Index by author
December 01, 2023; Volume 51,Issue 12
A
Abbasi, Armina
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Arya, Vikram
- You have accessInnovations, Opportunities, and Challenges for Predicting Alteration in Drug-Metabolizing Enzyme and Transporter Activity in Specific PopulationsParesh P. Chothe, Vikram Arya, Bhagwat Prasad, Diane Ramsden and Kunal TaskarDrug Metabolism and Disposition December 2023, 51 (12) 1547-1550; DOI: https://doi.org/10.1124/dmd.123.001453
B
Barber, Jill
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Bolleddula, Jayaprakasam
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Botha, Jean
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
C
Cao, Xiaolong
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Cha, David
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
Chen, Diyao
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Chen, Huohui
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Chen, Likun
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Chen, Weidong
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Chen, Youhao
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Chen, Yunna
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Cheruzel, Lionel
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Chothe, Paresh P.
- You have accessInnovations, Opportunities, and Challenges for Predicting Alteration in Drug-Metabolizing Enzyme and Transporter Activity in Specific PopulationsParesh P. Chothe, Vikram Arya, Bhagwat Prasad, Diane Ramsden and Kunal TaskarDrug Metabolism and Disposition December 2023, 51 (12) 1547-1550; DOI: https://doi.org/10.1124/dmd.123.001453
D
Di, Chanjuan
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Ding, Ke
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
E
Ellis, Ewa
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Etheredge, Harriet
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
F
Fabian, June
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Fujioka, Hijiri
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Fukami, Tatsuki
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
G
Galetin, Aleksandra
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Gu, Lijia
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Guan, Jin
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Guan, Shaoxing
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Guo, Huimin
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Guo, Yating
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
H
Hirasawa, Noriyasu
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Hiratsuka, Masahiro
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Hirosawa, Keiya
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Hishinuma, Eiji
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Houston, J. Brian
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Hsu, Mei-Hui
- You have accessDifferential Effects of Clotrimazole on X-Ray Crystal Structures of Human Cytochromes P450 3A5 and 3A4Mei-Hui Hsu and Eric F. JohnsonDrug Metabolism and Disposition December 2023, 51 (12) 1642-1650; DOI: https://doi.org/10.1124/dmd.123.001464
Hu, Wenjun
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Huang, Fang
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Huang, Min
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Hurrell, Tracey
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
I
Ishiguro, Naoki
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Izat, Nihan
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
J
Johnson, Eric F.
- You have accessDifferential Effects of Clotrimazole on X-Ray Crystal Structures of Human Cytochromes P450 3A5 and 3A4Mei-Hui Hsu and Eric F. JohnsonDrug Metabolism and Disposition December 2023, 51 (12) 1642-1650; DOI: https://doi.org/10.1124/dmd.123.001464
Jones, Robert S.
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
K
Kanji, Comfort Ropafadzo
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Kapungu, Nyasha Nicole
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Kearney, Brian P.
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
Kinoshita, Kengo
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Kishimoto, Wataru
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Kumondai, Masaki
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
L
Leeder, J. Steven
- You have accessOntogeny of Scaling Factors for Pediatric Physiologically Based Pharmacokinetic Modeling and Simulation: Cytosolic Protein Per Gram of LiverStephani L. Stancil, Robin E. Pearce, Vincent S. Staggs and J. Steven LeederDrug Metabolism and Disposition December 2023, 51 (12) 1578-1582; DOI: https://doi.org/10.1124/dmd.123.001417
Lei, Yuanyuan
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Li, Ning
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Li, Zhiyu
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Liang, Yan
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Lin, Daren
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Lin, Haishu
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Lin, Yaobin
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Lin, Zhichao
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Liu, Huafang
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Liu, Junling
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Long, Hao
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Loveland, Jerome
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
M
Ma, Shudong
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Maekawa, Masamitsu
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Maher, Heather
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Mano, Nariyasu
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Masimirembwa, Collen
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Meng, Haitao
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Meng, Xiangyun
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Mizuguchi, Hiroyuki
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Morinaga, Gaku
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Moss, Darren
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Mthembu, Busisiwe
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
N
Naidoo, Jerolen
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Nakajima, Miki
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Nakase, Hiroshi
- You have accessQuantitative Analysis of mRNA and Protein Expression Levels of Aldo-Keto Reductase and Short-Chain Dehydrogenase/Reductase Isoforms in the Human IntestineKeiya Hirosawa, Hijiri Fujioka, Gaku Morinaga, Tatsuki Fukami, Naoki Ishiguro, Wataru Kishimoto, Hiroshi Nakase, Hiroyuki Mizuguchi and Miki NakajimaDrug Metabolism and Disposition December 2023, 51 (12) 1569-1577; DOI: https://doi.org/10.1124/dmd.123.001402
Nakayoshi, Tomoki
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
O
Oda, Akifumi
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Ortega-Muro, Fatima
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
P
Pan, Jianquan
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Parmentier, Yannick
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Pearce, Robin E.
