Index by author
March 01, 2022; Volume 50,Issue 3
A
Ahire, Deepak
- You have accessInterindividual Variability and Differential Tissue Abundance of Mitochondrial Amidoxime Reducing Component Enzymes in HumansDeepak Ahire, Abdul Basit, Lisa J. Christopher, Ramaswamy Iyer, J. Steven Leeder and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 191-196; DOI: https://doi.org/10.1124/dmd.121.000805
Asano, Daigo
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
B
Basit, Abdul
- You have accessInterindividual Variability and Differential Tissue Abundance of Mitochondrial Amidoxime Reducing Component Enzymes in HumansDeepak Ahire, Abdul Basit, Lisa J. Christopher, Ramaswamy Iyer, J. Steven Leeder and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 191-196; DOI: https://doi.org/10.1124/dmd.121.000805
- You have accessComparison of Tissue Abundance of Non-Cytochrome P450 Drug-Metabolizing Enzymes by Quantitative Proteomics between Humans and Laboratory Animal SpeciesAbdul Basit, Peter W. Fan, S. Cyrus Khojasteh, Bernard P. Murray, Bill J. Smith, Scott Heyward and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 197-203; DOI: https://doi.org/10.1124/dmd.121.000774
C
Chiba, Koji
- Open AccessTransplacental Pharmacokinetic Model of Digoxin Based on Ex Vivo Human Placental Perfusion StudyKen Kurosawa, Saki Noguchi, Tomohiro Nishimura, Masatoshi Tomi and Koji ChibaDrug Metabolism and Disposition March 2022, 50 (3) 287-298; DOI: https://doi.org/10.1124/dmd.121.000648
Christopher, Lisa J.
- You have accessInterindividual Variability and Differential Tissue Abundance of Mitochondrial Amidoxime Reducing Component Enzymes in HumansDeepak Ahire, Abdul Basit, Lisa J. Christopher, Ramaswamy Iyer, J. Steven Leeder and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 191-196; DOI: https://doi.org/10.1124/dmd.121.000805
Cleary, Yumi
- You have accessAccelerating Clinical Development of Idasanutlin through a Physiologically Based Pharmacokinetic Modeling Risk Assessment for CYP450 Isoenzyme-Related Drug–Drug InteractionsKenichi Umehara, Yumi Cleary, Stephen Fowler, Neil Parrott and Dietrich TuerckDrug Metabolism and Disposition March 2022, 50 (3) 214-223; DOI: https://doi.org/10.1124/dmd.121.000720
D
Dalvie, Deepak
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
Dantonio, Alyssa L.
- You have accessIntersystem Extrapolation Factors Are Substrate-Dependent for CYP3A4: Impact on Cytochrome P450 Reaction PhenotypingAlyssa L. Dantonio, Angela C. Doran and R. Scott ObachDrug Metabolism and Disposition March 2022, 50 (3) 249-257; DOI: https://doi.org/10.1124/dmd.121.000758
Dhavaliker, Chinmayi
- You have accessExploring Drug Metabolism by the Gut Microbiota: Modes of Metabolism and Experimental ApproachesPooja Dhurjad, Chinmayi Dhavaliker, Kajal Gupta and Rajesh SontiDrug Metabolism and Disposition March 2022, 50 (3) 224-234; DOI: https://doi.org/10.1124/dmd.121.000669
Dhurjad, Pooja
- You have accessExploring Drug Metabolism by the Gut Microbiota: Modes of Metabolism and Experimental ApproachesPooja Dhurjad, Chinmayi Dhavaliker, Kajal Gupta and Rajesh SontiDrug Metabolism and Disposition March 2022, 50 (3) 224-234; DOI: https://doi.org/10.1124/dmd.121.000669
Doran, Angela C.
- You have accessIntersystem Extrapolation Factors Are Substrate-Dependent for CYP3A4: Impact on Cytochrome P450 Reaction PhenotypingAlyssa L. Dantonio, Angela C. Doran and R. Scott ObachDrug Metabolism and Disposition March 2022, 50 (3) 249-257; DOI: https://doi.org/10.1124/dmd.121.000758
E
Elmquist, William F.
