Index by author
September 01, 2015; Volume 43,Issue 9
A
Ajamie, Rose T.
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Azuma, Yoshiaki
- You have accessSUMOylation and Ubiquitylation Circuitry Controls Pregnane X Receptor Biology in HepatocytesWenqi Cui, Mengxi Sun, Nadezhda Galeva, Todd D. Williams, Yoshiaki Azuma and Jeff L. StaudingerDrug Metabolism and Disposition September 2015, 43 (9) 1316-1325; DOI: https://doi.org/10.1124/dmd.115.065201
B
Barbara, Joanna E.
- You have accessFurther Characterization of the Metabolism of Desloratadine and Its Cytochrome P450 and UDP-glucuronosyltransferase Inhibition Potential: Identification of Desloratadine as a Relatively Selective UGT2B10 InhibitorFaraz Kazmi, Phyllis Yerino, Joanna E. Barbara and Andrew ParkinsonDrug Metabolism and Disposition September 2015, 43 (9) 1294-1302; DOI: https://doi.org/10.1124/dmd.115.065011
Bian, Yicong
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
Boucaut, David
- You have accessCross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin AntagonistHugues Chanteux, Ludovicus Staelens, Valérie Mancel, Brigitte Gerin, David Boucaut, Chandra Prakash and Jean-Marie NicolasDrug Metabolism and Disposition September 2015, 43 (9) 1381-1391; DOI: https://doi.org/10.1124/dmd.115.064436
Bromek, Ewa
- You have accessDamage to the Brain Serotonergic System Increases the Expression of Liver Cytochrome P450Marta Rysz, Ewa Bromek, Anna Haduch, Anna Sadakierska-Chudy and Władysława A. DanielDrug Metabolism and Disposition September 2015, 43 (9) 1345-1352; DOI: https://doi.org/10.1124/dmd.115.064980
C
Caron, Patrick
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Chanteux, Hugues
- You have accessCross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin AntagonistHugues Chanteux, Ludovicus Staelens, Valérie Mancel, Brigitte Gerin, David Boucaut, Chandra Prakash and Jean-Marie NicolasDrug Metabolism and Disposition September 2015, 43 (9) 1381-1391; DOI: https://doi.org/10.1124/dmd.115.064436
Chen, Gang
- You have accessMilk Thistle Constituents Inhibit Raloxifene Intestinal Glucuronidation: A Potential Clinically Relevant Natural Product–Drug InteractionBrandon T. Gufford, Gang Chen, Ana G. Vergara, Philip Lazarus, Nicholas H. Oberlies and Mary F. PaineDrug Metabolism and Disposition September 2015, 43 (9) 1353-1359; DOI: https://doi.org/10.1124/dmd.115.065086
Cui, Wenqi
- You have accessSUMOylation and Ubiquitylation Circuitry Controls Pregnane X Receptor Biology in HepatocytesWenqi Cui, Mengxi Sun, Nadezhda Galeva, Todd D. Williams, Yoshiaki Azuma and Jeff L. StaudingerDrug Metabolism and Disposition September 2015, 43 (9) 1316-1325; DOI: https://doi.org/10.1124/dmd.115.065201
D
Daniel, Władysława A.
- You have accessDamage to the Brain Serotonergic System Increases the Expression of Liver Cytochrome P450Marta Rysz, Ewa Bromek, Anna Haduch, Anna Sadakierska-Chudy and Władysława A. DanielDrug Metabolism and Disposition September 2015, 43 (9) 1345-1352; DOI: https://doi.org/10.1124/dmd.115.064980
De Dios, Alfonso
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Ding, Xinxin
- You have accessOpioid Analgesia in P450 Gene Cluster Knockout Mice: A Search for Analgesia-Relevant IsoformsLindsay B. Hough, Julia W. Nalwalk, Xinxin Ding and Nico ScheerDrug Metabolism and Disposition September 2015, 43 (9) 1326-1330; DOI: https://doi.org/10.1124/dmd.115.065490
F
Fallon, John K.
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Fanslow, William C.
- You have accessIntracellular Catabolism of an Antibody Drug Conjugate with a Noncleavable LinkerBrooke M. Rock, Mark E. Tometsko, Sonal K. Patel, Kevin J. Hamblett, William C. Fanslow and Dan A. RockDrug Metabolism and Disposition September 2015, 43 (9) 1341-1344; DOI: https://doi.org/10.1124/dmd.115.064253
G
Galeva, Nadezhda
- You have accessSUMOylation and Ubiquitylation Circuitry Controls Pregnane X Receptor Biology in HepatocytesWenqi Cui, Mengxi Sun, Nadezhda Galeva, Todd D. Williams, Yoshiaki Azuma and Jeff L. StaudingerDrug Metabolism and Disposition September 2015, 43 (9) 1316-1325; DOI: https://doi.org/10.1124/dmd.115.065201
Gelbert, Lawrence M.
