Index by author
November 01, 2020; Volume 48,Issue 11
B
Balsitis, Scott
- You have accessCharacterization of Seasonal Pharmacokinetic Variability in WoodchucksJim Zheng, Scott Balsitis, Rex Santos, Bill J. Smith and Raju SubramanianDrug Metabolism and Disposition November 2020, 48 (11) 1199-1209; DOI: https://doi.org/10.1124/dmd.120.000140
Baudy, Andreas
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Beckers, Claire
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
Bolleddula, Jayaprakasam
- You have accessPharmacokinetics and Catabolism of [3H]TAK-164, a Guanylyl Cyclase C Targeted Antibody-Drug ConjugateJayaprakasam Bolleddula, Abhi Shah, Mohammad Shadid, Afrand Kamali, Michael D. Smith and Swapan K. ChowdhuryDrug Metabolism and Disposition November 2020, 48 (11) 1239-1245; DOI: https://doi.org/10.1124/dmd.120.000194
Bonnaillie, Pierre
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
C
Cai, Hao
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
Chanteux, Hugues
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
Chapron, Brian D.
- You have accessThe Respective Roles of CYP3A4 and CYP2D6 in the Metabolism of Pimozide to Established and Novel MetabolitesBrian D. Chapron, Jean C. Dinh, Paul C. Toren, Andrea Gaedigk and J. Steven LeederDrug Metabolism and Disposition November 2020, 48 (11) 1113-1120; DOI: https://doi.org/10.1124/dmd.120.000188
Chen, Ang
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
Chen, Qing
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Chowdhury, Swapan K.
- You have accessPharmacokinetics and Catabolism of [3H]TAK-164, a Guanylyl Cyclase C Targeted Antibody-Drug ConjugateJayaprakasam Bolleddula, Abhi Shah, Mohammad Shadid, Afrand Kamali, Michael D. Smith and Swapan K. ChowdhuryDrug Metabolism and Disposition November 2020, 48 (11) 1239-1245; DOI: https://doi.org/10.1124/dmd.120.000194
Cuypers, Marie-Lynn
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
D
Davies, Mari
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Delatour, Claude
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
Dell’Aiera, Sylvie
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
De Sousa Mendes, Mailys
- You have accessA Laboratory-Specific Scaling Factor to Predict the In Vivo Human Clearance of Aldehyde Oxidase SubstratesMailys De Sousa Mendes, Alexandra L. Orton, Helen E. Humphries, Barry Jones, Iain Gardner, Sibylle Neuhoff and Venkatesh Pilla ReddyDrug Metabolism and Disposition November 2020, 48 (11) 1231-1238; DOI: https://doi.org/10.1124/dmd.120.000082
Dinh, Jean C.
- You have accessThe Respective Roles of CYP3A4 and CYP2D6 in the Metabolism of Pimozide to Established and Novel MetabolitesBrian D. Chapron, Jean C. Dinh, Paul C. Toren, Andrea Gaedigk and J. Steven LeederDrug Metabolism and Disposition November 2020, 48 (11) 1113-1120; DOI: https://doi.org/10.1124/dmd.120.000188
E
Evers, Raymond
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
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Gaedigk, Andrea
- You have accessThe Respective Roles of CYP3A4 and CYP2D6 in the Metabolism of Pimozide to Established and Novel MetabolitesBrian D. Chapron, Jean C. Dinh, Paul C. Toren, Andrea Gaedigk and J. Steven LeederDrug Metabolism and Disposition November 2020, 48 (11) 1113-1120; DOI: https://doi.org/10.1124/dmd.120.000188
Gardner, Iain
- You have accessA Laboratory-Specific Scaling Factor to Predict the In Vivo Human Clearance of Aldehyde Oxidase SubstratesMailys De Sousa Mendes, Alexandra L. Orton, Helen E. Humphries, Barry Jones, Iain Gardner, Sibylle Neuhoff and Venkatesh Pilla ReddyDrug Metabolism and Disposition November 2020, 48 (11) 1231-1238; DOI: https://doi.org/10.1124/dmd.120.000082
Gillent, Eric
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
Golding, Melanie
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Gormsen, Lars C.