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
F
Fan, Peter W.
- You have accessComparison of Tissue Abundance of Non-Cytochrome P450 Drug-Metabolizing Enzymes by Quantitative Proteomics between Humans and Laboratory Animal SpeciesAbdul Basit, Peter W. Fan, S. Cyrus Khojasteh, Bernard P. Murray, Bill J. Smith, Scott Heyward and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 197-203; DOI: https://doi.org/10.1124/dmd.121.000774
Fowler, Stephen
- You have accessAccelerating Clinical Development of Idasanutlin through a Physiologically Based Pharmacokinetic Modeling Risk Assessment for CYP450 Isoenzyme-Related Drug–Drug InteractionsKenichi Umehara, Yumi Cleary, Stephen Fowler, Neil Parrott and Dietrich TuerckDrug Metabolism and Disposition March 2022, 50 (3) 214-223; DOI: https://doi.org/10.1124/dmd.121.000720
G
Guimaraes, Guilherme
- You have accessAntisense Oligonucleotide In Vitro Protein Binding Determination in Plasma, Brain, and Cerebral Spinal Fluid Using Hybridization LC-MS/MSGuilherme Guimaraes, Long Yuan and Pei LiDrug Metabolism and Disposition March 2022, 50 (3) 268-276; DOI: https://doi.org/10.1124/dmd.121.000751
Gupta, Kajal
- You have accessExploring Drug Metabolism by the Gut Microbiota: Modes of Metabolism and Experimental ApproachesPooja Dhurjad, Chinmayi Dhavaliker, Kajal Gupta and Rajesh SontiDrug Metabolism and Disposition March 2022, 50 (3) 224-234; DOI: https://doi.org/10.1124/dmd.121.000669
Gupta, Shiv K.
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
H
Hamaue, Syoya
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Hashimoto, Shinji
- You have accessUsefulness of Human Jejunal Spheroid–Derived Differentiated Intestinal Epithelial Cells for the Prediction of Intestinal Drug Absorption in HumansKazuyoshi Michiba, Kazuya Maeda, Osamu Shimomura, Yoshihiro Miyazaki, Shinji Hashimoto, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition March 2022, 50 (3) 204-213; DOI: https://doi.org/10.1124/dmd.121.000796
Heck, Carley J.S.
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
Heyward, Scott
- You have accessComparison of Tissue Abundance of Non-Cytochrome P450 Drug-Metabolizing Enzymes by Quantitative Proteomics between Humans and Laboratory Animal SpeciesAbdul Basit, Peter W. Fan, S. Cyrus Khojasteh, Bernard P. Murray, Bill J. Smith, Scott Heyward and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 197-203; DOI: https://doi.org/10.1124/dmd.121.000774
I
Ikeguchi, Marie
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Inoue, Shin-ichi
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Iyer, Ramaswamy
- You have accessInterindividual Variability and Differential Tissue Abundance of Mitochondrial Amidoxime Reducing Component Enzymes in HumansDeepak Ahire, Abdul Basit, Lisa J. Christopher, Ramaswamy Iyer, J. Steven Leeder and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 191-196; DOI: https://doi.org/10.1124/dmd.121.000805
K
Kalgutkar, Amit S.
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
Kazui, Miho
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Khojasteh, S. Cyrus
- You have accessComparison of Tissue Abundance of Non-Cytochrome P450 Drug-Metabolizing Enzymes by Quantitative Proteomics between Humans and Laboratory Animal SpeciesAbdul Basit, Peter W. Fan, S. Cyrus Khojasteh, Bernard P. Murray, Bill J. Smith, Scott Heyward and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 197-203; DOI: https://doi.org/10.1124/dmd.121.000774
Kim, Minjee
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Kimura, Takako
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Kramlinger, Valerie M.