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Gerin, Brigitte
- You have accessCross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin AntagonistHugues Chanteux, Ludovicus Staelens, Valérie Mancel, Brigitte Gerin, David Boucaut, Chandra Prakash and Jean-Marie NicolasDrug Metabolism and Disposition September 2015, 43 (9) 1381-1391; DOI: https://doi.org/10.1124/dmd.115.064436
Goldman, Jennifer L.
- You have accessIn Vitro Hepatic Oxidative Biotransformation of TrimethoprimJennifer L. Goldman, J. Steven Leeder, Leon Van Haandel and Robin E. PearceDrug Metabolism and Disposition September 2015, 43 (9) 1372-1380; DOI: https://doi.org/10.1124/dmd.115.065193
Gufford, Brandon T.
- You have accessMilk Thistle Constituents Inhibit Raloxifene Intestinal Glucuronidation: A Potential Clinically Relevant Natural Product–Drug InteractionBrandon T. Gufford, Gang Chen, Ana G. Vergara, Philip Lazarus, Nicholas H. Oberlies and Mary F. PaineDrug Metabolism and Disposition September 2015, 43 (9) 1353-1359; DOI: https://doi.org/10.1124/dmd.115.065086
Guillemette, Chantal
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Guo, Kenan
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
H
Haduch, Anna
- You have accessDamage to the Brain Serotonergic System Increases the Expression of Liver Cytochrome P450Marta Rysz, Ewa Bromek, Anna Haduch, Anna Sadakierska-Chudy and Władysława A. DanielDrug Metabolism and Disposition September 2015, 43 (9) 1345-1352; DOI: https://doi.org/10.1124/dmd.115.064980
Hamblett, Kevin J.
- You have accessIntracellular Catabolism of an Antibody Drug Conjugate with a Noncleavable LinkerBrooke M. Rock, Mark E. Tometsko, Sonal K. Patel, Kevin J. Hamblett, William C. Fanslow and Dan A. RockDrug Metabolism and Disposition September 2015, 43 (9) 1341-1344; DOI: https://doi.org/10.1124/dmd.115.064253
Hough, Lindsay B.
- You have accessOpioid Analgesia in P450 Gene Cluster Knockout Mice: A Search for Analgesia-Relevant IsoformsLindsay B. Hough, Julia W. Nalwalk, Xinxin Ding and Nico ScheerDrug Metabolism and Disposition September 2015, 43 (9) 1326-1330; DOI: https://doi.org/10.1124/dmd.115.065490
Hu, Haihong
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
J
Jiang, Huidi
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
K
Kazmi, Faraz
- You have accessFurther Characterization of the Metabolism of Desloratadine and Its Cytochrome P450 and UDP-glucuronosyltransferase Inhibition Potential: Identification of Desloratadine as a Relatively Selective UGT2B10 InhibitorFaraz Kazmi, Phyllis Yerino, Joanna E. Barbara and Andrew ParkinsonDrug Metabolism and Disposition September 2015, 43 (9) 1294-1302; DOI: https://doi.org/10.1124/dmd.115.065011
Kitagawara, Yumina
- You have accessNovel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450Yumina Kitagawara, Tomoyuki Ohe, Kumiko Tachibana, Kyoko Takahashi, Shigeo Nakamura and Tadahiko MashinoDrug Metabolism and Disposition September 2015, 43 (9) 1303-1306; DOI: https://doi.org/10.1124/dmd.115.065037
Klein, Kathrin
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Kulanthaivel, Palaniappan
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
L
Lazarus, Philip
- You have accessMilk Thistle Constituents Inhibit Raloxifene Intestinal Glucuronidation: A Potential Clinically Relevant Natural Product–Drug InteractionBrandon T. Gufford, Gang Chen, Ana G. Vergara, Philip Lazarus, Nicholas H. Oberlies and Mary F. PaineDrug Metabolism and Disposition September 2015, 43 (9) 1353-1359; DOI: https://doi.org/10.1124/dmd.115.065086
Leeder, J. Steven
- You have accessIn Vitro Hepatic Oxidative Biotransformation of TrimethoprimJennifer L. Goldman, J. Steven Leeder, Leon Van Haandel and Robin E. PearceDrug Metabolism and Disposition September 2015, 43 (9) 1372-1380; DOI: https://doi.org/10.1124/dmd.115.065193
