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Antibody Drug Conjugates Differentiate Uptake and DNA Alkylation of Pyrrolobenzodiazepines in Tumors from Organs of Xenograft Mice
Yong Ma, S. Cyrus Khojasteh, Cornelis E.C.A. Hop, Hans K. Erickson, Andrew Polson, Thomas H. Pillow, Shang-Fan Yu, Hong Wang, Peter S. Dragovich and Donglu Zhang
Drug Metabolism and Disposition December 2016, 44 (12) 1958-1962; DOI: https://doi.org/10.1124/dmd.116.073031
Yong Ma
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
S. Cyrus Khojasteh
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Cornelis E.C.A. Hop
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Hans K. Erickson
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Andrew Polson
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Thomas H. Pillow
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Shang-Fan Yu
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Hong Wang
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Peter S. Dragovich
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California
Donglu Zhang
Drug Metabolism & Pharmacokinetics (Y.M., S.C.K., C.E.C.A.H., D.Z.), Discovery Chemistry (T.H.P., P.S.D.), Translational Oncology (A.P., S.-F.Y.), Protein Chemistry (H.K.E.), and Development Toxicology (H.W.), Genentech, South San Francisco, California

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Rapid CommunicationShort Communication
Mechanism of Action of ADC Carrying Pyrrolobenzodiazepine
Yong Ma, S. Cyrus Khojasteh, Cornelis E.C.A. Hop, Hans K. Erickson, Andrew Polson, Thomas H. Pillow, Shang-Fan Yu, Hong Wang, Peter S. Dragovich and Donglu Zhang
Drug Metabolism and Disposition December 1, 2016, 44 (12) 1958-1962; DOI: https://doi.org/10.1124/dmd.116.073031
Rapid CommunicationShort Communication
Mechanism of Action of ADC Carrying Pyrrolobenzodiazepine
Yong Ma, S. Cyrus Khojasteh, Cornelis E.C.A. Hop, Hans K. Erickson, Andrew Polson, Thomas H. Pillow, Shang-Fan Yu, Hong Wang, Peter S. Dragovich and Donglu Zhang
Drug Metabolism and Disposition December 1, 2016, 44 (12) 1958-1962; DOI: https://doi.org/10.1124/dmd.116.073031
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