Index by author
May 01, 2014; Volume 42,Issue 5
A
Álvarez, Ana I.
- You have accessRole of ABCG2 in Transport of the Mammalian Lignan Enterolactone and its Secretion into Milk in Abcg2 Knockout MiceVerónica Miguel, Jon Andoni Otero, Rocío García-Villalba, Francisco Tomás-Barberán, Juan Carlos Espín, Gracia Merino and Ana I. ÁlvarezDrug Metabolism and Disposition May 2014, 42 (5) 943-946; DOI: https://doi.org/10.1124/dmd.113.055970
Atherton, James
- You have accessAssessment of the Mass Balance Recovery and Metabolite Profile of Avibactam in Humans and In Vitro Drug-Drug Interaction PotentialKarthick Vishwanathan, Stuart Mair, Anshul Gupta, James Atherton, Jacqueline Clarkson-Jones, Timi Edeki and Shampa DasDrug Metabolism and Disposition May 2014, 42 (5) 932-942; DOI: https://doi.org/10.1124/dmd.113.055335
B
Ballard, T. Eric
- You have accessGeneration of Major Human Excretory and Circulating Drug Metabolites Using a Hepatocyte Relay MethodT. Eric Ballard, Christine C. Orozco and R. Scott ObachDrug Metabolism and Disposition May 2014, 42 (5) 899-902; DOI: https://doi.org/10.1124/dmd.114.057026
Bi, Huichang
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Bu, Hai-Zhi
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
C
Challinor, Victoria L.
- You have accessCarbon-Carbon Bond Cleavage in Activation of the Prodrug NabumetoneFatbardha Varfaj, Siti N. A. Zulkifli, Hyoung-Goo Park, Victoria L. Challinor, James J. De Voss and Paul R. Ortiz de MontellanoDrug Metabolism and Disposition May 2014, 42 (5) 828-838; DOI: https://doi.org/10.1124/dmd.114.056903
Chen, Dongquan
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
Chen, Jie
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Chen, Pan
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Chen, Xiaoyan
- You have accessMetabolism and Pharmacokinetics of Allitinib in Cancer Patients: The Roles of Cytochrome P450s and Epoxide Hydrolase in its BiotransformationLishan Lin, Cen Xie, Zhiwei Gao, Xiaoyan Chen and Dafang ZhongDrug Metabolism and Disposition May 2014, 42 (5) 872-884; DOI: https://doi.org/10.1124/dmd.113.056341
Clarkson-Jones, Jacqueline
- You have accessAssessment of the Mass Balance Recovery and Metabolite Profile of Avibactam in Humans and In Vitro Drug-Drug Interaction PotentialKarthick Vishwanathan, Stuart Mair, Anshul Gupta, James Atherton, Jacqueline Clarkson-Jones, Timi Edeki and Shampa DasDrug Metabolism and Disposition May 2014, 42 (5) 932-942; DOI: https://doi.org/10.1124/dmd.113.055335
Crittenden, Frank
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
Cuyckens, Filip
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
D
Dalvie, Deepak K.
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Das, Shampa
- You have accessAssessment of the Mass Balance Recovery and Metabolite Profile of Avibactam in Humans and In Vitro Drug-Drug Interaction PotentialKarthick Vishwanathan, Stuart Mair, Anshul Gupta, James Atherton, Jacqueline Clarkson-Jones, Timi Edeki and Shampa DasDrug Metabolism and Disposition May 2014, 42 (5) 932-942; DOI: https://doi.org/10.1124/dmd.113.055335
Deese, Alan
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Deese, Alan J.
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Deng, Rongrong
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Devineni, Damayanthi
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
De Voss, James J.
