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Drug Metabolism & Disposition

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    • Current Issue
    • Fast Forward
    • Latest Articles
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Index by author

May 01, 2021; Volume 49,Issue 5
  • A
  • B
  • C
  • D
  • E
  • F
  • G
  • H
  • I
  • J
  • K
  • L
  • M
  • N
  • O
  • P
  • Q
  • R
  • S
  • T
  • U
  • V
  • W
  • X
  • Y
  • Z

B

  1. Bai, April

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220
  2. Boyer, Bert B.

    1. Open Access
      In Vivo Functional Effects of CYP2C9 M1L, a Novel and Common Variant in the Yup’ik Alaska Native Population
      Lindsay M. Henderson, Scarlett E. Hopkins, Bert B. Boyer, Timothy A. Thornton, Allan E. Rettie and Kenneth E. Thummel
      Drug Metabolism and Disposition May 2021, 49 (5) 345-352; DOI: https://doi.org/10.1124/dmd.120.000301
  3. Brooks, Jennifer

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220

C

  1. Cai, Hui

    1. Identification of Triterpene Acids in <em>Poria cocos</em> Extract as Bile Acid Uptake Transporter Inhibitors
      You have access
      Identification of Triterpene Acids in Poria cocos Extract as Bile Acid Uptake Transporter Inhibitors
      Hui Cai, Yujie Cheng, Qiunan Zhu, Dexuan Kong, Xijing Chen, Ikumi Tamai and Yang Lu
      Drug Metabolism and Disposition May 2021, 49 (5) 353-360; DOI: https://doi.org/10.1124/dmd.120.000308
  2. Cain, Meredith

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273
  3. Chen, Shitong

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  4. Chen, Xijing

    1. Identification of Triterpene Acids in <em>Poria cocos</em> Extract as Bile Acid Uptake Transporter Inhibitors
      You have access
      Identification of Triterpene Acids in Poria cocos Extract as Bile Acid Uptake Transporter Inhibitors
      Hui Cai, Yujie Cheng, Qiunan Zhu, Dexuan Kong, Xijing Chen, Ikumi Tamai and Yang Lu
      Drug Metabolism and Disposition May 2021, 49 (5) 353-360; DOI: https://doi.org/10.1124/dmd.120.000308
  5. Cheng, Yujie

    1. Identification of Triterpene Acids in <em>Poria cocos</em> Extract as Bile Acid Uptake Transporter Inhibitors
      You have access
      Identification of Triterpene Acids in Poria cocos Extract as Bile Acid Uptake Transporter Inhibitors
      Hui Cai, Yujie Cheng, Qiunan Zhu, Dexuan Kong, Xijing Chen, Ikumi Tamai and Yang Lu
      Drug Metabolism and Disposition May 2021, 49 (5) 353-360; DOI: https://doi.org/10.1124/dmd.120.000308

D

  1. Dalvie, Deepak

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220

G

  1. Gui, Lanlan

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385

H

  1. Han, Shengna

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  2. Hargreaves, Richard

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220
  3. Henderson, Lindsay M.

    1. Open Access
      In Vivo Functional Effects of CYP2C9 M1L, a Novel and Common Variant in the Yup’ik Alaska Native Population
      Lindsay M. Henderson, Scarlett E. Hopkins, Bert B. Boyer, Timothy A. Thornton, Allan E. Rettie and Kenneth E. Thummel
      Drug Metabolism and Disposition May 2021, 49 (5) 345-352; DOI: https://doi.org/10.1124/dmd.120.000301
  4. Ho, Ming-Fen

    1. Open Access
      SLCO1B1: Application and Limitations of Deep Mutational Scanning for Genomic Missense Variant Function
      Lingxin Zhang, Vivekananda Sarangi, Ming-Fen Ho, Irene Moon, Krishna R. Kalari, Liewei Wang and Richard M. Weinshilboum
      Drug Metabolism and Disposition May 2021, 49 (5) 395-404; DOI: https://doi.org/10.1124/dmd.120.000264
  5. Hopkins, Scarlett E.

