Index by author
April 01, 2015; Volume 43,Issue 4
A
Achour, Brahim
- You have accessMeta-Analysis of Expression of Hepatic Organic Anion–Transporting Polypeptide (OATP) Transporters in Cellular Systems Relative to Human Liver TissueJustine Badée, Brahim Achour, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition April 2015, 43 (4) 424-432; DOI: https://doi.org/10.1124/dmd.114.062034
Ando, Hirotaka
- You have accessA New Physiologically Based Pharmacokinetic Model for the Prediction of Gastrointestinal Drug Absorption: Translocation ModelHirotaka Ando, Akihiro Hisaka and Hiroshi SuzukiDrug Metabolism and Disposition April 2015, 43 (4) 590-602; DOI: https://doi.org/10.1124/dmd.114.060038
Asakura, Mitsutoshi
- You have accessDipeptidyl Peptidase-4 Greatly Contributes to the Hydrolysis of Vildagliptin in Human LiverMitsutoshi Asakura, Hideaki Fujii, Koichiro Atsuda, Tomoo Itoh and Ryoichi FujiwaraDrug Metabolism and Disposition April 2015, 43 (4) 477-484; DOI: https://doi.org/10.1124/dmd.114.062331
Atsuda, Koichiro
- You have accessDipeptidyl Peptidase-4 Greatly Contributes to the Hydrolysis of Vildagliptin in Human LiverMitsutoshi Asakura, Hideaki Fujii, Koichiro Atsuda, Tomoo Itoh and Ryoichi FujiwaraDrug Metabolism and Disposition April 2015, 43 (4) 477-484; DOI: https://doi.org/10.1124/dmd.114.062331
Avula, Bharathi
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
B
Badée, Justine
- You have accessMeta-Analysis of Expression of Hepatic Organic Anion–Transporting Polypeptide (OATP) Transporters in Cellular Systems Relative to Human Liver TissueJustine Badée, Brahim Achour, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition April 2015, 43 (4) 424-432; DOI: https://doi.org/10.1124/dmd.114.062034
Balani, Suresh K.
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Barbara, Joanna E.
- You have accessA Long-Standing Mystery Solved: The Formation of 3-Hydroxydesloratadine Is Catalyzed by CYP2C8 But Prior Glucuronidation of Desloratadine by UDP-Glucuronosyltransferase 2B10 Is an Obligatory RequirementFaraz Kazmi, Joanna E. Barbara, Phyllis Yerino and Andrew ParkinsonDrug Metabolism and Disposition April 2015, 43 (4) 523-533; DOI: https://doi.org/10.1124/dmd.114.062620
Barone, Gary
- You have accessHydrastine Pharmacokinetics and Metabolism after a Single Oral Dose of Goldenseal (Hydrastis canadensis) to HumansPrem K. Gupta, Gary Barone, Bill J. Gurley, E. Kim Fifer and Howard P. HendricksonDrug Metabolism and Disposition April 2015, 43 (4) 534-552; DOI: https://doi.org/10.1124/dmd.114.059410
Boulenc, Xavier
- You have accessPhysiologically Based Pharmacokinetic Modeling for Sequential Metabolism: Effect of CYP2C19 Genetic Polymorphism on Clopidogrel and Clopidogrel Active Metabolite PharmacokineticsNassim Djebli, David Fabre, Xavier Boulenc, Gérard Fabre, Eric Sultan and Fabrice HurbinDrug Metabolism and Disposition April 2015, 43 (4) 510-522; DOI: https://doi.org/10.1124/dmd.114.062596
C
Cai, Jian-Ping
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Cao, Lijuan
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Caron, Patrick
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
Chaurasiya, Narayan D.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Che, Yuan
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Chen, Weichao
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Cheng, Xuefang
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Chow, Edwin C. Y.