- You have accessCarbon-Carbon Bond Cleavage in Activation of the Prodrug NabumetoneFatbardha Varfaj, Siti N. A. Zulkifli, Hyoung-Goo Park, Victoria L. Challinor, James J. De Voss and Paul R. Ortiz de MontellanoDrug Metabolism and Disposition May 2014, 42 (5) 828-838; DOI: https://doi.org/10.1124/dmd.114.056903
Dixon, Russell
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
Dorko, Kenneth
- You have accessBedaquiline Metabolism: Enzymes and Novel MetabolitesKe Liu, Feng Li, Jie Lu, Shinlan Liu, Kenneth Dorko, Wen Xie and Xiaochao MaDrug Metabolism and Disposition May 2014, 42 (5) 863-866; DOI: https://doi.org/10.1124/dmd.113.056119
E
Edeki, Timi
- You have accessAssessment of the Mass Balance Recovery and Metabolite Profile of Avibactam in Humans and In Vitro Drug-Drug Interaction PotentialKarthick Vishwanathan, Stuart Mair, Anshul Gupta, James Atherton, Jacqueline Clarkson-Jones, Timi Edeki and Shampa DasDrug Metabolism and Disposition May 2014, 42 (5) 932-942; DOI: https://doi.org/10.1124/dmd.113.055335
Espín, Juan Carlos
- You have accessRole of ABCG2 in Transport of the Mammalian Lignan Enterolactone and its Secretion into Milk in Abcg2 Knockout MiceVerónica Miguel, Jon Andoni Otero, Rocío García-Villalba, Francisco Tomás-Barberán, Juan Carlos Espín, Gracia Merino and Ana I. ÁlvarezDrug Metabolism and Disposition May 2014, 42 (5) 943-946; DOI: https://doi.org/10.1124/dmd.113.055970
Ethen, Cheryl M.
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
Evans, David C.
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
F
Falany, Charles N.
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
Fan, Xiaomei
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Feng, Hao
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Ford, Kevin A.
- You have access1-Aminobenzotriazole Coincubated with (S)-Warfarin Results in Potent Inactivation of CYP2C9Jasleen K. Sodhi, Kevin A. Ford, Sophie Mukadam, Susan Wong, Cornelis E. C. A. Hop, S. Cyrus Khojasteh and Jason S. HalladayDrug Metabolism and Disposition May 2014, 42 (5) 813-817; DOI: https://doi.org/10.1124/dmd.113.055913
G
Gao, Zhiwei
- You have accessMetabolism and Pharmacokinetics of Allitinib in Cancer Patients: The Roles of Cytochrome P450s and Epoxide Hydrolase in its BiotransformationLishan Lin, Cen Xie, Zhiwei Gao, Xiaoyan Chen and Dafang ZhongDrug Metabolism and Disposition May 2014, 42 (5) 872-884; DOI: https://doi.org/10.1124/dmd.113.056341
García-Villalba, Rocío
- You have accessRole of ABCG2 in Transport of the Mammalian Lignan Enterolactone and its Secretion into Milk in Abcg2 Knockout MiceVerónica Miguel, Jon Andoni Otero, Rocío García-Villalba, Francisco Tomás-Barberán, Juan Carlos Espín, Gracia Merino and Ana I. ÁlvarezDrug Metabolism and Disposition May 2014, 42 (5) 943-946; DOI: https://doi.org/10.1124/dmd.113.055970
Gu, Zheming
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Gupta, Anshul
- You have accessAssessment of the Mass Balance Recovery and Metabolite Profile of Avibactam in Humans and In Vitro Drug-Drug Interaction PotentialKarthick Vishwanathan, Stuart Mair, Anshul Gupta, James Atherton, Jacqueline Clarkson-Jones, Timi Edeki and Shampa DasDrug Metabolism and Disposition May 2014, 42 (5) 932-942; DOI: https://doi.org/10.1124/dmd.113.055335
H
Halladay, Jason S.
- You have access1-Aminobenzotriazole Coincubated with (S)-Warfarin Results in Potent Inactivation of CYP2C9Jasleen K. Sodhi, Kevin A. Ford, Sophie Mukadam, Susan Wong, Cornelis E. C. A. Hop, S. Cyrus Khojasteh and Jason S. HalladayDrug Metabolism and Disposition May 2014, 42 (5) 813-817; DOI: https://doi.org/10.1124/dmd.113.055913
Han Hsu, Helen
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Hee, Brian
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Hop, Cornelis E. C. A.
- You have access1-Aminobenzotriazole Coincubated with (S)-Warfarin Results in Potent Inactivation of CYP2C9Jasleen K. Sodhi, Kevin A. Ford, Sophie Mukadam, Susan Wong, Cornelis E. C. A. Hop, S. Cyrus Khojasteh and Jason S. HalladayDrug Metabolism and Disposition May 2014, 42 (5) 813-817; DOI: https://doi.org/10.1124/dmd.113.055913
Hop, Cornelis E.C.A.
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Hu, Dong Gui
- You have accessPolymorphisms and Haplotypes of the UDP-Glucuronosyltransferase 2B7 Gene PromoterDong Gui Hu, Robyn Meech, Lu Lu, Ross A. McKinnon and Peter I. MackenzieDrug Metabolism and Disposition May 2014, 42 (5) 854-862; DOI: https://doi.org/10.1124/dmd.113.056630
Huang, Min
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Hunt, Kevin W.
