Index by author
June 01, 2017; Volume 45,Issue 6
A
Achour, Brahim
- You have accessGlobal Proteomic Analysis of Human Liver Microsomes: Rapid Characterization and Quantification of Hepatic Drug-Metabolizing EnzymesBrahim Achour, Hajar Al Feteisi, Francesco Lanucara, Amin Rostami-Hodjegan and Jill BarberDrug Metabolism and Disposition June 2017, 45 (6) 666-675; DOI: https://doi.org/10.1124/dmd.116.074732
Ahire, Deepak
- You have accessMetabolite Identification, Reaction Phenotyping, and Retrospective Drug-Drug Interaction Predictions of 17-Deacetylnorgestimate, the Active Component of the Oral Contraceptive NorgestimateDeepak Ahire, Sarmistha Sinha, Barry Brock, Ramaswamy Iyer, Sandhya Mandlekar and Murali SubramanianDrug Metabolism and Disposition June 2017, 45 (6) 676-685; DOI: https://doi.org/10.1124/dmd.116.073940
Al Feteisi, Hajar
- You have accessGlobal Proteomic Analysis of Human Liver Microsomes: Rapid Characterization and Quantification of Hepatic Drug-Metabolizing EnzymesBrahim Achour, Hajar Al Feteisi, Francesco Lanucara, Amin Rostami-Hodjegan and Jill BarberDrug Metabolism and Disposition June 2017, 45 (6) 666-675; DOI: https://doi.org/10.1124/dmd.116.074732
Amaral, Kirsten
- You have accessHuman Enterocytes as an In Vitro Model for the Evaluation of Intestinal Drug Metabolism: Characterization of Drug-Metabolizing Enzyme Activities of Cryopreserved Human Enterocytes from Twenty-Four DonorsMing-Chih David Ho, Nicholas Ring, Kirsten Amaral, Utkarsh Doshi and Albert P. LiDrug Metabolism and Disposition June 2017, 45 (6) 686-691; DOI: https://doi.org/10.1124/dmd.116.074377
Aubé, Jeffrey
- You have accessStructural and Functional Evaluation of Clinically Relevant Inhibitors of Steroidogenic Cytochrome P450 17A1Elyse M. Petrunak, Steven A. Rogers, Jeffrey Aubé and Emily E. ScottDrug Metabolism and Disposition June 2017, 45 (6) 635-645; DOI: https://doi.org/10.1124/dmd.117.075317
B
Bagul, Pravin
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
Barber, Jill
- You have accessGlobal Proteomic Analysis of Human Liver Microsomes: Rapid Characterization and Quantification of Hepatic Drug-Metabolizing EnzymesBrahim Achour, Hajar Al Feteisi, Francesco Lanucara, Amin Rostami-Hodjegan and Jill BarberDrug Metabolism and Disposition June 2017, 45 (6) 666-675; DOI: https://doi.org/10.1124/dmd.116.074732
Boer, Jason
- You have accessIn Vitro Interactions of Epacadostat and its Major Metabolites with Human Efflux and Uptake Transporters: Implications for Pharmacokinetics and Drug InteractionsQiang Zhang, Yan Zhang, Jason Boer, Jack G. Shi, Peidi Hu, Sharon Diamond and Swamy YeleswaramDrug Metabolism and Disposition June 2017, 45 (6) 612-623; DOI: https://doi.org/10.1124/dmd.116.074609
Brock, Barry
- You have accessMetabolite Identification, Reaction Phenotyping, and Retrospective Drug-Drug Interaction Predictions of 17-Deacetylnorgestimate, the Active Component of the Oral Contraceptive NorgestimateDeepak Ahire, Sarmistha Sinha, Barry Brock, Ramaswamy Iyer, Sandhya Mandlekar and Murali SubramanianDrug Metabolism and Disposition June 2017, 45 (6) 676-685; DOI: https://doi.org/10.1124/dmd.116.073940
C
Chang, Jae H.
