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Bioactivation of Trimethoprim to Protein-Reactive Metabolites in Human Liver Microsomes
Jennifer L. Goldman, Yakov M. Koen, Steven A. Rogers, Kelin Li, James S. Leeder and Robert P. Hanzlik
Drug Metabolism and Disposition October 2016, 44 (10) 1603-1607; DOI: https://doi.org/10.1124/dmd.116.072041
Jennifer L. Goldman
Divisions of Clinical Pharmacology, Toxicology, and Therapeutic Innovation, Children’s Mercy Hospital, University of Missouri, Kansas City, Missouri (J.L.G., J.S.L.); Department of Medicinal Chemistry, University of Kansas School of Pharmacy, Lawrence, Kansas (Y.M.K., R.P.H.); Baker & McKenzie LLP, Dallas, Texas (S.A.R.); and Center for Integrative Chemical Biology and Drug Discovery, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina (K.L.)
Yakov M. Koen
Divisions of Clinical Pharmacology, Toxicology, and Therapeutic Innovation, Children’s Mercy Hospital, University of Missouri, Kansas City, Missouri (J.L.G., J.S.L.); Department of Medicinal Chemistry, University of Kansas School of Pharmacy, Lawrence, Kansas (Y.M.K., R.P.H.); Baker & McKenzie LLP, Dallas, Texas (S.A.R.); and Center for Integrative Chemical Biology and Drug Discovery, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina (K.L.)
Steven A. Rogers
Divisions of Clinical Pharmacology, Toxicology, and Therapeutic Innovation, Children’s Mercy Hospital, University of Missouri, Kansas City, Missouri (J.L.G., J.S.L.); Department of Medicinal Chemistry, University of Kansas School of Pharmacy, Lawrence, Kansas (Y.M.K., R.P.H.); Baker & McKenzie LLP, Dallas, Texas (S.A.R.); and Center for Integrative Chemical Biology and Drug Discovery, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina (K.L.)
Kelin Li
Divisions of Clinical Pharmacology, Toxicology, and Therapeutic Innovation, Children’s Mercy Hospital, University of Missouri, Kansas City, Missouri (J.L.G., J.S.L.); Department of Medicinal Chemistry, University of Kansas School of Pharmacy, Lawrence, Kansas (Y.M.K., R.P.H.); Baker & McKenzie LLP, Dallas, Texas (S.A.R.); and Center for Integrative Chemical Biology and Drug Discovery, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina (K.L.)
James S. Leeder
Divisions of Clinical Pharmacology, Toxicology, and Therapeutic Innovation, Children’s Mercy Hospital, University of Missouri, Kansas City, Missouri (J.L.G., J.S.L.); Department of Medicinal Chemistry, University of Kansas School of Pharmacy, Lawrence, Kansas (Y.M.K., R.P.H.); Baker & McKenzie LLP, Dallas, Texas (S.A.R.); and Center for Integrative Chemical Biology and Drug Discovery, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina (K.L.)
Robert P. Hanzlik
Divisions of Clinical Pharmacology, Toxicology, and Therapeutic Innovation, Children’s Mercy Hospital, University of Missouri, Kansas City, Missouri (J.L.G., J.S.L.); Department of Medicinal Chemistry, University of Kansas School of Pharmacy, Lawrence, Kansas (Y.M.K., R.P.H.); Baker & McKenzie LLP, Dallas, Texas (S.A.R.); and Center for Integrative Chemical Biology and Drug Discovery, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina (K.L.)
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Rapid CommunicationShort Communication
Covalent Protein Binding of Trimethoprim In Vitro
Jennifer L. Goldman, Yakov M. Koen, Steven A. Rogers, Kelin Li, James S. Leeder and Robert P. Hanzlik
Drug Metabolism and Disposition October 1, 2016, 44 (10) 1603-1607; DOI: https://doi.org/10.1124/dmd.116.072041
Rapid CommunicationShort Communication
Covalent Protein Binding of Trimethoprim In Vitro
Jennifer L. Goldman, Yakov M. Koen, Steven A. Rogers, Kelin Li, James S. Leeder and Robert P. Hanzlik
Drug Metabolism and Disposition October 1, 2016, 44 (10) 1603-1607; DOI: https://doi.org/10.1124/dmd.116.072041
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