- You have accessPBPK Modeling to Unravel Nonlinear Pharmacokinetics of Verapamil to Estimate the Fractional Clearance for Verapamil N-Demethylation in the Recirculating Rat Liver PreparationQi Joy Yang, Luqin Si, Hui Tang, Helle H. Sveigaard, Edwin C. Y. Chow and K. Sandy PangDrug Metabolism and Disposition April 2015, 43 (4) 631-645; DOI: https://doi.org/10.1124/dmd.114.062265
Cook, Jack A.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Corbel, Tanguy
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Cui, Donghui
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
D
Dai, Da-Peng
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Degnan, Andrew P.
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
Diamond, Sharon
- You have accessImpact on Creatinine Renal Clearance by the Interplay of Multiple Renal Transporters: A Case Study with INCB039110Yan Zhang, Mark S. Warren, Xuexiang Zhang, Sharon Diamond, Bill Williams, Naresh Punwani, Jane Huang, Yong Huang and Swamy YeleswaramDrug Metabolism and Disposition April 2015, 43 (4) 485-489; DOI: https://doi.org/10.1124/dmd.114.060673
Djebli, Nassim
- You have accessPhysiologically Based Pharmacokinetic Modeling for Sequential Metabolism: Effect of CYP2C19 Genetic Polymorphism on Clopidogrel and Clopidogrel Active Metabolite PharmacokineticsNassim Djebli, David Fabre, Xavier Boulenc, Gérard Fabre, Eric Sultan and Fabrice HurbinDrug Metabolism and Disposition April 2015, 43 (4) 510-522; DOI: https://doi.org/10.1124/dmd.114.062596
Dong, Dong
- You have accessCharacterization of Chrysin Glucuronidation in UGT1A1-Overexpressing HeLa Cells: Elucidating the Transporters Responsible for Efflux of GlucuronideEnxi Quan, Huailing Wang, Dong Dong, Xingwang Zhang and Baojian WuDrug Metabolism and Disposition April 2015, 43 (4) 433-443; DOI: https://doi.org/10.1124/dmd.114.061598
E
Ellens, Harma
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
ElSohly, Mahmoud A.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
F
Fabre, David
- You have accessPhysiologically Based Pharmacokinetic Modeling for Sequential Metabolism: Effect of CYP2C19 Genetic Polymorphism on Clopidogrel and Clopidogrel Active Metabolite PharmacokineticsNassim Djebli, David Fabre, Xavier Boulenc, Gérard Fabre, Eric Sultan and Fabrice HurbinDrug Metabolism and Disposition April 2015, 43 (4) 510-522; DOI: https://doi.org/10.1124/dmd.114.062596
Fabre, Gérard
- You have accessPhysiologically Based Pharmacokinetic Modeling for Sequential Metabolism: Effect of CYP2C19 Genetic Polymorphism on Clopidogrel and Clopidogrel Active Metabolite PharmacokineticsNassim Djebli, David Fabre, Xavier Boulenc, Gérard Fabre, Eric Sultan and Fabrice HurbinDrug Metabolism and Disposition April 2015, 43 (4) 510-522; DOI: https://doi.org/10.1124/dmd.114.062596
Fallon, John K.
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
Fasinu, Pius S.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Feng, Bo
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Fifer, E. Kim
- You have accessHydrastine Pharmacokinetics and Metabolism after a Single Oral Dose of Goldenseal (Hydrastis canadensis) to HumansPrem K. Gupta, Gary Barone, Bill J. Gurley, E. Kim Fifer and Howard P. HendricksonDrug Metabolism and Disposition April 2015, 43 (4) 534-552; DOI: https://doi.org/10.1124/dmd.114.059410
Fu, Qian
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Fujii, Hideaki
- You have accessDipeptidyl Peptidase-4 Greatly Contributes to the Hydrolysis of Vildagliptin in Human LiverMitsutoshi Asakura, Hideaki Fujii, Koichiro Atsuda, Tomoo Itoh and Ryoichi FujiwaraDrug Metabolism and Disposition April 2015, 43 (4) 477-484; DOI: https://doi.org/10.1124/dmd.114.062331
Fujiwara, Ryoichi
- You have accessDipeptidyl Peptidase-4 Greatly Contributes to the Hydrolysis of Vildagliptin in Human LiverMitsutoshi Asakura, Hideaki Fujii, Koichiro Atsuda, Tomoo Itoh and Ryoichi FujiwaraDrug Metabolism and Disposition April 2015, 43 (4) 477-484; DOI: https://doi.org/10.1124/dmd.114.062331
G
Galetin, Aleksandra
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
- You have accessMeta-Analysis of Expression of Hepatic Organic Anion–Transporting Polypeptide (OATP) Transporters in Cellular Systems Relative to Human Liver TissueJustine Badée, Brahim Achour, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition April 2015, 43 (4) 424-432; DOI: https://doi.org/10.1124/dmd.114.062034
Gayrard, Véronique
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Ge, Guang-Bo
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Ge, Ren-Shan
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Guillemette, Chantal
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
Gupta, Prem K.