- You have accessApplying Stable Isotope Labeled Amino Acids in Micropatterned Hepatocyte Coculture to Directly Determine the Degradation Rate Constant for CYP3A4Ryan H. Takahashi, Sheerin K. Shahidi-Latham, Susan Wong and Jae H. ChangDrug Metabolism and Disposition June 2017, 45 (6) 581-585; DOI: https://doi.org/10.1124/dmd.116.074393
Chatterjee, Sagnik
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
Chen, Jiamei
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Chen, Liangfu
- You have accessPrediction of the Transporter-Mediated Drug-Drug Interaction Potential of Dabrafenib and Its Major Circulating MetabolitesHarma Ellens, Marta Johnson, Sarah K. Lawrence, Cory Watson, Liangfu Chen and Lauren E. Richards-PetersonDrug Metabolism and Disposition June 2017, 45 (6) 646-656; DOI: https://doi.org/10.1124/dmd.116.073932
Chen, Xiaoyan
- You have accessIncreased Plasma Exposures of Conjugated Metabolites of Morinidazole in Renal Failure Patients: A Critical Role of Uremic ToxinsFandi Kong, Xiaoyan Pang, Kan Zhong, Zitao Guo, Xiuli Li, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition June 2017, 45 (6) 593-603; DOI: https://doi.org/10.1124/dmd.116.074492
Cho, Takamasa
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
Chothe, Paresh P.
- You have accessQuantitative Prediction of CYP3A4 Induction: Impact of Measured, Free, and Intracellular Perpetrator Concentrations from Human Hepatocyte Induction Studies on Drug-Drug Interaction PredictionsYongkai Sun, Paresh P. Chothe, Jennifer E. Sager, Hong Tsao, Amanda Moore, Leena Laitinen and Niresh HariparsadDrug Metabolism and Disposition June 2017, 45 (6) 692-705; DOI: https://doi.org/10.1124/dmd.117.075481
D
Diamond, Sharon
- You have accessIn Vitro Interactions of Epacadostat and its Major Metabolites with Human Efflux and Uptake Transporters: Implications for Pharmacokinetics and Drug InteractionsQiang Zhang, Yan Zhang, Jason Boer, Jack G. Shi, Peidi Hu, Sharon Diamond and Swamy YeleswaramDrug Metabolism and Disposition June 2017, 45 (6) 612-623; DOI: https://doi.org/10.1124/dmd.116.074609
Doshi, Utkarsh
- You have accessHuman Enterocytes as an In Vitro Model for the Evaluation of Intestinal Drug Metabolism: Characterization of Drug-Metabolizing Enzyme Activities of Cryopreserved Human Enterocytes from Twenty-Four DonorsMing-Chih David Ho, Nicholas Ring, Kirsten Amaral, Utkarsh Doshi and Albert P. LiDrug Metabolism and Disposition June 2017, 45 (6) 686-691; DOI: https://doi.org/10.1124/dmd.116.074377
E
Ellens, Harma
- You have accessPrediction of the Transporter-Mediated Drug-Drug Interaction Potential of Dabrafenib and Its Major Circulating MetabolitesHarma Ellens, Marta Johnson, Sarah K. Lawrence, Cory Watson, Liangfu Chen and Lauren E. Richards-PetersonDrug Metabolism and Disposition June 2017, 45 (6) 646-656; DOI: https://doi.org/10.1124/dmd.116.073932
G
Gilibili, Ravindranath Reddy
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
Goto, Kei
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
Goto, Shin
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
Granica, Sebastian
- You have accessPhase II Conjugates of Urolithins Isolated from Human Urine and Potential Role of β-Glucuronidases in Their DispositionJakub P. Piwowarski, Iwona Stanisławska, Sebastian Granica, Joanna Stefańska and Anna K. KissDrug Metabolism and Disposition June 2017, 45 (6) 657-665; DOI: https://doi.org/10.1124/dmd.117.075200
Guo, Zitao
- You have accessIncreased Plasma Exposures of Conjugated Metabolites of Morinidazole in Renal Failure Patients: A Critical Role of Uremic ToxinsFandi Kong, Xiaoyan Pang, Kan Zhong, Zitao Guo, Xiuli Li, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition June 2017, 45 (6) 593-603; DOI: https://doi.org/10.1124/dmd.116.074492
H
Hariparsad, Niresh