- You have accessOntogeny of Scaling Factors for Pediatric Physiologically Based Pharmacokinetic Modeling and Simulation: Cytosolic Protein Per Gram of LiverStephani L. Stancil, Robin E. Pearce, Vincent S. Staggs and J. Steven LeederDrug Metabolism and Disposition December 2023, 51 (12) 1578-1582; DOI: https://doi.org/10.1124/dmd.123.001417
Peterkin, Vincent C.
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Plummer, Andrew
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
Prasad, Bhagwat
- You have accessInnovations, Opportunities, and Challenges for Predicting Alteration in Drug-Metabolizing Enzyme and Transporter Activity in Specific PopulationsParesh P. Chothe, Vikram Arya, Bhagwat Prasad, Diane Ramsden and Kunal TaskarDrug Metabolism and Disposition December 2023, 51 (12) 1547-1550; DOI: https://doi.org/10.1124/dmd.123.001453
Q
Qiu, Zhixia
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
R
Rambarran, Sharan
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Ramsay, Michele
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Ramsden, Diane
- You have accessInnovations, Opportunities, and Challenges for Predicting Alteration in Drug-Metabolizing Enzyme and Transporter Activity in Specific PopulationsParesh P. Chothe, Vikram Arya, Bhagwat Prasad, Diane Ramsden and Kunal TaskarDrug Metabolism and Disposition December 2023, 51 (12) 1547-1550; DOI: https://doi.org/10.1124/dmd.123.001453
S
Saito, Sakae
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Sato, Yu
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Scholefield, Janine
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Scotcher, Daniel
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Shang, Jianbiao
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Smyth, Natalie
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Staggs, Vincent S.
- You have accessOntogeny of Scaling Factors for Pediatric Physiologically Based Pharmacokinetic Modeling and Simulation: Cytosolic Protein Per Gram of LiverStephani L. Stancil, Robin E. Pearce, Vincent S. Staggs and J. Steven LeederDrug Metabolism and Disposition December 2023, 51 (12) 1578-1582; DOI: https://doi.org/10.1124/dmd.123.001417
Stancil, Stephani L.
- You have accessOntogeny of Scaling Factors for Pediatric Physiologically Based Pharmacokinetic Modeling and Simulation: Cytosolic Protein Per Gram of LiverStephani L. Stancil, Robin E. Pearce, Vincent S. Staggs and J. Steven LeederDrug Metabolism and Disposition December 2023, 51 (12) 1578-1582; DOI: https://doi.org/10.1124/dmd.123.001417
Strobele, Bernd
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Sun, Hong
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Sun, Qiushuang
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
T
Tadaka, Shu
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Taskar, Kunal
- You have accessInnovations, Opportunities, and Challenges for Predicting Alteration in Drug-Metabolizing Enzyme and Transporter Activity in Specific PopulationsParesh P. Chothe, Vikram Arya, Bhagwat Prasad, Diane Ramsden and Kunal TaskarDrug Metabolism and Disposition December 2023, 51 (12) 1547-1550; DOI: https://doi.org/10.1124/dmd.123.001453
Thelingwani, Roslyn Stella
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
Tian, Dan-Dan
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
Turnquist, David
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
U
Ueda, Akiko
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
V
van der Schyff, Francisca
- You have accessThe African Liver Tissue Biorepository Consortium: Capacitating Population-Appropriate Drug Metabolism, Pharmacokinetics, and Pharmacogenetics Research in Drug Discovery and DevelopmentCollen Masimirembwa, Michele Ramsay, Jean Botha, Ewa Ellis, Harriet Etheredge, Tracey Hurrell, Comfort Ropafadzo Kanji, Nyasha Nicole Kapungu, Heather Maher, Busisiwe Mthembu, Jerolen Naidoo, Janine Scholefield, Sharan Rambarran, Francisca van der Schyff, Natalie Smyth, Bernd Strobele, Roslyn Stella Thelingwani, Jerome Loveland and June FabianDrug Metabolism and Disposition December 2023, 51 (12) 1551-1560; DOI: https://doi.org/10.1124/dmd.123.001400
van Ingen, Eric
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
Venkatakrishnan, Karthik
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
W
Wang, Fengling
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Wang, Guangji
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Wang, Lei
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Wang, Shijiao
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Wang, Xueding
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Wilfret, David
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
Wong, Shekman L.