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
I
Iwasaki, Kazuhide
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
J
Johnson, Mark D.
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
K
Kalamaridis, Dennis
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Kallan, Nicholas C.
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Kang, Ping
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Kassahun, Kelem
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
Kawamura, Akio
- You have accessOptimized Methods for Targeted Peptide-Based Quantification of Human Uridine 5′-Diphosphate-Glucuronosyltransferases in Biological Specimens Using Liquid Chromatography–Tandem Mass SpectrometryYuichiro Sato, Masanori Nagata, Kazuhiro Tetsuka, Kouichi Tamura, Aiji Miyashita, Akio Kawamura and Takashi UsuiDrug Metabolism and Disposition May 2014, 42 (5) 885-889; DOI: https://doi.org/10.1124/dmd.113.056291
Kelley, Michael F.
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Khojasteh, S. Cyrus
- You have access1-Aminobenzotriazole Coincubated with (S)-Warfarin Results in Potent Inactivation of CYP2C9Jasleen K. Sodhi, Kevin A. Ford, Sophie Mukadam, Susan Wong, Cornelis E. C. A. Hop, S. Cyrus Khojasteh and Jason S. HalladayDrug Metabolism and Disposition May 2014, 42 (5) 813-817; DOI: https://doi.org/10.1124/dmd.113.055913
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Kim-Kang, Heasook
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Klamerus, Karen J.
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Koeplinger, Kenneth
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
Kraft, Timothy W.
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
Krauser, Joel A.
- You have accessApplication of a Deuterium Replacement Strategy to Modulate the Pharmacokinetics of 7-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)-3-(4-methoxy-2-methylphenyl)-2,6-dimethylpyrazolo[5,1-b]oxazole, a Novel CRF1 AntagonistRowan A. Stringer, Gareth Williams, Franck Picard, Bindi Sohal, Olivier Kretz, Jeff McKenna and Joel A. KrauserDrug Metabolism and Disposition May 2014, 42 (5) 954-962; DOI: https://doi.org/10.1124/dmd.114.057265
Kretz, Olivier
- You have accessApplication of a Deuterium Replacement Strategy to Modulate the Pharmacokinetics of 7-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)-3-(4-methoxy-2-methylphenyl)-2,6-dimethylpyrazolo[5,1-b]oxazole, a Novel CRF1 AntagonistRowan A. Stringer, Gareth Williams, Franck Picard, Bindi Sohal, Olivier Kretz, Jeff McKenna and Joel A. KrauserDrug Metabolism and Disposition May 2014, 42 (5) 954-962; DOI: https://doi.org/10.1124/dmd.114.057265
L
Li, Feng
- You have accessBedaquiline Metabolism: Enzymes and Novel MetabolitesKe Liu, Feng Li, Jie Lu, Shinlan Liu, Kenneth Dorko, Wen Xie and Xiaochao MaDrug Metabolism and Disposition May 2014, 42 (5) 863-866; DOI: https://doi.org/10.1124/dmd.113.056119
Li, Ke
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Lim, Heng Keang
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Lin, Lishan
- You have accessMetabolism and Pharmacokinetics of Allitinib in Cancer Patients: The Roles of Cytochrome P450s and Epoxide Hydrolase in its BiotransformationLishan Lin, Cen Xie, Zhiwei Gao, Xiaoyan Chen and Dafang ZhongDrug Metabolism and Disposition May 2014, 42 (5) 872-884; DOI: https://doi.org/10.1124/dmd.113.056341
Lin, Ronghui
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Liu, Ke
- You have accessBedaquiline Metabolism: Enzymes and Novel MetabolitesKe Liu, Feng Li, Jie Lu, Shinlan Liu, Kenneth Dorko, Wen Xie and Xiaochao MaDrug Metabolism and Disposition May 2014, 42 (5) 863-866; DOI: https://doi.org/10.1124/dmd.113.056119
Liu, Shinlan
- You have accessBedaquiline Metabolism: Enzymes and Novel MetabolitesKe Liu, Feng Li, Jie Lu, Shinlan Liu, Kenneth Dorko, Wen Xie and Xiaochao MaDrug Metabolism and Disposition May 2014, 42 (5) 863-866; DOI: https://doi.org/10.1124/dmd.113.056119
Liu, Xingrong
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Lu, Jie
- You have accessBedaquiline Metabolism: Enzymes and Novel MetabolitesKe Liu, Feng Li, Jie Lu, Shinlan Liu, Kenneth Dorko, Wen Xie and Xiaochao MaDrug Metabolism and Disposition May 2014, 42 (5) 863-866; DOI: https://doi.org/10.1124/dmd.113.056119
Lu, Lu
- You have accessPolymorphisms and Haplotypes of the UDP-Glucuronosyltransferase 2B7 Gene PromoterDong Gui Hu, Robyn Meech, Lu Lu, Ross A. McKinnon and Peter I. MackenzieDrug Metabolism and Disposition May 2014, 42 (5) 854-862; DOI: https://doi.org/10.1124/dmd.113.056630
M
Ma, Shuguang
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Ma, Xiaochao
- You have accessBedaquiline Metabolism: Enzymes and Novel MetabolitesKe Liu, Feng Li, Jie Lu, Shinlan Liu, Kenneth Dorko, Wen Xie and Xiaochao MaDrug Metabolism and Disposition May 2014, 42 (5) 863-866; DOI: https://doi.org/10.1124/dmd.113.056119
Mackenzie, Peter I.