- You have accessSuccessful Prediction of Positron Emission Tomography–Imaged Metformin Hepatic Uptake Clearance in Humans Using the Quantitative Proteomics–Informed Relative Expression Factor ApproachMadhav Sachar, Vineet Kumar, Lars C. Gormsen, Ole Lajord Munk and Jashvant D. UnadkatDrug Metabolism and Disposition November 2020, 48 (11) 1210-1216; DOI: https://doi.org/10.1124/dmd.120.000156
Guo, Yuanqing
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
H
Hafey, Michael J.
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Hagenbuch, Bruno
- You have accessFunctional Consequences of Pravastatin Isomerization on OATP1B1-Mediated TransportJonathan B. Wagner, Melissa Ruggiero, J. Steven Leeder and Bruno HagenbuchDrug Metabolism and Disposition November 2020, 48 (11) 1192-1198; DOI: https://doi.org/10.1124/dmd.120.000122
Harlfinger, Stephanie
- You have accessEvaluation of the Disconnect between Hepatocyte and Microsome Intrinsic Clearance and In Vitro In Vivo Extrapolation PerformanceBeth Williamson, Stephanie Harlfinger and Dermot F. McGinnityDrug Metabolism and Disposition November 2020, 48 (11) 1137-1146; DOI: https://doi.org/10.1124/dmd.120.000131
Horne, Lloyd P.
- You have accessExposure of Rats to Multiple Oral Doses of Dichloroacetate Results in Upregulation of Hepatic Glutathione Transferases and NAD(P)H Dehydrogenase [Quinone] 1Edwin J. Squirewell, Ricky Mareus, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1224-1230; DOI: https://doi.org/10.1124/dmd.120.000143
- You have accessEffects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult RatsEdwin J. Squirewell, Marci G. Smeltz, Laura Rowland-Faux, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1217-1223; DOI: https://doi.org/10.1124/dmd.120.000142
Houle, Robert
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Humphries, Helen E.
- You have accessA Laboratory-Specific Scaling Factor to Predict the In Vivo Human Clearance of Aldehyde Oxidase SubstratesMailys De Sousa Mendes, Alexandra L. Orton, Helen E. Humphries, Barry Jones, Iain Gardner, Sibylle Neuhoff and Venkatesh Pilla ReddyDrug Metabolism and Disposition November 2020, 48 (11) 1231-1238; DOI: https://doi.org/10.1124/dmd.120.000082
J
James, Margaret O.
- You have accessExposure of Rats to Multiple Oral Doses of Dichloroacetate Results in Upregulation of Hepatic Glutathione Transferases and NAD(P)H Dehydrogenase [Quinone] 1Edwin J. Squirewell, Ricky Mareus, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1224-1230; DOI: https://doi.org/10.1124/dmd.120.000143
- You have accessEffects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult RatsEdwin J. Squirewell, Marci G. Smeltz, Laura Rowland-Faux, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1217-1223; DOI: https://doi.org/10.1124/dmd.120.000142
Jones, Barry
- You have accessA Laboratory-Specific Scaling Factor to Predict the In Vivo Human Clearance of Aldehyde Oxidase SubstratesMailys De Sousa Mendes, Alexandra L. Orton, Helen E. Humphries, Barry Jones, Iain Gardner, Sibylle Neuhoff and Venkatesh Pilla ReddyDrug Metabolism and Disposition November 2020, 48 (11) 1231-1238; DOI: https://doi.org/10.1124/dmd.120.000082
K
Kamali, Afrand
- You have accessPharmacokinetics and Catabolism of [3H]TAK-164, a Guanylyl Cyclase C Targeted Antibody-Drug ConjugateJayaprakasam Bolleddula, Abhi Shah, Mohammad Shadid, Afrand Kamali, Michael D. Smith and Swapan K. ChowdhuryDrug Metabolism and Disposition November 2020, 48 (11) 1239-1245; DOI: https://doi.org/10.1124/dmd.120.000194
Kamath, Amrita V.