- You have accessHydrastine Pharmacokinetics and Metabolism after a Single Oral Dose of Goldenseal (Hydrastis canadensis) to HumansPrem K. Gupta, Gary Barone, Bill J. Gurley, E. Kim Fifer and Howard P. HendricksonDrug Metabolism and Disposition April 2015, 43 (4) 534-552; DOI: https://doi.org/10.1124/dmd.114.059410
Gurley, Bill J.
- You have accessHydrastine Pharmacokinetics and Metabolism after a Single Oral Dose of Goldenseal (Hydrastis canadensis) to HumansPrem K. Gupta, Gary Barone, Bill J. Gurley, E. Kim Fifer and Howard P. HendricksonDrug Metabolism and Disposition April 2015, 43 (4) 534-552; DOI: https://doi.org/10.1124/dmd.114.059410
H
Hao, Haiping
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
He, Ling
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
He, Yu-Qi
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Hendrickson, Howard P.
- You have accessHydrastine Pharmacokinetics and Metabolism after a Single Oral Dose of Goldenseal (Hydrastis canadensis) to HumansPrem K. Gupta, Gary Barone, Bill J. Gurley, E. Kim Fifer and Howard P. HendricksonDrug Metabolism and Disposition April 2015, 43 (4) 534-552; DOI: https://doi.org/10.1124/dmd.114.059410
Herath, H.M.T. Bandara
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Hisaka, Akihiro
- You have accessA New Physiologically Based Pharmacokinetic Model for the Prediction of Gastrointestinal Drug Absorption: Translocation ModelHirotaka Ando, Akihiro Hisaka and Hiroshi SuzukiDrug Metabolism and Disposition April 2015, 43 (4) 590-602; DOI: https://doi.org/10.1124/dmd.114.060038
Horikawa, Takashi
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
Hu, Guo-Xin
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Huang, Hong
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
Huang, Jane
- You have accessImpact on Creatinine Renal Clearance by the Interplay of Multiple Renal Transporters: A Case Study with INCB039110Yan Zhang, Mark S. Warren, Xuexiang Zhang, Sharon Diamond, Bill Williams, Naresh Punwani, Jane Huang, Yong Huang and Swamy YeleswaramDrug Metabolism and Disposition April 2015, 43 (4) 485-489; DOI: https://doi.org/10.1124/dmd.114.060673
Huang, Min
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Huang, Xiaohua Stella
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
Huang, Yong
- You have accessImpact on Creatinine Renal Clearance by the Interplay of Multiple Renal Transporters: A Case Study with INCB039110Yan Zhang, Mark S. Warren, Xuexiang Zhang, Sharon Diamond, Bill Williams, Naresh Punwani, Jane Huang, Yong Huang and Swamy YeleswaramDrug Metabolism and Disposition April 2015, 43 (4) 485-489; DOI: https://doi.org/10.1124/dmd.114.060673
Humphreys, W. Griffith
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Hurbin, Fabrice
- You have accessPhysiologically Based Pharmacokinetic Modeling for Sequential Metabolism: Effect of CYP2C19 Genetic Polymorphism on Clopidogrel and Clopidogrel Active Metabolite PharmacokineticsNassim Djebli, David Fabre, Xavier Boulenc, Gérard Fabre, Eric Sultan and Fabrice HurbinDrug Metabolism and Disposition April 2015, 43 (4) 510-522; DOI: https://doi.org/10.1124/dmd.114.062596
I
Itoh, Tomoo
- You have accessDipeptidyl Peptidase-4 Greatly Contributes to the Hydrolysis of Vildagliptin in Human LiverMitsutoshi Asakura, Hideaki Fujii, Koichiro Atsuda, Tomoo Itoh and Ryoichi FujiwaraDrug Metabolism and Disposition April 2015, 43 (4) 477-484; DOI: https://doi.org/10.1124/dmd.114.062331
Iwao, Takahiro
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
J
Jain, Surendra
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Johnson, Benjamin M.