Lei, Jinxiu
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
Li, Hui
- You have accessInfluence of ABCB1 Genotype in Collies on the Pharmacokinetics and Pharmacodynamics of Loperamide in a Dose-Escalation StudyMichael J. Myers, Marilyn Martinez, Hui Li, Junshan Qiu, Lisa Troutman, Michele Sharkey and Haile F. YancyDrug Metabolism and Disposition September 2015, 43 (9) 1392-1407; DOI: https://doi.org/10.1124/dmd.115.063735
M
Mancel, Valérie
- You have accessCross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin AntagonistHugues Chanteux, Ludovicus Staelens, Valérie Mancel, Brigitte Gerin, David Boucaut, Chandra Prakash and Jean-Marie NicolasDrug Metabolism and Disposition September 2015, 43 (9) 1381-1391; DOI: https://doi.org/10.1124/dmd.115.064436
Margaillan, Guillaume
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Martinez, Marilyn
- You have accessInfluence of ABCB1 Genotype in Collies on the Pharmacokinetics and Pharmacodynamics of Loperamide in a Dose-Escalation StudyMichael J. Myers, Marilyn Martinez, Hui Li, Junshan Qiu, Lisa Troutman, Michele Sharkey and Haile F. YancyDrug Metabolism and Disposition September 2015, 43 (9) 1392-1407; DOI: https://doi.org/10.1124/dmd.115.063735
Mashino, Tadahiko
- You have accessNovel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450Yumina Kitagawara, Tomoyuki Ohe, Kumiko Tachibana, Kyoko Takahashi, Shigeo Nakamura and Tadahiko MashinoDrug Metabolism and Disposition September 2015, 43 (9) 1303-1306; DOI: https://doi.org/10.1124/dmd.115.065037
Myers, Michael J.
- You have accessInfluence of ABCB1 Genotype in Collies on the Pharmacokinetics and Pharmacodynamics of Loperamide in a Dose-Escalation StudyMichael J. Myers, Marilyn Martinez, Hui Li, Junshan Qiu, Lisa Troutman, Michele Sharkey and Haile F. YancyDrug Metabolism and Disposition September 2015, 43 (9) 1392-1407; DOI: https://doi.org/10.1124/dmd.115.063735
N
Nakamura, Shigeo
- You have accessNovel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450Yumina Kitagawara, Tomoyuki Ohe, Kumiko Tachibana, Kyoko Takahashi, Shigeo Nakamura and Tadahiko MashinoDrug Metabolism and Disposition September 2015, 43 (9) 1303-1306; DOI: https://doi.org/10.1124/dmd.115.065037
Nalwalk, Julia W.
- You have accessOpioid Analgesia in P450 Gene Cluster Knockout Mice: A Search for Analgesia-Relevant IsoformsLindsay B. Hough, Julia W. Nalwalk, Xinxin Ding and Nico ScheerDrug Metabolism and Disposition September 2015, 43 (9) 1326-1330; DOI: https://doi.org/10.1124/dmd.115.065490
Nicolas, Jean-Marie
- You have accessCross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin AntagonistHugues Chanteux, Ludovicus Staelens, Valérie Mancel, Brigitte Gerin, David Boucaut, Chandra Prakash and Jean-Marie NicolasDrug Metabolism and Disposition September 2015, 43 (9) 1381-1391; DOI: https://doi.org/10.1124/dmd.115.064436
O
Oberlies, Nicholas H.
- You have accessMilk Thistle Constituents Inhibit Raloxifene Intestinal Glucuronidation: A Potential Clinically Relevant Natural Product–Drug InteractionBrandon T. Gufford, Gang Chen, Ana G. Vergara, Philip Lazarus, Nicholas H. Oberlies and Mary F. PaineDrug Metabolism and Disposition September 2015, 43 (9) 1353-1359; DOI: https://doi.org/10.1124/dmd.115.065086
Ohe, Tomoyuki
- You have accessNovel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450Yumina Kitagawara, Tomoyuki Ohe, Kumiko Tachibana, Kyoko Takahashi, Shigeo Nakamura and Tadahiko MashinoDrug Metabolism and Disposition September 2015, 43 (9) 1303-1306; DOI: https://doi.org/10.1124/dmd.115.065037
P
Paine, Mary F.
