Research ArticleArticle
Metabolic Disposition of Osimertinib in Rats, Dogs, and Humans: Insights into a Drug Designed to Bind Covalently to a Cysteine Residue of Epidermal Growth Factor Receptor
Paul A. Dickinson, Mireille V. Cantarini, Jo Collier, Paul Frewer, Scott Martin, Kathryn Pickup and Peter Ballard
Drug Metabolism and Disposition August 2016, 44 (8) 1201-1212; DOI: https://doi.org/10.1124/dmd.115.069203
Paul A. Dickinson
AstraZeneca, Macclesfield (M.V.C., P.F., S.M., K.P., P.B.), Seda Pharmaceutical Development Services, Cheshire (P.A.D), and Quotient Clinical Ltd., Ruddington, United Kingdom (J.C.)
Mireille V. Cantarini
AstraZeneca, Macclesfield (M.V.C., P.F., S.M., K.P., P.B.), Seda Pharmaceutical Development Services, Cheshire (P.A.D), and Quotient Clinical Ltd., Ruddington, United Kingdom (J.C.)
Jo Collier
AstraZeneca, Macclesfield (M.V.C., P.F., S.M., K.P., P.B.), Seda Pharmaceutical Development Services, Cheshire (P.A.D), and Quotient Clinical Ltd., Ruddington, United Kingdom (J.C.)
Paul Frewer
AstraZeneca, Macclesfield (M.V.C., P.F., S.M., K.P., P.B.), Seda Pharmaceutical Development Services, Cheshire (P.A.D), and Quotient Clinical Ltd., Ruddington, United Kingdom (J.C.)
Scott Martin
AstraZeneca, Macclesfield (M.V.C., P.F., S.M., K.P., P.B.), Seda Pharmaceutical Development Services, Cheshire (P.A.D), and Quotient Clinical Ltd., Ruddington, United Kingdom (J.C.)
Kathryn Pickup
AstraZeneca, Macclesfield (M.V.C., P.F., S.M., K.P., P.B.), Seda Pharmaceutical Development Services, Cheshire (P.A.D), and Quotient Clinical Ltd., Ruddington, United Kingdom (J.C.)
Peter Ballard
AstraZeneca, Macclesfield (M.V.C., P.F., S.M., K.P., P.B.), Seda Pharmaceutical Development Services, Cheshire (P.A.D), and Quotient Clinical Ltd., Ruddington, United Kingdom (J.C.)

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Research ArticleArticle
Metabolic Disposition of Osimertinib in Rats, Dogs, and Humans
Paul A. Dickinson, Mireille V. Cantarini, Jo Collier, Paul Frewer, Scott Martin, Kathryn Pickup and Peter Ballard
Drug Metabolism and Disposition August 1, 2016, 44 (8) 1201-1212; DOI: https://doi.org/10.1124/dmd.115.069203
Research ArticleArticle
Metabolic Disposition of Osimertinib in Rats, Dogs, and Humans
Paul A. Dickinson, Mireille V. Cantarini, Jo Collier, Paul Frewer, Scott Martin, Kathryn Pickup and Peter Ballard
Drug Metabolism and Disposition August 1, 2016, 44 (8) 1201-1212; DOI: https://doi.org/10.1124/dmd.115.069203