- You have accessPolymorphisms and Haplotypes of the UDP-Glucuronosyltransferase 2B7 Gene PromoterDong Gui Hu, Robyn Meech, Lu Lu, Ross A. McKinnon and Peter I. MackenzieDrug Metabolism and Disposition May 2014, 42 (5) 854-862; DOI: https://doi.org/10.1124/dmd.113.056630
Mair, Stuart
- You have accessAssessment of the Mass Balance Recovery and Metabolite Profile of Avibactam in Humans and In Vitro Drug-Drug Interaction PotentialKarthick Vishwanathan, Stuart Mair, Anshul Gupta, James Atherton, Jacqueline Clarkson-Jones, Timi Edeki and Shampa DasDrug Metabolism and Disposition May 2014, 42 (5) 932-942; DOI: https://doi.org/10.1124/dmd.113.055335
Mamidi, Rao N. V. S.
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
McIntosh, Ian
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
McKenna, Jeff
- You have accessApplication of a Deuterium Replacement Strategy to Modulate the Pharmacokinetics of 7-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)-3-(4-methoxy-2-methylphenyl)-2,6-dimethylpyrazolo[5,1-b]oxazole, a Novel CRF1 AntagonistRowan A. Stringer, Gareth Williams, Franck Picard, Bindi Sohal, Olivier Kretz, Jeff McKenna and Joel A. KrauserDrug Metabolism and Disposition May 2014, 42 (5) 954-962; DOI: https://doi.org/10.1124/dmd.114.057265
McKinnon, Ross A.
- You have accessPolymorphisms and Haplotypes of the UDP-Glucuronosyltransferase 2B7 Gene PromoterDong Gui Hu, Robyn Meech, Lu Lu, Ross A. McKinnon and Peter I. MackenzieDrug Metabolism and Disposition May 2014, 42 (5) 854-862; DOI: https://doi.org/10.1124/dmd.113.056630
Meech, Robyn
- You have accessPolymorphisms and Haplotypes of the UDP-Glucuronosyltransferase 2B7 Gene PromoterDong Gui Hu, Robyn Meech, Lu Lu, Ross A. McKinnon and Peter I. MackenzieDrug Metabolism and Disposition May 2014, 42 (5) 854-862; DOI: https://doi.org/10.1124/dmd.113.056630
Merino, Gracia
- You have accessRole of ABCG2 in Transport of the Mammalian Lignan Enterolactone and its Secretion into Milk in Abcg2 Knockout MiceVerónica Miguel, Jon Andoni Otero, Rocío García-Villalba, Francisco Tomás-Barberán, Juan Carlos Espín, Gracia Merino and Ana I. ÁlvarezDrug Metabolism and Disposition May 2014, 42 (5) 943-946; DOI: https://doi.org/10.1124/dmd.113.055970
Miguel, Verónica
- You have accessRole of ABCG2 in Transport of the Mammalian Lignan Enterolactone and its Secretion into Milk in Abcg2 Knockout MiceVerónica Miguel, Jon Andoni Otero, Rocío García-Villalba, Francisco Tomás-Barberán, Juan Carlos Espín, Gracia Merino and Ana I. ÁlvarezDrug Metabolism and Disposition May 2014, 42 (5) 943-946; DOI: https://doi.org/10.1124/dmd.113.055970
Miller, Deborah L.
