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Drug Metabolism & Disposition

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  • Articles
    • Current Issue
    • Fast Forward
    • Latest Articles
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Index by author

June 01, 2023; Volume 51,Issue 6
  • A
  • B
  • C
  • D
  • E
  • F
  • G
  • H
  • I
  • J
  • K
  • L
  • M
  • N
  • O
  • P
  • Q
  • R
  • S
  • T
  • U
  • V
  • W
  • X
  • Y
  • Z

B

  1. Baillie, Thomas A.

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  2. Bansal, Sumit

    1. You have access
      A Physiologically-Based Pharmacokinetic Model for Cannabidiol in Healthy Adults, Hepatically-Impaired Adults, and Children
      Sumit Bansal, Mayur K. Ladumor, Mary F. Paine and Jashvant D. Unadkat
      Drug Metabolism and Disposition June 2023, 51 (6) 743-752; DOI: https://doi.org/10.1124/dmd.122.001128
  3. Barnes, J. Paige

    1. You have access
      Mechanistic Investigation of the Time-Dependent Aldehyde Oxidase Inhibitor Hydralazine
      J. Paige Barnes, Shaoyun M. Yang, Taylor S. Thompson, Caithlyne M. Guevarra, Shaniya S. Pleasant, Tri Q. Do and Rachel D. Crouch
      Drug Metabolism and Disposition June 2023, 51 (6) 782-791; DOI: https://doi.org/10.1124/dmd.123.001257
  4. Busse, Gregory

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218

C

  1. Carter, Adam

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  2. Cerny, Matthew A.

    1. You have access
      Human Absorption, Distribution, Metabolism, and Excretion Studies: Origins, Innovations, and Importance
      Matthew A. Cerny, Douglas K. Spracklin and R. Scott Obach
      Drug Metabolism and Disposition June 2023, 51 (6) 647-656; DOI: https://doi.org/10.1124/dmd.122.001006
  3. Chen, Huili

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  4. Chen, Xiang

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  5. Chen, Xijing

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  6. Cronin, Joseph M.

    1. Open Access
      Recombinant Technologies Facilitate Drug Metabolism, Pharmacokinetics, and General Biomedical Research
      Joseph M. Cronin and Ai-Ming Yu
      Drug Metabolism and Disposition June 2023, 51 (6) 685-699; DOI: https://doi.org/10.1124/dmd.122.001008
  7. Crouch, Rachel D.

    1. You have access
      Mechanistic Investigation of the Time-Dependent Aldehyde Oxidase Inhibitor Hydralazine
      J. Paige Barnes, Shaoyun M. Yang, Taylor S. Thompson, Caithlyne M. Guevarra, Shaniya S. Pleasant, Tri Q. Do and Rachel D. Crouch
      Drug Metabolism and Disposition June 2023, 51 (6) 782-791; DOI: https://doi.org/10.1124/dmd.123.001257

D

  1. Ding, Xinxin

    1. You have access
      Special Section on Perspectives on Drug Metabolism and Disposition, Part I—Editorial
      Yurong Lai and Xinxin Ding
      Drug Metabolism and Disposition June 2023, 51 (6) 645-646; DOI: https://doi.org/10.1124/dmd.123.001352
  2. Do, Tri Q.

    1. You have access
      Mechanistic Investigation of the Time-Dependent Aldehyde Oxidase Inhibitor Hydralazine
      J. Paige Barnes, Shaoyun M. Yang, Taylor S. Thompson, Caithlyne M. Guevarra, Shaniya S. Pleasant, Tri Q. Do and Rachel D. Crouch
      Drug Metabolism and Disposition June 2023, 51 (6) 782-791; DOI: https://doi.org/10.1124/dmd.123.001257

E

  1. Ebner, Thomas

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  2. English, Stephen

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  3. Esmaeeli, Mariam

    1. Open Access
      Inactivation of Human Aldehyde Oxidase by Small Sulfhydryl-Containing Reducing Agents
      Mariam Esmaeeli, Manfred Nimtz, Lothar Jänsch, Lloyd W. Ruddock and Silke Leimkühler
      Drug Metabolism and Disposition June 2023, 51 (6) 764-770; DOI: https://doi.org/10.1124/dmd.122.001244

F

  1. Fitch, William L.

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  2. Fitzsimmons, Michael E.

