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Exposure-Efficacy Analysis of Antibody-Drug Conjugates Delivering an Excessive Level of Payload to Tissues
Donglu Zhang, Peter S. Dragovich, Shang-Fan Yu, Yong Ma, Thomas H. Pillow, Jack D. Sadowsky, Dian Su, Wei Wang, Andrew Polson, S. Cyrus Khojasteh and Cornelis E.C.A. Hop
Drug Metabolism and Disposition October 2019, 47 (10) 1146-1155; DOI: https://doi.org/10.1124/dmd.119.087023
Donglu Zhang
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Peter S. Dragovich
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Shang-Fan Yu
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Yong Ma
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Thomas H. Pillow
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Jack D. Sadowsky
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Dian Su
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Wei Wang
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Andrew Polson
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
S. Cyrus Khojasteh
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California
Cornelis E.C.A. Hop
Drug Metabolism & Pharmacokinetics (D.Z., Y.M., D.S., W.W., S.C.K., C.E.C.A.H.), Discovery Chemistry (P.S.D., T.H.P.), Translational Oncology (S.-F.Y., A.P.), and Protein Chemistry (J.D.S.), Genentech, South San Francisco, California

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Research ArticleArticle
ADCs Can Deliver Excess Payload to Tumors
Donglu Zhang, Peter S. Dragovich, Shang-Fan Yu, Yong Ma, Thomas H. Pillow, Jack D. Sadowsky, Dian Su, Wei Wang, Andrew Polson, S. Cyrus Khojasteh and Cornelis E.C.A. Hop
Drug Metabolism and Disposition October 1, 2019, 47 (10) 1146-1155; DOI: https://doi.org/10.1124/dmd.119.087023
Research ArticleArticle
ADCs Can Deliver Excess Payload to Tumors
Donglu Zhang, Peter S. Dragovich, Shang-Fan Yu, Yong Ma, Thomas H. Pillow, Jack D. Sadowsky, Dian Su, Wei Wang, Andrew Polson, S. Cyrus Khojasteh and Cornelis E.C.A. Hop
Drug Metabolism and Disposition October 1, 2019, 47 (10) 1146-1155; DOI: https://doi.org/10.1124/dmd.119.087023
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