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
Joy, Melanie S.
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
K
Kabeya, Tomoki
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
Kamezawa, Miho
- You have accessUtility of Bilirubins and Bile Acids as Endogenous Biomarkers for the Inhibition of Hepatic TransportersTomoko Watanabe, Manami Miyake, Toshinobu Shimizu, Miho Kamezawa, Naoya Masutomi, Takesada Shimura and Rikiya OhashiDrug Metabolism and Disposition April 2015, 43 (4) 459-466; DOI: https://doi.org/10.1124/dmd.114.061051
Kazmi, Faraz
- You have accessA Long-Standing Mystery Solved: The Formation of 3-Hydroxydesloratadine Is Catalyzed by CYP2C8 But Prior Glucuronidation of Desloratadine by UDP-Glucuronosyltransferase 2B10 Is an Obligatory RequirementFaraz Kazmi, Joanna E. Barbara, Phyllis Yerino and Andrew ParkinsonDrug Metabolism and Disposition April 2015, 43 (4) 523-533; DOI: https://doi.org/10.1124/dmd.114.062620
Khan, Ikhlas A.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Khan, Shabana I.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Kodama, Nao
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
Kondo, Yuki
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
Kurose, Kouichi
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
L
Lacroix, Marlène Z.
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Lai, W. George
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Lee, Anthony J.
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Lee, Caroline A.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Li, Feiyan
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Li, Jiali
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Li, Jun
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Li, Yan
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Lian, Qing-Quan
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Liang, Si-Cheng
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Lim, Heng-Keang
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Liu, Huiying
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Liu, Shu
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Liu, Xiaoman
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Luo, Jun
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
M
MacLauchlin, Christopher
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Mao, Jialin
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Margaillan, Guillaume
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
Masutomi, Naoya
- You have accessUtility of Bilirubins and Bile Acids as Endogenous Biomarkers for the Inhibition of Hepatic TransportersTomoko Watanabe, Manami Miyake, Toshinobu Shimizu, Miho Kamezawa, Naoya Masutomi, Takesada Shimura and Rikiya OhashiDrug Metabolism and Disposition April 2015, 43 (4) 459-466; DOI: https://doi.org/10.1124/dmd.114.061051
Matsunaga, Tamihide
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
McChesney, James D.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Miyake, Manami
- You have accessUtility of Bilirubins and Bile Acids as Endogenous Biomarkers for the Inhibition of Hepatic TransportersTomoko Watanabe, Manami Miyake, Toshinobu Shimizu, Miho Kamezawa, Naoya Masutomi, Takesada Shimura and Rikiya OhashiDrug Metabolism and Disposition April 2015, 43 (4) 459-466; DOI: https://doi.org/10.1124/dmd.114.061051
N
Nakamura, Katsunori
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
Nanayakkara, N.P. Dhammika
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Ning, Jing
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Niwa, Takuro
- You have accessGeneration of Enterocyte-Like Cells with Pharmacokinetic Functions from Human Induced Pluripotent Stem Cells Using Small-Molecule CompoundsTakahiro Iwao, Nao Kodama, Yuki Kondo, Tomoki Kabeya, Katsunori Nakamura, Takashi Horikawa, Takuro Niwa, Kouichi Kurose and Tamihide MatsunagaDrug Metabolism and Disposition April 2015, 43 (4) 603-610; DOI: https://doi.org/10.1124/dmd.114.062604
O
O’Connor, Meeghan A.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Ohashi, Rikiya
