Research ArticleArticle
Metabolic Profiling of the Novel Hypoxia-Inducible Factor 2α Inhibitor PT2385 In Vivo and In Vitro
Cen Xie, Xiaoxia Gao, Dongxue Sun, Youbo Zhang, Kristopher W. Krausz, Xuemei Qin and Frank J. Gonzalez
Drug Metabolism and Disposition April 2018, 46 (4) 336-345; DOI: https://doi.org/10.1124/dmd.117.079723
Cen Xie
Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland (C.X., X.G., D.S., Y.Z., K.W.K., F.J.G.); and Modern Research Center for Traditional Chinese Medicine, Shanxi University, Taiyuan, Shanxi, People’s Republic of China (X.G., X.Q.)
Xiaoxia Gao
Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland (C.X., X.G., D.S., Y.Z., K.W.K., F.J.G.); and Modern Research Center for Traditional Chinese Medicine, Shanxi University, Taiyuan, Shanxi, People’s Republic of China (X.G., X.Q.)
Dongxue Sun
Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland (C.X., X.G., D.S., Y.Z., K.W.K., F.J.G.); and Modern Research Center for Traditional Chinese Medicine, Shanxi University, Taiyuan, Shanxi, People’s Republic of China (X.G., X.Q.)
Youbo Zhang
Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland (C.X., X.G., D.S., Y.Z., K.W.K., F.J.G.); and Modern Research Center for Traditional Chinese Medicine, Shanxi University, Taiyuan, Shanxi, People’s Republic of China (X.G., X.Q.)
Kristopher W. Krausz
Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland (C.X., X.G., D.S., Y.Z., K.W.K., F.J.G.); and Modern Research Center for Traditional Chinese Medicine, Shanxi University, Taiyuan, Shanxi, People’s Republic of China (X.G., X.Q.)
Xuemei Qin
Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland (C.X., X.G., D.S., Y.Z., K.W.K., F.J.G.); and Modern Research Center for Traditional Chinese Medicine, Shanxi University, Taiyuan, Shanxi, People’s Republic of China (X.G., X.Q.)
Frank J. Gonzalez
Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland (C.X., X.G., D.S., Y.Z., K.W.K., F.J.G.); and Modern Research Center for Traditional Chinese Medicine, Shanxi University, Taiyuan, Shanxi, People’s Republic of China (X.G., X.Q.)
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Research ArticleArticle
Metabolic Profiling of PT2385
Cen Xie, Xiaoxia Gao, Dongxue Sun, Youbo Zhang, Kristopher W. Krausz, Xuemei Qin and Frank J. Gonzalez
Drug Metabolism and Disposition April 1, 2018, 46 (4) 336-345; DOI: https://doi.org/10.1124/dmd.117.079723
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