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Hepatocellular Disposition and Transporter Interactions with Tolvaptan and Metabolites in Sandwich-Cultured Human Hepatocytes
Yang Lu, Jason R. Slizgi, Kenneth R. Brouwer, Robert L. St. Claire, Kimberly M. Freeman, Maxwell Pan, William J. Brock and Kim L. R. Brouwer
Drug Metabolism and Disposition June 2016, 44 (6) 867-870; DOI: https://doi.org/10.1124/dmd.115.067629
Yang Lu
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)
Jason R. Slizgi
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)
Kenneth R. Brouwer
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)
Robert L. St. Claire
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)
Kimberly M. Freeman
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)
Maxwell Pan
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)
William J. Brock
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)
Kim L. R. Brouwer
Division of Pharmacotherapy and Experimental Therapeutics, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina (Y.L., J.R.S., K.L.R.B); Qualyst Transporter Solutions, Durham, North Carolina (K.R.B., R.L.S.C., K.M.F); Otsuka PDC, Inc., Rockville, Maryland (M.P.); Brock Scientific Consulting, Montgomery Village, Maryland (W.J.B.)

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Rapid CommunicationShort Communication
Tolvaptan Disposition and DDIs in SCHH
Yang Lu, Jason R. Slizgi, Kenneth R. Brouwer, Robert L. St. Claire, Kimberly M. Freeman, Maxwell Pan, William J. Brock and Kim L. R. Brouwer
Drug Metabolism and Disposition June 1, 2016, 44 (6) 867-870; DOI: https://doi.org/10.1124/dmd.115.067629
Rapid CommunicationShort Communication
Tolvaptan Disposition and DDIs in SCHH
Yang Lu, Jason R. Slizgi, Kenneth R. Brouwer, Robert L. St. Claire, Kimberly M. Freeman, Maxwell Pan, William J. Brock and Kim L. R. Brouwer
Drug Metabolism and Disposition June 1, 2016, 44 (6) 867-870; DOI: https://doi.org/10.1124/dmd.115.067629
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