Research ArticleArticle
Simple Evaluation Method for CYP3A4 Induction from Human Hepatocytes: The Relative Factor Approach with an Induction Detection Limit Concentration Based on the Emax Model
Shino Kuramoto, Motohiro Kato, Hidetoshi Shindoh, Akihisa Kaneko, Masaki Ishigai and Seiji Miyauchi
Drug Metabolism and Disposition November 2017, 45 (11) 1139-1145; DOI: https://doi.org/10.1124/dmd.117.076349
Shino Kuramoto
Research Division, Chugai Pharmaceutical Co. Ltd., Kanagawa, Japan (S.K., M.K., H.S., A.K., M.I.); and Department of Pharmacokinetics, Toho University School of Pharmaceutical Sciences, Chiba, Japan (S.M.)
Motohiro Kato
Research Division, Chugai Pharmaceutical Co. Ltd., Kanagawa, Japan (S.K., M.K., H.S., A.K., M.I.); and Department of Pharmacokinetics, Toho University School of Pharmaceutical Sciences, Chiba, Japan (S.M.)
Hidetoshi Shindoh
Research Division, Chugai Pharmaceutical Co. Ltd., Kanagawa, Japan (S.K., M.K., H.S., A.K., M.I.); and Department of Pharmacokinetics, Toho University School of Pharmaceutical Sciences, Chiba, Japan (S.M.)
Akihisa Kaneko
Research Division, Chugai Pharmaceutical Co. Ltd., Kanagawa, Japan (S.K., M.K., H.S., A.K., M.I.); and Department of Pharmacokinetics, Toho University School of Pharmaceutical Sciences, Chiba, Japan (S.M.)
Masaki Ishigai
Research Division, Chugai Pharmaceutical Co. Ltd., Kanagawa, Japan (S.K., M.K., H.S., A.K., M.I.); and Department of Pharmacokinetics, Toho University School of Pharmaceutical Sciences, Chiba, Japan (S.M.)
Seiji Miyauchi
Research Division, Chugai Pharmaceutical Co. Ltd., Kanagawa, Japan (S.K., M.K., H.S., A.K., M.I.); and Department of Pharmacokinetics, Toho University School of Pharmaceutical Sciences, Chiba, Japan (S.M.)
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Research ArticleArticle
The Relative Factor Approach Based on the Emax Model
Shino Kuramoto, Motohiro Kato, Hidetoshi Shindoh, Akihisa Kaneko, Masaki Ishigai and Seiji Miyauchi
Drug Metabolism and Disposition November 1, 2017, 45 (11) 1139-1145; DOI: https://doi.org/10.1124/dmd.117.076349
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