- You have accessQuantitative Prediction of CYP3A4 Induction: Impact of Measured, Free, and Intracellular Perpetrator Concentrations from Human Hepatocyte Induction Studies on Drug-Drug Interaction PredictionsYongkai Sun, Paresh P. Chothe, Jennifer E. Sager, Hong Tsao, Amanda Moore, Leena Laitinen and Niresh HariparsadDrug Metabolism and Disposition June 2017, 45 (6) 692-705; DOI: https://doi.org/10.1124/dmd.117.075481
Ho, Ming-Chih David
- You have accessHuman Enterocytes as an In Vitro Model for the Evaluation of Intestinal Drug Metabolism: Characterization of Drug-Metabolizing Enzyme Activities of Cryopreserved Human Enterocytes from Twenty-Four DonorsMing-Chih David Ho, Nicholas Ring, Kirsten Amaral, Utkarsh Doshi and Albert P. LiDrug Metabolism and Disposition June 2017, 45 (6) 686-691; DOI: https://doi.org/10.1124/dmd.116.074377
Hu, Ming
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Hu, Peidi
- You have accessIn Vitro Interactions of Epacadostat and its Major Metabolites with Human Efflux and Uptake Transporters: Implications for Pharmacokinetics and Drug InteractionsQiang Zhang, Yan Zhang, Jason Boer, Jack G. Shi, Peidi Hu, Sharon Diamond and Swamy YeleswaramDrug Metabolism and Disposition June 2017, 45 (6) 612-623; DOI: https://doi.org/10.1124/dmd.116.074609
I
Iyer, Ramaswamy
- You have accessMetabolite Identification, Reaction Phenotyping, and Retrospective Drug-Drug Interaction Predictions of 17-Deacetylnorgestimate, the Active Component of the Oral Contraceptive NorgestimateDeepak Ahire, Sarmistha Sinha, Barry Brock, Ramaswamy Iyer, Sandhya Mandlekar and Murali SubramanianDrug Metabolism and Disposition June 2017, 45 (6) 676-685; DOI: https://doi.org/10.1124/dmd.116.073940
J
Jiang, Huangyu
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Johnson, Marta
- You have accessPrediction of the Transporter-Mediated Drug-Drug Interaction Potential of Dabrafenib and Its Major Circulating MetabolitesHarma Ellens, Marta Johnson, Sarah K. Lawrence, Cory Watson, Liangfu Chen and Lauren E. Richards-PetersonDrug Metabolism and Disposition June 2017, 45 (6) 646-656; DOI: https://doi.org/10.1124/dmd.116.073932
K
Kaneko, Yoshikatsu
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
Kiss, Anna K.
- You have accessPhase II Conjugates of Urolithins Isolated from Human Urine and Potential Role of β-Glucuronidases in Their DispositionJakub P. Piwowarski, Iwona Stanisławska, Sebastian Granica, Joanna Stefańska and Anna K. KissDrug Metabolism and Disposition June 2017, 45 (6) 657-665; DOI: https://doi.org/10.1124/dmd.117.075200
Kong, Fandi
- You have accessIncreased Plasma Exposures of Conjugated Metabolites of Morinidazole in Renal Failure Patients: A Critical Role of Uremic ToxinsFandi Kong, Xiaoyan Pang, Kan Zhong, Zitao Guo, Xiuli Li, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition June 2017, 45 (6) 593-603; DOI: https://doi.org/10.1124/dmd.116.074492
L
Lai, Yurong
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
Laitinen, Leena
- You have accessQuantitative Prediction of CYP3A4 Induction: Impact of Measured, Free, and Intracellular Perpetrator Concentrations from Human Hepatocyte Induction Studies on Drug-Drug Interaction PredictionsYongkai Sun, Paresh P. Chothe, Jennifer E. Sager, Hong Tsao, Amanda Moore, Leena Laitinen and Niresh HariparsadDrug Metabolism and Disposition June 2017, 45 (6) 692-705; DOI: https://doi.org/10.1124/dmd.117.075481
Lanucara, Francesco
- You have accessGlobal Proteomic Analysis of Human Liver Microsomes: Rapid Characterization and Quantification of Hepatic Drug-Metabolizing EnzymesBrahim Achour, Hajar Al Feteisi, Francesco Lanucara, Amin Rostami-Hodjegan and Jill BarberDrug Metabolism and Disposition June 2017, 45 (6) 666-675; DOI: https://doi.org/10.1124/dmd.116.074732
Lawrence, Sarah K.
