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Drug Metabolism & Disposition

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    • Current Issue
    • Fast Forward
    • Latest Articles
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Index by author

December 01, 2021; Volume 49,Issue 12
  • A
  • B
  • C
  • D
  • E
  • F
  • G
  • H
  • I
  • J
  • K
  • L
  • M
  • N
  • O
  • P
  • Q
  • R
  • S
  • T
  • U
  • V
  • W
  • X
  • Y
  • Z

A

  1. Allinder, Matthew

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

B

  1. Bardhi, Keti

    1. Open Access
      Inhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their Metabolites
      Shamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
  2. Barnouin, Karin

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
  3. Bershas, David A.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

C

  1. Chan, Tom S.

    1. You have access
      HLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable Beads
      Ting Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. Chan
      Drug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
  2. Chen, Gang

    1. Open Access
      Characterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, Exemestane
      Irina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
    2. Open Access
      Inhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their Metabolites
      Shamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
  3. Crossman, Lee

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
  4. Cutler, Paul

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559

D

  1. Dennison, Jeremy M.T.J.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
  2. de Wildt, Saskia N.

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559

F

  1. Fort, Gabriela

    1. Open Access
      Inhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their Metabolites
      Shamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530

H

  1. Holenarsipur, Vinay K.

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  2. Humphreys, W. Griffith

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486

K

  1. Keith-Luzzi, Monica

    1. You have access
      HLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable Beads
      Ting Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. Chan
      Drug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
  2. Kenworthy, David

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
  3. Kiss, Márton

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
  4. Kist, Nico

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
  5. Korzekwa, Ken

    1. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical Considerations
      Zeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken Korzekwa
      Drug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
    2. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental Data
      Erickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati Nagar
      Drug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
  6. Kotian, Apoorva

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559

L

  1. Lai, Yurong

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  2. Lazarus, Philip

    1. Open Access
      Characterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, Exemestane
      Irina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
    2. Open Access
      Inhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their Metabolites
      Shamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
    3. Open Access
      Cannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug Interactions
      Shamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442

M

  1. Mariappan, T. Thanga

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  2. Mbasu, Richard

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
  3. McLaughlin, Megan M.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
  4. Mooij, Miriam G.

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559
  5. Mudunuru, Jennypher

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

N

  1. Nagar, Swati

    1. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical Considerations
      Zeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken Korzekwa
      Drug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
    2. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental Data
      Erickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati Nagar
      Drug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
  2. Nasrin, Shamema

    1. Open Access
      Inhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their Metabolites
      Shamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
    2. Open Access
      Cannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug Interactions
      Shamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442
  3. Nicolaï, Johan

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559

O

  1. O’Connor-Semmes, Robin L.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

P

  1. Panfen, Erika

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  2. Paragas, Erickson M.

    1. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical Considerations
      Zeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken Korzekwa
      Drug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
    2. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental Data
      Erickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati Nagar
      Drug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
  3. Pereira, Adrian I.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
  4. Perez-Paramo, Yadira X

    1. Open Access
      Cannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug Interactions
      Shamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442
  5. Pirhalla, Jill L.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

R

  1. Russel, Frans G. M.

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559

S

  1. Sanghvi, Mitesh

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
  2. Shen, Hong

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  3. Swift, Brandon

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

T

  1. Tang, Jennifer

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  2. Teslenko, Irina

    1. Open Access
      Characterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, Exemestane
      Irina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
  3. Thorpe, Karl M.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

U

  1. Ungell, Anna-Lena

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559

W

  1. Wang, Ting

    1. You have access
      HLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable Beads
      Ting Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. Chan
      Drug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
  2. Wang, Zeyuan

    1. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 1. Theoretical Considerations
      Zeyuan Wang, Erickson M. Paragas, Swati Nagar and Ken Korzekwa
      Drug Metabolism and Disposition December 2021, 49 (12) 1090-1099; DOI: https://doi.org/10.1124/dmd.121.000553
    2. You have access
      Complex Cytochrome P450 Kinetics Due to Multisubstrate Binding and Sequential Metabolism. Part 2. Modeling of Experimental Data
      Erickson M. Paragas, Zeyuan Wang, Ken Korzekwa and Swati Nagar
      Drug Metabolism and Disposition December 2021, 49 (12) 1100-1108; DOI: https://doi.org/10.1124/dmd.121.000554
  3. Watson, Christy J.W.

