Index by author
January 01, 2021; Volume 49,Issue 1
A
Achour, Brahim
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Al-Majdoub, Zubida M.
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Aluri, Jagadeesh
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
Asakura, Shoji
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
B
Barber, Jill
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Beuckmann, Carsten T.
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
Bi, Yi-an
- You have accessEffect of Human Plasma on Hepatic Uptake of Organic Anion–Transporting Polypeptide 1B Substrates: Studies Using Transfected Cells and Primary Human HepatocytesYi-an Bi, Sangwoo Ryu, David A. Tess, A. David Rodrigues and Manthena V. S. VarmaDrug Metabolism and Disposition January 2021, 49 (1) 72-83; DOI: https://doi.org/10.1124/dmd.120.000134
C
Chen, Liangfu
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Chen, Shujuan
- You have accessRegulation of Intestinal UDP-Glucuronosyltransferase 1A1 by the Farnesoid X Receptor Agonist Obeticholic Acid Is Controlled by Constitutive Androstane Receptor through Intestinal MaturationAndré A. Weber, Elvira Mennillo, Xiaojing Yang, Lori W.E. van der Schoor, Johan W. Jonker, Shujuan Chen and Robert H. TukeyDrug Metabolism and Disposition January 2021, 49 (1) 12-19; DOI: https://doi.org/10.1124/dmd.120.000240
Clench, Malcolm R.
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Corton, J. Christopher
- You have accessSex-, Age-, and Race/Ethnicity-Dependent Variations in Drug-Processing and NRF2-Regulated Genes in Human LiversJie Liu, Julia Yue Cui, Yuan-Fu Lu, J. Christopher Corton and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 111-119; DOI: https://doi.org/10.1124/dmd.120.000181
Couto, Narciso
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Cui, Julia Yue
- You have accessSex-, Age-, and Race/Ethnicity-Dependent Variations in Drug-Processing and NRF2-Regulated Genes in Human LiversJie Liu, Julia Yue Cui, Yuan-Fu Lu, J. Christopher Corton and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 111-119; DOI: https://doi.org/10.1124/dmd.120.000181
D
Dallas, Shannon
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Deguchi, Yoshiharu
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
Ding, Xinxin
- You have accessEditorialXinxin DingDrug Metabolism and Disposition January 2021, 49 (1) 1-2; DOI: https://doi.org/10.1124/dmd.120.000298
E
Einolf, Heidi J.
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Endo, Hiromi
- You have accessDownregulation of CYP1A2, CYP2B6, and CYP3A4 in Human Hepatocytes by Prolyl Hydroxylase Domain 2 Inhibitors via Hypoxia-Inducible Factor-α StabilizationHiroki Takano, Jun-ichi Yamaguchi, Sota Kato, Makoto Hamada, Mika Tada and Hiromi EndoDrug Metabolism and Disposition January 2021, 49 (1) 20-30; DOI: https://doi.org/10.1124/dmd.120.000124
Enomoto, Tsuyoshi
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
F
Fricker, Gert
- You have accessExtension of the Mechanistic Tissue Distribution Model of Rodgers and Rowland by Systematic Incorporation of Lysosomal Trapping: Impact on Unbound Partition Coefficient and Volume of Distribution Predictions in the RatMaximilian V. Schmitt, Andreas Reichel, Xiaohui Liu, Gert Fricker and Philip LienauDrug Metabolism and Disposition January 2021, 49 (1) 53-61; DOI: https://doi.org/10.1124/dmd.120.000161
Fung, Conrad
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
G
Goosen, Theunis C.
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Guo, Ying
- You have accessEffect of Gender and Various Diets on Bile Acid Profile and Related Genes in MiceChong Ma, Ying Guo and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 62-71; DOI: https://doi.org/10.1124/dmd.120.000166
H
Hamada, Makoto
- You have accessDownregulation of CYP1A2, CYP2B6, and CYP3A4 in Human Hepatocytes by Prolyl Hydroxylase Domain 2 Inhibitors via Hypoxia-Inducible Factor-α StabilizationHiroki Takano, Jun-ichi Yamaguchi, Sota Kato, Makoto Hamada, Mika Tada and Hiromi EndoDrug Metabolism and Disposition January 2021, 49 (1) 20-30; DOI: https://doi.org/10.1124/dmd.120.000124
Hariparsad, Niresh
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Higuchi, Kei
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
I
Ishida, Tomomi
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
J
Jones, Barry
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Jonker, Johan W.
