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Role of epoxide hydrolases and cytochrome P450s on metabolism of KZR-616, a first-in-class selective inhibitor of the immunoproteasome
Ying Fang, Henry Johnson, Janet L. Anderl, Tony Muchamuel, Dustin McMinn, Christophe Morisseau, Bruce D. Hammock, Christopher Kirk and Jinhai Wang
Drug Metabolism and Disposition July 7, 2021, DMD-AR-2020-000307; DOI: https://doi.org/10.1124/dmd.120.000307
Ying Fang
1Kezar Life Sciences, United States
Henry Johnson
1Kezar Life Sciences, United States
Janet L. Anderl
1Kezar Life Sciences, United States
Tony Muchamuel
1Kezar Life Sciences, United States
Dustin McMinn
1Kezar Life Sciences, United States
Christophe Morisseau
2Entomology, UC Davis, United States
Bruce D. Hammock
3Department of Entomology, University of California - Davis, United States
Christopher Kirk
1Kezar Life Sciences, United States
Jinhai Wang
1Kezar Life Sciences, United States

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In this issue
Drug Metabolism and Disposition
Vol. 50, Issue 5
1 May 2022
OtherArticle
Microsomal epoxide hydrolase on metabolism of KZR-616
Ying Fang, Henry Johnson, Janet L. Anderl, Tony Muchamuel, Dustin McMinn, Christophe Morisseau, Bruce D. Hammock, Christopher Kirk and Jinhai Wang
Drug Metabolism and Disposition July 7, 2021, DMD-AR-2020-000307; DOI: https://doi.org/10.1124/dmd.120.000307
OtherArticle
Microsomal epoxide hydrolase on metabolism of KZR-616
Ying Fang, Henry Johnson, Janet L. Anderl, Tony Muchamuel, Dustin McMinn, Christophe Morisseau, Bruce D. Hammock, Christopher Kirk and Jinhai Wang
Drug Metabolism and Disposition July 7, 2021, DMD-AR-2020-000307; DOI: https://doi.org/10.1124/dmd.120.000307
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