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
Katayama, Kazuhide
- You have accessImpact of P-Glycoprotein–Mediated Active Efflux on Drug Distribution into Lumbar Cerebrospinal Fluid in Nonhuman PrimatesYoko Nagaya, Kazuhide Katayama, Hiroyuki Kusuhara and Yoshitane NozakiDrug Metabolism and Disposition November 2020, 48 (11) 1183-1190; DOI: https://doi.org/10.1124/dmd.120.000099
Khojasteh, S. Cyrus
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
King, Lloyd
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Knemeyer, Ian
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Kotian, Apoorva
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Kumar, Vineet
- You have accessSuccessful Prediction of Positron Emission Tomography–Imaged Metformin Hepatic Uptake Clearance in Humans Using the Quantitative Proteomics–Informed Relative Expression Factor ApproachMadhav Sachar, Vineet Kumar, Lars C. Gormsen, Ole Lajord Munk and Jashvant D. UnadkatDrug Metabolism and Disposition November 2020, 48 (11) 1210-1216; DOI: https://doi.org/10.1124/dmd.120.000156
Kusuhara, Hiroyuki
- You have accessImpact of P-Glycoprotein–Mediated Active Efflux on Drug Distribution into Lumbar Cerebrospinal Fluid in Nonhuman PrimatesYoko Nagaya, Kazuhide Katayama, Hiroyuki Kusuhara and Yoshitane NozakiDrug Metabolism and Disposition November 2020, 48 (11) 1183-1190; DOI: https://doi.org/10.1124/dmd.120.000099
L
L. Orton, Alexandra
- You have accessA Laboratory-Specific Scaling Factor to Predict the In Vivo Human Clearance of Aldehyde Oxidase SubstratesMailys De Sousa Mendes, Alexandra L. Orton, Helen E. Humphries, Barry Jones, Iain Gardner, Sibylle Neuhoff and Venkatesh Pilla ReddyDrug Metabolism and Disposition November 2020, 48 (11) 1231-1238; DOI: https://doi.org/10.1124/dmd.120.000082
Lee, M. Violet
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
Leeder, J. Steven
- You have accessThe Respective Roles of CYP3A4 and CYP2D6 in the Metabolism of Pimozide to Established and Novel MetabolitesBrian D. Chapron, Jean C. Dinh, Paul C. Toren, Andrea Gaedigk and J. Steven LeederDrug Metabolism and Disposition November 2020, 48 (11) 1113-1120; DOI: https://doi.org/10.1124/dmd.120.000188
- You have accessFunctional Consequences of Pravastatin Isomerization on OATP1B1-Mediated TransportJonathan B. Wagner, Melissa Ruggiero, J. Steven Leeder and Bruno HagenbuchDrug Metabolism and Disposition November 2020, 48 (11) 1192-1198; DOI: https://doi.org/10.1124/dmd.120.000122
Liu, Mingyao
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
Ljumanovic, Nina
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
Lu, Jian
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
M
Ma, Shuguang
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
Ma, Xinrun
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
Manevski, Nenad
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Mareus, Ricky
- You have accessExposure of Rats to Multiple Oral Doses of Dichloroacetate Results in Upregulation of Hepatic Glutathione Transferases and NAD(P)H Dehydrogenase [Quinone] 1Edwin J. Squirewell, Ricky Mareus, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1224-1230; DOI: https://doi.org/10.1124/dmd.120.000143
McGinnity, Dermot F.