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  3. Fukami, Tatsuki

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113

G

  1. Guevarra, Caithlyne M.

    1. You have access
      Mechanistic Investigation of the Time-Dependent Aldehyde Oxidase Inhibitor Hydralazine
      J. Paige Barnes, Shaoyun M. Yang, Taylor S. Thompson, Caithlyne M. Guevarra, Shaniya S. Pleasant, Tri Q. Do and Rachel D. Crouch
      Drug Metabolism and Disposition June 2023, 51 (6) 782-791; DOI: https://doi.org/10.1124/dmd.123.001257

H

  1. Han, Luyao

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  2. Hashiba, Shiori

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  3. Huang, Haoyan

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245

I

  1. Ishiguro, Naoki

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  2. Isoherranen, Nina

    1. Open Access
      Impact of Intracellular Lipid Binding Proteins on Endogenous and Xenobiotic Ligand Metabolism and Disposition
      King Clyde B. Yabut and Nina Isoherranen
      Drug Metabolism and Disposition June 2023, 51 (6) 700-717; DOI: https://doi.org/10.1124/dmd.122.001010

J

  1. Jänsch, Lothar

    1. Open Access
      Inactivation of Human Aldehyde Oxidase by Small Sulfhydryl-Containing Reducing Agents
      Mariam Esmaeeli, Manfred Nimtz, Lothar Jänsch, Lloyd W. Ruddock and Silke Leimkühler
      Drug Metabolism and Disposition June 2023, 51 (6) 764-770; DOI: https://doi.org/10.1124/dmd.122.001244
  2. Jin, Jing

    1. Epigenetic Mechanisms Contribute to Intraindividual Variations of Drug Metabolism Mediated by Cytochrome P450 Enzymes
      You have access
      Epigenetic Mechanisms Contribute to Intraindividual Variations of Drug Metabolism Mediated by Cytochrome P450 Enzymes
      Jing Jin and Xiao-bo Zhong
      Drug Metabolism and Disposition June 2023, 51 (6) 672-684; DOI: https://doi.org/10.1124/dmd.122.001007

K

  1. Kudo, Takashi

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113

L

  1. Ladumor, Mayur K.

    1. You have access
      A Physiologically-Based Pharmacokinetic Model for Cannabidiol in Healthy Adults, Hepatically-Impaired Adults, and Children
      Sumit Bansal, Mayur K. Ladumor, Mary F. Paine and Jashvant D. Unadkat
      Drug Metabolism and Disposition June 2023, 51 (6) 743-752; DOI: https://doi.org/10.1124/dmd.122.001128
  2. Lai, Yurong

    1. You have access
      Special Section on Perspectives on Drug Metabolism and Disposition, Part I—Editorial
      Yurong Lai and Xinxin Ding
      Drug Metabolism and Disposition June 2023, 51 (6) 645-646; DOI: https://doi.org/10.1124/dmd.123.001352
  3. Leimkühler, Silke

    1. Open Access
      Inactivation of Human Aldehyde Oxidase by Small Sulfhydryl-Containing Reducing Agents
      Mariam Esmaeeli, Manfred Nimtz, Lothar Jänsch, Lloyd W. Ruddock and Silke Leimkühler
      Drug Metabolism and Disposition June 2023, 51 (6) 764-770; DOI: https://doi.org/10.1124/dmd.122.001244
  4. Li, Li

    1. You have access
      Combined Oral Contraceptives As Victims of Drug Interactions
      Li Li, Xinning Yang, Doanh Tran, Shirley K. Seo and Yanhui Lu
      Drug Metabolism and Disposition June 2023, 51 (6) 718-732; DOI: https://doi.org/10.1124/dmd.122.000854
  5. Lu, Yanhui

    1. You have access
      Combined Oral Contraceptives As Victims of Drug Interactions
      Li Li, Xinning Yang, Doanh Tran, Shirley K. Seo and Yanhui Lu
      Drug Metabolism and Disposition June 2023, 51 (6) 718-732; DOI: https://doi.org/10.1124/dmd.122.000854
  6. Ludwig-Schwellinger, Eva

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113

M

  1. Matsui, Akiko

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  2. Morinaga, Gaku

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113

N

  1. Nakajima, Miki

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  2. Nakano, Masataka

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  3. Nakashima, Shimon

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  4. Nimtz, Manfred

    1. Open Access
      Inactivation of Human Aldehyde Oxidase by Small Sulfhydryl-Containing Reducing Agents
      Mariam Esmaeeli, Manfred Nimtz, Lothar Jänsch, Lloyd W. Ruddock and Silke Leimkühler
      Drug Metabolism and Disposition June 2023, 51 (6) 764-770; DOI: https://doi.org/10.1124/dmd.122.001244