- You have accessPrediction of the Transporter-Mediated Drug-Drug Interaction Potential of Dabrafenib and Its Major Circulating MetabolitesHarma Ellens, Marta Johnson, Sarah K. Lawrence, Cory Watson, Liangfu Chen and Lauren E. Richards-PetersonDrug Metabolism and Disposition June 2017, 45 (6) 646-656; DOI: https://doi.org/10.1124/dmd.116.073932
Li, Albert P.
- You have accessHuman Enterocytes as an In Vitro Model for the Evaluation of Intestinal Drug Metabolism: Characterization of Drug-Metabolizing Enzyme Activities of Cryopreserved Human Enterocytes from Twenty-Four DonorsMing-Chih David Ho, Nicholas Ring, Kirsten Amaral, Utkarsh Doshi and Albert P. LiDrug Metabolism and Disposition June 2017, 45 (6) 686-691; DOI: https://doi.org/10.1124/dmd.116.074377
Li, Xiaoyan
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Li, Xiuli
- You have accessIncreased Plasma Exposures of Conjugated Metabolites of Morinidazole in Renal Failure Patients: A Critical Role of Uremic ToxinsFandi Kong, Xiaoyan Pang, Kan Zhong, Zitao Guo, Xiuli Li, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition June 2017, 45 (6) 593-603; DOI: https://doi.org/10.1124/dmd.116.074492
Liu, Zhongqiu
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Lu, Linlin
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
M
Mandlekar, Sandhya
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
- You have accessMetabolite Identification, Reaction Phenotyping, and Retrospective Drug-Drug Interaction Predictions of 17-Deacetylnorgestimate, the Active Component of the Oral Contraceptive NorgestimateDeepak Ahire, Sarmistha Sinha, Barry Brock, Ramaswamy Iyer, Sandhya Mandlekar and Murali SubramanianDrug Metabolism and Disposition June 2017, 45 (6) 676-685; DOI: https://doi.org/10.1124/dmd.116.073940
Mariappan, T. Thanga
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
Maruyama, Hiroki
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
Moore, Amanda
- You have accessQuantitative Prediction of CYP3A4 Induction: Impact of Measured, Free, and Intracellular Perpetrator Concentrations from Human Hepatocyte Induction Studies on Drug-Drug Interaction PredictionsYongkai Sun, Paresh P. Chothe, Jennifer E. Sager, Hong Tsao, Amanda Moore, Leena Laitinen and Niresh HariparsadDrug Metabolism and Disposition June 2017, 45 (6) 692-705; DOI: https://doi.org/10.1124/dmd.117.075481
Mosure, Kathleen W.
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
Murali, Bokka Venkata
- You have accessCoproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition AssayRavindranath Reddy Gilibili, Sagnik Chatterjee, Pravin Bagul, Kathleen W. Mosure, Bokka Venkata Murali, T. Thanga Mariappan, Sandhya Mandlekar and Yurong LaiDrug Metabolism and Disposition June 2017, 45 (6) 604-611; DOI: https://doi.org/10.1124/dmd.116.074740
N
Narita, Ichiei
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
O
Otsuka, Tadashi
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
P
Pang, Xiaoyan
- You have accessIncreased Plasma Exposures of Conjugated Metabolites of Morinidazole in Renal Failure Patients: A Critical Role of Uremic ToxinsFandi Kong, Xiaoyan Pang, Kan Zhong, Zitao Guo, Xiuli Li, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition June 2017, 45 (6) 593-603; DOI: https://doi.org/10.1124/dmd.116.074492
Petrunak, Elyse M.