- You have accessUtility of Bilirubins and Bile Acids as Endogenous Biomarkers for the Inhibition of Hepatic TransportersTomoko Watanabe, Manami Miyake, Toshinobu Shimizu, Miho Kamezawa, Naoya Masutomi, Takesada Shimura and Rikiya OhashiDrug Metabolism and Disposition April 2015, 43 (4) 459-466; DOI: https://doi.org/10.1124/dmd.114.061051
P
Paine, Mary F.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Pan, Pei-Pei
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Pang, K. Sandy
- You have accessPBPK Modeling to Unravel Nonlinear Pharmacokinetics of Verapamil to Estimate the Fractional Clearance for Verapamil N-Demethylation in the Recirculating Rat Liver PreparationQi Joy Yang, Luqin Si, Hui Tang, Helle H. Sveigaard, Edwin C. Y. Chow and K. Sandy PangDrug Metabolism and Disposition April 2015, 43 (4) 631-645; DOI: https://doi.org/10.1124/dmd.114.062265
Parkinson, Andrew
- You have accessA Long-Standing Mystery Solved: The Formation of 3-Hydroxydesloratadine Is Catalyzed by CYP2C8 But Prior Glucuronidation of Desloratadine by UDP-Glucuronosyltransferase 2B10 Is an Obligatory RequirementFaraz Kazmi, Joanna E. Barbara, Phyllis Yerino and Andrew ParkinsonDrug Metabolism and Disposition April 2015, 43 (4) 523-533; DOI: https://doi.org/10.1124/dmd.114.062620
Perdu, Elisabeth
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Picard-Hagen, Nicole
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Polli, Joseph W.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Prakash, Chandra
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Puel, Sylvie
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Punwani, Naresh
- You have accessImpact on Creatinine Renal Clearance by the Interplay of Multiple Renal Transporters: A Case Study with INCB039110Yan Zhang, Mark S. Warren, Xuexiang Zhang, Sharon Diamond, Bill Williams, Naresh Punwani, Jane Huang, Yong Huang and Swamy YeleswaramDrug Metabolism and Disposition April 2015, 43 (4) 485-489; DOI: https://doi.org/10.1124/dmd.114.060673
Q
Qi, Qu
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Qian, Xing-Kai
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Qiu, Xiang-Jun
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Quan, Enxi
- You have accessCharacterization of Chrysin Glucuronidation in UGT1A1-Overexpressing HeLa Cells: Elucidating the Transporters Responsible for Efflux of GlucuronideEnxi Quan, Huailing Wang, Dong Dong, Xingwang Zhang and Baojian WuDrug Metabolism and Disposition April 2015, 43 (4) 433-443; DOI: https://doi.org/10.1124/dmd.114.061598
R
Ragueneau-Majlessi, Isabelle
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Ritchie, Tasha K.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Rostami-Hodjegan, Amin
- You have accessMeta-Analysis of Expression of Hepatic Organic Anion–Transporting Polypeptide (OATP) Transporters in Cellular Systems Relative to Human Liver TissueJustine Badée, Brahim Achour, Amin Rostami-Hodjegan and Aleksandra GaletinDrug Metabolism and Disposition April 2015, 43 (4) 424-432; DOI: https://doi.org/10.1124/dmd.114.062034
Rouleau, Michèle
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
S
Sahu, Rajnish
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Shimizu, Toshinobu
- You have accessUtility of Bilirubins and Bile Acids as Endogenous Biomarkers for the Inhibition of Hepatic TransportersTomoko Watanabe, Manami Miyake, Toshinobu Shimizu, Miho Kamezawa, Naoya Masutomi, Takesada Shimura and Rikiya OhashiDrug Metabolism and Disposition April 2015, 43 (4) 459-466; DOI: https://doi.org/10.1124/dmd.114.061051
Shimura, Takesada
- You have accessUtility of Bilirubins and Bile Acids as Endogenous Biomarkers for the Inhibition of Hepatic TransportersTomoko Watanabe, Manami Miyake, Toshinobu Shimizu, Miho Kamezawa, Naoya Masutomi, Takesada Shimura and Rikiya OhashiDrug Metabolism and Disposition April 2015, 43 (4) 459-466; DOI: https://doi.org/10.1124/dmd.114.061051
Shu, Yue-Zhong
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
Si, Luqin
- You have accessPBPK Modeling to Unravel Nonlinear Pharmacokinetics of Verapamil to Estimate the Fractional Clearance for Verapamil N-Demethylation in the Recirculating Rat Liver PreparationQi Joy Yang, Luqin Si, Hui Tang, Helle H. Sveigaard, Edwin C. Y. Chow and K. Sandy PangDrug Metabolism and Disposition April 2015, 43 (4) 631-645; DOI: https://doi.org/10.1124/dmd.114.062265
Smith, Philip C.
