Cells: Findings in an Orthotopic Rat Xenograft Model of GliomaSagar Agarwal, Pooja Manchanda, Michael A. Vogelbaum, John R. Ohlfest and William F. ElmquistDrug Metabolism and Disposition January 2013, 41 (1) 33-39; DOI: https://doi.org/10.1124/dmd.112.048322
W
Wada, Taira
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Wang, Lei
- You have accessCharacterization of Differential Cocaine Metabolism in Mouse and Rat through Metabolomics-Guided Metabolite ProfilingDan Yao, Xiaolei Shi, Lei Wang, Blake A. Gosnell and Chi ChenDrug Metabolism and Disposition January 2013, 41 (1) 79-88; DOI: https://doi.org/10.1124/dmd.112.048678
Wang, Zhengping
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Watanabe, Hiroshi
- You have accessCarbon Monoxide–Bound Red Blood Cells Protect Red Blood Cell Transfusion-Induced Hepatic Cytochrome P450 Impairment in Hemorrhagic-Shock RatsShigeru Ogaki, Kazuaki Taguchi, Hiroshi Watanabe, Masaki Otagiri and Toru MaruyamaDrug Metabolism and Disposition January 2013, 41 (1) 141-148; DOI: https://doi.org/10.1124/dmd.112.048744
Watkins, Paul B.
- You have accessCombination Lopinavir and Ritonavir Alter Exogenous and Endogenous Bile Acid Disposition in Sandwich-Cultured Rat HepatocytesLaToya M. Griffin, Paul B. Watkins, Cassandra H. Perry, Robert L. St. Claire and Kim L. R. BrouwerDrug Metabolism and Disposition January 2013, 41 (1) 188-196; DOI: https://doi.org/10.1124/dmd.112.047225
Wei, Yuan
- You have accessGeneration and Characterization of a Novel Cyp2a(4/5)bgs-Null Mouse ModelYuan Wei, Lei Li, Xin Zhou, Qing-Yu Zhang, Anwar Dunbar, Fang Liu, Kerri Kluetzman, Weizhu Yang and Xinxin DingDrug Metabolism and Disposition January 2013, 41 (1) 132-140; DOI: https://doi.org/10.1124/dmd.112.048736
Weisell, Janne
- You have accessMetabolism of Triethylenetetramine and 1,12-Diamino-3,6,9-Triazadodecane by the Spermidine/Spermine-N1-Acetyltransferase and Thialysine AcetyltransferaseMervi T. Hyvönen, Janne Weisell, Alex R. Khomutov, Leena Alhonen, Jouko Vepsäläinen and Tuomo A. KeinänenDrug Metabolism and Disposition January 2013, 41 (1) 30-32; DOI: https://doi.org/10.1124/dmd.112.047274
Wojnicz, Aneta
- You have accessEvaluation of the Relationship between Sex, Polymorphisms in CYP2C8 and CYP2C9, and Pharmacokinetics of Angiotensin Receptor BlockersTeresa Cabaleiro, Manuel Román, Dolores Ochoa, María Talegón, Rocío Prieto-Pérez, Aneta Wojnicz, Rosario López-Rodríguez, Jesús Novalbos and Francisco Abad-SantosDrug Metabolism and Disposition January 2013, 41 (1) 224-229; DOI: https://doi.org/10.1124/dmd.112.046292
Wolf, C. Roland
- You have accessNADPH–Cytochrome P450 Oxidoreductase: Roles in Physiology, Pharmacology, and ToxicologyDavid S. Riddick, Xinxin Ding, C. Roland Wolf, Todd D. Porter, Amit V. Pandey, Qing-Yu Zhang, Jun Gu, Robert D. Finn, Sebastien Ronseaux, Lesley A. McLaughlin, Colin J. Henderson, Ling Zou and Christa E. FlückDrug Metabolism and Disposition January 2013, 41 (1) 12-23; DOI: https://doi.org/10.1124/dmd.112.048991
Wong, Alvin
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Woo, Tina
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
X
Xie, Wen
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Y
Yan, S. Frank
- You have accessDiscovery and Characterization of Novel, Potent, and Selective Cytochrome P450 2J2 InhibitorsShuang Ren, Juan Zeng, Ye Mei, John Z. H. Zhang, S. Frank Yan, Jian Fei and Li ChenDrug Metabolism and Disposition January 2013, 41 (1) 60-71; DOI: https://doi.org/10.1124/dmd.112.048264
Yang, Jinfu