    1. Open Access
      Characterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, Exemestane
      Irina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635
    2. Open Access
      Cannabinoid Metabolites as Inhibitors of Major Hepatic CYP450 Enzymes, with Implications for Cannabis-Drug Interactions
      Shamema Nasrin, Christy J.W. Watson, Yadira X Perez-Paramo and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1070-1080; DOI: https://doi.org/10.1124/dmd.121.000442
  4. Watson, Christy J. W.

    1. Open Access
      Inhibition of UDP-Glucuronosyltransferase Enzymes by Major Cannabinoids and Their Metabolites
      Shamema Nasrin, Christy J. W. Watson, Keti Bardhi, Gabriela Fort, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1081-1089; DOI: https://doi.org/10.1124/dmd.121.000530
  5. Whitcher-Johnstone, Andrea

    1. You have access
      HLM-beads: Rapid Assessment of Nonspecific Binding to Human Liver Microsomes Using Magnetizable Beads
      Ting Wang, Andrea Whitcher-Johnstone, Monica Keith-Luzzi and Tom S. Chan
      Drug Metabolism and Disposition December 2021, 49 (12) 1056-1062; DOI: https://doi.org/10.1124/dmd.121.000575
  6. Wijnen, Rene M. H.

    1. Open Access
      Ontogeny of Small Intestinal Drug Transporters and Metabolizing Enzymes Based on Targeted Quantitative Proteomics
      Márton Kiss, Richard Mbasu, Johan Nicolaï, Karin Barnouin, Apoorva Kotian, Miriam G. Mooij, Nico Kist, Rene M. H. Wijnen, Anna-Lena Ungell, Paul Cutler, Frans G. M. Russel and Saskia N. de Wildt
      Drug Metabolism and Disposition December 2021, 49 (12) 1038-1046; DOI: https://doi.org/10.1124/dmd.121.000559

X

  1. Xia, Zuping

    1. Open Access
      Characterization of Cytosolic Glutathione S-Transferases Involved in the Metabolism of the Aromatase Inhibitor, Exemestane
      Irina Teslenko, Christy J.W. Watson, Zuping Xia, Gang Chen and Philip Lazarus
      Drug Metabolism and Disposition December 2021, 49 (12) 1047-1055; DOI: https://doi.org/10.1124/dmd.121.000635

Y

  1. Young, Graeme C.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595

Z

  1. Zamek-Gliszczynski, Maciej J.

    1. Pharmacokinetics and ADME Characterization of Intravenous and Oral [<sup>14</sup>C]-Linerixibat in Healthy Male Volunteers
      Open Access
      Pharmacokinetics and ADME Characterization of Intravenous and Oral [14C]-Linerixibat in Healthy Male Volunteers
      Maciej J. Zamek-Gliszczynski, David Kenworthy, David A. Bershas, Mitesh Sanghvi, Adrian I. Pereira, Jennypher Mudunuru, Lee Crossman, Jill L. Pirhalla, Karl M. Thorpe, Jeremy M.T.J. Dennison, Megan M. McLaughlin, Matthew Allinder, Brandon Swift, Robin L. O’Connor-Semmes and Graeme C. Young
      Drug Metabolism and Disposition December 2021, 49 (12) 1109-1117; DOI: https://doi.org/10.1124/dmd.121.000595
  2. Zhang, Yueping

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  3. Zhao, Xiaofeng

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
  4. Zheng, Jim

    1. You have access
      Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
      Jennifer Tang, Hong Shen, Xiaofeng Zhao, Vinay K. Holenarsipur, T. Thanga Mariappan, Yueping Zhang, Erika Panfen, Jim Zheng, W. Griffith Humphreys and Yurong Lai
      Drug Metabolism and Disposition December 2021, 49 (12) 1063-1069; DOI: https://doi.org/10.1124/dmd.121.000486
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Drug Metabolism and Disposition: 49 (12)
Drug Metabolism and Disposition
Vol. 49, Issue 12
1 Dec 2021
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  • Cytochrome P450 inhibitors. Evaluation of specificities in the in vitrometabolism of therapeutic agents by human liver microsomes.
  • Prediction of Human Clearance of Twenty-Nine Drugs from Hepatic Microsomal Intrinsic Clearance Data: An Examination of In Vitro Half-Life Approach and Nonspecific Binding to Microsomes
  • THE HUMAN INTESTINAL CYTOCHROME P450 “PIE”
  • DRUG-DRUG INTERACTIONS FOR UDP-GLUCURONOSYLTRANSFERASE SUBSTRATES: A PHARMACOKINETIC EXPLANATION FOR TYPICALLY OBSERVED LOW EXPOSURE (AUCI/AUC) RATIOS
  • In Vitro-In Vivo Scaling of CYP Kinetic Data Not Consistent with the Classical Michaelis-Menten Model
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