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
Miyashita, Aiji
- You have accessOptimized Methods for Targeted Peptide-Based Quantification of Human Uridine 5′-Diphosphate-Glucuronosyltransferases in Biological Specimens Using Liquid Chromatography–Tandem Mass SpectrometryYuichiro Sato, Masanori Nagata, Kazuhiro Tetsuka, Kouichi Tamura, Aiji Miyashita, Akio Kawamura and Takashi UsuiDrug Metabolism and Disposition May 2014, 42 (5) 885-889; DOI: https://doi.org/10.1124/dmd.113.056291
Mukadam, Sophie
- You have access1-Aminobenzotriazole Coincubated with (S)-Warfarin Results in Potent Inactivation of CYP2C9Jasleen K. Sodhi, Kevin A. Ford, Sophie Mukadam, Susan Wong, Cornelis E. C. A. Hop, S. Cyrus Khojasteh and Jason S. HalladayDrug Metabolism and Disposition May 2014, 42 (5) 813-817; DOI: https://doi.org/10.1124/dmd.113.055913
Murayama, Norie
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
N
Nagata, Masanori
- You have accessOptimized Methods for Targeted Peptide-Based Quantification of Human Uridine 5′-Diphosphate-Glucuronosyltransferases in Biological Specimens Using Liquid Chromatography–Tandem Mass SpectrometryYuichiro Sato, Masanori Nagata, Kazuhiro Tetsuka, Kouichi Tamura, Aiji Miyashita, Akio Kawamura and Takashi UsuiDrug Metabolism and Disposition May 2014, 42 (5) 885-889; DOI: https://doi.org/10.1124/dmd.113.056291
Nakamura, Chika
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
O
Obach, R. Scott
- You have accessGeneration of Major Human Excretory and Circulating Drug Metabolites Using a Hepatocyte Relay MethodT. Eric Ballard, Christine C. Orozco and R. Scott ObachDrug Metabolism and Disposition May 2014, 42 (5) 899-902; DOI: https://doi.org/10.1124/dmd.114.057026
Orozco, Christine C.
- You have accessGeneration of Major Human Excretory and Circulating Drug Metabolites Using a Hepatocyte Relay MethodT. Eric Ballard, Christine C. Orozco and R. Scott ObachDrug Metabolism and Disposition May 2014, 42 (5) 899-902; DOI: https://doi.org/10.1124/dmd.114.057026
Ortiz de Montellano, Paul R.
- You have accessCarbon-Carbon Bond Cleavage in Activation of the Prodrug NabumetoneFatbardha Varfaj, Siti N. A. Zulkifli, Hyoung-Goo Park, Victoria L. Challinor, James J. De Voss and Paul R. Ortiz de MontellanoDrug Metabolism and Disposition May 2014, 42 (5) 828-838; DOI: https://doi.org/10.1124/dmd.114.056903
Otero, Jon Andoni
- You have accessRole of ABCG2 in Transport of the Mammalian Lignan Enterolactone and its Secretion into Milk in Abcg2 Knockout MiceVerónica Miguel, Jon Andoni Otero, Rocío García-Villalba, Francisco Tomás-Barberán, Juan Carlos Espín, Gracia Merino and Ana I. ÁlvarezDrug Metabolism and Disposition May 2014, 42 (5) 943-946; DOI: https://doi.org/10.1124/dmd.113.055970
P
Parant, John M.
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
Park, Hyoung-Goo
- You have accessCarbon-Carbon Bond Cleavage in Activation of the Prodrug NabumetoneFatbardha Varfaj, Siti N. A. Zulkifli, Hyoung-Goo Park, Victoria L. Challinor, James J. De Voss and Paul R. Ortiz de MontellanoDrug Metabolism and Disposition May 2014, 42 (5) 828-838; DOI: https://doi.org/10.1124/dmd.114.056903
Picard, Franck
- You have accessApplication of a Deuterium Replacement Strategy to Modulate the Pharmacokinetics of 7-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)-3-(4-methoxy-2-methylphenyl)-2,6-dimethylpyrazolo[5,1-b]oxazole, a Novel CRF1 AntagonistRowan A. Stringer, Gareth Williams, Franck Picard, Bindi Sohal, Olivier Kretz, Jeff McKenna and Joel A. KrauserDrug Metabolism and Disposition May 2014, 42 (5) 954-962; DOI: https://doi.org/10.1124/dmd.114.057265
Pithavala, Yazdi
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Pool, William F.