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
Snyder, Lawrence B.
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
Stanford, Donald
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Sultan, Eric
- You have accessPhysiologically Based Pharmacokinetic Modeling for Sequential Metabolism: Effect of CYP2C19 Genetic Polymorphism on Clopidogrel and Clopidogrel Active Metabolite PharmacokineticsNassim Djebli, David Fabre, Xavier Boulenc, Gérard Fabre, Eric Sultan and Fabrice HurbinDrug Metabolism and Disposition April 2015, 43 (4) 510-522; DOI: https://doi.org/10.1124/dmd.114.062596
Surapaneni, Sekhar
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Suzuki, Hiroshi
- You have accessA New Physiologically Based Pharmacokinetic Model for the Prediction of Gastrointestinal Drug Absorption: Translocation ModelHirotaka Ando, Akihiro Hisaka and Hiroshi SuzukiDrug Metabolism and Disposition April 2015, 43 (4) 590-602; DOI: https://doi.org/10.1124/dmd.114.060038
Sveigaard, Helle H.
- You have accessPBPK Modeling to Unravel Nonlinear Pharmacokinetics of Verapamil to Estimate the Fractional Clearance for Verapamil N-Demethylation in the Recirculating Rat Liver PreparationQi Joy Yang, Luqin Si, Hui Tang, Helle H. Sveigaard, Edwin C. Y. Chow and K. Sandy PangDrug Metabolism and Disposition April 2015, 43 (4) 631-645; DOI: https://doi.org/10.1124/dmd.114.062265
T
Tang, Hui
- You have accessPBPK Modeling to Unravel Nonlinear Pharmacokinetics of Verapamil to Estimate the Fractional Clearance for Verapamil N-Demethylation in the Recirculating Rat Liver PreparationQi Joy Yang, Luqin Si, Hui Tang, Helle H. Sveigaard, Edwin C. Y. Chow and K. Sandy PangDrug Metabolism and Disposition April 2015, 43 (4) 631-645; DOI: https://doi.org/10.1124/dmd.114.062265
Taub, Mitchell E.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Tekwani, Babu L.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Toutain, Pierre-Louis
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Tse, Susanna
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Turcotte, Véronique
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
U
Upthagrove, Alana
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
V
Viguié, Catherine
- You have accessConjugation and Deconjugation Reactions within the Fetoplacental Compartment in a Sheep Model: A Key Factor Determining Bisphenol A Fetal ExposureTanguy Corbel, Elisabeth Perdu, Véronique Gayrard, Sylvie Puel, Marlène Z. Lacroix, Catherine Viguié, Pierre-Louis Toutain, Daniel Zalko and Nicole Picard-HagenDrug Metabolism and Disposition April 2015, 43 (4) 467-476; DOI: https://doi.org/10.1124/dmd.114.061291
Villeneuve, Lyne
- You have accessQuantitative Profiling of Human Renal UDP-glucuronosyltransferases and Glucuronidation Activity: A Comparison of Normal and Tumoral Kidney TissuesGuillaume Margaillan, Michèle Rouleau, John K. Fallon, Patrick Caron, Lyne Villeneuve, Véronique Turcotte, Philip C. Smith, Melanie S. Joy and Chantal GuillemetteDrug Metabolism and Disposition April 2015, 43 (4) 611-619; DOI: https://doi.org/10.1124/dmd.114.062877
W
Walker, Larry A.
