Research ArticleArticle
Amide Hydrolysis of a Novel Chemical Series of Microsomal Prostaglandin E Synthase-1 Inhibitors Induces Kidney Toxicity in the Rat
Johan Bylund, Anita Annas, Dennis Hellgren, Sivert Bjurström, Håkan Andersson and Alexander Svanhagen
Drug Metabolism and Disposition March 2013, 41 (3) 634-641; DOI: https://doi.org/10.1124/dmd.112.048983
Johan Bylund
Drug Metabolism and Pharmacokinetics, CNSP iMed Science (J.B.), and Safety Assessment (A.A., D.H., S.B., H.A., A.S.), AstraZeneca R&D, Innovative Medicines, Södertälje, Sweden; and Department of Pharmaceutical Biosciences, Uppsala Biomedical Centre, Uppsala University, Uppsala, Sweden (J.B.)
Anita Annas
Drug Metabolism and Pharmacokinetics, CNSP iMed Science (J.B.), and Safety Assessment (A.A., D.H., S.B., H.A., A.S.), AstraZeneca R&D, Innovative Medicines, Södertälje, Sweden; and Department of Pharmaceutical Biosciences, Uppsala Biomedical Centre, Uppsala University, Uppsala, Sweden (J.B.)
Dennis Hellgren
Drug Metabolism and Pharmacokinetics, CNSP iMed Science (J.B.), and Safety Assessment (A.A., D.H., S.B., H.A., A.S.), AstraZeneca R&D, Innovative Medicines, Södertälje, Sweden; and Department of Pharmaceutical Biosciences, Uppsala Biomedical Centre, Uppsala University, Uppsala, Sweden (J.B.)
Sivert Bjurström
Drug Metabolism and Pharmacokinetics, CNSP iMed Science (J.B.), and Safety Assessment (A.A., D.H., S.B., H.A., A.S.), AstraZeneca R&D, Innovative Medicines, Södertälje, Sweden; and Department of Pharmaceutical Biosciences, Uppsala Biomedical Centre, Uppsala University, Uppsala, Sweden (J.B.)
Håkan Andersson
Drug Metabolism and Pharmacokinetics, CNSP iMed Science (J.B.), and Safety Assessment (A.A., D.H., S.B., H.A., A.S.), AstraZeneca R&D, Innovative Medicines, Södertälje, Sweden; and Department of Pharmaceutical Biosciences, Uppsala Biomedical Centre, Uppsala University, Uppsala, Sweden (J.B.)
Alexander Svanhagen
Drug Metabolism and Pharmacokinetics, CNSP iMed Science (J.B.), and Safety Assessment (A.A., D.H., S.B., H.A., A.S.), AstraZeneca R&D, Innovative Medicines, Södertälje, Sweden; and Department of Pharmaceutical Biosciences, Uppsala Biomedical Centre, Uppsala University, Uppsala, Sweden (J.B.)

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Research ArticleArticle
Amide Hydrolysis-Induced Kidney Toxicity
Johan Bylund, Anita Annas, Dennis Hellgren, Sivert Bjurström, Håkan Andersson and Alexander Svanhagen
Drug Metabolism and Disposition March 1, 2013, 41 (3) 634-641; DOI: https://doi.org/10.1124/dmd.112.048983
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