    1. Open Access
      In Vivo Functional Effects of CYP2C9 M1L, a Novel and Common Variant in the Yup’ik Alaska Native Population
      Lindsay M. Henderson, Scarlett E. Hopkins, Bert B. Boyer, Timothy A. Thornton, Allan E. Rettie and Kenneth E. Thummel
      Drug Metabolism and Disposition May 2021, 49 (5) 345-352; DOI: https://doi.org/10.1124/dmd.120.000301
  6. Hu, Yiting

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385

J

  1. Jia, Wei

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385

K

  1. Kalari, Krishna R.

    1. Open Access
      SLCO1B1: Application and Limitations of Deep Mutational Scanning for Genomic Missense Variant Function
      Lingxin Zhang, Vivekananda Sarangi, Ming-Fen Ho, Irene Moon, Krishna R. Kalari, Liewei Wang and Richard M. Weinshilboum
      Drug Metabolism and Disposition May 2021, 49 (5) 395-404; DOI: https://doi.org/10.1124/dmd.120.000264
  2. Kong, Dexuan

    1. Identification of Triterpene Acids in <em>Poria cocos</em> Extract as Bile Acid Uptake Transporter Inhibitors
      You have access
      Identification of Triterpene Acids in Poria cocos Extract as Bile Acid Uptake Transporter Inhibitors
      Hui Cai, Yujie Cheng, Qiunan Zhu, Dexuan Kong, Xijing Chen, Ikumi Tamai and Yang Lu
      Drug Metabolism and Disposition May 2021, 49 (5) 353-360; DOI: https://doi.org/10.1124/dmd.120.000308
  3. Kulkarni, Swarupa

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273
  4. Kumar, Gondi

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220

L

  1. Lan, Ke

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385
  2. Langenickel, Thomas

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273
  3. Li, Xuejing

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385
  4. Liu, Changxiao

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385
  5. Liu, Huixiang

    1. You have access
      Metabolic Retroversion of Piperaquine (PQ) via Hepatic Cytochrome P450–Mediated N-Oxidation and Reduction: Not an Important Contributor to the Prolonged Elimination of PQ
      Yuewu Xie, Yunrui Zhang, Huixiang Liu and Jie Xing
      Drug Metabolism and Disposition May 2021, 49 (5) 379-388; DOI: https://doi.org/10.1124/dmd.120.000306
  6. Lu, Yang

    1. Identification of Triterpene Acids in <em>Poria cocos</em> Extract as Bile Acid Uptake Transporter Inhibitors
      You have access
      Identification of Triterpene Acids in Poria cocos Extract as Bile Acid Uptake Transporter Inhibitors
      Hui Cai, Yujie Cheng, Qiunan Zhu, Dexuan Kong, Xijing Chen, Ikumi Tamai and Yang Lu
      Drug Metabolism and Disposition May 2021, 49 (5) 353-360; DOI: https://doi.org/10.1124/dmd.120.000308

M

  1. Moon, Irene

    1. Open Access
      SLCO1B1: Application and Limitations of Deep Mutational Scanning for Genomic Missense Variant Function
      Lingxin Zhang, Vivekananda Sarangi, Ming-Fen Ho, Irene Moon, Krishna R. Kalari, Liewei Wang and Richard M. Weinshilboum
      Drug Metabolism and Disposition May 2021, 49 (5) 395-404; DOI: https://doi.org/10.1124/dmd.120.000264

P

  1. Palmisano, Maria

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220
  2. Poller, Birk

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273

R

  1. Rahmanzadeh, Gholamreza

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273
  2. Rettie, Allan E.

    1. Open Access
      In Vivo Functional Effects of CYP2C9 M1L, a Novel and Common Variant in the Yup’ik Alaska Native Population
      Lindsay M. Henderson, Scarlett E. Hopkins, Bert B. Boyer, Timothy A. Thornton, Allan E. Rettie and Kenneth E. Thummel
      Drug Metabolism and Disposition May 2021, 49 (5) 345-352; DOI: https://doi.org/10.1124/dmd.120.000301

S

  1. Sarangi, Vivekananda

    1. Open Access
      SLCO1B1: Application and Limitations of Deep Mutational Scanning for Genomic Missense Variant Function
      Lingxin Zhang, Vivekananda Sarangi, Ming-Fen Ho, Irene Moon, Krishna R. Kalari, Liewei Wang and Richard M. Weinshilboum
      Drug Metabolism and Disposition May 2021, 49 (5) 395-404; DOI: https://doi.org/10.1124/dmd.120.000264
  2. Selkirk, Julie V.