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
Kurosawa, Ken
- Open AccessTransplacental Pharmacokinetic Model of Digoxin Based on Ex Vivo Human Placental Perfusion StudyKen Kurosawa, Saki Noguchi, Tomohiro Nishimura, Masatoshi Tomi and Koji ChibaDrug Metabolism and Disposition March 2022, 50 (3) 287-298; DOI: https://doi.org/10.1124/dmd.121.000648
Kusuhara, Hiroyuki
- You have accessUsefulness of Human Jejunal Spheroid–Derived Differentiated Intestinal Epithelial Cells for the Prediction of Intestinal Drug Absorption in HumansKazuyoshi Michiba, Kazuya Maeda, Osamu Shimomura, Yoshihiro Miyazaki, Shinji Hashimoto, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition March 2022, 50 (3) 204-213; DOI: https://doi.org/10.1124/dmd.121.000796
L
Laramy, Janice
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Leeder, J. Steven
- You have accessInterindividual Variability and Differential Tissue Abundance of Mitochondrial Amidoxime Reducing Component Enzymes in HumansDeepak Ahire, Abdul Basit, Lisa J. Christopher, Ramaswamy Iyer, J. Steven Leeder and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 191-196; DOI: https://doi.org/10.1124/dmd.121.000805
Li, Jiapeng
- You have accessContributions of Cathepsin A and Carboxylesterase 1 to the Hydrolysis of Tenofovir Alafenamide in the Human Liver, and the Effect of CES1 Genetic Variation on Tenofovir Alafenamide HydrolysisJiapeng Li, Jian Shi, Jingcheng Xiao, Lana Tran, Xinwen Wang and Hao-Jie ZhuDrug Metabolism and Disposition March 2022, 50 (3) 243-248; DOI: https://doi.org/10.1124/dmd.120.000323
Li, Pei
- You have accessAntisense Oligonucleotide In Vitro Protein Binding Determination in Plasma, Brain, and Cerebral Spinal Fluid Using Hybridization LC-MS/MSGuilherme Guimaraes, Long Yuan and Pei LiDrug Metabolism and Disposition March 2022, 50 (3) 268-276; DOI: https://doi.org/10.1124/dmd.121.000751
M
Maeda, Kazuya
- You have accessUsefulness of Human Jejunal Spheroid–Derived Differentiated Intestinal Epithelial Cells for the Prediction of Intestinal Drug Absorption in HumansKazuyoshi Michiba, Kazuya Maeda, Osamu Shimomura, Yoshihiro Miyazaki, Shinji Hashimoto, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition March 2022, 50 (3) 204-213; DOI: https://doi.org/10.1124/dmd.121.000796
Michiba, Kazuyoshi
- You have accessUsefulness of Human Jejunal Spheroid–Derived Differentiated Intestinal Epithelial Cells for the Prediction of Intestinal Drug Absorption in HumansKazuyoshi Michiba, Kazuya Maeda, Osamu Shimomura, Yoshihiro Miyazaki, Shinji Hashimoto, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition March 2022, 50 (3) 204-213; DOI: https://doi.org/10.1124/dmd.121.000796
Miyazaki, Yoshihiro
- You have accessUsefulness of Human Jejunal Spheroid–Derived Differentiated Intestinal Epithelial Cells for the Prediction of Intestinal Drug Absorption in HumansKazuyoshi Michiba, Kazuya Maeda, Osamu Shimomura, Yoshihiro Miyazaki, Shinji Hashimoto, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition March 2022, 50 (3) 204-213; DOI: https://doi.org/10.1124/dmd.121.000796
Mladek, Ann C.
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Mohammad, Afroz S.
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Murray, Bernard P.
