| | pmol/min per milligram | μM | nM | ml/min per milligram |
THC depletiona | P450s | — | — | — | 235.6 (48%) |
11-OH-THC formation | CYP2C9 | 624 (2%) | 0.07 (4%) | 3 (36%) | 214.4 (34%) |
Unknown THC metabolite formationb | CYP2D6 | 4905 (17%) | 5.48 (20%) | 231 (44%) | 21.3 (34%) |
11-OH-THC depletiona | P450s/UGTs | — | — | — | 12.3 (26%) |
COOH-THC formation | CYP2C9 | 5 (2%) | 0.50 (4%) | 32 (44%) | 0.15 (34%) |
Unknown 11-OH-THC metabolite formationb | CYP2C9 | 54 (6%) | 0.50 (4%) | 32 (44%) | 1.7 (34%) |
Unknown 11-OH-THC metabolite formationb | CYP3A | 1826 (6%) | 12.8 (8%) | 824 (59%) | 2.2 (34%) |
Unknown 11-OH-THC metabolite formationb | UGT2B7/1A9 | 343 (4%) | 0.64 (4%) | 39 (44%) | 8.8 (44%) |