- You have accessEnantioselective Pharmacokinetics of Primaquine in Healthy Human VolunteersBabu L. Tekwani, Bharathi Avula, Rajnish Sahu, Narayan D. Chaurasiya, Shabana I. Khan, Surendra Jain, Pius S. Fasinu, H.M.T. Bandara Herath, Donald Stanford, N.P. Dhammika Nanayakkara, James D. McChesney, Travis W. Yates, Mahmoud A. ElSohly, Ikhlas A. Khan and Larry A. WalkerDrug Metabolism and Disposition April 2015, 43 (4) 571-577; DOI: https://doi.org/10.1124/dmd.114.061127
Walsky, Robert L.
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Wang, Changxi
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Wang, Guangji
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Wang, Hong
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Wang, Hongyang
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Wang, Huailing
- You have accessCharacterization of Chrysin Glucuronidation in UGT1A1-Overexpressing HeLa Cells: Elucidating the Transporters Responsible for Efflux of GlucuronideEnxi Quan, Huailing Wang, Dong Dong, Xingwang Zhang and Baojian WuDrug Metabolism and Disposition April 2015, 43 (4) 433-443; DOI: https://doi.org/10.1124/dmd.114.061598
Wang, Ping
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Wang, Shuang-Hu
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Wang, Xueding
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Wang, Zeng-Shou
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Ware, Joseph A.
- You have accessBreast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study DesignCaroline A. Lee, Meeghan A. O’Connor, Tasha K. Ritchie, Aleksandra Galetin, Jack A. Cook, Isabelle Ragueneau-Majlessi, Harma Ellens, Bo Feng, Mitchell E. Taub, Mary F. Paine, Joseph W. Polli, Joseph A. Ware and Maciej J. Zamek-GliszczynskiDrug Metabolism and Disposition April 2015, 43 (4) 490-509; DOI: https://doi.org/10.1124/dmd.114.062174
Warren, Mark S.
- You have accessImpact on Creatinine Renal Clearance by the Interplay of Multiple Renal Transporters: A Case Study with INCB039110Yan Zhang, Mark S. Warren, Xuexiang Zhang, Sharon Diamond, Bill Williams, Naresh Punwani, Jane Huang, Yong Huang and Swamy YeleswaramDrug Metabolism and Disposition April 2015, 43 (4) 485-489; DOI: https://doi.org/10.1124/dmd.114.060673
Watanabe, Tomoko
- You have accessUtility of Bilirubins and Bile Acids as Endogenous Biomarkers for the Inhibition of Hepatic TransportersTomoko Watanabe, Manami Miyake, Toshinobu Shimizu, Miho Kamezawa, Naoya Masutomi, Takesada Shimura and Rikiya OhashiDrug Metabolism and Disposition April 2015, 43 (4) 459-466; DOI: https://doi.org/10.1124/dmd.114.061051
Wen, Bo
- You have accessContribution of Metabolites to P450 Inhibition–Based Drug–Drug Interactions: Scholarship from the Drug Metabolism Leadership Group of the Innovation and Quality Consortium Metabolite GroupHongbin Yu, Suresh K. Balani, Weichao Chen, Donghui Cui, Ling He, W. Griffith Humphreys, Jialin Mao, W. George Lai, Anthony J. Lee, Heng-Keang Lim, Christopher MacLauchlin, Chandra Prakash, Sekhar Surapaneni, Susanna Tse, Alana Upthagrove, Robert L. Walsky, Bo Wen and Zhaopie ZengDrug Metabolism and Disposition April 2015, 43 (4) 620-630; DOI: https://doi.org/10.1124/dmd.114.059345
Williams, Bill
- You have accessImpact on Creatinine Renal Clearance by the Interplay of Multiple Renal Transporters: A Case Study with INCB039110Yan Zhang, Mark S. Warren, Xuexiang Zhang, Sharon Diamond, Bill Williams, Naresh Punwani, Jane Huang, Yong Huang and Swamy YeleswaramDrug Metabolism and Disposition April 2015, 43 (4) 485-489; DOI: https://doi.org/10.1124/dmd.114.060673
Wu, Baojian