- You have accessComparison of Tissue Abundance of Non-Cytochrome P450 Drug-Metabolizing Enzymes by Quantitative Proteomics between Humans and Laboratory Animal SpeciesAbdul Basit, Peter W. Fan, S. Cyrus Khojasteh, Bernard P. Murray, Bill J. Smith, Scott Heyward and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 197-203; DOI: https://doi.org/10.1124/dmd.121.000774
N
Nishimura, Tomohiro
- Open AccessTransplacental Pharmacokinetic Model of Digoxin Based on Ex Vivo Human Placental Perfusion StudyKen Kurosawa, Saki Noguchi, Tomohiro Nishimura, Masatoshi Tomi and Koji ChibaDrug Metabolism and Disposition March 2022, 50 (3) 287-298; DOI: https://doi.org/10.1124/dmd.121.000648
Nishiya, Yumi
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Noguchi, Saki
- Open AccessTransplacental Pharmacokinetic Model of Digoxin Based on Ex Vivo Human Placental Perfusion StudyKen Kurosawa, Saki Noguchi, Tomohiro Nishimura, Masatoshi Tomi and Koji ChibaDrug Metabolism and Disposition March 2022, 50 (3) 287-298; DOI: https://doi.org/10.1124/dmd.121.000648
O
O’Neill, James
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
Obach, R. Scott
- You have accessIntersystem Extrapolation Factors Are Substrate-Dependent for CYP3A4: Impact on Cytochrome P450 Reaction PhenotypingAlyssa L. Dantonio, Angela C. Doran and R. Scott ObachDrug Metabolism and Disposition March 2022, 50 (3) 249-257; DOI: https://doi.org/10.1124/dmd.121.000758
Oda, Tatsuya
- You have accessUsefulness of Human Jejunal Spheroid–Derived Differentiated Intestinal Epithelial Cells for the Prediction of Intestinal Drug Absorption in HumansKazuyoshi Michiba, Kazuya Maeda, Osamu Shimomura, Yoshihiro Miyazaki, Shinji Hashimoto, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition March 2022, 50 (3) 204-213; DOI: https://doi.org/10.1124/dmd.121.000796
P
Parrott, Neil
- You have accessAccelerating Clinical Development of Idasanutlin through a Physiologically Based Pharmacokinetic Modeling Risk Assessment for CYP450 Isoenzyme-Related Drug–Drug InteractionsKenichi Umehara, Yumi Cleary, Stephen Fowler, Neil Parrott and Dietrich TuerckDrug Metabolism and Disposition March 2022, 50 (3) 214-223; DOI: https://doi.org/10.1124/dmd.121.000720
Prasad, Bhagwat
- You have accessInterindividual Variability and Differential Tissue Abundance of Mitochondrial Amidoxime Reducing Component Enzymes in HumansDeepak Ahire, Abdul Basit, Lisa J. Christopher, Ramaswamy Iyer, J. Steven Leeder and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 191-196; DOI: https://doi.org/10.1124/dmd.121.000805
- You have accessComparison of Tissue Abundance of Non-Cytochrome P450 Drug-Metabolizing Enzymes by Quantitative Proteomics between Humans and Laboratory Animal SpeciesAbdul Basit, Peter W. Fan, S. Cyrus Khojasteh, Bernard P. Murray, Bill J. Smith, Scott Heyward and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 197-203; DOI: https://doi.org/10.1124/dmd.121.000774
R
Rodrigues, A. David
- You have accessCynomolgus Monkey as an Emerging Animal Model to Study Drug Transporters: In Vitro, In Vivo, In Vitro-to-In Vivo TranslationHong Shen, Zheng Yang and A. David RodriguesDrug Metabolism and Disposition March 2022, 50 (3) 299-319; DOI: https://doi.org/10.1124/dmd.121.000695
S
Sarkaria, Jann N.