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220
  3. Shah, Bharti

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273
  4. Surapaneni, Sekhar

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220

T

  1. Tamai, Ikumi

    1. Identification of Triterpene Acids in <em>Poria cocos</em> Extract as Bile Acid Uptake Transporter Inhibitors
      You have access
      Identification of Triterpene Acids in Poria cocos Extract as Bile Acid Uptake Transporter Inhibitors
      Hui Cai, Yujie Cheng, Qiunan Zhu, Dexuan Kong, Xijing Chen, Ikumi Tamai and Yang Lu
      Drug Metabolism and Disposition May 2021, 49 (5) 353-360; DOI: https://doi.org/10.1124/dmd.120.000308
  2. Tan, Xianwen

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385
  3. Thornton, Timothy A.

    1. Open Access
      In Vivo Functional Effects of CYP2C9 M1L, a Novel and Common Variant in the Yup’ik Alaska Native Population
      Lindsay M. Henderson, Scarlett E. Hopkins, Bert B. Boyer, Timothy A. Thornton, Allan E. Rettie and Kenneth E. Thummel
      Drug Metabolism and Disposition May 2021, 49 (5) 345-352; DOI: https://doi.org/10.1124/dmd.120.000301
  4. Thummel, Kenneth E.

    1. Open Access
      In Vivo Functional Effects of CYP2C9 M1L, a Novel and Common Variant in the Yup’ik Alaska Native Population
      Lindsay M. Henderson, Scarlett E. Hopkins, Bert B. Boyer, Timothy A. Thornton, Allan E. Rettie and Kenneth E. Thummel
      Drug Metabolism and Disposition May 2021, 49 (5) 345-352; DOI: https://doi.org/10.1124/dmd.120.000301
  5. Tran, Jonathan Q.

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220

V

  1. Vemula, Janardhana

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273

W

  1. Wang, Liewei

    1. Open Access
      SLCO1B1: Application and Limitations of Deep Mutational Scanning for Genomic Missense Variant Function
      Lingxin Zhang, Vivekananda Sarangi, Ming-Fen Ho, Irene Moon, Krishna R. Kalari, Liewei Wang and Richard M. Weinshilboum
      Drug Metabolism and Disposition May 2021, 49 (5) 395-404; DOI: https://doi.org/10.1124/dmd.120.000264
  2. Wang, Pei

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  3. Wang, Xiaofei

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  4. Wang, Xiaomin

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220
  5. Wang, Yiting

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  6. Weinshilboum, Richard M.

    1. Open Access
      SLCO1B1: Application and Limitations of Deep Mutational Scanning for Genomic Missense Variant Function
      Lingxin Zhang, Vivekananda Sarangi, Ming-Fen Ho, Irene Moon, Krishna R. Kalari, Liewei Wang and Richard M. Weinshilboum
      Drug Metabolism and Disposition May 2021, 49 (5) 395-404; DOI: https://doi.org/10.1124/dmd.120.000264
  7. Weiss, H. Markus

    1. Open Access
      Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
      H. Markus Weiss, Thomas Langenickel, Meredith Cain, Swarupa Kulkarni, Bharti Shah, Janardhana Vemula, Gholamreza Rahmanzadeh and Birk Poller
      Drug Metabolism and Disposition May 2021, 49 (5) 389-394; DOI: https://doi.org/10.1124/dmd.120.000273
  8. Wu, Qingliang

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385

X

  1. Xie, Yuewu

    1. You have access
      Metabolic Retroversion of Piperaquine (PQ) via Hepatic Cytochrome P450–Mediated N-Oxidation and Reduction: Not an Important Contributor to the Prolonged Elimination of PQ
      Yuewu Xie, Yunrui Zhang, Huixiang Liu and Jie Xing
      Drug Metabolism and Disposition May 2021, 49 (5) 379-388; DOI: https://doi.org/10.1124/dmd.120.000306
  2. Xing, Jie