- You have accessRegulation of Intestinal UDP-Glucuronosyltransferase 1A1 by the Farnesoid X Receptor Agonist Obeticholic Acid Is Controlled by Constitutive Androstane Receptor through Intestinal MaturationAndré A. Weber, Elvira Mennillo, Xiaojing Yang, Lori W.E. van der Schoor, Johan W. Jonker, Shujuan Chen and Robert H. TukeyDrug Metabolism and Disposition January 2021, 49 (1) 12-19; DOI: https://doi.org/10.1124/dmd.120.000240
K
Kameyama, Takaaki
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
Karunakaran, Esther
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Kato, Sota
- You have accessDownregulation of CYP1A2, CYP2B6, and CYP3A4 in Human Hepatocytes by Prolyl Hydroxylase Domain 2 Inhibitors via Hypoxia-Inducible Factor-α StabilizationHiroki Takano, Jun-ichi Yamaguchi, Sota Kato, Makoto Hamada, Mika Tada and Hiromi EndoDrug Metabolism and Disposition January 2021, 49 (1) 20-30; DOI: https://doi.org/10.1124/dmd.120.000124
Kawabata, Kenji
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
Klaassen, Curtis D.
- You have accessEffect of Gender and Various Diets on Bile Acid Profile and Related Genes in MiceChong Ma, Ying Guo and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 62-71; DOI: https://doi.org/10.1124/dmd.120.000166
- You have accessSex-, Age-, and Race/Ethnicity-Dependent Variations in Drug-Processing and NRF2-Regulated Genes in Human LiversJie Liu, Julia Yue Cui, Yuan-Fu Lu, J. Christopher Corton and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 111-119; DOI: https://doi.org/10.1124/dmd.120.000181
Kurimori, Ko
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
Kurosawa, Toshiki
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
Kusano, Kazutomi
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
Kusuhara, Hiroyuki
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
L
Lienau, Philip
- You have accessExtension of the Mechanistic Tissue Distribution Model of Rodgers and Rowland by Systematic Incorporation of Lysosomal Trapping: Impact on Unbound Partition Coefficient and Volume of Distribution Predictions in the RatMaximilian V. Schmitt, Andreas Reichel, Xiaohui Liu, Gert Fricker and Philip LienauDrug Metabolism and Disposition January 2021, 49 (1) 53-61; DOI: https://doi.org/10.1124/dmd.120.000161
Liu, Jie
- You have accessSex-, Age-, and Race/Ethnicity-Dependent Variations in Drug-Processing and NRF2-Regulated Genes in Human LiversJie Liu, Julia Yue Cui, Yuan-Fu Lu, J. Christopher Corton and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 111-119; DOI: https://doi.org/10.1124/dmd.120.000181
Liu, Xiaohui
- You have accessExtension of the Mechanistic Tissue Distribution Model of Rodgers and Rowland by Systematic Incorporation of Lysosomal Trapping: Impact on Unbound Partition Coefficient and Volume of Distribution Predictions in the RatMaximilian V. Schmitt, Andreas Reichel, Xiaohui Liu, Gert Fricker and Philip LienauDrug Metabolism and Disposition January 2021, 49 (1) 53-61; DOI: https://doi.org/10.1124/dmd.120.000161
Lu, Yuan-Fu
- You have accessSex-, Age-, and Race/Ethnicity-Dependent Variations in Drug-Processing and NRF2-Regulated Genes in Human LiversJie Liu, Julia Yue Cui, Yuan-Fu Lu, J. Christopher Corton and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 111-119; DOI: https://doi.org/10.1124/dmd.120.000181
M
Ma, Chong
- You have accessEffect of Gender and Various Diets on Bile Acid Profile and Related Genes in MiceChong Ma, Ying Guo and Curtis D. KlaassenDrug Metabolism and Disposition January 2021, 49 (1) 62-71; DOI: https://doi.org/10.1124/dmd.120.000166
Maeda, Kazuya
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
Mennillo, Elvira
- You have accessRegulation of Intestinal UDP-Glucuronosyltransferase 1A1 by the Farnesoid X Receptor Agonist Obeticholic Acid Is Controlled by Constitutive Androstane Receptor through Intestinal MaturationAndré A. Weber, Elvira Mennillo, Xiaojing Yang, Lori W.E. van der Schoor, Johan W. Jonker, Shujuan Chen and Robert H. TukeyDrug Metabolism and Disposition January 2021, 49 (1) 12-19; DOI: https://doi.org/10.1124/dmd.120.000240
Michiba, Kazuyoshi
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
Mizuno, Tadahaya
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
Mochizuki, Tatsuki
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
N
Newton, Jillian R.A.