- You have accessStructural and Functional Evaluation of Clinically Relevant Inhibitors of Steroidogenic Cytochrome P450 17A1Elyse M. Petrunak, Steven A. Rogers, Jeffrey Aubé and Emily E. ScottDrug Metabolism and Disposition June 2017, 45 (6) 635-645; DOI: https://doi.org/10.1124/dmd.117.075317
Piwowarski, Jakub P.
- You have accessPhase II Conjugates of Urolithins Isolated from Human Urine and Potential Role of β-Glucuronidases in Their DispositionJakub P. Piwowarski, Iwona Stanisławska, Sebastian Granica, Joanna Stefańska and Anna K. KissDrug Metabolism and Disposition June 2017, 45 (6) 657-665; DOI: https://doi.org/10.1124/dmd.117.075200
Q
Qi, Xiaoxiao
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
R
Richards-Peterson, Lauren E.
- You have accessPrediction of the Transporter-Mediated Drug-Drug Interaction Potential of Dabrafenib and Its Major Circulating MetabolitesHarma Ellens, Marta Johnson, Sarah K. Lawrence, Cory Watson, Liangfu Chen and Lauren E. Richards-PetersonDrug Metabolism and Disposition June 2017, 45 (6) 646-656; DOI: https://doi.org/10.1124/dmd.116.073932
Ring, Nicholas
- You have accessHuman Enterocytes as an In Vitro Model for the Evaluation of Intestinal Drug Metabolism: Characterization of Drug-Metabolizing Enzyme Activities of Cryopreserved Human Enterocytes from Twenty-Four DonorsMing-Chih David Ho, Nicholas Ring, Kirsten Amaral, Utkarsh Doshi and Albert P. LiDrug Metabolism and Disposition June 2017, 45 (6) 686-691; DOI: https://doi.org/10.1124/dmd.116.074377
Rogers, Steven A.
- You have accessStructural and Functional Evaluation of Clinically Relevant Inhibitors of Steroidogenic Cytochrome P450 17A1Elyse M. Petrunak, Steven A. Rogers, Jeffrey Aubé and Emily E. ScottDrug Metabolism and Disposition June 2017, 45 (6) 635-645; DOI: https://doi.org/10.1124/dmd.117.075317
Rostami-Hodjegan, Amin
- You have accessGlobal Proteomic Analysis of Human Liver Microsomes: Rapid Characterization and Quantification of Hepatic Drug-Metabolizing EnzymesBrahim Achour, Hajar Al Feteisi, Francesco Lanucara, Amin Rostami-Hodjegan and Jill BarberDrug Metabolism and Disposition June 2017, 45 (6) 666-675; DOI: https://doi.org/10.1124/dmd.116.074732
S
Sager, Jennifer E.
- You have accessQuantitative Prediction of CYP3A4 Induction: Impact of Measured, Free, and Intracellular Perpetrator Concentrations from Human Hepatocyte Induction Studies on Drug-Drug Interaction PredictionsYongkai Sun, Paresh P. Chothe, Jennifer E. Sager, Hong Tsao, Amanda Moore, Leena Laitinen and Niresh HariparsadDrug Metabolism and Disposition June 2017, 45 (6) 692-705; DOI: https://doi.org/10.1124/dmd.117.075481
Sato, Yuya
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
Scott, Emily E.
- You have accessStructural and Functional Evaluation of Clinically Relevant Inhibitors of Steroidogenic Cytochrome P450 17A1Elyse M. Petrunak, Steven A. Rogers, Jeffrey Aubé and Emily E. ScottDrug Metabolism and Disposition June 2017, 45 (6) 635-645; DOI: https://doi.org/10.1124/dmd.117.075317
Shahidi-Latham, Sheerin K.
- You have accessApplying Stable Isotope Labeled Amino Acids in Micropatterned Hepatocyte Coculture to Directly Determine the Degradation Rate Constant for CYP3A4Ryan H. Takahashi, Sheerin K. Shahidi-Latham, Susan Wong and Jae H. ChangDrug Metabolism and Disposition June 2017, 45 (6) 581-585; DOI: https://doi.org/10.1124/dmd.116.074393
Shi, Jack G.