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Shen, Hong
- You have accessCynomolgus Monkey as an Emerging Animal Model to Study Drug Transporters: In Vitro, In Vivo, In Vitro-to-In Vivo TranslationHong Shen, Zheng Yang and A. David RodriguesDrug Metabolism and Disposition March 2022, 50 (3) 299-319; DOI: https://doi.org/10.1124/dmd.121.000695
Shi, Jian
- You have accessContributions of Cathepsin A and Carboxylesterase 1 to the Hydrolysis of Tenofovir Alafenamide in the Human Liver, and the Effect of CES1 Genetic Variation on Tenofovir Alafenamide HydrolysisJiapeng Li, Jian Shi, Jingcheng Xiao, Lana Tran, Xinwen Wang and Hao-Jie ZhuDrug Metabolism and Disposition March 2022, 50 (3) 243-248; DOI: https://doi.org/10.1124/dmd.120.000323
Shibayama, Takahiro
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Shimomura, Osamu
- You have accessUsefulness of Human Jejunal Spheroid–Derived Differentiated Intestinal Epithelial Cells for the Prediction of Intestinal Drug Absorption in HumansKazuyoshi Michiba, Kazuya Maeda, Osamu Shimomura, Yoshihiro Miyazaki, Shinji Hashimoto, Tatsuya Oda and Hiroyuki KusuharaDrug Metabolism and Disposition March 2022, 50 (3) 204-213; DOI: https://doi.org/10.1124/dmd.121.000796
Shinozuka, Tsuyoshi
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Shiozawa, Hideyuki
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Smith, Bill J.
- You have accessComparison of Tissue Abundance of Non-Cytochrome P450 Drug-Metabolizing Enzymes by Quantitative Proteomics between Humans and Laboratory Animal SpeciesAbdul Basit, Peter W. Fan, S. Cyrus Khojasteh, Bernard P. Murray, Bill J. Smith, Scott Heyward and Bhagwat PrasadDrug Metabolism and Disposition March 2022, 50 (3) 197-203; DOI: https://doi.org/10.1124/dmd.121.000774
Sonti, Rajesh
- You have accessExploring Drug Metabolism by the Gut Microbiota: Modes of Metabolism and Experimental ApproachesPooja Dhurjad, Chinmayi Dhavaliker, Kajal Gupta and Rajesh SontiDrug Metabolism and Disposition March 2022, 50 (3) 224-234; DOI: https://doi.org/10.1124/dmd.121.000669
Su, Dian
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
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Talele, Surabhi
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Teitelbaum, Aaron M.
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
Tomi, Masatoshi
- Open AccessTransplacental Pharmacokinetic Model of Digoxin Based on Ex Vivo Human Placental Perfusion StudyKen Kurosawa, Saki Noguchi, Tomohiro Nishimura, Masatoshi Tomi and Koji ChibaDrug Metabolism and Disposition March 2022, 50 (3) 287-298; DOI: https://doi.org/10.1124/dmd.121.000648
Totah, Rheem A.
- You have accessFuture of Biotransformation Science in the Pharmaceutical IndustryValerie M. Kramlinger, Deepak Dalvie, Carley J.S. Heck, Amit S. Kalgutkar, James O’Neill, Dian Su, Aaron M. Teitelbaum and Rheem A. TotahDrug Metabolism and Disposition March 2022, 50 (3) 258-267; DOI: https://doi.org/10.1124/dmd.121.000658
Tran, Lana
- You have accessContributions of Cathepsin A and Carboxylesterase 1 to the Hydrolysis of Tenofovir Alafenamide in the Human Liver, and the Effect of CES1 Genetic Variation on Tenofovir Alafenamide HydrolysisJiapeng Li, Jian Shi, Jingcheng Xiao, Lana Tran, Xinwen Wang and Hao-Jie ZhuDrug Metabolism and Disposition March 2022, 50 (3) 243-248; DOI: https://doi.org/10.1124/dmd.120.000323
Tuerck, Dietrich
- You have accessAccelerating Clinical Development of Idasanutlin through a Physiologically Based Pharmacokinetic Modeling Risk Assessment for CYP450 Isoenzyme-Related Drug–Drug InteractionsKenichi Umehara, Yumi Cleary, Stephen Fowler, Neil Parrott and Dietrich TuerckDrug Metabolism and Disposition March 2022, 50 (3) 214-223; DOI: https://doi.org/10.1124/dmd.121.000720