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Nishiyama, Hiroyuki
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
Nozaki, Yoshitane
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
O
Oda, Tatsuya
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
P
Palamanda, Jairam
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
R
Ramsden, Diane
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Reichel, Andreas
- You have accessExtension of the Mechanistic Tissue Distribution Model of Rodgers and Rowland by Systematic Incorporation of Lysosomal Trapping: Impact on Unbound Partition Coefficient and Volume of Distribution Predictions in the RatMaximilian V. Schmitt, Andreas Reichel, Xiaohui Liu, Gert Fricker and Philip LienauDrug Metabolism and Disposition January 2021, 49 (1) 53-61; DOI: https://doi.org/10.1124/dmd.120.000161
Rodrigues, A. David
- You have accessEffect of Human Plasma on Hepatic Uptake of Organic Anion–Transporting Polypeptide 1B Substrates: Studies Using Transfected Cells and Primary Human HepatocytesYi-an Bi, Sangwoo Ryu, David A. Tess, A. David Rodrigues and Manthena V. S. VarmaDrug Metabolism and Disposition January 2021, 49 (1) 72-83; DOI: https://doi.org/10.1124/dmd.120.000134
Rostami-Hodjegan, Amin
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Russo, Cristina
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Ryu, Sangwoo
- You have accessEffect of Human Plasma on Hepatic Uptake of Organic Anion–Transporting Polypeptide 1B Substrates: Studies Using Transfected Cells and Primary Human HepatocytesYi-an Bi, Sangwoo Ryu, David A. Tess, A. David Rodrigues and Manthena V. S. VarmaDrug Metabolism and Disposition January 2021, 49 (1) 72-83; DOI: https://doi.org/10.1124/dmd.120.000134
S
Schmitt, Maximilian V.
- You have accessExtension of the Mechanistic Tissue Distribution Model of Rodgers and Rowland by Systematic Incorporation of Lysosomal Trapping: Impact on Unbound Partition Coefficient and Volume of Distribution Predictions in the RatMaximilian V. Schmitt, Andreas Reichel, Xiaohui Liu, Gert Fricker and Philip LienauDrug Metabolism and Disposition January 2021, 49 (1) 53-61; DOI: https://doi.org/10.1124/dmd.120.000161
Shimomura, Osamu
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
Sidaway, James
- You have accessLabel-Free Quantitative Proteomics and Substrate-Based Mass Spectrometry Imaging of Xenobiotic Metabolizing Enzymes in Ex Vivo Human Skin and a Human Living Skin Equivalent ModelNarciso Couto, Jillian R.A. Newton, Cristina Russo, Esther Karunakaran, Brahim Achour, Zubida M. Al-Majdoub, James Sidaway, Amin Rostami-Hodjegan, Malcolm R. Clench and Jill BarberDrug Metabolism and Disposition January 2021, 49 (1) 39-52; DOI: https://doi.org/10.1124/dmd.120.000168
Siu, Y. Amy
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Suzuki, Michiyuki
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
T
Tada, Mika
- You have accessDownregulation of CYP1A2, CYP2B6, and CYP3A4 in Human Hepatocytes by Prolyl Hydroxylase Domain 2 Inhibitors via Hypoxia-Inducible Factor-α StabilizationHiroki Takano, Jun-ichi Yamaguchi, Sota Kato, Makoto Hamada, Mika Tada and Hiromi EndoDrug Metabolism and Disposition January 2021, 49 (1) 20-30; DOI: https://doi.org/10.1124/dmd.120.000124
Takano, Hiroki
- You have accessDownregulation of CYP1A2, CYP2B6, and CYP3A4 in Human Hepatocytes by Prolyl Hydroxylase Domain 2 Inhibitors via Hypoxia-Inducible Factor-α StabilizationHiroki Takano, Jun-ichi Yamaguchi, Sota Kato, Makoto Hamada, Mika Tada and Hiromi EndoDrug Metabolism and Disposition January 2021, 49 (1) 20-30; DOI: https://doi.org/10.1124/dmd.120.000124
Takeuchi, Tomoyo
- You have accessCharacterization of the Human Intestinal Drug Transport with Ussing Chamber System Incorporating Freshly Isolated Human JejunumKazuyoshi Michiba, Kazuya Maeda, Ko Kurimori, Tsuyoshi Enomoto, Osamu Shimomura, Tomoyo Takeuchi, Hiroyuki Nishiyama, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 84-93; DOI: https://doi.org/10.1124/dmd.120.000138
Tega, Yuma
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
Tess, David A.
- You have accessEffect of Human Plasma on Hepatic Uptake of Organic Anion–Transporting Polypeptide 1B Substrates: Studies Using Transfected Cells and Primary Human HepatocytesYi-an Bi, Sangwoo Ryu, David A. Tess, A. David Rodrigues and Manthena V. S. VarmaDrug Metabolism and Disposition January 2021, 49 (1) 72-83; DOI: https://doi.org/10.1124/dmd.120.000134
Tukey, Robert H.
