Saracatinib | 293 cells regulated expression | pEBTetD | Unlabeled compound HPLC + UV detector at 259 nm | 10 µM/10 min | Harrach et al. (2017) |
Cytarabine, gemcitabine | 293 cells, sorted by FACS permanent expression | Retroviral vector pMIG II | Radiotracer / LC-MS/MS | 1 µM/5 min | Drenberg et al., 2017 |
Ipratropium | 293 cells permanent expression | pcDNA3 | Radiotracer | 0.015 µM/10 min | Nakamura et al. (2010) |
Oxaliplatin | 293 cells permanent expression | pcDNA3 | Radiotracer | 1 µM/60 min | Jong et al. (2011) |
Metformin | MDCKII cells permanent expression | pcDNA3 | Unlabeled compound HPLC + UV detector at 236 nm | 3 mM/80 min | Nakamichi et al. (2013) |
Gabapentin | 293 cells permanent expression | (Flp-In system) | Radiotracer | 10 µM/10 min | Urban et al. (2008) |
All | 293 cells regulated expression | pEBTetD | Unlabeled compounds LC-MS/MS | 0.1/1/10 µM/1 min | This study |