Index by author
December 01, 2021; Volume 49,Issue 12
A
Allinder, Matthew
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
B
Bardhi, Keti
- Open AccessInhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their MetabolitesShamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
Barnouin, Karin
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
Bershas, David A.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
C
Chan, Tom S.
- You have accessHLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable BeadsTing Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. ChanDrug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
Chen, Gang
- Open AccessCharacterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, ExemestaneIrina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
- Open AccessInhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their MetabolitesShamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
Crossman, Lee
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
Cutler, Paul
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
D
Dennison, Jeremy M.T.J.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
de Wildt, Saskia N.
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
F
Fort, Gabriela
- Open AccessInhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their MetabolitesShamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
H
Holenarsipur, Vinay K.
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Humphreys, W. Griffith
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
K
Keith-Luzzi, Monica
- You have accessHLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable BeadsTing Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. ChanDrug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
Kenworthy, David
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
Kiss, Márton
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
Kist, Nico
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
Korzekwa, Ken
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical ConsiderationsZeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken KorzekwaDrug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental DataErickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati NagarDrug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
Kotian, Apoorva
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
L
Lai, Yurong
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Lazarus, Philip
- Open AccessCharacterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, ExemestaneIrina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
- Open AccessInhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their MetabolitesShamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
- Open AccessCannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug InteractionsShamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442
M
Mariappan, T. Thanga
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Mbasu, Richard
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
McLaughlin, Megan M.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
Mooij, Miriam G.
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
Mudunuru, Jennypher
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
N
Nagar, Swati
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical ConsiderationsZeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken KorzekwaDrug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental DataErickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati NagarDrug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
Nasrin, Shamema
- Open AccessInhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their MetabolitesShamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
- Open AccessCannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug InteractionsShamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442
Nicolaï, Johan
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
O
O’Connor-Semmes, Robin L.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
P
Panfen, Erika
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Paragas, Erickson M.
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical ConsiderationsZeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken KorzekwaDrug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental DataErickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati NagarDrug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
Pereira, Adrian I.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
Perez-Paramo, Yadira X
- Open AccessCannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug InteractionsShamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442
Pirhalla, Jill L.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
R
Russel, Frans G. M.
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
S
Sanghvi, Mitesh
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
Shen, Hong
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Swift, Brandon
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
T
Tang, Jennifer
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Teslenko, Irina
- Open AccessCharacterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, ExemestaneIrina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
Thorpe, Karl M.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
U
Ungell, Anna-Lena
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
W
Wang, Ting
- You have accessHLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable BeadsTing Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. ChanDrug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
Wang, Zeyuan
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical ConsiderationsZeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken KorzekwaDrug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
- You have accessComplex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental DataErickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati NagarDrug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
Watson, Christy J.W.
- Open AccessCharacterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, ExemestaneIrina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
- Open AccessCannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug InteractionsShamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442
Watson, Christy J. W.
- Open AccessInhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their MetabolitesShamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
Whitcher-Johnstone, Andrea
- You have accessHLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable BeadsTing Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. ChanDrug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
Wijnen, Rene M. H.
- Open AccessOntogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative ProteomicsMárton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de WildtDrug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
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Xia, Zuping
- Open AccessCharacterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, ExemestaneIrina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip LazarusDrug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
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Young, Graeme C.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
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Zamek-Gliszczynski, Maciej J.
- Open AccessPharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male VolunteersMaciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. YoungDrug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
Zhang, Yueping
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Zhao, Xiaofeng
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
Zheng, Jim
- You have accessEndogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 InhibitionJennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong LaiDrug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
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