- You have accessClinical Pharmacokinetics, Metabolism, and Drug-Drug Interaction of CarfilzomibZhengping Wang, Jinfu Yang, Christopher Kirk, Ying Fang, Melissa Alsina, Ashraf Badros, Kyriakos Papadopoulos, Alvin Wong, Tina Woo, Darrin Bomba, Jin Li and Jeffrey R. InfanteDrug Metabolism and Disposition January 2013, 41 (1) 230-237; DOI: https://doi.org/10.1124/dmd.112.047662
Yang, Weizhu
- You have accessGeneration and Characterization of a Novel Cyp2a(4/5)bgs-Null Mouse ModelYuan Wei, Lei Li, Xin Zhou, Qing-Yu Zhang, Anwar Dunbar, Fang Liu, Kerri Kluetzman, Weizhu Yang and Xinxin DingDrug Metabolism and Disposition January 2013, 41 (1) 132-140; DOI: https://doi.org/10.1124/dmd.112.048736
Yao, Dan
- You have accessCharacterization of Differential Cocaine Metabolism in Mouse and Rat through Metabolomics-Guided Metabolite ProfilingDan Yao, Xiaolei Shi, Lei Wang, Blake A. Gosnell and Chi ChenDrug Metabolism and Disposition January 2013, 41 (1) 79-88; DOI: https://doi.org/10.1124/dmd.112.048678
Yasui-Furukori, Norio
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
Yepuru, Muralimohan
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Yokochi, Miyu
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
Yoshida, Kenta
- You have accessEffect of Coadministration of Single and Multiple Doses of Rifampicin on the Pharmacokinetics of Fexofenadine Enantiomers in Healthy SubjectsHiroyuki Kusuhara, Masatomo Miura, Norio Yasui-Furukori, Kenta Yoshida, Yumiko Akamine, Miyu Yokochi, Shinya Fukizawa, Kazuaki Ikejiri, Kayoko Kanamitsu, Tsukasa Uno and Yuichi SugiyamaDrug Metabolism and Disposition January 2013, 41 (1) 206-213; DOI: https://doi.org/10.1124/dmd.112.048330
Young, Graeme C.
- You have accessMetabolism and Disposition of Vilanterol, a Long-Acting β2-Adrenoceptor Agonist for Inhalation Use in HumansAndrew W. Harrell, Sarah K. Siederer, Jo Bal, Nainesh H. Patel, Graeme C. Young, Clive C. Felgate, Sebastian J. Pearce, Andy D. Roberts, Claire Beaumont, Amanda J. Emmons, Adrian I. Pereira and Rodger D. KempsfordDrug Metabolism and Disposition January 2013, 41 (1) 89-100; DOI: https://doi.org/10.1124/dmd.112.048603
Z
Zampella, Angela
- You have accessRole of Nuclear Receptors in Lipid Dysfunction and Obesity-Related DiseasesHollie I. Swanson, Taira Wada, Wen Xie, Barbara Renga, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci, Bo Kong, Ann M. Thomas, Grace L. Guo, Ramesh Narayanan, Muralimohan Yepuru, James T. Dalton and John Y. L. ChiangDrug Metabolism and Disposition January 2013, 41 (1) 1-11; DOI: https://doi.org/10.1124/dmd.112.048694
Zeng, Juan
- You have accessDiscovery and Characterization of Novel, Potent, and Selective Cytochrome P450 2J2 InhibitorsShuang Ren, Juan Zeng, Ye Mei, John Z. H. Zhang, S. Frank Yan, Jian Fei and Li ChenDrug Metabolism and Disposition January 2013, 41 (1) 60-71; DOI: https://doi.org/10.1124/dmd.112.048264
Zhang, Haoming
- You have accessInteractions between CYP2E1 and CYP2B4: Effects on Affinity for NADPH-Cytochrome P450 Reductase and Substrate MetabolismCesar Kenaan, Erin V. Shea, Hsia-lien Lin, Haoming Zhang, Matthew J. Pratt-Hyatt and Paul F. HollenbergDrug Metabolism and Disposition January 2013, 41 (1) 101-110; DOI: https://doi.org/10.1124/dmd.112.046094
Zhang, John Z. H.
- You have accessDiscovery and Characterization of Novel, Potent, and Selective Cytochrome P450 2J2 InhibitorsShuang Ren, Juan Zeng, Ye Mei, John Z. H. Zhang, S. Frank Yan, Jian Fei and Li ChenDrug Metabolism and Disposition January 2013, 41 (1) 60-71; DOI: https://doi.org/10.1124/dmd.112.048264
Zhang, Qing-Yu
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