| | | | | | | | | |
Ambrisentan | Negative | >100 | >100 | >100 | >100 | 10 | 9.8 | 0.01 | 0.12 |
Amoxicillin | Negative | >100 | >100 | >100 | >100 | 500 | 4.93 | 0.83 | 79.80 |
Amprenavir | Negative | 98 | >100 | 45.7 | >100 | 1200 | 18 | 0.10 | 17.62 |
Aripiprazole | Negative | 42.1 | >100 | >100 | >100 | 15 | 0.13 | 0.01 | 0.02 |
Aspirin | Negative | >100 | >100 | 45 | >100 | 2000 | 77.7 | 0.004 | 3.27 |
Atorvastatin | Negative | 6.3 | >100 | 3.8 | 19.8 | 80 | 0.1 | 0.02 | 0.19 |
Buspirone | Negative | >100 | >100 | >100 | >100 | 30 | 0.01 | 0.05 | 0.26 |
Caffeine | Negative | >100 | >100 | >100 | >100 | 200 | 11.7 | 0.83 | 66.70 |
Carisoprodol | Negative | >100 | >100 | >100 | >100 | 350 | 23 | 0.40 | 45.05 |
Cefprozil | Negative | 38.2 | >100 | >100 | >100 | 500 | 24.7 | 0.64 | 70.65 |
Cefuroxime | Negative | >100 | 33 | >100 | 9 | 500 | 41.3 | 0.50 | 59.92 |
Chloramphenicol | Negative | >100 | >100 | >100 | >100 | 666 | 10.3 | 0.47 | 69.27 |
Chlorpropamide | Negative | >100 | >100 | >100 | >100 | 500 | 275 | 0.10 | 39.55 |
Cimetidine | Negative | >100 | >100 | >100 | >100 | 1600 | 36.5 | 0.85 | 390.33 |
Ciprofloxacin | Negative | >100 | >100 | 73 | >100 | 600 | 9.66 | 0.80 | 104.30 |
Clarithromycin | Negative | >100 | >100 | 71 | 34.9 | 500 | 5 | 0.41 | 20.32 |
Clofibrate | Negative | >100 | >100 | >100 | >100 | 1000 | 404 | 0.08 | 54.30 |
Clotrimazole | Negative | 10 | >100 | >100 | >100 | 50 | 0.12 | 0.02 | 0.20 |
Diltiazem | Negative | >100 | >100 | >100 | >100 | 500 | 0.3 | 0.30 | 24.21 |
Diphenhydramine | Negative | 73 | >100 | >100 | 43 | 50 | 0.33 | 0.02 | 0.27 |
Dipyridamole | Negative | 0.8 | >100 | >100 | 2.8 | 100 | 3.67 | 0.009 | 0.15 |
Disopyramide | Negative | >100 | >100 | >100 | >100 | 800 | 22.4 | 0.50 | 89.75 |
Entacapone | Negative | 11.4 | 52 | 9 | 0.7 | 200 | 3.28 | 0.02 | 0.94 |
Erythromycin | Negative | >100 | >100 | >100 | >100 | 250 | 1.91 | 0.10 | 2.46 |
Esomeprasole | Negative | >100 | >100 | >100 | >100 | 40 | 7 | 0.03 | 0.44 |
Famotidine | Negative | >100 | >100 | >100 | >100 | 160 | 0.47 | 0.20 | 5.75 |
Fluoxetine | Negative | >100 | 43 | 32 | >100 | 80 | 0.98 | 0.06 | 1.09 |
Furosemide | Negative | >100 | >100 | >100 | 1.7 | 480 | 32.7 | 0.02 | 2.07 |
Hydroxyzine | Negative | >100 | >100 | >100 | >100 | 100 | 0.35 | 0.07 | 1.27 |
Levofloxacin | Negative | >100 | >100 | >100 | >100 | 750 | 25.7 | 0.27 | 44.30 |
Lopinavir | Negative | 7.4 | >100 | 81 | >100 | 800 | 18.8 | 0.02 | 2.07 |
Loracarbef | Negative | >100 | >100 | >100 | >100 | 625 | 56.8 | 0.08 | 13.19 |
Megestrol | Negative | 14.4 | >100 | >100 | >100 | 800 | 2.73 | 0.02 | 3.39 |
Meloxicam | Negative | 34 | >100 | >100 | >100 | 15 | 9.1 | 0.01 | 0.07 |
Metformin | Negative | >100 | >100 | >100 | >100 | 850 | 9.4 | 1.00 | 448.13 |
Nabumetone | Negative | >100 | >100 | >100 | 30.3 | 2000 | 315 | 0.01 | 8.99 |
Nadolol | Negative | 84 | >100 | >100 | >100 | 240 | 2.9 | 0.70 | 38.23 |
Naproxen | Negative | >100 | >100 | >100 | 25 | 500 | 423 | 0.01 | 5.68 |
Nifedipine | Negative | 23 | >100 | >100 | >100 | 30 | 0.26 | 0.08 | 0.48 |
Olanzapine | Negative | >100 | >100 | >100 | >100 | 20 | 0.26 | 0.07 | 0.32 |