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
S
Sato, Yuichiro
- You have accessOptimized Methods for Targeted Peptide-Based Quantification of Human Uridine 5′-Diphosphate-Glucuronosyltransferases in Biological Specimens Using Liquid Chromatography–Tandem Mass SpectrometryYuichiro Sato, Masanori Nagata, Kazuhiro Tetsuka, Kouichi Tamura, Aiji Miyashita, Akio Kawamura and Takashi UsuiDrug Metabolism and Disposition May 2014, 42 (5) 885-889; DOI: https://doi.org/10.1124/dmd.113.056291
Scheers, Ellen
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Sha, Sue
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Shimizu, Makiko
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
Shu, Pan
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Silva, Jose
- You have accessMetabolism and Excretion of Canagliflozin in Mice, Rats, Dogs, and HumansRao N. V. S. Mamidi, Filip Cuyckens, Jie Chen, Ellen Scheers, Dennis Kalamaridis, Ronghui Lin, Jose Silva, Sue Sha, David C. Evans, Michael F. Kelley, Damayanthi Devineni, Mark D. Johnson and Heng Keang LimDrug Metabolism and Disposition May 2014, 42 (5) 903-916; DOI: https://doi.org/10.1124/dmd.113.056440
Siu, Michael
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Smith, Bill J.
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Sodhi, Jasleen K.
- You have access1-Aminobenzotriazole Coincubated with (S)-Warfarin Results in Potent Inactivation of CYP2C9Jasleen K. Sodhi, Kevin A. Ford, Sophie Mukadam, Susan Wong, Cornelis E. C. A. Hop, S. Cyrus Khojasteh and Jason S. HalladayDrug Metabolism and Disposition May 2014, 42 (5) 813-817; DOI: https://doi.org/10.1124/dmd.113.055913
Sohal, Bindi
- You have accessApplication of a Deuterium Replacement Strategy to Modulate the Pharmacokinetics of 7-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)-3-(4-methoxy-2-methylphenyl)-2,6-dimethylpyrazolo[5,1-b]oxazole, a Novel CRF1 AntagonistRowan A. Stringer, Gareth Williams, Franck Picard, Bindi Sohal, Olivier Kretz, Jeff McKenna and Joel A. KrauserDrug Metabolism and Disposition May 2014, 42 (5) 954-962; DOI: https://doi.org/10.1124/dmd.114.057265
Stoch, S. Aubrey
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
Stringer, Rowan A.
- You have accessApplication of a Deuterium Replacement Strategy to Modulate the Pharmacokinetics of 7-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)-3-(4-methoxy-2-methylphenyl)-2,6-dimethylpyrazolo[5,1-b]oxazole, a Novel CRF1 AntagonistRowan A. Stringer, Gareth Williams, Franck Picard, Bindi Sohal, Olivier Kretz, Jeff McKenna and Joel A. KrauserDrug Metabolism and Disposition May 2014, 42 (5) 954-962; DOI: https://doi.org/10.1124/dmd.114.057265
Sun, Li
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
T
Takahashi, Ryan
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Talaty, Jennifer E.