- You have accessIn Vitro Interactions of Epacadostat and its Major Metabolites with Human Efflux and Uptake Transporters: Implications for Pharmacokinetics and Drug InteractionsQiang Zhang, Yan Zhang, Jason Boer, Jack G. Shi, Peidi Hu, Sharon Diamond and Swamy YeleswaramDrug Metabolism and Disposition June 2017, 45 (6) 612-623; DOI: https://doi.org/10.1124/dmd.116.074609
Sinha, Sarmistha
- You have accessMetabolite Identification, Reaction Phenotyping, and Retrospective Drug-Drug Interaction Predictions of 17-Deacetylnorgestimate, the Active Component of the Oral Contraceptive NorgestimateDeepak Ahire, Sarmistha Sinha, Barry Brock, Ramaswamy Iyer, Sandhya Mandlekar and Murali SubramanianDrug Metabolism and Disposition June 2017, 45 (6) 676-685; DOI: https://doi.org/10.1124/dmd.116.073940
Stanisławska, Iwona
- You have accessPhase II Conjugates of Urolithins Isolated from Human Urine and Potential Role of β-Glucuronidases in Their DispositionJakub P. Piwowarski, Iwona Stanisławska, Sebastian Granica, Joanna Stefańska and Anna K. KissDrug Metabolism and Disposition June 2017, 45 (6) 657-665; DOI: https://doi.org/10.1124/dmd.117.075200
Stefańska, Joanna
- You have accessPhase II Conjugates of Urolithins Isolated from Human Urine and Potential Role of β-Glucuronidases in Their DispositionJakub P. Piwowarski, Iwona Stanisławska, Sebastian Granica, Joanna Stefańska and Anna K. KissDrug Metabolism and Disposition June 2017, 45 (6) 657-665; DOI: https://doi.org/10.1124/dmd.117.075200
Subramanian, Murali
- You have accessMetabolite Identification, Reaction Phenotyping, and Retrospective Drug-Drug Interaction Predictions of 17-Deacetylnorgestimate, the Active Component of the Oral Contraceptive NorgestimateDeepak Ahire, Sarmistha Sinha, Barry Brock, Ramaswamy Iyer, Sandhya Mandlekar and Murali SubramanianDrug Metabolism and Disposition June 2017, 45 (6) 676-685; DOI: https://doi.org/10.1124/dmd.116.073940
Sun, Yongkai
- You have accessQuantitative Prediction of CYP3A4 Induction: Impact of Measured, Free, and Intracellular Perpetrator Concentrations from Human Hepatocyte Induction Studies on Drug-Drug Interaction PredictionsYongkai Sun, Paresh P. Chothe, Jennifer E. Sager, Hong Tsao, Amanda Moore, Leena Laitinen and Niresh HariparsadDrug Metabolism and Disposition June 2017, 45 (6) 692-705; DOI: https://doi.org/10.1124/dmd.117.075481
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Takahashi, Ryan H.
- You have accessApplying Stable Isotope Labeled Amino Acids in Micropatterned Hepatocyte Coculture to Directly Determine the Degradation Rate Constant for CYP3A4Ryan H. Takahashi, Sheerin K. Shahidi-Latham, Susan Wong and Jae H. ChangDrug Metabolism and Disposition June 2017, 45 (6) 581-585; DOI: https://doi.org/10.1124/dmd.116.074393
Tsao, Hong
- You have accessQuantitative Prediction of CYP3A4 Induction: Impact of Measured, Free, and Intracellular Perpetrator Concentrations from Human Hepatocyte Induction Studies on Drug-Drug Interaction PredictionsYongkai Sun, Paresh P. Chothe, Jennifer E. Sager, Hong Tsao, Amanda Moore, Leena Laitinen and Niresh HariparsadDrug Metabolism and Disposition June 2017, 45 (6) 692-705; DOI: https://doi.org/10.1124/dmd.117.075481
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Wang, Ying
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Watson, Cory
- You have accessPrediction of the Transporter-Mediated Drug-Drug Interaction Potential of Dabrafenib and Its Major Circulating MetabolitesHarma Ellens, Marta Johnson, Sarah K. Lawrence, Cory Watson, Liangfu Chen and Lauren E. Richards-PetersonDrug Metabolism and Disposition June 2017, 45 (6) 646-656; DOI: https://doi.org/10.1124/dmd.116.073932
