Research ArticleArticle
Biotransformation of Two β-Secretase Inhibitors Including Ring Opening and Contraction of a Pyrimidine Ring
Anders Lindgren, Göran Eklund, Dominika Turek, Jonas Malmquist, Britt-Marie Swahn, Jörg Holenz, Stefan von Berg, Sofia Karlström and Tjerk Bueters
Drug Metabolism and Disposition May 2013, 41 (5) 1134-1147; DOI: https://doi.org/10.1124/dmd.112.050351
Anders Lindgren
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Göran Eklund
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Dominika Turek
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Jonas Malmquist
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Britt-Marie Swahn
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Jörg Holenz
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Stefan von Berg
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Sofia Karlström
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
Tjerk Bueters
Drug Metabolism and Pharmacokinetics (A.L., G.E., T.B.) and Medicinal Chemistry, Central Nervous System and Pain iMed Science (D.T., B.-M.S., J.H., S.v.B., S.K.), Medicinal Chemistry, Respiratory Inflammatory and Autoimmunity iMed Science (S.v.B.), and Global Drug Metabolism and Pharmacokinetics Screening and Profiling, AstraZeneca R&D (J.M.), Novandi Chemistry AB (J.M.), and MetaSafe AB (G.E.), Södertälje, Sweden
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Research ArticleArticle
Biotransformation of Pyrimidine Ring
Anders Lindgren, Göran Eklund, Dominika Turek, Jonas Malmquist, Britt-Marie Swahn, Jörg Holenz, Stefan von Berg, Sofia Karlström and Tjerk Bueters
Drug Metabolism and Disposition May 1, 2013, 41 (5) 1134-1147; DOI: https://doi.org/10.1124/dmd.112.050351
Research ArticleArticle
Biotransformation of Pyrimidine Ring
Anders Lindgren, Göran Eklund, Dominika Turek, Jonas Malmquist, Britt-Marie Swahn, Jörg Holenz, Stefan von Berg, Sofia Karlström and Tjerk Bueters
Drug Metabolism and Disposition May 1, 2013, 41 (5) 1134-1147; DOI: https://doi.org/10.1124/dmd.112.050351
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