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
Tamura, Kouichi
- You have accessOptimized Methods for Targeted Peptide-Based Quantification of Human Uridine 5′-Diphosphate-Glucuronosyltransferases in Biological Specimens Using Liquid Chromatography–Tandem Mass SpectrometryYuichiro Sato, Masanori Nagata, Kazuhiro Tetsuka, Kouichi Tamura, Aiji Miyashita, Akio Kawamura and Takashi UsuiDrug Metabolism and Disposition May 2014, 42 (5) 885-889; DOI: https://doi.org/10.1124/dmd.113.056291
Tetsuka, Kazuhiro
- You have accessOptimized Methods for Targeted Peptide-Based Quantification of Human Uridine 5′-Diphosphate-Glucuronosyltransferases in Biological Specimens Using Liquid Chromatography–Tandem Mass SpectrometryYuichiro Sato, Masanori Nagata, Kazuhiro Tetsuka, Kouichi Tamura, Aiji Miyashita, Akio Kawamura and Takashi UsuiDrug Metabolism and Disposition May 2014, 42 (5) 885-889; DOI: https://doi.org/10.1124/dmd.113.056291
Thomas, Holly
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
Tomás-Barberán, Francisco
- You have accessRole of ABCG2 in Transport of the Mammalian Lignan Enterolactone and its Secretion into Milk in Abcg2 Knockout MiceVerónica Miguel, Jon Andoni Otero, Rocío García-Villalba, Francisco Tomás-Barberán, Juan Carlos Espín, Gracia Merino and Ana I. ÁlvarezDrug Metabolism and Disposition May 2014, 42 (5) 943-946; DOI: https://doi.org/10.1124/dmd.113.055970
U
Uehara, Shotaro
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
Uno, Yasuhiro
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
Usui, Takashi
- You have accessOptimized Methods for Targeted Peptide-Based Quantification of Human Uridine 5′-Diphosphate-Glucuronosyltransferases in Biological Specimens Using Liquid Chromatography–Tandem Mass SpectrometryYuichiro Sato, Masanori Nagata, Kazuhiro Tetsuka, Kouichi Tamura, Aiji Miyashita, Akio Kawamura and Takashi UsuiDrug Metabolism and Disposition May 2014, 42 (5) 885-889; DOI: https://doi.org/10.1124/dmd.113.056291
Utoh, Masahiro
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
V
Varfaj, Fatbardha
- You have accessCarbon-Carbon Bond Cleavage in Activation of the Prodrug NabumetoneFatbardha Varfaj, Siti N. A. Zulkifli, Hyoung-Goo Park, Victoria L. Challinor, James J. De Voss and Paul R. Ortiz de MontellanoDrug Metabolism and Disposition May 2014, 42 (5) 828-838; DOI: https://doi.org/10.1124/dmd.114.056903
Vishwanathan, Karthick
- You have accessAssessment of the Mass Balance Recovery and Metabolite Profile of Avibactam in Humans and In Vitro Drug-Drug Interaction PotentialKarthick Vishwanathan, Stuart Mair, Anshul Gupta, James Atherton, Jacqueline Clarkson-Jones, Timi Edeki and Shampa DasDrug Metabolism and Disposition May 2014, 42 (5) 932-942; DOI: https://doi.org/10.1124/dmd.113.055335
W
Wang, Yang
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Wang, Yongtao
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Williams, Gareth
- You have accessApplication of a Deuterium Replacement Strategy to Modulate the Pharmacokinetics of 7-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)-3-(4-methoxy-2-methylphenyl)-2,6-dimethylpyrazolo[5,1-b]oxazole, a Novel CRF1 AntagonistRowan A. Stringer, Gareth Williams, Franck Picard, Bindi Sohal, Olivier Kretz, Jeff McKenna and Joel A. KrauserDrug Metabolism and Disposition May 2014, 42 (5) 954-962; DOI: https://doi.org/10.1124/dmd.114.057265
Wong, Susan
- You have access1-Aminobenzotriazole Coincubated with (S)-Warfarin Results in Potent Inactivation of CYP2C9Jasleen K. Sodhi, Kevin A. Ford, Sophie Mukadam, Susan Wong, Cornelis E. C. A. Hop, S. Cyrus Khojasteh and Jason S. HalladayDrug Metabolism and Disposition May 2014, 42 (5) 813-817; DOI: https://doi.org/10.1124/dmd.113.055913
Wu, Ellen Y.
- You have accessPharmacokinetics, Metabolism, and Excretion of [14C]Axitinib, a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor, in HumansBill J. Smith, Yazdi Pithavala, Hai-Zhi Bu, Ping Kang, Brian Hee, Alan J. Deese, William F. Pool, Karen J. Klamerus, Ellen Y. Wu and Deepak K. DalvieDrug Metabolism and Disposition May 2014, 42 (5) 918-931; DOI: https://doi.org/10.1124/dmd.113.056531
Wu, Xiaoyun
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Wu, Zhengliang L.
