Article Figures & Data
Figures
Tables
Data Supplement
- Supplemental Data -
Supplementary Figure 1 - OATP1B1 activity after preincubation with regorafenib, nilotinib, and asunaprevir.
Supplementary Figure 2 - Observed kobs,app values for OATP1B1-mediated transport of [3H]E1S versus OATP1B1 inhibitor concentration.
Supplementary Figure 3 - Recovery of OATP1B1 activity after preincubation with OATP1B1 inhibitors.
Supplementary Table 1 - Validation of bioanalytical methods.
Supplementary Table 2 - Concentrations used in in vitro study and reported Km values of OATP1B1 substrates.
Supplementary Table 3 - Pharmacokinetic parameters of preincubation-dependent OATP1B1 inhibitors.
Supplementary Table 4 - Effect of preincubation with regorafenib, nilotinib, pazopanib, and asunaprevir on OATP1B1-mediated uptake.
Supplementary References
- Supplemental Data -