Omeprazole | Negative | 22.5 | >100 | >100 | >100 | 40 | 5.41 | 0.05 | 0.66 |
Paroxetine | Negative | >100 | >100 | 59.5 | >100 | 60 | 0.05 | 0.05 | 0.61 |
Pentoxyfilline | Negative | >100 | >100 | 32.9 | >100 | 400 | 0.3 | 0.30 | 28.87 |
Probenecid | Negative | 68.5 | >100 | >100 | >100 | 500 | 122 | 0.25 | 59.70 |
Propranolol | Negative | >100 | >100 | >100 | >100 | 160 | 3.86 | 0.10 | 4.50 |
Quinidine | Negative | 49.3 | >100 | >100 | >100 | 400 | 4.84 | 0.20 | 17.43 |
Raloxifene | Negative | 37 | >100 | >100 | 30.5 | 60 | 0 | 0.05 | 0.42 |
Ranitidine | Negative | >100 | 91 | >100 | >100 | 150 | 1.5 | 0.15 | 5.00 |
Rosiglitazone | Negative | 0.6 | >100 | >100 | 4.3 | 8 | 1.4 | 0.002 | 0.01 |
Sumatriptan | Negative | >100 | >100 | >100 | >100 | 200 | 0.2 | 0.86 | 39.12 |
Tacrine | Negative | >100 | >100 | >100 | >100 | 160 | 0.17 | 0.45 | 24.29 |
Tetracycline | Negative | >100 | >100 | >100 | >100 | 500 | 9 | 0.45 | 37.80 |
Tramadol | Negative | >100 | >100 | >100 | >100 | 100 | 1.01 | 0.80 | 21.06 |
Trimethobenzamide | Negative | >100 | >100 | 48.8 | >100 | 300 | 10 | 1.00 | 61.49 |
Valsartan | Negative | 16.2 | >100 | >100 | >100 | 320 | 0.14 | 0.05 | 2.46 |
Verapamil | Negative | >100 | >100 | >100 | 52.7 | 120 | 0.6 | 0.10 | 1.82 |
Zolpidem | Negative | 97 | >100 | 56 | >100 | 10 | 0.39 | 0.08 | 0.205 |
Acetaminophen | Positive | >100 | >100 | >100 | >100 | 1000 | 64.6 | 0.90 | 455.04 |
Almorexant | Positive | 1.7 | >100 | >100 | >100 | 400 | 0.22 | 0.01 | 0.52 |
Alpidem | Positive | 9.3 | >100 | >100 | >100 | 50 | 0.07 | 0.01 | 0.05 |
Amiodarone | Positive | >100 | >100 | 58 | >100 | 600 | 0.7 | 0.04 | 2.51 |
Amoxicillin*-clavulanate** | Positive | >100 | >100 | >100 | 40 | 300*/75** | 9*/7.5** | 0.88*/0.75** | 56*/24** |
Azithromycin | Positive | >100 | >100 | 22.4 | >100 | 2000 | 2.36 | 0.93 | 167.75 |
Benzbromarone | Positive | 4.6 | 1.04 | >100 | 1 | 300 | 42.4 | 0.01 | 0.90 |
Bosentan | Positive | 37 | >100 | >100 | 22.2 | 125 | 2.54 | 0.02 | 0.35 |
Bromfenac | Positive | >100 | >100 | >100 | 1 | 50 | 12 | 0.001 | 0.02 |
Carbamazepine | Positive | >100 | >100 | >100 | >100 | 200 | 11.6 | 0.24 | 16.33 |
Chlormezanone | Positive | >100 | >100 | >100 | >100 | 600 | 32.9 | 0.52 | 93.09 |
Clopidogrel | Positive | 36 | >100 | >100 | >100 | 75 | 0.01 | 0.06 | 0.93 |
Clozapine | Positive | >100 | >100 | 38 | >100 | 300 | 3.67 | 0.03 | 1.95 |
Cyproterone acetate | Positive | 6.7 | >100 | >100 | >100 | 100 | 0.53 | 0.04 | 0.66 |
Diclofenac | Positive | >100 | >100 | >100 | 30 | 100 | 0.84 | 0.01 | 0.23 |
Dilevalol | Positive | >100 | >100 | >100 | >100 | 1200 | 1.12 | 0.50 | 122.40 |
Ethambutol | Positive | >100 | >100 | 35 | >100 | 2500 | 8.4 | 0.80 | 659.32 |
Felbamate | Positive | >100 | >100 | >100 | >100 | 1200 | 192 | 0.78 | 411.68 |
Flucloxacillin | Positive | 50.1 | >100 | >100 | >100 | 250 | 16 | 0.05 | 2.64 |
Flutamide | Positive | >100 | >100 | >100 | 10.9 | 250 | 0.36 | 0.06 | 3.64 |
HCV-796 | Positive | >100 | >100 | >100 | >100 | 1000 | 4.93 | 0.48 | 73.26 |
Isoniazid | Positive | >100 | >100 | >100 | >100 | 300 | 26.3 | 1.00 | 172.14 |