O

  1. Obach, R. Scott

    1. You have access
      Human Absorption, Distribution, Metabolism, and Excretion Studies: Origins, Innovations, and Importance
      Matthew A. Cerny, Douglas K. Spracklin and R. Scott Obach
      Drug Metabolism and Disposition June 2023, 51 (6) 647-656; DOI: https://doi.org/10.1124/dmd.122.001006

P

  1. Paine, Mary F.

    1. You have access
      A Physiologically-Based Pharmacokinetic Model for Cannabidiol in Healthy Adults, Hepatically-Impaired Adults, and Children
      Sumit Bansal, Mayur K. Ladumor, Mary F. Paine and Jashvant D. Unadkat
      Drug Metabolism and Disposition June 2023, 51 (6) 743-752; DOI: https://doi.org/10.1124/dmd.122.001128
  2. Pan, He

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  3. Pleasant, Shaniya S.

    1. You have access
      Mechanistic Investigation of the Time-Dependent Aldehyde Oxidase Inhibitor Hydralazine
      J. Paige Barnes, Shaoyun M. Yang, Taylor S. Thompson, Caithlyne M. Guevarra, Shaniya S. Pleasant, Tri Q. Do and Rachel D. Crouch
      Drug Metabolism and Disposition June 2023, 51 (6) 782-791; DOI: https://doi.org/10.1124/dmd.123.001257

R

  1. Ren, Julie

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  2. Riddick, David S.

    1. You have access
      Fifty Years of Aryl Hydrocarbon Receptor Research as Reflected in the Pages of Drug Metabolism and Disposition
      David S. Riddick
      Drug Metabolism and Disposition June 2023, 51 (6) 657-671; DOI: https://doi.org/10.1124/dmd.122.001009
  3. Ruddock, Lloyd W.

    1. Open Access
      Inactivation of Human Aldehyde Oxidase by Small Sulfhydryl-Containing Reducing Agents
      Mariam Esmaeeli, Manfred Nimtz, Lothar Jänsch, Lloyd W. Ruddock and Silke Leimkühler
      Drug Metabolism and Disposition June 2023, 51 (6) 764-770; DOI: https://doi.org/10.1124/dmd.122.001244

S

  1. Saporito, Michael

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  2. Sato, Rei

    1. You have access
      Characterization of Enzymes Involved in Nintedanib Metabolism in Humans
      Shimon Nakashima, Rei Sato, Tatsuki Fukami, Takashi Kudo, Shiori Hashiba, Gaku Morinaga, Masataka Nakano, Eva Ludwig-Schwellinger, Akiko Matsui, Naoki Ishiguro, Thomas Ebner and Miki Nakajima
      Drug Metabolism and Disposition June 2023, 51 (6) 733-742; DOI: https://doi.org/10.1124/dmd.122.001113
  3. Seo, Shirley K.

    1. You have access
      Combined Oral Contraceptives As Victims of Drug Interactions
      Li Li, Xinning Yang, Doanh Tran, Shirley K. Seo and Yanhui Lu
      Drug Metabolism and Disposition June 2023, 51 (6) 718-732; DOI: https://doi.org/10.1124/dmd.122.000854
  4. Smith, Steven

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  5. Spracklin, Douglas K.

    1. You have access
      Human Absorption, Distribution, Metabolism, and Excretion Studies: Origins, Innovations, and Importance
      Matthew A. Cerny, Douglas K. Spracklin and R. Scott Obach
      Drug Metabolism and Disposition June 2023, 51 (6) 647-656; DOI: https://doi.org/10.1124/dmd.122.001006
  6. Sun, Shanliang

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245

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  1. Thompson, Taylor S.

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      Mechanistic Investigation of the Time-Dependent Aldehyde Oxidase Inhibitor Hydralazine
      J. Paige Barnes, Shaoyun M. Yang, Taylor S. Thompson, Caithlyne M. Guevarra, Shaniya S. Pleasant, Tri Q. Do and Rachel D. Crouch
      Drug Metabolism and Disposition June 2023, 51 (6) 782-791; DOI: https://doi.org/10.1124/dmd.123.001257
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      Combined Oral Contraceptives As Victims of Drug Interactions
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      Drug Metabolism and Disposition June 2023, 51 (6) 718-732; DOI: https://doi.org/10.1124/dmd.122.000854

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  1. Unadkat, Jashvant D.