- You have accessCharacterization of Chrysin Glucuronidation in UGT1A1-Overexpressing HeLa Cells: Elucidating the Transporters Responsible for Efflux of GlucuronideEnxi Quan, Huailing Wang, Dong Dong, Xingwang Zhang and Baojian WuDrug Metabolism and Disposition April 2015, 43 (4) 433-443; DOI: https://doi.org/10.1124/dmd.114.061598
X
Xia, Yang-Liu
- You have accessStructural Modifications at the C-4 Position Strongly Affect the Glucuronidation of 6,7-DihydroxycoumarinsYang-Liu Xia, Guang-Bo Ge, Ping Wang, Si-Cheng Liang, Yu-Qi He, Jing Ning, Xing-Kai Qian, Yan Li and Ling YangDrug Metabolism and Disposition April 2015, 43 (4) 553-560; DOI: https://doi.org/10.1124/dmd.114.060681
Xie, Yang
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Xie, Yuan
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Xu, Tao
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Y
Yan, Tingting
- You have accessMechanism-Based Inhibitory and Peroxisome Proliferator-Activated Receptor α–Dependent Modulating Effects of Silybin on Principal Hepatic Drug-Metabolizing EnzymesHong Wang, Tingting Yan, Yuan Xie, Min Zhao, Yuan Che, Jun Zhang, Huiying Liu, Lijuan Cao, Xuefang Cheng, Yang Xie, Feiyan Li, Qu Qi, Guangji Wang and Haiping HaoDrug Metabolism and Disposition April 2015, 43 (4) 444-454; DOI: https://doi.org/10.1124/dmd.114.061622
Yang, Fukang
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
Yang, Li-Ping
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Yang, Ling
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Yang, Qi Joy
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Yates, Travis W.
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Yeleswaram, Swamy
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Yerino, Phyllis
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Yu, Hongbin
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Zamek-Gliszczynski, Maciej J.
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Zeng, Zhaopie
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Zhang, Jun
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Zhang, Yan
- You have accessImpact on Creatinine Renal Clearance by the Interplay of Multiple Renal Transporters: A Case Study with INCB039110Yan Zhang, Mark S. Warren, Xuexiang Zhang, Sharon Diamond, Bill Williams, Naresh Punwani, Jane Huang, Yong Huang and Swamy YeleswaramDrug Metabolism and Disposition April 2015, 43 (4) 485-489; DOI: https://doi.org/10.1124/dmd.114.060673
Zhang, Yu
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Zhu, Chen
- You have accessAssociations of HSD11B1 Polymorphisms with Tacrolimus Concentrations in Chinese Renal Transplant Recipients with Prednisone Combined TherapyXiaoman Liu, Jiali Li, Qian Fu, Shu Liu, Yu Zhang, Xueding Wang, Hongyang Wang, Jun Li, Chen Zhu, Changxi Wang and Min HuangDrug Metabolism and Disposition April 2015, 43 (4) 455-458; DOI: https://doi.org/10.1124/dmd.114.062117
Zhu, Guang-Hui
- You have accessIn Vitro and In Vivo Characterization of 13 CYP2C9 Allelic Variants Found in Chinese Han PopulationGuo-Xin Hu, Pei-Pei Pan, Zeng-Shou Wang, Li-Ping Yang, Da-Peng Dai, Shuang-Hu Wang, Guang-Hui Zhu, Xiang-Jun Qiu, Tao Xu, Jun Luo, Qing-Quan Lian, Ren-Shan Ge and Jian-Ping CaiDrug Metabolism and Disposition April 2015, 43 (4) 561-569; DOI: https://doi.org/10.1124/dmd.114.061200
Zhuo, Xiaoliang
- You have accessIdentification of Glutathione Conjugates of Acetylene-Containing Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5Xiaoliang Zhuo, Xiaohua Stella Huang, Andrew P. Degnan, Lawrence B. Snyder, Fukang Yang, Hong Huang, Yue-Zhong Shu and Benjamin M. JohnsonDrug Metabolism and Disposition April 2015, 43 (4) 578-589; DOI: https://doi.org/10.1124/dmd.114.061879
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