    1. You have access
      Metabolic Retroversion of Piperaquine (PQ) via Hepatic Cytochrome P450–Mediated N-Oxidation and Reduction: Not an Important Contributor to the Prolonged Elimination of PQ
      Yuewu Xie, Yunrui Zhang, Huixiang Liu and Jie Xing
      Drug Metabolism and Disposition May 2021, 49 (5) 379-388; DOI: https://doi.org/10.1124/dmd.120.000306

Y

  1. Yan, Liang

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  2. Yan, Yingzhuo Grace

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220
  3. Yang, Kun

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  4. Yang, Lian

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385
  5. Yerramilli, Usha

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220

Z

  1. Zeng, Wushuang

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385
  2. Zhang, Lingxin

    1. Open Access
      SLCO1B1: Application and Limitations of Deep Mutational Scanning for Genomic Missense Variant Function
      Lingxin Zhang, Vivekananda Sarangi, Ming-Fen Ho, Irene Moon, Krishna R. Kalari, Liewei Wang and Richard M. Weinshilboum
      Drug Metabolism and Disposition May 2021, 49 (5) 395-404; DOI: https://doi.org/10.1124/dmd.120.000264
  3. Zhang, Lirong

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  4. Zhang, Peijin

    1. Open Access
      Absorption, Metabolism, and Excretion, In Vitro Pharmacology, and Clinical Pharmacokinetics of Ozanimod, a Novel Sphingosine 1-Phosphate Receptor Modulator
      Sekhar Surapaneni, Usha Yerramilli, April Bai, Deepak Dalvie, Jennifer Brooks, Xiaomin Wang, Julie V. Selkirk, Yingzhuo Grace Yan, Peijin Zhang, Richard Hargreaves, Gondi Kumar, Maria Palmisano and Jonathan Q. Tran
      Drug Metabolism and Disposition May 2021, 49 (5) 405-419; DOI: https://doi.org/10.1124/dmd.120.000220
  5. Zhang, Yunrui

    1. You have access
      Metabolic Retroversion of Piperaquine (PQ) via Hepatic Cytochrome P450–Mediated N-Oxidation and Reduction: Not an Important Contributor to the Prolonged Elimination of PQ
      Yuewu Xie, Yunrui Zhang, Huixiang Liu and Jie Xing
      Drug Metabolism and Disposition May 2021, 49 (5) 379-388; DOI: https://doi.org/10.1124/dmd.120.000306
  6. Zhong, Xiao-bo

    1. You have access
      The Long Noncoding RNA Hepatocyte Nuclear Factor 4α Antisense RNA 1 Negatively Regulates Cytochrome P450 Enzymes in Huh7 Cells via Histone Modifications
      Pei Wang, Shitong Chen, Yiting Wang, Xiaofei Wang, Liang Yan, Kun Yang, Xiao-bo Zhong, Shengna Han and Lirong Zhang
      Drug Metabolism and Disposition May 2021, 49 (5) 361-368; DOI: https://doi.org/10.1124/dmd.120.000316
  7. Zhu, Pingping

    1. Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      You have access
      Tertiary Oxidation of Deoxycholate Is Predictive of CYP3A Activity in Dogs
      Wushuang Zeng, Lanlan Gui, Xianwen Tan, Pingping Zhu, Yiting Hu, Qingliang Wu, Xuejing Li, Lian Yang, Wei Jia, Changxiao Liu and Ke Lan
      Drug Metabolism and Disposition May 2021, 49 (5) 369-378; DOI: https://doi.org/10.1124/dmd.121.000385
  8. Zhu, Qiunan

    1. Identification of Triterpene Acids in <em>Poria cocos</em> Extract as Bile Acid Uptake Transporter Inhibitors
      You have access
      Identification of Triterpene Acids in Poria cocos Extract as Bile Acid Uptake Transporter Inhibitors
      Hui Cai, Yujie Cheng, Qiunan Zhu, Dexuan Kong, Xijing Chen, Ikumi Tamai and Yang Lu
      Drug Metabolism and Disposition May 2021, 49 (5) 353-360; DOI: https://doi.org/10.1124/dmd.120.000308
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Drug Metabolism and Disposition: 49 (5)
Drug Metabolism and Disposition
Vol. 49, Issue 5
1 May 2021
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  • Cannabinoid Metabolites as CYP450 Inhibitors
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