- You have accessEvaluation of the Disconnect between Hepatocyte and Microsome Intrinsic Clearance and In Vitro In Vivo Extrapolation PerformanceBeth Williamson, Stephanie Harlfinger and Dermot F. McGinnityDrug Metabolism and Disposition November 2020, 48 (11) 1137-1146; DOI: https://doi.org/10.1124/dmd.120.000131
Monroe, James
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Munk, Ole Lajord
- You have accessSuccessful Prediction of Positron Emission Tomography–Imaged Metformin Hepatic Uptake Clearance in Humans Using the Quantitative Proteomics–Informed Relative Expression Factor ApproachMadhav Sachar, Vineet Kumar, Lars C. Gormsen, Ole Lajord Munk and Jashvant D. UnadkatDrug Metabolism and Disposition November 2020, 48 (11) 1210-1216; DOI: https://doi.org/10.1124/dmd.120.000156
N
Nagaya, Yoko
- You have accessImpact of P-Glycoprotein–Mediated Active Efflux on Drug Distribution into Lumbar Cerebrospinal Fluid in Nonhuman PrimatesYoko Nagaya, Kazuhide Katayama, Hiroyuki Kusuhara and Yoshitane NozakiDrug Metabolism and Disposition November 2020, 48 (11) 1183-1190; DOI: https://doi.org/10.1124/dmd.120.000099
Neuhoff, Sibylle
- You have accessA Laboratory-Specific Scaling Factor to Predict the In Vivo Human Clearance of Aldehyde Oxidase SubstratesMailys De Sousa Mendes, Alexandra L. Orton, Helen E. Humphries, Barry Jones, Iain Gardner, Sibylle Neuhoff and Venkatesh Pilla ReddyDrug Metabolism and Disposition November 2020, 48 (11) 1231-1238; DOI: https://doi.org/10.1124/dmd.120.000082
Nicolaï, Johan
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
Nozaki, Yoshitane
- You have accessImpact of P-Glycoprotein–Mediated Active Efflux on Drug Distribution into Lumbar Cerebrospinal Fluid in Nonhuman PrimatesYoko Nagaya, Kazuhide Katayama, Hiroyuki Kusuhara and Yoshitane NozakiDrug Metabolism and Disposition November 2020, 48 (11) 1183-1190; DOI: https://doi.org/10.1124/dmd.120.000099
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Penney, Mark
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Peramuhendige, Prabha
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Pilla Reddy, Venkatesh
- You have accessA Laboratory-Specific Scaling Factor to Predict the In Vivo Human Clearance of Aldehyde Oxidase SubstratesMailys De Sousa Mendes, Alexandra L. Orton, Helen E. Humphries, Barry Jones, Iain Gardner, Sibylle Neuhoff and Venkatesh Pilla ReddyDrug Metabolism and Disposition November 2020, 48 (11) 1231-1238; DOI: https://doi.org/10.1124/dmd.120.000082
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Rowland-Faux, Laura
- You have accessEffects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult RatsEdwin J. Squirewell, Marci G. Smeltz, Laura Rowland-Faux, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1217-1223; DOI: https://doi.org/10.1124/dmd.120.000142
Ruggiero, Melissa
- You have accessFunctional Consequences of Pravastatin Isomerization on OATP1B1-Mediated TransportJonathan B. Wagner, Melissa Ruggiero, J. Steven Leeder and Bruno HagenbuchDrug Metabolism and Disposition November 2020, 48 (11) 1192-1198; DOI: https://doi.org/10.1124/dmd.120.000122
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Saad, Ola
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
Sachar, Madhav
- You have accessSuccessful Prediction of Positron Emission Tomography–Imaged Metformin Hepatic Uptake Clearance in Humans Using the Quantitative Proteomics–Informed Relative Expression Factor ApproachMadhav Sachar, Vineet Kumar, Lars C. Gormsen, Ole Lajord Munk and Jashvant D. UnadkatDrug Metabolism and Disposition November 2020, 48 (11) 1210-1216; DOI: https://doi.org/10.1124/dmd.120.000156
Santos, Rex
- You have accessCharacterization of Seasonal Pharmacokinetic Variability in WoodchucksJim Zheng, Scott Balsitis, Rex Santos, Bill J. Smith and Raju SubramanianDrug Metabolism and Disposition November 2020, 48 (11) 1199-1209; DOI: https://doi.org/10.1124/dmd.120.000140
Saunders, Kenneth
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
Scott, Dr. Emily E.