U
Umehara, Kenichi
- You have accessAccelerating Clinical Development of Idasanutlin through a Physiologically Based Pharmacokinetic Modeling Risk Assessment for CYP450 Isoenzyme-Related Drug–Drug InteractionsKenichi Umehara, Yumi Cleary, Stephen Fowler, Neil Parrott and Dietrich TuerckDrug Metabolism and Disposition March 2022, 50 (3) 214-223; DOI: https://doi.org/10.1124/dmd.121.000720
W
Wang, Xinwen
- You have accessContributions of Cathepsin A and Carboxylesterase 1 to the Hydrolysis of Tenofovir Alafenamide in the Human Liver, and the Effect of CES1 Genetic Variation on Tenofovir Alafenamide HydrolysisJiapeng Li, Jian Shi, Jingcheng Xiao, Lana Tran, Xinwen Wang and Hao-Jie ZhuDrug Metabolism and Disposition March 2022, 50 (3) 243-248; DOI: https://doi.org/10.1124/dmd.120.000323
Watanabe, Nobuaki
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Watanabe, Toshiyuki
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
X
Xiao, Jingcheng
- You have accessContributions of Cathepsin A and Carboxylesterase 1 to the Hydrolysis of Tenofovir Alafenamide in the Human Liver, and the Effect of CES1 Genetic Variation on Tenofovir Alafenamide HydrolysisJiapeng Li, Jian Shi, Jingcheng Xiao, Lana Tran, Xinwen Wang and Hao-Jie ZhuDrug Metabolism and Disposition March 2022, 50 (3) 243-248; DOI: https://doi.org/10.1124/dmd.120.000323
Y
Yahara, Chizuko
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Yamamura, Naotoshi
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Yang, Zheng
- You have accessCynomolgus Monkey as an Emerging Animal Model to Study Drug Transporters: In Vitro, In Vivo, In Vitro-to-In Vivo TranslationHong Shen, Zheng Yang and A. David RodriguesDrug Metabolism and Disposition March 2022, 50 (3) 299-319; DOI: https://doi.org/10.1124/dmd.121.000695
Yoshinari, Kouichi
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Yuan, Long
- You have accessAntisense Oligonucleotide In Vitro Protein Binding Determination in Plasma, Brain, and Cerebral Spinal Fluid Using Hybridization LC-MS/MSGuilherme Guimaraes, Long Yuan and Pei LiDrug Metabolism and Disposition March 2022, 50 (3) 268-276; DOI: https://doi.org/10.1124/dmd.121.000751
Z
Zahir, Hamim
- You have accessCYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective NaV1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase SubstrateDaigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe and Kouichi YoshinariDrug Metabolism and Disposition March 2022, 50 (3) 235-242; DOI: https://doi.org/10.1124/dmd.121.000665
Zhang, Shuangling
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Zhang, Wenjuan
- You have accessFactors Influencing Luciferase-Based Bioluminescent Imaging in Preclinical Models of Brain TumorMinjee Kim, Shiv K. Gupta, Wenjuan Zhang, Surabhi Talele, Afroz S. Mohammad, Janice Laramy, Ann C. Mladek, Shuangling Zhang, Jann N. Sarkaria and William F. ElmquistDrug Metabolism and Disposition March 2022, 50 (3) 277-286; DOI: https://doi.org/10.1124/dmd.121.000597
Zhu, Hao-Jie
- You have accessContributions of Cathepsin A and Carboxylesterase 1 to the Hydrolysis of Tenofovir Alafenamide in the Human Liver, and the Effect of CES1 Genetic Variation on Tenofovir Alafenamide HydrolysisJiapeng Li, Jian Shi, Jingcheng Xiao, Lana Tran, Xinwen Wang and Hao-Jie ZhuDrug Metabolism and Disposition March 2022, 50 (3) 243-248; DOI: https://doi.org/10.1124/dmd.120.000323
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