- You have accessMilk Thistle Constituents Inhibit Raloxifene Intestinal Glucuronidation: A Potential Clinically Relevant Natural Product–Drug InteractionBrandon T. Gufford, Gang Chen, Ana G. Vergara, Philip Lazarus, Nicholas H. Oberlies and Mary F. PaineDrug Metabolism and Disposition September 2015, 43 (9) 1353-1359; DOI: https://doi.org/10.1124/dmd.115.065086
Parkinson, Andrew
- You have accessFurther Characterization of the Metabolism of Desloratadine and Its Cytochrome P450 and UDP-glucuronosyltransferase Inhibition Potential: Identification of Desloratadine as a Relatively Selective UGT2B10 InhibitorFaraz Kazmi, Phyllis Yerino, Joanna E. Barbara and Andrew ParkinsonDrug Metabolism and Disposition September 2015, 43 (9) 1294-1302; DOI: https://doi.org/10.1124/dmd.115.065011
Patel, Sonal K.
- You have accessIntracellular Catabolism of an Antibody Drug Conjugate with a Noncleavable LinkerBrooke M. Rock, Mark E. Tometsko, Sonal K. Patel, Kevin J. Hamblett, William C. Fanslow and Dan A. RockDrug Metabolism and Disposition September 2015, 43 (9) 1341-1344; DOI: https://doi.org/10.1124/dmd.115.064253
Pearce, Robin E.
- You have accessIn Vitro Hepatic Oxidative Biotransformation of TrimethoprimJennifer L. Goldman, J. Steven Leeder, Leon Van Haandel and Robin E. PearceDrug Metabolism and Disposition September 2015, 43 (9) 1372-1380; DOI: https://doi.org/10.1124/dmd.115.065193
Prakash, Chandra
- You have accessCross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin AntagonistHugues Chanteux, Ludovicus Staelens, Valérie Mancel, Brigitte Gerin, David Boucaut, Chandra Prakash and Jean-Marie NicolasDrug Metabolism and Disposition September 2015, 43 (9) 1381-1391; DOI: https://doi.org/10.1124/dmd.115.064436
Q
Qiu, Junshan
- You have accessInfluence of ABCB1 Genotype in Collies on the Pharmacokinetics and Pharmacodynamics of Loperamide in a Dose-Escalation StudyMichael J. Myers, Marilyn Martinez, Hui Li, Junshan Qiu, Lisa Troutman, Michele Sharkey and Haile F. YancyDrug Metabolism and Disposition September 2015, 43 (9) 1392-1407; DOI: https://doi.org/10.1124/dmd.115.063735
R
Ramsden, Diane
- You have accessDetermination of a Degradation Constant for CYP3A4 by Direct Suppression of mRNA in a Novel Human Hepatocyte Model, HepatoPacDiane Ramsden, Jin Zhou and Donald J. TweedieDrug Metabolism and Disposition September 2015, 43 (9) 1307-1315; DOI: https://doi.org/10.1124/dmd.115.065326
Raub, Thomas J.
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Rock, Brooke M.
- You have accessIntracellular Catabolism of an Antibody Drug Conjugate with a Noncleavable LinkerBrooke M. Rock, Mark E. Tometsko, Sonal K. Patel, Kevin J. Hamblett, William C. Fanslow and Dan A. RockDrug Metabolism and Disposition September 2015, 43 (9) 1341-1344; DOI: https://doi.org/10.1124/dmd.115.064253
Rock, Dan A.
- You have accessIntracellular Catabolism of an Antibody Drug Conjugate with a Noncleavable LinkerBrooke M. Rock, Mark E. Tometsko, Sonal K. Patel, Kevin J. Hamblett, William C. Fanslow and Dan A. RockDrug Metabolism and Disposition September 2015, 43 (9) 1341-1344; DOI: https://doi.org/10.1124/dmd.115.064253
Rouleau, Michèle
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Rysz, Marta
- You have accessDamage to the Brain Serotonergic System Increases the Expression of Liver Cytochrome P450Marta Rysz, Ewa Bromek, Anna Haduch, Anna Sadakierska-Chudy and Władysława A. DanielDrug Metabolism and Disposition September 2015, 43 (9) 1345-1352; DOI: https://doi.org/10.1124/dmd.115.064980
S
Sadakierska-Chudy, Anna
- You have accessDamage to the Brain Serotonergic System Increases the Expression of Liver Cytochrome P450Marta Rysz, Ewa Bromek, Anna Haduch, Anna Sadakierska-Chudy and Władysława A. DanielDrug Metabolism and Disposition September 2015, 43 (9) 1345-1352; DOI: https://doi.org/10.1124/dmd.115.064980
Sanchez-Martinez, Concepcion
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Sawada, Geri A.