- You have accessInhibition of SULT4A1 Expression Induces Up-Regulation of Phototransduction Gene Expression in 72-Hour Postfertilization Zebrafish LarvaeFrank Crittenden, Holly Thomas, Cheryl M. Ethen, Zhengliang L. Wu, Dongquan Chen, Timothy W. Kraft, John M. Parant and Charles N. FalanyDrug Metabolism and Disposition May 2014, 42 (5) 947-953; DOI: https://doi.org/10.1124/dmd.114.057042
X
Xie, Cen
- You have accessMetabolism and Pharmacokinetics of Allitinib in Cancer Patients: The Roles of Cytochrome P450s and Epoxide Hydrolase in its BiotransformationLishan Lin, Cen Xie, Zhiwei Gao, Xiaoyan Chen and Dafang ZhongDrug Metabolism and Disposition May 2014, 42 (5) 872-884; DOI: https://doi.org/10.1124/dmd.113.056341
Xie, Wen
- You have accessBedaquiline Metabolism: Enzymes and Novel MetabolitesKe Liu, Feng Li, Jie Lu, Shinlan Liu, Kenneth Dorko, Wen Xie and Xiaochao MaDrug Metabolism and Disposition May 2014, 42 (5) 863-866; DOI: https://doi.org/10.1124/dmd.113.056119
Xu, Chenshu
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Y
Yajima, Kanako
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
Yamazaki, Hiroshi
- You have accessEvaluation of 23 Lots of Commercially Available Cryopreserved Hepatocytes for Induction Assays of Human Cytochromes P450Kanako Yajima, Yasuhiro Uno, Norie Murayama, Shotaro Uehara, Makiko Shimizu, Chika Nakamura, Kazuhide Iwasaki, Masahiro Utoh and Hiroshi YamazakiDrug Metabolism and Disposition May 2014, 42 (5) 867-871; DOI: https://doi.org/10.1124/dmd.113.056804
Yi, Yijun
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Yue, Qin
- You have accessElucidating the Mechanism of Cytochrome P450–Mediated Pyrimidine Ring Conversion to Pyrazole Metabolites with the BACE1 Inhibitor GNE-892 in RatsRyan Takahashi, Shuguang Ma, Alan Deese, Qin Yue, Heasook Kim-Kang, Yijun Yi, Michael Siu, Kevin W. Hunt, Nicholas C. Kallan, Cornelis E.C.A. Hop, Xingrong Liu and S. Cyrus KhojastehDrug Metabolism and Disposition May 2014, 42 (5) 890-898; DOI: https://doi.org/10.1124/dmd.114.057141
Z
Zajic, Stefan
- You have accessDisposition and Metabolism of the Cathepsin K Inhibitor Odanacatib in HumansKelem Kassahun, Ian McIntosh, Kenneth Koeplinger, Li Sun, Jennifer E. Talaty, Deborah L. Miller, Russell Dixon, Stefan Zajic and S. Aubrey StochDrug Metabolism and Disposition May 2014, 42 (5) 818-827; DOI: https://doi.org/10.1124/dmd.113.056580
Zeng, Hang
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Zhang, Lingling
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Zhao, Sylvia
- You have access4β-Hydroxycholesterol as an Endogenous Biomarker of CYP3A Activity in Cynomolgus MonkeysKe Li, Sylvia Zhao, Lingling Zhang, Xiaoyun Wu, Pan Shu, Yang Wang, Hao Feng, Zheming Gu and Helen Han HsuDrug Metabolism and Disposition May 2014, 42 (5) 839-843; DOI: https://doi.org/10.1124/dmd.114.057224
Zhong, Dafang
- You have accessMetabolism and Pharmacokinetics of Allitinib in Cancer Patients: The Roles of Cytochrome P450s and Epoxide Hydrolase in its BiotransformationLishan Lin, Cen Xie, Zhiwei Gao, Xiaoyan Chen and Dafang ZhongDrug Metabolism and Disposition May 2014, 42 (5) 872-884; DOI: https://doi.org/10.1124/dmd.113.056341
Zhou, Xunian
- You have accessLow Dose of Oleanolic Acid Protects against Lithocholic Acid–Induced Cholestasis in Mice: Potential Involvement of Nuclear Factor-E2-Related Factor 2-Mediated Upregulation of Multidrug Resistance-Associated ProteinsPan Chen, Hang Zeng, Yongtao Wang, Xiaomei Fan, Chenshu Xu, Rongrong Deng, Xunian Zhou, Huichang Bi and Min HuangDrug Metabolism and Disposition May 2014, 42 (5) 844-852; DOI: https://doi.org/10.1124/dmd.113.056549
Zulkifli, Siti N. A.
- You have accessCarbon-Carbon Bond Cleavage in Activation of the Prodrug NabumetoneFatbardha Varfaj, Siti N. A. Zulkifli, Hyoung-Goo Park, Victoria L. Challinor, James J. De Voss and Paul R. Ortiz de MontellanoDrug Metabolism and Disposition May 2014, 42 (5) 828-838; DOI: https://doi.org/10.1124/dmd.114.056903
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