Research ArticleArticle
Open Access
Bioavailability, Biotransformation, and Excretion of the Covalent Bruton Tyrosine Kinase Inhibitor Acalabrutinib in Rats, Dogs, and Humans
Terry Podoll, Paul G. Pearson, Jerry Evarts, Tim Ingallinera, Elena Bibikova, Hao Sun, Mark Gohdes, Kristen Cardinal, Mitesh Sanghvi and J. Greg Slatter
Drug Metabolism and Disposition February 2019, 47 (2) 145-154; DOI: https://doi.org/10.1124/dmd.118.084459
Terry Podoll
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Paul G. Pearson
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Jerry Evarts
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Tim Ingallinera
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Elena Bibikova
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Hao Sun
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Mark Gohdes
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Kristen Cardinal
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
Mitesh Sanghvi
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)
J. Greg Slatter
Acerta Pharma, South San Francisco, California (T.P., J.E., T.I., E.B., J.G.S.); Pearson Pharma Partners, Westlake Village, California (P.G.P.); Covance, Madison, Wisconsin (H.S., M.G., K.C.); and Xceleron, Germantown, Maryland (M.S.)

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Research ArticleArticle
Bioavailability, Metabolism, and Excretion of [14C]Acalabrutinib
Terry Podoll, Paul G. Pearson, Jerry Evarts, Tim Ingallinera, Elena Bibikova, Hao Sun, Mark Gohdes, Kristen Cardinal, Mitesh Sanghvi and J. Greg Slatter
Drug Metabolism and Disposition February 1, 2019, 47 (2) 145-154; DOI: https://doi.org/10.1124/dmd.118.084459
Research ArticleArticle
Bioavailability, Metabolism, and Excretion of [14C]Acalabrutinib
Terry Podoll, Paul G. Pearson, Jerry Evarts, Tim Ingallinera, Elena Bibikova, Hao Sun, Mark Gohdes, Kristen Cardinal, Mitesh Sanghvi and J. Greg Slatter
Drug Metabolism and Disposition February 1, 2019, 47 (2) 145-154; DOI: https://doi.org/10.1124/dmd.118.084459