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Scheer, Nico
- You have accessOpioid Analgesia in P450 Gene Cluster Knockout Mice: A Search for Analgesia-Relevant IsoformsLindsay B. Hough, Julia W. Nalwalk, Xinxin Ding and Nico ScheerDrug Metabolism and Disposition September 2015, 43 (9) 1326-1330; DOI: https://doi.org/10.1124/dmd.115.065490
Shang, Haitao
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
Shannon, Harlan E.
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Sharkey, Michele
- You have accessInfluence of ABCB1 Genotype in Collies on the Pharmacokinetics and Pharmacodynamics of Loperamide in a Dose-Escalation StudyMichael J. Myers, Marilyn Martinez, Hui Li, Junshan Qiu, Lisa Troutman, Michele Sharkey and Haile F. YancyDrug Metabolism and Disposition September 2015, 43 (9) 1392-1407; DOI: https://doi.org/10.1124/dmd.115.063735
Smith, Philip C.
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Staelens, Ludovicus
- You have accessCross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin AntagonistHugues Chanteux, Ludovicus Staelens, Valérie Mancel, Brigitte Gerin, David Boucaut, Chandra Prakash and Jean-Marie NicolasDrug Metabolism and Disposition September 2015, 43 (9) 1381-1391; DOI: https://doi.org/10.1124/dmd.115.064436
Staton, Brian A.
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Staudinger, Jeff L.
- You have accessSUMOylation and Ubiquitylation Circuitry Controls Pregnane X Receptor Biology in HepatocytesWenqi Cui, Mengxi Sun, Nadezhda Galeva, Todd D. Williams, Yoshiaki Azuma and Jeff L. StaudingerDrug Metabolism and Disposition September 2015, 43 (9) 1316-1325; DOI: https://doi.org/10.1124/dmd.115.065201
Sun, Mengxi
- You have accessSUMOylation and Ubiquitylation Circuitry Controls Pregnane X Receptor Biology in HepatocytesWenqi Cui, Mengxi Sun, Nadezhda Galeva, Todd D. Williams, Yoshiaki Azuma and Jeff L. StaudingerDrug Metabolism and Disposition September 2015, 43 (9) 1316-1325; DOI: https://doi.org/10.1124/dmd.115.065201
T
Tachibana, Kumiko
- You have accessNovel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450Yumina Kitagawara, Tomoyuki Ohe, Kumiko Tachibana, Kyoko Takahashi, Shigeo Nakamura and Tadahiko MashinoDrug Metabolism and Disposition September 2015, 43 (9) 1303-1306; DOI: https://doi.org/10.1124/dmd.115.065037
Takahashi, Kyoko
- You have accessNovel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450Yumina Kitagawara, Tomoyuki Ohe, Kumiko Tachibana, Kyoko Takahashi, Shigeo Nakamura and Tadahiko MashinoDrug Metabolism and Disposition September 2015, 43 (9) 1303-1306; DOI: https://doi.org/10.1124/dmd.115.065037
Tometsko, Mark E.
- You have accessIntracellular Catabolism of an Antibody Drug Conjugate with a Noncleavable LinkerBrooke M. Rock, Mark E. Tometsko, Sonal K. Patel, Kevin J. Hamblett, William C. Fanslow and Dan A. RockDrug Metabolism and Disposition September 2015, 43 (9) 1341-1344; DOI: https://doi.org/10.1124/dmd.115.064253
Troutman, Lisa
- You have accessInfluence of ABCB1 Genotype in Collies on the Pharmacokinetics and Pharmacodynamics of Loperamide in a Dose-Escalation StudyMichael J. Myers, Marilyn Martinez, Hui Li, Junshan Qiu, Lisa Troutman, Michele Sharkey and Haile F. YancyDrug Metabolism and Disposition September 2015, 43 (9) 1392-1407; DOI: https://doi.org/10.1124/dmd.115.063735
Tweedie, Donald J.
