Research ArticleArticle
Pharmacokinetics, Metabolism, and Excretion of the Antidiabetic Agent Ertugliflozin (PF-04971729) in Healthy Male Subjects
Zhuang Miao, Gianluca Nucci, Neeta Amin, Raman Sharma, Vincent Mascitti, Meera Tugnait, Alfin D. Vaz, Ernesto Callegari and Amit S. Kalgutkar
Drug Metabolism and Disposition February 2013, 41 (2) 445-456; DOI: https://doi.org/10.1124/dmd.112.049551
Zhuang Miao
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Gianluca Nucci
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Neeta Amin
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Raman Sharma
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Vincent Mascitti
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Meera Tugnait
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Alfin D. Vaz
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Ernesto Callegari
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).
Amit S. Kalgutkar
Pharmacokinetics, Dynamics and Metabolism, New Chemical Entities, Groton, Connecticut (Z.M., R.S., M.T., A.D.V., E.C.) and Cambridge, Massachusetts (A.S.K.); Cardiovascular, Metabolic and Endocrine Diseases Research Unit (N.A.); Clinical Pharmacology, Cambridge, Massachusetts (G.N.); and Worldwide Medicinal Chemistry, Pfizer Inc., Groton, Connecticut (V.M.).

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Research ArticleArticle
Disposition of Ertugliflozin in Humans
Zhuang Miao, Gianluca Nucci, Neeta Amin, Raman Sharma, Vincent Mascitti, Meera Tugnait, Alfin D. Vaz, Ernesto Callegari and Amit S. Kalgutkar
Drug Metabolism and Disposition February 1, 2013, 41 (2) 445-456; DOI: https://doi.org/10.1124/dmd.112.049551
Research ArticleArticle
Disposition of Ertugliflozin in Humans
Zhuang Miao, Gianluca Nucci, Neeta Amin, Raman Sharma, Vincent Mascitti, Meera Tugnait, Alfin D. Vaz, Ernesto Callegari and Amit S. Kalgutkar
Drug Metabolism and Disposition February 1, 2013, 41 (2) 445-456; DOI: https://doi.org/10.1124/dmd.112.049551
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