- You have accessAnnouncementDr. Emily E. ScottDrug Metabolism and Disposition November 2020, 48 (11) 1191; DOI: https://doi.org/10.1124/dmd.120.000249
Shadid, Mohammad
- You have accessPharmacokinetics and Catabolism of [3H]TAK-164, a Guanylyl Cyclase C Targeted Antibody-Drug ConjugateJayaprakasam Bolleddula, Abhi Shah, Mohammad Shadid, Afrand Kamali, Michael D. Smith and Swapan K. ChowdhuryDrug Metabolism and Disposition November 2020, 48 (11) 1239-1245; DOI: https://doi.org/10.1124/dmd.120.000194
Shah, Abhi
- You have accessPharmacokinetics and Catabolism of [3H]TAK-164, a Guanylyl Cyclase C Targeted Antibody-Drug ConjugateJayaprakasam Bolleddula, Abhi Shah, Mohammad Shadid, Afrand Kamali, Michael D. Smith and Swapan K. ChowdhuryDrug Metabolism and Disposition November 2020, 48 (11) 1239-1245; DOI: https://doi.org/10.1124/dmd.120.000194
Shah, Syeda
- You have accessEvaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug DiscoveryMari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda Shah and Nenad ManevskiDrug Metabolism and Disposition November 2020, 48 (11) 1169-1182; DOI: https://doi.org/10.1124/dmd.120.000111
Shang, Jackie
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Shang, Xuyang
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
Shen, Ben-Quan
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
Sistare, Frank D.
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Smeltz, Marci G.
- You have accessEffects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult RatsEdwin J. Squirewell, Marci G. Smeltz, Laura Rowland-Faux, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1217-1223; DOI: https://doi.org/10.1124/dmd.120.000142
Smith, Bill J.
- You have accessCharacterization of Seasonal Pharmacokinetic Variability in WoodchucksJim Zheng, Scott Balsitis, Rex Santos, Bill J. Smith and Raju SubramanianDrug Metabolism and Disposition November 2020, 48 (11) 1199-1209; DOI: https://doi.org/10.1124/dmd.120.000140
Smith, Michael D.
- You have accessPharmacokinetics and Catabolism of [3H]TAK-164, a Guanylyl Cyclase C Targeted Antibody-Drug ConjugateJayaprakasam Bolleddula, Abhi Shah, Mohammad Shadid, Afrand Kamali, Michael D. Smith and Swapan K. ChowdhuryDrug Metabolism and Disposition November 2020, 48 (11) 1239-1245; DOI: https://doi.org/10.1124/dmd.120.000194
Squirewell, Edwin J.
- You have accessExposure of Rats to Multiple Oral Doses of Dichloroacetate Results in Upregulation of Hepatic Glutathione Transferases and NAD(P)H Dehydrogenase [Quinone] 1Edwin J. Squirewell, Ricky Mareus, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1224-1230; DOI: https://doi.org/10.1124/dmd.120.000143
- You have accessEffects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult RatsEdwin J. Squirewell, Marci G. Smeltz, Laura Rowland-Faux, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1217-1223; DOI: https://doi.org/10.1124/dmd.120.000142
Stacpoole, Peter W.
- You have accessExposure of Rats to Multiple Oral Doses of Dichloroacetate Results in Upregulation of Hepatic Glutathione Transferases and NAD(P)H Dehydrogenase [Quinone] 1Edwin J. Squirewell, Ricky Mareus, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1224-1230; DOI: https://doi.org/10.1124/dmd.120.000143
- You have accessEffects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult RatsEdwin J. Squirewell, Marci G. Smeltz, Laura Rowland-Faux, Lloyd P. Horne, Peter W. Stacpoole and Margaret O. JamesDrug Metabolism and Disposition November 2020, 48 (11) 1217-1223; DOI: https://doi.org/10.1124/dmd.120.000142
Subramanian, Raju
- You have accessCharacterization of Seasonal Pharmacokinetic Variability in WoodchucksJim Zheng, Scott Balsitis, Rex Santos, Bill J. Smith and Raju SubramanianDrug Metabolism and Disposition November 2020, 48 (11) 1199-1209; DOI: https://doi.org/10.1124/dmd.120.000140
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Tanis, Keith Q.