- You have accessDetermination of a Degradation Constant for CYP3A4 by Direct Suppression of mRNA in a Novel Human Hepatocyte Model, HepatoPacDiane Ramsden, Jin Zhou and Donald J. TweedieDrug Metabolism and Disposition September 2015, 43 (9) 1307-1315; DOI: https://doi.org/10.1124/dmd.115.065326
V
Van Haandel, Leon
- You have accessIn Vitro Hepatic Oxidative Biotransformation of TrimethoprimJennifer L. Goldman, J. Steven Leeder, Leon Van Haandel and Robin E. PearceDrug Metabolism and Disposition September 2015, 43 (9) 1372-1380; DOI: https://doi.org/10.1124/dmd.115.065193
Vergara, Ana G.
- You have accessMilk Thistle Constituents Inhibit Raloxifene Intestinal Glucuronidation: A Potential Clinically Relevant Natural Product–Drug InteractionBrandon T. Gufford, Gang Chen, Ana G. Vergara, Philip Lazarus, Nicholas H. Oberlies and Mary F. PaineDrug Metabolism and Disposition September 2015, 43 (9) 1353-1359; DOI: https://doi.org/10.1124/dmd.115.065086
Villeneuve, Lyne
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
W
Wei, Hong
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
Williams, Todd D.
- You have accessSUMOylation and Ubiquitylation Circuitry Controls Pregnane X Receptor Biology in HepatocytesWenqi Cui, Mengxi Sun, Nadezhda Galeva, Todd D. Williams, Yoshiaki Azuma and Jeff L. StaudingerDrug Metabolism and Disposition September 2015, 43 (9) 1316-1325; DOI: https://doi.org/10.1124/dmd.115.065201
Wishart, Graham N.
- You have accessBrain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma XenograftThomas J. Raub, Graham N. Wishart, Palaniappan Kulanthaivel, Brian A. Staton, Rose T. Ajamie, Geri A. Sawada, Lawrence M. Gelbert, Harlan E. Shannon, Concepcion Sanchez-Martinez and Alfonso De DiosDrug Metabolism and Disposition September 2015, 43 (9) 1360-1371; DOI: https://doi.org/10.1124/dmd.114.062745
Y
Yancy, Haile F.
- You have accessInfluence of ABCB1 Genotype in Collies on the Pharmacokinetics and Pharmacodynamics of Loperamide in a Dose-Escalation StudyMichael J. Myers, Marilyn Martinez, Hui Li, Junshan Qiu, Lisa Troutman, Michele Sharkey and Haile F. YancyDrug Metabolism and Disposition September 2015, 43 (9) 1392-1407; DOI: https://doi.org/10.1124/dmd.115.063735
Yao, Qingqing
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
Yerino, Phyllis
- You have accessFurther Characterization of the Metabolism of Desloratadine and Its Cytochrome P450 and UDP-glucuronosyltransferase Inhibition Potential: Identification of Desloratadine as a Relatively Selective UGT2B10 InhibitorFaraz Kazmi, Phyllis Yerino, Joanna E. Barbara and Andrew ParkinsonDrug Metabolism and Disposition September 2015, 43 (9) 1294-1302; DOI: https://doi.org/10.1124/dmd.115.065011
Yu, Lushan
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
Z
Zanger, Ulrich M.
- You have accessMultiplexed Targeted Quantitative Proteomics Predicts Hepatic Glucuronidation PotentialGuillaume Margaillan, Michèle Rouleau, Kathrin Klein, John K. Fallon, Patrick Caron, Lyne Villeneuve, Philip C. Smith, Ulrich M. Zanger and Chantal GuillemetteDrug Metabolism and Disposition September 2015, 43 (9) 1331-1335; DOI: https://doi.org/10.1124/dmd.115.065391
Zeng, Su
- You have accessExpression of Bama Minipig and Human CYP3A Enzymes: Comparison of the Catalytic Characteristics with Each Other and Their Liver MicrosomesYicong Bian, Qingqing Yao, Haitao Shang, Jinxiu Lei, Haihong Hu, Kenan Guo, Huidi Jiang, Lushan Yu, Hong Wei and Su ZengDrug Metabolism and Disposition September 2015, 43 (9) 1336-1340; DOI: https://doi.org/10.1124/dmd.115.064717
Zhou, Jin
- You have accessDetermination of a Degradation Constant for CYP3A4 by Direct Suppression of mRNA in a Novel Human Hepatocyte Model, HepatoPacDiane Ramsden, Jin Zhou and Donald J. TweedieDrug Metabolism and Disposition September 2015, 43 (9) 1307-1315; DOI: https://doi.org/10.1124/dmd.115.065326
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