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      Drug Metabolism and Disposition June 2023, 51 (6) 743-752; DOI: https://doi.org/10.1124/dmd.122.001128

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  1. Yabut, King Clyde B.

    1. Open Access
      Impact of Intracellular Lipid Binding Proteins on Endogenous and Xenobiotic Ligand Metabolism and Disposition
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      Drug Metabolism and Disposition June 2023, 51 (6) 700-717; DOI: https://doi.org/10.1124/dmd.122.001010
  2. Yang, Shaoyun M.

    1. You have access
      Mechanistic Investigation of the Time-Dependent Aldehyde Oxidase Inhibitor Hydralazine
      J. Paige Barnes, Shaoyun M. Yang, Taylor S. Thompson, Caithlyne M. Guevarra, Shaniya S. Pleasant, Tri Q. Do and Rachel D. Crouch
      Drug Metabolism and Disposition June 2023, 51 (6) 782-791; DOI: https://doi.org/10.1124/dmd.123.001257
  3. Yang, Xinning

    1. You have access
      Combined Oral Contraceptives As Victims of Drug Interactions
      Li Li, Xinning Yang, Doanh Tran, Shirley K. Seo and Yanhui Lu
      Drug Metabolism and Disposition June 2023, 51 (6) 718-732; DOI: https://doi.org/10.1124/dmd.122.000854
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    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
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      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
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      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
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  6. Yu, Ai-Ming

    1. Open Access
      Recombinant Technologies Facilitate Drug Metabolism, Pharmacokinetics, and General Biomedical Research
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  1. Zhang, Chenmeng

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  2. Zhang, Mingbao

    1. Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      You have access
      Complex Metabolism of the Novel Neurosteroid, Ganaxolone, in Humans: A Unique Challenge for Metabolites in Safety Testing Assessment
      William L. Fitch, Steven Smith, Michael Saporito, Gregory Busse, Mingbao Zhang, Julie Ren, Michael E. Fitzsimmons, Ping Yi, Stephen English, Adam Carter and Thomas A. Baillie
      Drug Metabolism and Disposition June 2023, 51 (6) 753-763; DOI: https://doi.org/10.1124/dmd.122.001218
  3. Zhang, Yongjie

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  4. Zhao, Yulin

    1. Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      You have access
      Mechanistic Study of Icaritin-Induced Inactivation of Cytochrome P450 2C9
      Xiang Chen, Luyao Han, Yulin Zhao, Haoyan Huang, He Pan, Chenmeng Zhang, Huili Chen, Shanliang Sun, Sihui Yao, Xijing Chen and Yongjie Zhang
      Drug Metabolism and Disposition June 2023, 51 (6) 771-781; DOI: https://doi.org/10.1124/dmd.122.001245
  5. Zhong, Xiao-bo

    1. Epigenetic Mechanisms Contribute to Intraindividual Variations of Drug Metabolism Mediated by Cytochrome P450 Enzymes
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      Epigenetic Mechanisms Contribute to Intraindividual Variations of Drug Metabolism Mediated by Cytochrome P450 Enzymes
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      Drug Metabolism and Disposition June 2023, 51 (6) 672-684; DOI: https://doi.org/10.1124/dmd.122.001007
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Drug Metabolism and Disposition: 51 (6)
Drug Metabolism and Disposition
Vol. 51, Issue 6
1 Jun 2023
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  • Cytochrome P450 inhibitors. Evaluation of specificities in the in vitrometabolism of therapeutic agents by human liver microsomes.
  • Prediction of Human Clearance of Twenty-Nine Drugs from Hepatic Microsomal Intrinsic Clearance Data: An Examination of In Vitro Half-Life Approach and Nonspecific Binding to Microsomes
  • DRUG-DRUG INTERACTIONS FOR UDP-GLUCURONOSYLTRANSFERASE SUBSTRATES: A PHARMACOKINETIC EXPLANATION FOR TYPICALLY OBSERVED LOW EXPOSURE (AUCI/AUC) RATIOS
  • In Vitro-In Vivo Scaling of CYP Kinetic Data Not Consistent with the Classical Michaelis-Menten Model
  • THE HUMAN INTESTINAL CYTOCHROME P450 “PIE”
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