- You have accessRegulation of Intestinal UDP-Glucuronosyltransferase 1A1 by the Farnesoid X Receptor Agonist Obeticholic Acid Is Controlled by Constitutive Androstane Receptor through Intestinal MaturationAndré A. Weber, Elvira Mennillo, Xiaojing Yang, Lori W.E. van der Schoor, Johan W. Jonker, Shujuan Chen and Robert H. TukeyDrug Metabolism and Disposition January 2021, 49 (1) 12-19; DOI: https://doi.org/10.1124/dmd.120.000240
Tweedie, Donald
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
U
Ueno, Takashi
- You have accessDisposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating MetabolitesTakashi Ueno, Tomomi Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura and Kazutomi KusanoDrug Metabolism and Disposition January 2021, 49 (1) 31-38; DOI: https://doi.org/10.1124/dmd.120.000229
V
van der Schoor, Lori W.E.
- You have accessRegulation of Intestinal UDP-Glucuronosyltransferase 1A1 by the Farnesoid X Receptor Agonist Obeticholic Acid Is Controlled by Constitutive Androstane Receptor through Intestinal MaturationAndré A. Weber, Elvira Mennillo, Xiaojing Yang, Lori W.E. van der Schoor, Johan W. Jonker, Shujuan Chen and Robert H. TukeyDrug Metabolism and Disposition January 2021, 49 (1) 12-19; DOI: https://doi.org/10.1124/dmd.120.000240
Varma, Manthena V. S.
- You have accessEffect of Human Plasma on Hepatic Uptake of Organic Anion–Transporting Polypeptide 1B Substrates: Studies Using Transfected Cells and Primary Human HepatocytesYi-an Bi, Sangwoo Ryu, David A. Tess, A. David Rodrigues and Manthena V. S. VarmaDrug Metabolism and Disposition January 2021, 49 (1) 72-83; DOI: https://doi.org/10.1124/dmd.120.000134
W
Weber, André A.
- You have accessRegulation of Intestinal UDP-Glucuronosyltransferase 1A1 by the Farnesoid X Receptor Agonist Obeticholic Acid Is Controlled by Constitutive Androstane Receptor through Intestinal MaturationAndré A. Weber, Elvira Mennillo, Xiaojing Yang, Lori W.E. van der Schoor, Johan W. Jonker, Shujuan Chen and Robert H. TukeyDrug Metabolism and Disposition January 2021, 49 (1) 12-19; DOI: https://doi.org/10.1124/dmd.120.000240
Wong, Simon G.
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Y
Yamaguchi, Jun-ichi
- You have accessDownregulation of CYP1A2, CYP2B6, and CYP3A4 in Human Hepatocytes by Prolyl Hydroxylase Domain 2 Inhibitors via Hypoxia-Inducible Factor-α StabilizationHiroki Takano, Jun-ichi Yamaguchi, Sota Kato, Makoto Hamada, Mika Tada and Hiromi EndoDrug Metabolism and Disposition January 2021, 49 (1) 20-30; DOI: https://doi.org/10.1124/dmd.120.000124
Yamaguchi, Tomoko
- You have accessFunctional Investigation of Solute Carrier Family 35, Member F2, in Three Cellular Models of the Primate Blood-Brain BarrierTatsuki Mochizuki, Tadahaya Mizuno, Toshiki Kurosawa, Tomoko Yamaguchi, Kei Higuchi, Yuma Tega, Yoshitane Nozaki, Kenji Kawabata, Yoshiharu Deguchi and Hiroyuki KusuharaDrug Metabolism and Disposition January 2021, 49 (1) 3-11; DOI: https://doi.org/10.1124/dmd.120.000115
Yang, Xiaojing
- You have accessRegulation of Intestinal UDP-Glucuronosyltransferase 1A1 by the Farnesoid X Receptor Agonist Obeticholic Acid Is Controlled by Constitutive Androstane Receptor through Intestinal MaturationAndré A. Weber, Elvira Mennillo, Xiaojing Yang, Lori W.E. van der Schoor, Johan W. Jonker, Shujuan Chen and Robert H. TukeyDrug Metabolism and Disposition January 2021, 49 (1) 12-19; DOI: https://doi.org/10.1124/dmd.120.000240
Yates, Phillip D.
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
Z
Zhang, George
- You have accessConsiderations from the Innovation and Quality Induction Working Group in Response to Drug-Drug Interaction Guidance from Regulatory Agencies: Guidelines on Model Fitting and Recommendations on Time Course for In Vitro Cytochrome P450 Induction Studies Including Impact on Drug Interaction Risk AssessmentSimon G. Wong, Diane Ramsden, Shannon Dallas, Conrad Fung, Heidi J. Einolf, Jairam Palamanda, Liangfu Chen, Theunis C. Goosen, Y. Amy Siu, George Zhang, Donald Tweedie, Niresh Hariparsad, Barry Jones and Phillip D. YatesDrug Metabolism and Disposition January 2021, 49 (1) 94-110; DOI: https://doi.org/10.1124/dmd.120.000055
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