- You have accessA Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug DiscoveryMichael J. Hafey, Robert Houle, Keith Q. Tanis, Ian Knemeyer, Jackie Shang, Qing Chen, Andreas Baudy, James Monroe, Frank D. Sistare and Raymond EversDrug Metabolism and Disposition November 2020, 48 (11) 1147-1160; DOI: https://doi.org/10.1124/dmd.120.000086
Toren, Paul C.
- You have accessThe Respective Roles of CYP3A4 and CYP2D6 in the Metabolism of Pimozide to Established and Novel MetabolitesBrian D. Chapron, Jean C. Dinh, Paul C. Toren, Andrea Gaedigk and J. Steven LeederDrug Metabolism and Disposition November 2020, 48 (11) 1113-1120; DOI: https://doi.org/10.1124/dmd.120.000188
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Unadkat, Jashvant D.
- You have accessSuccessful Prediction of Positron Emission Tomography–Imaged Metformin Hepatic Uptake Clearance in Humans Using the Quantitative Proteomics–Informed Relative Expression Factor ApproachMadhav Sachar, Vineet Kumar, Lars C. Gormsen, Ole Lajord Munk and Jashvant D. UnadkatDrug Metabolism and Disposition November 2020, 48 (11) 1210-1216; DOI: https://doi.org/10.1124/dmd.120.000156
Ungell, Anna-Lena
- You have access(–)-N-3-Benzylphenobarbital Is Superior to Omeprazole and (+)-N-3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human HepatocytesMarie-Lynn Cuypers, Hugues Chanteux, Eric Gillent, Pierre Bonnaillie, Kenneth Saunders, Claire Beckers, Claude Delatour, Sylvie Dell’Aiera, Anna-Lena Ungell and Johan NicolaïDrug Metabolism and Disposition November 2020, 48 (11) 1121-1128; DOI: https://doi.org/10.1124/dmd.120.000089
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Wagner, Jonathan B.
- You have accessFunctional Consequences of Pravastatin Isomerization on OATP1B1-Mediated TransportJonathan B. Wagner, Melissa Ruggiero, J. Steven Leeder and Bruno HagenbuchDrug Metabolism and Disposition November 2020, 48 (11) 1192-1198; DOI: https://doi.org/10.1124/dmd.120.000122
Wang, Xin
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
Williamson, Beth
- You have accessEvaluation of the Disconnect between Hepatocyte and Microsome Intrinsic Clearance and In Vitro In Vivo Extrapolation PerformanceBeth Williamson, Stephanie Harlfinger and Dermot F. McGinnityDrug Metabolism and Disposition November 2020, 48 (11) 1137-1146; DOI: https://doi.org/10.1124/dmd.120.000131
Wong, Sylvia
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
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Yip, Victor
- Open AccessCharacterization of Tissue Distribution, Catabolism, and Elimination of an Anti–Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in RatsHao Cai, Victor Yip, M. Violet Lee, Sylvia Wong, Ola Saad, Shuguang Ma, Nina Ljumanovic, S. Cyrus Khojasteh, Amrita V. Kamath and Ben-Quan ShenDrug Metabolism and Disposition November 2020, 48 (11) 1161-1168; DOI: https://doi.org/10.1124/dmd.120.000092
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Zhang, Yuanjin
- You have accessGeneration and Characterization of Cytochrome P450 2J3/10 CRISPR/Cas9 Knockout Rat ModelJian Lu, Ang Chen, Xinrun Ma, Xuyang Shang, Yuanjin Zhang, Yuanqing Guo, Mingyao Liu and Xin WangDrug Metabolism and Disposition November 2020, 48 (11) 1129-1136; DOI: https://doi.org/10.1124/dmd.120.000114
Zheng, Jim
- You have accessCharacterization of Seasonal Pharmacokinetic Variability in WoodchucksJim Zheng, Scott Balsitis, Rex Santos, Bill J. Smith and Raju SubramanianDrug Metabolism and Disposition November 2020, 48 (11) 1199-1209; DOI: https://doi.org/10.1124/dmd.120.000140
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