Research ArticleArticle
Pharmacokinetics, Metabolism, and Excretion of the Glycogen Synthase Kinase-3 Inhibitor LY2090314 in Rats, Dogs, and Humans: A Case Study in Rapid Clearance by Extensive Metabolism with Low Circulating Metabolite Exposure
Maciej J. Zamek-Gliszczynski, Trent L. Abraham, Jeffrey J. Alberts, Palaniappan Kulanthaivel, Kimberley A. Jackson, Kay H. Chow, Denis J. McCann, Haitao Hu, Shelby Anderson, Nathan A. Furr, Robert J. Barbuch and Kenneth C. Cassidy
Drug Metabolism and Disposition April 2013, 41 (4) 714-726; DOI: https://doi.org/10.1124/dmd.112.048488
Maciej J. Zamek-Gliszczynski
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Trent L. Abraham
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Jeffrey J. Alberts
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Palaniappan Kulanthaivel
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Kimberley A. Jackson
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Kay H. Chow
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Denis J. McCann
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Haitao Hu
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Shelby Anderson
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Nathan A. Furr
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Robert J. Barbuch
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
Kenneth C. Cassidy
Drug Disposition/Pharmacokinetics/Pharmacodynamics (M.J.Z.-G., T.L.A., J.J.A., P.K., K.A.J., K.H.C., D.J.M., S.A., N.A.F., R.J.B., K.C.C.), Discovery Chemistry and Research Technologies (H.H.), Lilly Research Laboratories, Indianapolis, Indiana
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Research ArticleArticle
PK, Metabolism, and Excretion of LY2090314
Maciej J. Zamek-Gliszczynski, Trent L. Abraham, Jeffrey J. Alberts, Palaniappan Kulanthaivel, Kimberley A. Jackson, Kay H. Chow, Denis J. McCann, Haitao Hu, Shelby Anderson, Nathan A. Furr, Robert J. Barbuch and Kenneth C. Cassidy
Drug Metabolism and Disposition April 1, 2013, 41 (4) 714-726; DOI: https://doi.org/10.1124/dmd.112.048488
Research ArticleArticle
PK, Metabolism, and Excretion of LY2090314
Maciej J. Zamek-Gliszczynski, Trent L. Abraham, Jeffrey J. Alberts, Palaniappan Kulanthaivel, Kimberley A. Jackson, Kay H. Chow, Denis J. McCann, Haitao Hu, Shelby Anderson, Nathan A. Furr, Robert J. Barbuch and Kenneth C. Cassidy
Drug Metabolism and Disposition April 1, 2013, 41 (4) 714-726; DOI: https://doi.org/10.1124/dmd.112.048488
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