Labetalol | Positive | >100 | >100 | >100 | >100 | 600 | 1.36 | 0.50 | 61.66 |
Lapatanib | Positive | 1.2 | >100 | 57.1 | 1.6 | 1250 | 2.12 | 0.01 | 0.92 |
Lumiracoxib | Positive | >100 | >100 | >100 | 9 | 400 | 25 | 0.02 | 2.32 |
Methimazole | Positive | 56.1 | >100 | >100 | >100 | 20 | 3.5 | 0.05 | 0.76 |
Methyldopa | Positive | >100 | >100 | >100 | >100 | 500 | 10.4 | 0.90 | 151.40 |
Metiamide | Positive | >100 | >100 | 100 | >100 | | | | |
MK-0377 | Positive | >100 | >100 | 30 | >100 | | | | |
MK-0536 | Positive | >100 | >100 | >100 | >100 | 400 | 9.9 | 0.01 | 0.71 |
MK-0571 | Positive | 1.2 | 8.58 | 17.2 | 0.4 | | | | |
MK-0633 | Positive | 7.4 | >100 | >100 | 16.6 | 100 | 4 | 0.08 | 1.49 |
MK-0773 | Positive | 1.1 | >100 | >100 | 18.1 | 200 | 31.3 | 0.01 | 0.71 |
MK-0974 | Positive | 26.3 | >100 | >100 | 61.4 | 280 | 4 | 0.04 | 1.5 |
MK-A | Positive | >100 | 43 | 82 | >100 | 400 | 0.6 | 0.26 | 12.26 |
MK-2461 | Positive | 4.1 | 48 | >100 | 0.7 | 60 | 0.37 | 0.05 | 0.40 |
MK-2764 | Positive | >100 | >100 | 33 | >100 | 600 | 0.93 | 0.14 | 10.20 |
MK-3207 | Positive | 0.5 | >100 | >100 | >100 | 900 | 5 | 0.1 | 11.3 |
MK-3984 | Positive | >100 | >100 | >100 | >100 | 125 | 1.8 | 0.03 | 250.05 |
Nefazodone | Positive | 2.8 | >100 | >100 | >100 | 300 | 6.12 | 0.01 | 0.49 |
Nelfinavir | Positive | 22.8 | >100 | >100 | >100 | 250 | 5.3 | 0.02 | 0.69 |
Nevirapine | Positive | 72 | >100 | >100 | >100 | 200 | 5.81 | 0.40 | 22.31 |
Nitrofurantoin | Positive | >100 | >100 | >100 | 1.3 | 100 | 4.2 | 0.80 | 25.75 |
Nomifensine | Positive | >100 | >100 | >100 | >100 | 200 | 18 | 0.40 | 29.58 |
Oxandrolone | Positive | >100 | >100 | 67 | >100 | 20 | 1.30 | 0.05 | 0.28 |
Panadiplon | Positive | >100 | >100 | >100 | >100 | | | | |
Pemoline | Positive | 78 | >100 | 55 | >100 | 112 | 15.26 | 0.50 | 28.82 |
Perhexiline maleate | Positive | >100 | >100 | 30.2 | >100 | 200 | 0.24 | 0.10 | 4.83 |
Ritonavir | Positive | 0.7 | 85 | 31 | 25.5 | 600 | 15.3 | 0.02 | 1.42 |
Saquinavir | Positive | 11 | >100 | 23.9 | >100 | 1000 | 8.25 | 0.02 | 2.15 |
Sitaxsentan | Positive | 4.3 | >100 | >100 | 13.3 | 100 | 30.6 | 0.01 | 0.45 |
Sudoxicam | Positive | 33 | >100 | >100 | 60 | | | | |
Tasosartan | Positive | 1.7 | >100 | >100 | 30.8 | 300 | 12.7 | 0.01 | 0.31 |
Telithromycin | Positive | 4.2 | >100 | >100 | >100 | 400 | 1.02 | 0.40 | 13.54 |
Ticlopidine | Positive | 73 | >100 | >100 | >100 | 250 | 3.8 | 0.02 | 1.34 |
Ticrynafen | Positive | 41 | >100 | 80.6 | 13 | 500 | 42.3 | 0.02 | 2.14 |
Tolcapone | Positive | 12.1 | 46 | >100 | 0.6 | 200 | 20.9 | 0.001 | 0.07 |
Troglitazone | Positive | 1.3 | 6.3 | >100 | 21.3 | 600 | 7.5 | 0.01 | 0.98 |
Trovafloxacin mesylate | Positive | >100 | >100 | >100 | >100 | 200 | 5 | 0.30 | 11.11 |
Valproate | Positive | >100 | >100 | >100 | >100 | 650 | 477 | 0.19 | 143.83 |
Verlukast | Positive | 0.9 | 11.1 | 20.1 | 0.8 | 1500 | 241 | 0.001 | 0.44 |
Ximelagatran | Positive | >100 | 38 | >100 | >100 | | | | |
Zafirlukast | Positive | 4.5 | 11.5 | >100 | 5.8 | 20 | 0.65 | 0.01 | 0.03 |
Zimelidine | Positive | >100 | 58.3 | >100 | >100 | 600 | 1.64 | 0.09 | 10.99 |