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
Wu, Linlin
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
X
Xie, Lin
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Xu, Feng
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Xu, Pengfei
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Xu, Yexin
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Y
Yamazaki, Shuki
- You have accessFunctional Characterization of 29 Cytochrome P450 4F2 Variants Identified in a Population of 8380 Japanese Subjects and Assessment of Arachidonic Acid ω-HydroxylationYu Sato, Eiji Hishinuma, Shuki Yamazaki, Akiko Ueda, Masaki Kumondai, Sakae Saito, Shu Tadaka, Kengo Kinoshita, Tomoki Nakayoshi, Akifumi Oda, Masamitsu Maekawa, Nariyasu Mano, Noriyasu Hirasawa and Masahiro HiratsukaDrug Metabolism and Disposition December 2023, 51 (12) 1561-1568; DOI: https://doi.org/10.1124/dmd.123.001389
Yang, Huizhu
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Yang, Ziping
- You have accessCharacterization of Pharmacokinetics, Biotransformation and Elimination of Pomotrelvir Orally Administered in Healthy Male Adults Using Two [14C]-Labeled Microtracers with Separate Labeling PositionsZiping Yang, Shekman L. Wong, David Cha, David Wilfret, David Turnquist, Andrew Plummer, Eric van Ingen and Brian P. KearneyDrug Metabolism and Disposition December 2023, 51 (12) 1607-1614; DOI: https://doi.org/10.1124/dmd.123.001439
Ye, Xi
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Z
Zhang, Mengdi
- You have accessBempedoic Acid Unveils Therapeutic Potential in Non-Alcoholic Fatty Liver Disease: Suppression of the Hepatic PXR-SLC13A5/ACLY Signaling AxisQiushuang Sun, Yating Guo, Wenjun Hu, Mengdi Zhang, Shijiao Wang, Yuanyuan Lei, Haitao Meng, Ning Li, Pengfei Xu, Zhiyu Li, Haishu Lin, Fang Huang and Zhixia QiuDrug Metabolism and Disposition December 2023, 51 (12) 1628-1641; DOI: https://doi.org/10.1124/dmd.123.001449
Zhang, Tingting
- You have accessIdentification and Validation of Active Ingredient in Cerebrotein Hydrolysate-I Based on Pharmacokinetic and Pharmacodynamic StudiesHuimin Guo, Huizhu Yang, Chanjuan Di, Feng Xu, Hong Sun, Yexin Xu, Huafang Liu, Linlin Wu, Ke Ding, Tingting Zhang, Lin Xie, Guangji Wang and Yan LiangDrug Metabolism and Disposition December 2023, 51 (12) 1615-1627; DOI: https://doi.org/10.1124/dmd.123.001443
Zhang, Weijian
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Zhang, Xue
- You have accessActivation of CYP3A by Accelerated Blood Clearance Phenomenon Potentiates the Hepatocellular Carcinoma-Targeting Therapeutic Effects of PEGylated Anticancer Prodrug LiposomesXue Zhang, Jianquan Pan, Xi Ye, Yunna Chen, Lei Wang, Xiangyun Meng, Weidong Chen and Fengling WangDrug Metabolism and Disposition December 2023, 51 (12) 1651-1662; DOI: https://doi.org/10.1124/dmd.123.001496
Zhao, Jian
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Zhao, Zerui
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Zhou, Chengzhi
- You have accessThe Effects of Drug Exposure and Single Nucleotide Polymorphisms on Aaptinib-Induced Severe Toxicities in Solid TumorsYouhao Chen, Yaobin Lin, Shaoxing Guan, Zerui Zhao, Daren Lin, Jin Guan, Chengzhi Zhou, Junling Liu, Xiaolong Cao, Zhichao Lin, Diyao Chen, Jianbiao Shang, Weijian Zhang, Huohui Chen, Likun Chen, Shudong Ma, Lijia Gu, Jian Zhao, Min Huang, Xueding Wang and Hao LongDrug Metabolism and Disposition December 2023, 51 (12) 1583-1590; DOI: https://doi.org/10.1124/dmd.123.001428
Zientek, Michael A.
- Open AccessChallenges and Opportunities for In Vitro–In Vivo Extrapolation of Aldehyde Oxidase-Mediated Clearance: Toward a Roadmap for Quantitative TranslationNihan Izat, Jayaprakasam Bolleddula, Armina Abbasi, Lionel Cheruzel, Robert S. Jones, Darren Moss, Fatima Ortega-Muro, Yannick Parmentier, Vincent C. Peterkin, Dan-Dan Tian, Karthik Venkatakrishnan, Michael A. Zientek, Jill Barber, J. Brian Houston, Aleksandra Galetin and Daniel ScotcherDrug Metabolism and Disposition December 2023, 51 (12) 1591-1606; DOI: https://doi.org/10.1124/dmd.123.001436
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