Research ArticleArticles
The Phenomenon of Albumin-Mediated Hepatic Uptake of Organic Anion Transport Polypeptide Substrates: Prediction of the In Vivo Uptake Clearance from the In Vitro Uptake by Isolated Hepatocytes Using a Facilitated-Dissociation Model
Seiji Miyauchi, Masayuki Masuda, Soo-Jin Kim, Yuudai Tanaka, Kyeong-Ryoon Lee, Shouko Iwakado, Momoko Nemoto, Shotaro Sasaki, Kazumi Shimono, Yoshio Tanaka and Yuichi Sugiyama
Drug Metabolism and Disposition March 2018, 46 (3) 259-267; DOI: https://doi.org/10.1124/dmd.117.077115
Seiji Miyauchi
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Masayuki Masuda
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Soo-Jin Kim
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Yuudai Tanaka
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Kyeong-Ryoon Lee
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Shouko Iwakado
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Momoko Nemoto
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Shotaro Sasaki
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Kazumi Shimono
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Yoshio Tanaka
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
Yuichi Sugiyama
Faculty of Pharmaceutical Sciences, Toho University, 2-2-1 Miyama, Funabashi, Chiba, Japan (S.M., M.M., Y.T., S.I., M.N., S.S., K.S., Y.T.) and Sugiyama Laboratory, RIKEN Innovation Center, RIKEN Cluster for Industry Partnerships, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Japan (S.-J.K., K.-R.L., Y.S.)
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In this issue
Research ArticleArticles
IVIVE for Albumin-Mediated Hepatic Uptake
Seiji Miyauchi, Masayuki Masuda, Soo-Jin Kim, Yuudai Tanaka, Kyeong-Ryoon Lee, Shouko Iwakado, Momoko Nemoto, Shotaro Sasaki, Kazumi Shimono, Yoshio Tanaka and Yuichi Sugiyama
Drug Metabolism and Disposition March 1, 2018, 46 (3) 259-267; DOI: https://doi.org/10.1124/dmd.117.077115
Research ArticleArticles
IVIVE for Albumin-Mediated Hepatic Uptake
Seiji Miyauchi, Masayuki Masuda, Soo-Jin Kim, Yuudai Tanaka, Kyeong-Ryoon Lee, Shouko Iwakado, Momoko Nemoto, Shotaro Sasaki, Kazumi Shimono, Yoshio Tanaka and Yuichi Sugiyama
Drug Metabolism and Disposition March 1, 2018, 46 (3) 259-267; DOI: https://doi.org/10.1124/dmd.117.077115
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