Wong, Susan
- You have accessApplying Stable Isotope Labeled Amino Acids in Micropatterned Hepatocyte Coculture to Directly Determine the Degradation Rate Constant for CYP3A4Ryan H. Takahashi, Sheerin K. Shahidi-Latham, Susan Wong and Jae H. ChangDrug Metabolism and Disposition June 2017, 45 (6) 581-585; DOI: https://doi.org/10.1124/dmd.116.074393
X
Xie, Cong
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Y
Yamamoto, Suguru
- You have accessProlactin Upregulates Female-Predominant P450 Gene Expressions and Downregulates Male-Predominant Gene Expressions in Mouse LiverYuya Sato, Yoshikatsu Kaneko, Takamasa Cho, Kei Goto, Tadashi Otsuka, Suguru Yamamoto, Shin Goto, Hiroki Maruyama and Ichiei NaritaDrug Metabolism and Disposition June 2017, 45 (6) 586-592; DOI: https://doi.org/10.1124/dmd.116.074658
Yan, Tongmeng
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Yeleswaram, Swamy
- You have accessIn Vitro Interactions of Epacadostat and its Major Metabolites with Human Efflux and Uptake Transporters: Implications for Pharmacokinetics and Drug InteractionsQiang Zhang, Yan Zhang, Jason Boer, Jack G. Shi, Peidi Hu, Sharon Diamond and Swamy YeleswaramDrug Metabolism and Disposition June 2017, 45 (6) 612-623; DOI: https://doi.org/10.1124/dmd.116.074609
Yu, Jia
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Z
Zeng, Sijing
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Zhang, Qiang
- You have accessIn Vitro Interactions of Epacadostat and its Major Metabolites with Human Efflux and Uptake Transporters: Implications for Pharmacokinetics and Drug InteractionsQiang Zhang, Yan Zhang, Jason Boer, Jack G. Shi, Peidi Hu, Sharon Diamond and Swamy YeleswaramDrug Metabolism and Disposition June 2017, 45 (6) 612-623; DOI: https://doi.org/10.1124/dmd.116.074609
Zhang, Yan
- You have accessIn Vitro Interactions of Epacadostat and its Major Metabolites with Human Efflux and Uptake Transporters: Implications for Pharmacokinetics and Drug InteractionsQiang Zhang, Yan Zhang, Jason Boer, Jack G. Shi, Peidi Hu, Sharon Diamond and Swamy YeleswaramDrug Metabolism and Disposition June 2017, 45 (6) 612-623; DOI: https://doi.org/10.1124/dmd.116.074609
Zheng, Haihui
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
Zhong, Dafang
- You have accessIncreased Plasma Exposures of Conjugated Metabolites of Morinidazole in Renal Failure Patients: A Critical Role of Uremic ToxinsFandi Kong, Xiaoyan Pang, Kan Zhong, Zitao Guo, Xiuli Li, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition June 2017, 45 (6) 593-603; DOI: https://doi.org/10.1124/dmd.116.074492
Zhong, Kan
- You have accessIncreased Plasma Exposures of Conjugated Metabolites of Morinidazole in Renal Failure Patients: A Critical Role of Uremic ToxinsFandi Kong, Xiaoyan Pang, Kan Zhong, Zitao Guo, Xiuli Li, Dafang Zhong and Xiaoyan ChenDrug Metabolism and Disposition June 2017, 45 (6) 593-603; DOI: https://doi.org/10.1124/dmd.116.074492
Zhu, Lijun
- You have accessHigh-Throughput and Reliable Isotope Label-free Approach for Profiling 24 Metabolic Enzymes in FVB Mice and Sex DifferencesJiamei Chen, Lijun Zhu, Xiaoyan Li, Haihui Zheng, Tongmeng Yan, Cong Xie, Sijing Zeng, Jia Yu, Huangyu Jiang, Linlin Lu, Xiaoxiao Qi, Ying Wang, Ming Hu and Zhongqiu LiuDrug Metabolism and Disposition June 2017, 45 (6) 624-634; DOI: https://doi.org/10.1124/dmd.116.074682
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