Research ArticleArticle
Static Model–Based Assessment of OATP1B1-Mediated Drug Interactions with Preincubation-Dependent Inhibitors Based on Inactivation and Recovery Kinetics
Takayuki Taguchi, Yusuke Masuo, Azusa Futatsugi and Yukio Kato
Drug Metabolism and Disposition September 2020, 48 (9) 750-758; DOI: https://doi.org/10.1124/dmd.120.000020
Takayuki Taguchi
Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.)
Yusuke Masuo
Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.)
Azusa Futatsugi
Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.)
Yukio Kato
Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.)
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Prediction of OATP1B1-Mediated Preincubation-Dependent DDIs
Takayuki Taguchi, Yusuke Masuo, Azusa Futatsugi and Yukio Kato
Drug Metabolism and Disposition September 1, 2020, 48 (9) 750-758; DOI: https://doi.org/10.1124/dmd.120.000020
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